Receptor
PDB id Resolution Class Description Source Keywords
5F6X 1.56 Å EC: 6.3.2.- CRYSTAL STRUCTURE OF UBC9 (K48/K49A/E54A) COMPLEXED WITH FRA (MERCAPTOBENZOXAZOLE FROM COCKTAIL SCREEN) HOMO SAPIENS UBC9 FRAGMENT DRUG DESIGN SUMOYLATION LIGASE-LIGASE INHIBCOMPLEX
Ref.: INSIGHTS INTO THE ALLOSTERIC INHIBITION OF THE SUMO ENZYME UBC9. ANGEW.CHEM.INT.ED.ENGL. V. 55 5703 2016
Ligand
Ligand Chain:Residue Validity Ligand Warnings Binding Data NGL Viewer Molecular Weight (Da) Formula SMILES
5VM A:201;
Valid;
none;
submit data
185.631 C7 H4 Cl N O S c1cc2...
View in 3D viewer
90% Homology Family
Leader
PDB id Resolution Class Description Source Keywords
5F6U 1.55 Å EC: 6.3.2.- CRYSTAL STRUCTURE OF UBC9 (K48A/K49A/E54A) COMPLEXED WITH FR (JSS190B146) HOMO SAPIENS UBC9 SUMOYLATION DRUG DISCOVERY LIGASE-LIGASE INHIBITOR C
Ref.: INSIGHTS INTO THE ALLOSTERIC INHIBITION OF THE SUMO ENZYME UBC9. ANGEW.CHEM.INT.ED.ENGL. V. 55 5703 2016
Members (6)
No: PDB id Binding Data Representative ligand Formula Smiles
The Class containing this family consists of a total of 41 families.
1 5F6W ic50 = 5.8 mM 5VL C12 H10 O2 c1ccc(c(c1....
2 5F6X - 5VM C7 H4 Cl N O S c1cc2c(cc1....
3 5F6D - 5VJ C12 H9 N O2 S c1ccc2c(c1....
4 5F6V ic50 = 5.8 mM 5VL C12 H10 O2 c1ccc(c(c1....
5 5F6Y - 5VM C7 H4 Cl N O S c1cc2c(cc1....
6 5F6U ic50 = 3 mM 5VK C17 H18 O4 CCOC(=O)CC....
70% Homology Family (6)
No: PDB id Binding Data Representative ligand Formula Smiles
The Class containing this family consists of a total of 27 families.
1 5F6W ic50 = 5.8 mM 5VL C12 H10 O2 c1ccc(c(c1....
2 5F6X - 5VM C7 H4 Cl N O S c1cc2c(cc1....
3 5F6D - 5VJ C12 H9 N O2 S c1ccc2c(c1....
4 5F6V ic50 = 5.8 mM 5VL C12 H10 O2 c1ccc(c(c1....
5 5F6Y - 5VM C7 H4 Cl N O S c1cc2c(cc1....
6 5F6U ic50 = 3 mM 5VK C17 H18 O4 CCOC(=O)CC....
50% Homology Family (6)
No: PDB id Binding Data Representative ligand Formula Smiles
The Class containing this family consists of a total of 21 families.
1 5F6W ic50 = 5.8 mM 5VL C12 H10 O2 c1ccc(c(c1....
2 5F6X - 5VM C7 H4 Cl N O S c1cc2c(cc1....
3 5F6D - 5VJ C12 H9 N O2 S c1ccc2c(c1....
4 5F6V ic50 = 5.8 mM 5VL C12 H10 O2 c1ccc(c(c1....
5 5F6Y - 5VM C7 H4 Cl N O S c1cc2c(cc1....
6 5F6U ic50 = 3 mM 5VK C17 H18 O4 CCOC(=O)CC....
