Receptor
PDB id Resolution Class Description Source Keywords
4a6w 1.46 Å EC: 3.4.11.18 X-RAY STRUCTURES OF OXAZOLE HYDROXAMATE ECMETAP-MN COMPLEXES ESCHERICHIA COLI TRANSFERASE
Ref.: HYDROXAMIC ACIDS AS POTENT INHIBITORS OF FE(II) AND E. COLI METHIONINE AMINOPEPTIDASE: BIOLOGICAL ACTIV AND X-RAY STRUCTURES OF OXAZOLE HYDROXAMATE-ECMETAP COMPLEXES. CHEMMEDCHEM V. 7 1020 2012
Ligand
Ligand Chain:Residue Validity Ligand Warnings Binding Data NGL Viewer Molecular Weight (Da) Formula SMILES
5C1 A:1265;
Valid;
none;
ic50 = 1.9 uM
238.627 C10 H7 Cl N2 O3 c1ccc...
MN A:1264;
A:1266;
Part of Protein;
Part of Protein;
none;
none;
submit data
54.938 Mn [Mn+2...
View in 3D viewer
90% Homology Family
Leader
PDB id Resolution Class Description Source Keywords
1YVM 1.6 Å EC: 3.4.11.18 E. COLI METHIONINE AMINOPEPTIDASE IN COMPLEX WITH THIABENDAZOLE ESCHERICHIA COLI HYDROLASE(ALPHA-AMINOACYLPEPTIDE) METAL COMPLEX THIABENDAZOLE METHIONINE AMINOPEPTIDASE INHIBITOR
Ref.: METAL IONS AS COFACTORS FOR THE BINDING OF INHIBITORS TO METHIONINE AMINOPEPTIDASE: A CRITICAL VIEW OF THE RELEVANCE OF IN VITRO METALLOENZYME ASSAYS. ANGEW.CHEM.INT.ED.ENGL. V. 44 3620 2005
Members (36)
No: PDB id Binding Data Representative ligand Formula Smiles
The Class containing this family consists of a total of 8 families.
1 2GG0 ic50 = 1.7 uM U11 C16 H20 F3 N3 O5 C[C@@H](C(....
2 1YVM Ki = 0.4 uM TMG C10 H7 N3 S c1ccc2c(c1....
3 2GU6 - NLP C5 H14 N O3 P CCCC[C@H](....
4 2Q95 ic50 = 1.6 uM A05 C11 H6 Cl N O5 c1cc(c(cc1....
5 2GG8 ic50 = 25 uM U15 C20 H31 N3 O5 Cc1ccc(cc1....
6 2GTX - NLP C5 H14 N O3 P CCCC[C@H](....
7 2EVC ic50 = 0.29 uM FC3 C12 H7 F3 O3 c1ccc(c(c1....
8 4A6W ic50 = 1.9 uM 5C1 C10 H7 Cl N2 O3 c1ccc(c(c1....
9 2GG3 ic50 = 0.58 uM U13 C9 H7 F N6 [H]/N=C/1C....
10 3D27 ic50 = 55.7 uM W29 C12 H12 O2 S CCc1ccsc1c....
11 2GG7 ic50 = 1.75 uM U14 C10 H8 N6 O2 [H]/N=C1/C....
12 2GU5 - NLP C5 H14 N O3 P CCCC[C@H](....
13 1XNZ ic50 = 0.24 uM FCD C11 H7 Cl O3 c1ccc(c(c1....
14 4A6V ic50 = 1.9 uM IKY C11 H7 F3 N2 O3 c1ccc(c(c1....
15 1C21 - MET C5 H11 N O2 S CSCC[C@@H]....
16 2Q92 ic50 = 1.1 uM B23 C11 H7 N O5 c1ccc(c(c1....
17 1C27 - NLP C5 H14 N O3 P CCCC[C@H](....
18 1C24 - MPJ C4 H12 N O2 P S CSCC[C@H](....
19 2EVO ic50 = 0.067 uM CT0 C10 H13 N3 O2 S c1csc(n1)N....
20 2P99 ic50 = 1.16 uM YE6 C11 H9 Cl N2 O2 c1ccc(c(c1....
21 2GG9 ic50 = 3.5 uM U16 C22 H35 N3 O5 CC(C)C[C@H....
22 2Q94 ic50 = 0.37 uM A04 C12 H7 F3 O4 c1ccc(c(c1....
23 2P98 ic50 = 0.64 uM YE7 C12 H10 N4 O c1ccc2c(c1....
