4H5D | 2.02 | HOMO SAPIENS | ENZYME 2.5.1.10 | YS4, POP, MG | Kd = 0.58 uM | 402.276, 175.959, 24.305 |
4H5E | 2.04 | HOMO SAPIENS | ENZYME 2.5.1.10 | YS4, MG, IPR | Kd = 0.86 uM | 402.276, 24.305, 248.108 |
4LFV | 2 | HOMO SAPIENS | ENZYME 2.5.1.10 | YS4, CL, PO4, MG | | 402.276, 35.453, 94.971, 24.305 |
4P0V | 2.4 | HOMO SAPIENS | ENZYME 2.5.1.10 | 1WO, ZOL, MG | | 314.419, 272.09, 24.305 |
4P0W | 2.41 | HOMO SAPIENS | ENZYME 2.5.1.10 | ZOL, MG, 1XH | | 272.09, 24.305, 312.446 |
4RXC | 2.31 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | HRX, MG | ic50 ~ 33 uM | 297.139, 24.305 |
4RXD | 2 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | RIS, MG | ic50 = 300 nM | 283.112, 24.305 |
4RXE | 2.5 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | 3YQ, MG | ic50 = 230 nM | 282.128, 24.305 |
4UMJ | 1.85 | PSEUDOMONAS AERUGINOSA | ENZYME 2.5.1.10 | BFQ, MG | ic50 = 2.7 uM | 319.229, 24.305 |
5AFX | 2.39 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | PVZ, MG | ic50 = 1.2 uM | 399.337, 24.305 |
4DWB | 2.1 | TRYPANOSOMA CRUZI | ENZYME 2.5.1.10 | NA, 0M7, SO4, ACT, IPE, MG | ic50 = 1840 nM | 22.99, 275.176, 96.063, 59.044, 246.092, 24.305 |
4DWG | 2.01 | TRYPANOSOMA CRUZI | ENZYME 2.5.1.10 | NA, PEG, ACT, MG, 0M8, SO4 | ic50 = 58 nM | 22.99, 106.12, 59.044, 24.305, 303.23, 96.063 |