Polypharmacology
Similar Ligands (2D)
Ligand no: 1; Ligand: 5VM; Similar ligands found: 3
No: Ligand ECFP6 Tc MDL keys Tc
1 5VM 1 1
2 CLW 0.511111 0.756098
3 P92 0.409091 0.888889
Similar Ligands (3D)
Ligand no: 1; Ligand: 5VM; Similar ligands found: 1160
No: Ligand Similarity coefficient
1 36R 1.0000
2 VGD 1.0000
3 1P8 0.9987
4 ES2 0.9976
5 ET2 0.9943
6 K2T 0.9909
7 FBB 0.9869
8 JA8 0.9867
9 H42 0.9762
10 5MI 0.9717
11 11S 0.9712
12 AX7 0.9705
13 XAZ 0.9699
14 CWJ 0.9692
15 J6W 0.9692
16 H4N 0.9689
17 BZX 0.9689
18 ES9 0.9686
19 F60 0.9684
20 5H1 0.9678
21 6AI 0.9675
22 FK1 0.9674
23 2K4 0.9673
24 14O 0.9673
25 5JL 0.9673
26 5MB 0.9672
27 2HQ 0.9669
28 2MI 0.9664
29 270 0.9658
30 4FS 0.9657
31 5JQ 0.9656
32 COU 0.9653
33 6RQ 0.9650
34 8NY 0.9648
35 MQN 0.9648
36 URC 0.9647
37 2AQ 0.9640
38 ES5 0.9638
39 03V 0.9635
40 B55 0.9634
41 75K 0.9632
42 94W 0.9626
43 ABV 0.9624
44 XQ0 0.9613
45 86J 0.9612
46 OCH 0.9611
47 0TU 0.9607
48 9R5 0.9605
49 SYV 0.9596
50 BTY 0.9592
51 8TX 0.9592
52 IV2 0.9588
53 4JQ 0.9573
54 BZ3 0.9559
55 NPO 0.9557
56 4YO 0.9556
57 1M2 0.9555
58 PHB 0.9553
59 5WV 0.9550
60 8IG 0.9542
61 KJU 0.9541
62 5OB 0.9536
63 4FA 0.9534
64 XIY 0.9530
65 5XC 0.9529
66 8ZE 0.9516
67 F9Y 0.9508
68 HDH 0.9502
69 JB5 0.9490
70 7MU 0.9485
71 4HM 0.9482
72 HBD 0.9476
73 2BG 0.9474
74 HMH 0.9472
75 MS9 0.9470
76 3PF 0.9469
77 RM1 0.9468
78 JAE 0.9465
79 GLC 0.9464
80 MR1 0.9463
81 3ID 0.9461
82 DMD 0.9459
83 OTR 0.9457
84 5GU 0.9455
85 5QY 0.9455
86 QWN 0.9454
87 E7S 0.9452
88 Z82 0.9450
89 67N 0.9447
90 1P7 0.9443
91 G3E 0.9443
92 KDV 0.9442
93 PAB 0.9441
94 I3A 0.9441
95 7W4 0.9440
96 1Y6 0.9440
97 4M0 0.9438
98 ISN 0.9438
99 N2I 0.9435
100 HBA 0.9430
101 BHA 0.9429
102 TH7 0.9429
103 4XR 0.9428
104 1PT 0.9426
105 ODO 0.9424
106 DOB 0.9422
107 FA0 0.9420
108 XM0 0.9419
109 8H8 0.9414
110 Q88 0.9412
111 CWM 0.9410
112 FYU 0.9409
113 ES0 0.9399
114 5NU 0.9398
115 ES7 0.9397
116 3DM 0.9397
117 4BZ 0.9397
118 5CU 0.9396
119 KOJ 0.9394
120 174 0.9393
121 5B1 0.9393
122 DHR 0.9392
123 D48 0.9392
124 TTL 0.9392
125 YRL 0.9390
126 BGC 0.9389
127 M1A 0.9386
128 717 0.9385
129 9DG 0.9385
130 AHR 0.9385
131 QUZ 0.9384
132 4MA 0.9382
133 R8S 0.9381
134 QXW 0.9381
135 KKN 0.9380
136 826 0.9378
137 PBZ 0.9378
138 8WO 0.9374
139 P72 0.9372
140 2FY 0.9369
141 B62 0.9368
142 GUN 0.9367
143 J5I 0.9366
144 PNZ 0.9364
145 XYP 0.9363
146 4BY 0.9362
147 4VP 0.9360
148 E5X 0.9360
149 AZA 0.9359
150 NPY 0.9358
151 YH7 0.9357
152 7W1 0.9357
153 173 0.9356
154 CTL 0.9356
155 4JT 0.9350
156 0FO 0.9348
157 6M9 0.9347
158 7HQ 0.9345
159 AEF 0.9345
160 OTW 0.9342
161 PKU 0.9341
162 NOJ 0.9341
163 TGX 0.9340
164 6KT 0.9340
165 ZZT 0.9338
166 1DW 0.9338
167 SE2 0.9337
168 ANN 0.9337
169 ISZ 0.9336
170 DHB 0.9335
171 SKA 0.9333
172 BPN 0.9330
173 XAN 0.9329
174 J9Q 0.9329
175 4AA 0.9327
176 KUF 0.9327
177 1XM 0.9326
178 AC6 0.9326
179 DEN 0.9326
180 AZ8 0.9326
181 2EC 0.9322
182 2A9 0.9320
183 A7W 0.9320
184 HX3 0.9319
185 MEW 0.9319
186 XHP 0.9317
187 BZI 0.9317
188 NSP 0.9317
189 BZF 0.9317
190 3ZB 0.9316
191 A2F 0.9314
192 12Q 0.9312
193 MUA 0.9312
194 2D0 0.9311
195 0CT 0.9311
196 H8N 0.9311
197 0HO 0.9306
198 4JP 0.9306
199 0JD 0.9305
200 KJH 0.9303
201 0CU 0.9302
202 PZM 0.9302
203 M5K 0.9300
204 IND 0.9300
205 BCP 0.9299
206 IGA 0.9299
207 6NT 0.9299
208 6AP 0.9297
209 LZ1 0.9295
210 0RW 0.9294
211 TYL 0.9293
212 INO 0.9292
213 4TU 0.9291
214 UNJ 0.9291
215 BHO 0.9291
216 DQU 0.9290
217 AJ2 0.9290
218 Q24 0.9289
219 141 0.9289
220 HQT 0.9289
221 DX4 0.9287
222 A29 0.9286
223 BOA 0.9284
224 CWS 0.9283
225 4NC 0.9282
226 NIZ 0.9281
227 LXC 0.9280
228 4JM 0.9279
229 4CS 0.9279
230 AZG 0.9278
231 5QX 0.9278
232 XRG 0.9277
233 0R1 0.9274
234 4HC 0.9274
235 HMU 0.9273
236 SW7 0.9268
237 HH5 0.9267
238 0HN 0.9267
239 3NT 0.9267
240 3NY 0.9267
241 HIS 0.9267
242 3F0 0.9266
243 9FL 0.9266
244 DIN 0.9265
245 PXL 0.9264
246 44W 0.9263
247 1F1 0.9263
248 8GC 0.9263
249 EA1 0.9261
250 97T 0.9261
251 I1E 0.9260
252 MRW 0.9259
253 MPI 0.9259
254 42J 0.9258
255 EUG 0.9257
256 428 0.9257
257 GVH 0.9256
258 3HM 0.9256
259 4A3 0.9255
260 3HA 0.9254
261 WCE 0.9254
262 F81 0.9253
263 4BL 0.9253
264 AQO 0.9252
265 OAA 0.9252
266 24B 0.9252
267 15E 0.9251
268 P9P 0.9251
269 MVN 0.9250
270 9EW 0.9249
271 5NI 0.9249
272 4P5 0.9248
273 NNO 0.9247
274 JND 0.9247
275 PQ0 0.9246
276 F05 0.9246
277 3MB 0.9244
278 2AK 0.9244
279 2ZM 0.9243
280 FDB 0.9242
281 BEZ 0.9242
282 FHB 0.9241
283 0P6 0.9240
284 BZ2 0.9240
285 OVM 0.9239
286 PH2 0.9239
287 PE0 0.9238
288 93K 0.9238
289 2HU 0.9236
290 LDP 0.9235
291 GAB 0.9234
292 6NI 0.9233
293 TH0 0.9232
294 2CK 0.9230
295 XX2 0.9229
296 3M0 0.9228
297 QBK 0.9228
298 JAW 0.9226
299 GCS 0.9226
300 CFI 0.9225
301 5UC 0.9225
302 SOE 0.9225
303 TSS 0.9225
304 3HB 0.9224
305 BEN 0.9224
306 1MC 0.9223
307 HQJ 0.9222
308 5RN 0.9221
309 MSR 0.9220
310 JBK 0.9219
311 6ME 0.9219
312 FE DB1 0.9218
313 7B4 0.9216
314 3AB 0.9216
315 TDR 0.9215
316 PRF 0.9213
317 4WL 0.9212
318 BAM 0.9212
319 290 0.9211
320 LZM 0.9210
321 42A 0.9209
322 14J 0.9208
323 G3F 0.9208
324 PEA 0.9207
325 2HO 0.9206
326 F4E 0.9204
327 23A 0.9204
328 MYJ 0.9203
329 6M4 0.9203
330 DBH 0.9202
331 8CM 0.9202
332 NCA 0.9202
333 069 0.9201
334 3A9 0.9200
335 92K 0.9199
336 B57 0.9199
337 CFP 0.9198
338 JFJ 0.9196
339 C2B 0.9196
340 9CA 0.9195
341 5MH 0.9193
342 NMJ 0.9191
343 ICB 0.9189
344 HC4 0.9186
345 BCU 0.9184
346 5HN 0.9184
347 IDM 0.9183
348 OVV 0.9183
349 8WT 0.9182
350 44V 0.9182
351 6PC 0.9181
352 1SQ 0.9180
353 BRT 0.9179
354 4NM 0.9179
355 24W 0.9178
356 GTQ 0.9175
357 AZ9 0.9175
358 R8V 0.9173
359 5RO 0.9171
360 ABI 0.9170
361 R9Y 0.9170
362 5RG 0.9169
363 4JL 0.9167
364 FBM 0.9166
365 TZF 0.9165
366 5LA 0.9164
367 SNU 0.9162
368 5Q0 0.9161
369 82I 0.9161
370 MCT 0.9161
371 LT2 0.9160
372 ICP 0.9159
373 SN4 0.9158
374 NIO 0.9158
375 3QV 0.9157
376 XBT 0.9157
377 5SG 0.9156
378 4JU 0.9156
379 SHA 0.9153
380 4HO 0.9153
381 NBZ 0.9153
382 OW4 0.9152
383 B53 0.9152
384 URF 0.9151
385 6FZ 0.9151
386 5IQ 0.9150
387 J9T 0.9150
388 SVN 0.9150
389 53C 0.9150
390 YCP 0.9150
391 FBA 0.9148
392 2F6 0.9147
393 NTN 0.9144
394 1IT 0.9143
395 1NP 0.9142
396 4YS 0.9140
397 SNO 0.9140
398 3BZ 0.9139
399 MLT 0.9139
400 54G 0.9138
401 261 0.9138
402 FQI 0.9137
403 JB8 0.9136
404 HQY 0.9135
405 4ZA 0.9134
406 WBU 0.9134
407 5M0 0.9133
408 FUD 0.9131
409 XBZ 0.9130
410 TPA 0.9129
411 3OC 0.9129
412 SX1 0.9128
413 DGJ 0.9128
414 259 0.9128
415 BEA 0.9128
416 I3E 0.9128
417 ADZ 0.9127
418 SAL 0.9127
419 NDH 0.9123
420 N5J 0.9122
421 IUR 0.9121
422 1LQ 0.9121
423 ESP 0.9121
424 GXY 0.9121
425 27Y 0.9121
426 JZ9 0.9120
427 ASO 0.9120
428 M4T 0.9120
429 GAL 0.9120
430 43M 0.9118
431 4MU 0.9118
432 ICO 0.9118
433 5MK 0.9117
434 HPA 0.9117
435 6GU 0.9115
436 K34 0.9113
437 JZ2 0.9113
438 CHB 0.9113
439 15N 0.9113
440 BE2 0.9111
441 QX2 0.9110
442 E7Z 0.9108
443 F31 0.9107
444 4ME 0.9107
445 RSF 0.9107
446 ES1 0.9106
447 4SV 0.9106
448 DRL 0.9104
449 MZG 0.9103
450 PHU 0.9102
451 VGL 0.9101
452 TSU 0.9101
453 F9P 0.9101
454 PIM 0.9101
455 7VS 0.9100
456 MO8 0.9099
457 NAG 0.9099
458 JDN 0.9098
459 QWW 0.9098
460 AC0 0.9098
461 PZA 0.9098
462 BSX 0.9097
463 P3K 0.9097
464 6CS 0.9096
465 PYD 0.9095
466 8S0 0.9095
467 2MH 0.9094
468 4JO 0.9093
469 JPZ 0.9092
470 BR9 0.9092
471 K97 0.9091
472 AMH 0.9090
473 CH9 0.9090
474 1KP 0.9089
475 E1T 0.9089
476 XYD 0.9088
477 HLR 0.9087
478 4CL 0.9087
479 4Z4 0.9086
480 4JJ 0.9086
481 MWM 0.9086
482 6VD 0.9086
483 IWT 0.9084
484 9TW 0.9084
485 2AL 0.9084
486 3XX 0.9083
487 GZL 0.9083
488 CLZ 0.9082
489 DE5 0.9081
490 OK7 0.9081
491 4NB 0.9081
492 SAN 0.9081
493 92P 0.9080
494 IPB 0.9080
495 N8Y 0.9080
496 HQD 0.9077
497 XQG 0.9076
498 RSO 0.9075
499 KT7 0.9074
500 ZBT 0.9074
501 34A 0.9073
502 ADE 0.9073
503 4ZE 0.9071
504 FDR 0.9071
505 C2Y 0.9070
506 IDH 0.9070
507 JLZ 0.9069
508 GOJ 0.9068
509 FPY 0.9068
510 3Z8 0.9067
511 52C 0.9067
512 CPZ 0.9066
513 PZI 0.9065
514 M1Q 0.9064
515 2AC 0.9063
516 MWJ 0.9063
517 UNU 0.9061
518 TT4 0.9060
519 A1U 0.9059
520 LG4 0.9059
521 2MP 0.9057
522 PBC 0.9055
523 NK 0.9053
524 9MG 0.9053
525 GVG 0.9051
526 IHB 0.9050
527 0N7 0.9049
528 10L 0.9048
529 8W9 0.9048
530 SLS 0.9048
531 8NX 0.9044
532 PXY 0.9044
533 SS1 0.9043
534 FCR 0.9042
535 DVQ 0.9042
536 0FN 0.9040
537 HHA 0.9040
538 3U4 0.9039
539 FAN 0.9037
540 5JC 0.9037
541 VNL 0.9037
542 8OZ 0.9037
543 FP1 0.9037
544 EV0 0.9035
545 FUL 0.9034
546 INE 0.9033
547 AMC 0.9033
548 AKG 0.9032
549 XYS 0.9032
550 6MP 0.9030
551 9TZ 0.9030
552 ES6 0.9029
553 2H5 0.9029
554 OVP 0.9028
555 A7H 0.9025
556 L5V 0.9025
557 NOY 0.9025
558 25R 0.9023
559 H33 0.9022
560 G5V 0.9021
561 9ZE 0.9020
562 PCR 0.9020
563 IFL 0.9020
564 PIY 0.9020
565 12T 0.9019
566 HQE 0.9019
567 BE7 0.9018
568 0W8 0.9018
569 L99 0.9016
570 2CQ 0.9016
571 6TZ 0.9016
572 JBE 0.9014
573 VK3 0.9012
574 IF7 0.9011
575 2YU 0.9011
576 4J8 0.9011
577 IFP 0.9010
578 QSB 0.9008
579 4VY 0.9007
580 9DA 0.9005
581 NQ 0.9003
582 FPI 0.9003
583 4XH 0.9001
584 GLA 0.9001
585 DHK 0.9001
586 HH8 0.8999
587 SWA 0.8998
588 RHU 0.8996
589 RD4 0.8995
590 209 0.8995
591 BML 0.8995
592 BDP 0.8995
593 ESX 0.8994
594 DFB 0.8994
595 O72 0.8993
596 JBH 0.8993
597 2FQ 0.8991
598 RNO 0.8990
599 GDE 0.8990
600 4ZC 0.8989
601 RIP 0.8988
602 DA1 0.8987
603 EKZ 0.8987
604 PLQ 0.8986
605 7HP 0.8985
606 K22 0.8984
607 PBA 0.8983
608 PDC 0.8983
609 DBX 0.8982
610 4HS 0.8981
611 1LM 0.8980
612 JZ3 0.8980
613 1P3 0.8980
614 G6D 0.8980
615 KJY 0.8979
616 C1M 0.8977
617 1WG 0.8977
618 39O 0.8975
619 FPN 0.8975
620 9HX 0.8973
621 TLD 0.8973
622 KTJ 0.8971
623 BP1 0.8970
624 AJV 0.8968
625 AGK 0.8968
626 0MK 0.8968
627 FA1 0.8968
628 DIE 0.8967
629 DNF 0.8965
630 TM7 0.8965
631 QX4 0.8965
632 DYA 0.8965
633 GJP 0.8964
634 M1E 0.8964
635 G2F 0.8964
636 SRO 0.8964
637 M2K 0.8963
638 AAS 0.8963
639 4JN 0.8961
640 149 0.8961
641 GCU 0.8961
642 GIF 0.8960
643 BTE 0.8959
644 OW7 0.8958
645 SKM 0.8958
646 PM6 0.8957
647 37T 0.8955
648 7WA 0.8953
649 0R0 0.8953
650 J1Z 0.8952
651 F0J 0.8951
652 AN3 0.8951
653 150 0.8951
654 HT4 0.8951
655 4CH 0.8951
656 HHR 0.8950
657 V55 0.8950
658 RXA 0.8948
659 51R 0.8948
660 1DV 0.8945
661 PEY 0.8945
662 HLZ 0.8944
663 K32 0.8943
664 EN1 0.8943
665 FUC 0.8942
666 JKE 0.8940
667 0F9 0.8940
668 NID 0.8939
669 XYL 0.8936
670 RB5 0.8936
671 LQ2 0.8936
672 7WG 0.8935
673 MNM 0.8935
674 4RU 0.8933
675 X0V 0.8932
676 GIV 0.8931
677 SWD 0.8928
678 42C 0.8927
679 OHG 0.8927
680 EUE 0.8925
681 HBX 0.8924
682 GAF 0.8923
683 JG8 0.8922
684 A7N 0.8921
685 ES4 0.8920
686 8NB 0.8920
687 IOL 0.8920
688 3FH 0.8919
689 P9E 0.8919
690 1HN 0.8918
691 DIU 0.8917
692 SRT 0.8915
693 DFU 0.8913
694 TWO 0.8913
695 PAC 0.8912
696 1WD 0.8911
697 MBG 0.8911
698 QSC 0.8910
699 PCA 0.8908
700 282 0.8906
701 MAE 0.8905
702 S76 0.8904
703 2KA 0.8903
704 RBL 0.8903
705 LNR 0.8902
706 AX3 0.8902
707 B60 0.8901
708 PD2 0.8900
709 7NI 0.8900
710 TTY 0.8900
711 GRE 0.8899
712 NCT 0.8897
713 JTH 0.8897
714 X6X 0.8896
715 ESI 0.8895
716 1GN 0.8895
717 PRZ 0.8894
718 4XS 0.8893
719 20J 0.8893
720 PRO 0.8892
721 TIU 0.8891
722 7WV 0.8891
723 ASC 0.8890
724 X0U 0.8890
725 3R6 0.8890
726 CTS 0.8888
727 MWP 0.8888
728 Q6T 0.8887
729 2LP 0.8886
730 4XV 0.8885
731 275 0.8884
732 27B 0.8884
733 ZYR 0.8883
734 45C 0.8882
735 SYN 0.8882
736 TEP 0.8880
737 A5E 0.8880
738 MPV 0.8880
739 4I8 0.8879
740 GYE 0.8879
741 GF4 0.8879
742 KIB 0.8878
743 IT2 0.8877
744 Y8I 0.8876
745 GXL 0.8875
746 EQT 0.8874
747 MAQ 0.8874
748 7ME 0.8873
749 HX4 0.8872
750 IAC 0.8872
751 7VP 0.8870
752 KBZ 0.8870
753 FGZ 0.8869
754 FBS 0.8868
755 F4Z 0.8867
756 J9N 0.8867
757 PY7 0.8867
758 PYQ 0.8866
759 ZXD 0.8866
760 36E 0.8866
761 LPK 0.8865
762 PYF 0.8865
763 BNL 0.8865
764 3DO 0.8864
765 FOA 0.8864
766 ABN 0.8864
767 ARB 0.8864
768 25W 0.8864
769 M58 0.8862
770 3R4 0.8861
771 PQK 0.8861
772 SR1 0.8860
773 0BP 0.8860
774 J9W 0.8859
775 OXC 0.8859
776 PXM 0.8859
777 N3W 0.8859
778 TC7 0.8856
779 NBE 0.8855
780 LCN 0.8855
781 AJY 0.8854
782 6F0 0.8854
783 KYA 0.8854
784 S0E 0.8854
785 LYL 0.8853
786 TYR 0.8853
787 RIB 0.8851
788 1A7 0.8850
789 LMR 0.8850
790 3WA 0.8850
791 0TR 0.8849
792 OXQ 0.8849
793 LDU 0.8849
794 FRU 0.8849
795 RMN 0.8849
796 GO2 0.8849
797 Z5P 0.8848
798 7CZ 0.8848
799 K17 0.8848
800 CRS 0.8848
801 APZ 0.8845
802 2BX 0.8844
803 AMS 0.8843
804 R20 0.8843
805 2FG 0.8842
806 CXF 0.8842
807 VOH 0.8841
808 2GS 0.8840
809 DHQ 0.8840
810 HSO 0.8839
811 HA5 0.8839
812 4JC 0.8839
813 JBZ 0.8838
814 YPN 0.8838
815 6M1 0.8837
816 HIO 0.8836
817 M4E 0.8836
818 SHG 0.8835
819 8XL 0.8834
820 X0W 0.8833
821 D07 0.8832
822 2ZV 0.8831
823 M6N 0.8831
824 TP5 0.8831
825 WOT 0.8830
826 H4E 0.8830
827 FCA 0.8830
828 PYC 0.8830
829 36Y 0.8828
830 GBD 0.8827
831 LGC 0.8827
832 268 0.8825
833 XUL 0.8824
834 39A 0.8823
835 32X 0.8822
836 2HC 0.8822
837 MAN 0.8820
838 DBJ 0.8820
839 9FE 0.8820
840 GLL 0.8820
841 DEE 0.8820
842 C2U 0.8819
843 CIT 0.8819
844 DRG 0.8818
845 K82 0.8817
846 PHE 0.8815
847 NDG 0.8815
848 TLA 0.8814
849 GAG 0.8812
850 JIF 0.8812
851 VNJ 0.8812
852 FDK 0.8812
853 GWM 0.8811
854 1XN 0.8809
855 3V4 0.8807
856 AEH 0.8806
857 SJ5 0.8806
858 NDM 0.8804
859 3BU 0.8803
860 X05 0.8800
861 T6C 0.8800
862 2K8 0.8800
863 MZW 0.8799
864 G4D 0.8798
865 M4S 0.8798
866 EYK 0.8796
867 344 0.8796
868 BDF 0.8795
869 4FH 0.8794
870 1DU 0.8794
871 BPY 0.8794
872 2PC 0.8793
873 8G0 0.8792
874 JU2 0.8790
875 B5D 0.8790
876 ORO 0.8790
877 45L 0.8790
878 L14 0.8790
879 AKH 0.8788
880 AL0 0.8788
881 3SK 0.8784
882 W81 0.8782
883 PJW 0.8781
884 UEG 0.8781
885 XLS 0.8780
886 AA 0.8780
887 60P 0.8779
888 L22 0.8779
889 QSH 0.8779
890 JBQ 0.8777
891 9KT 0.8777
892 DOR 0.8777
893 GIO 0.8777
894 MT0 0.8776
895 QPR 0.8775
896 SOR 0.8775
897 4V2 0.8773
898 FBW 0.8773
899 258 0.8772
900 PYG 0.8772
901 3Z7 0.8772
902 3IT 0.8772
903 FH2 0.8771
904 PEL 0.8771
905 CN0 0.8771
906 MAJ 0.8771
907 M6W 0.8770
908 7MX 0.8768
909 PFL 0.8767
910 JFD 0.8766
911 M0W 0.8766
912 0FK 0.8765
913 OGA 0.8764
914 RCO 0.8763
915 HHS 0.8762
916 FOT 0.8761
917 4SX 0.8760
918 JAB 0.8758
919 P4B 0.8758
920 UNC 0.8757
921 WOO 0.8757
922 F4K 0.8757
923 5WY 0.8754
924 K5W 0.8753
925 M2H 0.8753
926 KTW 0.8753
927 VXX 0.8752
928 UAN 0.8752
929 ABE 0.8752
930 DTU 0.8752
931 M3H 0.8751
932 ALL 0.8751
933 PFB 0.8751
934 1MR 0.8750
935 HHH 0.8750
936 BP9 0.8748
937 JXN 0.8748
938 C21 0.8748
939 7ZE 0.8747
940 2ZQ 0.8747
941 K37 0.8747
942 5WX 0.8747
943 C2A 0.8747
944 RNS 0.8744
945 HJP 0.8744
946 LKA 0.8743
947 BPU 0.8742
948 ADK 0.8742
949 R8A 0.8742
950 HY3 0.8741
951 HZQ 0.8740
952 JZ5 0.8740
953 TZC 0.8740
954 F5B 0.8739
955 3CH 0.8739
956 HGQ 0.8739
957 JYB 0.8739
958 URP 0.8737
959 FHC 0.8737
960 L3Q 0.8736
961 QIV 0.8736
962 Q71 0.8735
963 495 0.8733
964 7B3 0.8733
965 36M 0.8732
966 265 0.8731
967 1SA 0.8731
968 DMJ 0.8730
969 OXZ 0.8729
970 XCZ 0.8728
971 M0Q 0.8728
972 DHS 0.8727
973 RAM 0.8726
974 0W1 0.8725
975 7MH 0.8724
976 SMV 0.8724
977 4M4 0.8723
978 TOF 0.8722
979 7N0 0.8722
980 68A 0.8720
981 7O4 0.8719
982 BNF 0.8718
983 GNM 0.8718
984 5TY 0.8717
985 ADA 0.8717
986 TAR 0.8716
987 GOO 0.8716
988 TBS 0.8715
989 ANF 0.8714
990 PRA 0.8712
991 1L5 0.8712
992 IFM 0.8711
993 EMZ 0.8710
994 Y3L 0.8710
995 ONR 0.8708
996 23W 0.8708
997 AZF 0.8707
998 M1H 0.8706
999 BBK 0.8706
1000 CXH 0.8704
1001 HSM 0.8704
1002 LI6 0.8703
1003 PPY 0.8703
1004 9X7 0.8703
1005 FBJ 0.8701
1006 NGO 0.8701
1007 HA7 0.8701
1008 8HC 0.8699
1009 CYT 0.8699
1010 293 0.8699
1011 LG3 0.8698
1012 LG5 0.8698
1013 N4E 0.8698
1014 V1T 0.8696
1015 AEG 0.8692
1016 CFF 0.8692
1017 D1X 0.8692
1018 286 0.8690
1019 XXR 0.8690
1020 2QC 0.8688
1021 ZZ3 0.8686
1022 URA 0.8684
1023 GMN 0.8684
1024 SXS 0.8683
1025 EXO 0.8683
1026 DS0 0.8682
1027 549 0.8681
1028 JBN 0.8680
1029 FB2 0.8678
1030 3MC 0.8677
1031 BVF 0.8676
1032 3VX 0.8675
1033 HEW 0.8674
1034 3SL 0.8672
1035 AW5 0.8670
1036 3MG 0.8666
1037 IJZ 0.8664
1038 MBD 0.8663
1039 R2B 0.8662
1040 QMP 0.8661
1041 M45 0.8661
1042 FBV 0.8660
1043 OA3 0.8660
1044 NGT 0.8660
1045 8K2 0.8659
1046 PA1 0.8658
1047 EXD 0.8658
1048 GLO 0.8657
1049 QOS 0.8656
1050 H76 0.8656
1051 OMD 0.8656
1052 FB1 0.8656
1053 6MH 0.8655
1054 Q02 0.8654
1055 THA 0.8654
1056 K8X 0.8653
1057 ZB1 0.8652
1058 1Z6 0.8650
1059 QY9 0.8650
1060 OKG 0.8649
1061 TBP 0.8648
1062 6FB 0.8647
1063 F12 0.8647
1064 26D 0.8647
1065 HHI 0.8643
1066 RA7 0.8643
1067 680 0.8643
1068 MAK 0.8642
1069 3CE 0.8641
1070 GJZ 0.8641
1071 3AE 0.8641
1072 B2J 0.8641
1073 TM4 0.8640
1074 PRY 0.8640
1075 X09 0.8640
1076 ZEC 0.8640
1077 95Z 0.8639
1078 FUF 0.8638
1079 NSG 0.8638
1080 DA4 0.8637
1081 PMB 0.8637
1082 MEV 0.8636
1083 N91 0.8635
1084 HYP 0.8633
1085 S7J 0.8631
1086 RAT 0.8631
1087 FBF 0.8631
1088 KYD 0.8630
1089 QIC 0.8630
1090 A13 0.8630
1091 JP2 0.8628
1092 M3T 0.8628
1093 ASN 0.8628
1094 2FT 0.8627
1095 P80 0.8626
1096 1DQ 0.8625
1097 3FA 0.8624
1098 EVF 0.8622
1099 PO6 0.8620
1100 HBO 0.8620
1101 363 0.8620
1102 4H2 0.8618
1103 G12 0.8618
1104 KBB 0.8615
1105 8GF 0.8614
1106 2MY 0.8611
1107 7VJ 0.8611
1108 DNA 0.8610
1109 2C9 0.8610
1110 6QF 0.8609
1111 B3R 0.8608
1112 UFV 0.8608
1113 FFP 0.8606
1114 12B 0.8605
1115 SMN 0.8603
1116 TAG 0.8602
1117 7MW 0.8602
1118 CIG 0.8601
1119 LSA 0.8597
1120 3MA 0.8596
1121 9RW 0.8593
1122 UY7 0.8592
1123 TMZ 0.8591
1124 47J 0.8590
1125 FLM 0.8590
1126 PHH 0.8590
1127 LR5 0.8586
1128 H5B 0.8585
1129 2CM 0.8584
1130 35C 0.8584
1131 SD4 0.8579
1132 SS2 0.8579
1133 GVY 0.8578
1134 URS 0.8577
1135 F1A 0.8576
1136 GLT 0.8573
1137 ZZZ 0.8572
1138 TXW 0.8569
1139 P84 0.8568
1140 HXX 0.8568
1141 H3M 0.8565
1142 HHQ 0.8565
1143 DUB 0.8563
1144 K6X 0.8563
1145 F2W 0.8559
1146 091 0.8552
1147 BNS 0.8550
1148 BZJ 0.8548
1149 QAT 0.8546
1150 94N 0.8545
1151 BEW 0.8538
1152 GLU 0.8537
1153 N0Z 0.8536
1154 CKA 0.8532
1155 T9G 0.8530
1156 492 0.8530
1157 GJS 0.8525
1158 0XT 0.8524
1159 ORN 0.8520
1160 3MH 0.8517
Similar Binding Sites (Proteins are less than 50% similar to leader)
Pocket No.: 1; Query (leader) PDB : 5F6U; Ligand: 5VK; Similar sites found with APoc: No similar binding sites found, or similarity not calculated due to duplicate pocket.
This union binding pocket(no: 1) in the query (biounit: 5f6u.bio1) has 10 residues
No: Leader PDB Ligand Sequence Similarity
APoc FAQ
Feedback