24 2GGB ic50 = 12 uM U17 C17 H33 N3 O6 CCCC[C@H](....
25 2EVM ic50 = 0.693 uM FC2 C11 H6 Cl2 O3 c1cc(c(cc1....
26 1C22 - MF3 C5 H8 F3 N O2 S C(CSC(F)(F....
27 1C23 - MPH C4 H12 N O3 P S CSCC[C@H](....
28 2Q96 ic50 = 1.2 uM A18 C12 H9 Cl O3 c1ccc(c(c1....
29 2BB7 ic50 = 2.14 uM QMS C10 H10 N2 O2 S CS(=O)(=O)....
30 2GG2 ic50 = 0.25 uM U12 C10 H7 F3 N6 c1cc(cc(c1....
31 2GGC - MET C5 H11 N O2 S CSCC[C@@H]....
32 2GU4 - NLP C5 H14 N O3 P CCCC[C@H](....
33 2Q93 ic50 = 0.56 uM B21 C12 H10 O4 COc1ccccc1....
34 2GG5 ic50 = 0.25 uM U19 C10 H7 F3 N6 [H]/N=C1/C....
35 3MAT - AHH ALA LEU VAL 0A9 n/a n/a
36 2P9A ic50 = 6.56 uM YE6 C11 H9 Cl N2 O2 c1ccc(c(c1....
70% Homology Family (36)
No: PDB id Binding Data Representative ligand Formula Smiles
The Class containing this family consists of a total of 6 families.
1 2GG0 ic50 = 1.7 uM U11 C16 H20 F3 N3 O5 C[C@@H](C(....
2 1YVM Ki = 0.4 uM TMG C10 H7 N3 S c1ccc2c(c1....
3 2GU6 - NLP C5 H14 N O3 P CCCC[C@H](....
4 2Q95 ic50 = 1.6 uM A05 C11 H6 Cl N O5 c1cc(c(cc1....
5 2GG8 ic50 = 25 uM U15 C20 H31 N3 O5 Cc1ccc(cc1....
6 2GTX - NLP C5 H14 N O3 P CCCC[C@H](....
7 2EVC ic50 = 0.29 uM FC3 C12 H7 F3 O3 c1ccc(c(c1....
8 4A6W ic50 = 1.9 uM 5C1 C10 H7 Cl N2 O3 c1ccc(c(c1....
9 2GG3 ic50 = 0.58 uM U13 C9 H7 F N6 [H]/N=C/1C....
10 3D27 ic50 = 55.7 uM W29 C12 H12 O2 S CCc1ccsc1c....
11 2GG7 ic50 = 1.75 uM U14 C10 H8 N6 O2 [H]/N=C1/C....
12 2GU5 - NLP C5 H14 N O3 P CCCC[C@H](....
13 1XNZ ic50 = 0.24 uM FCD C11 H7 Cl O3 c1ccc(c(c1....
14 4A6V ic50 = 1.9 uM IKY C11 H7 F3 N2 O3 c1ccc(c(c1....
15 1C21 - MET C5 H11 N O2 S CSCC[C@@H]....
16 2Q92 ic50 = 1.1 uM B23 C11 H7 N O5 c1ccc(c(c1....
17 1C27 - NLP C5 H14 N O3 P CCCC[C@H](....
18 1C24 - MPJ C4 H12 N O2 P S CSCC[C@H](....
19 2EVO ic50 = 0.067 uM CT0 C10 H13 N3 O2 S c1csc(n1)N....
20 2P99 ic50 = 1.16 uM YE6 C11 H9 Cl N2 O2 c1ccc(c(c1....
21 2GG9 ic50 = 3.5 uM U16 C22 H35 N3 O5 CC(C)C[C@H....
22 2Q94 ic50 = 0.37 uM A04 C12 H7 F3 O4 c1ccc(c(c1....
23 2P98 ic50 = 0.64 uM YE7 C12 H10 N4 O c1ccc2c(c1....
24 2GGB ic50 = 12 uM U17 C17 H33 N3 O6 CCCC[C@H](....
25 2EVM ic50 = 0.693 uM FC2 C11 H6 Cl2 O3 c1cc(c(cc1....
26 1C22 - MF3 C5 H8 F3 N O2 S C(CSC(F)(F....
27 1C23 - MPH C4 H12 N O3 P S CSCC[C@H](....
28 2Q96 ic50 = 1.2 uM A18 C12 H9 Cl O3 c1ccc(c(c1....
29 2BB7 ic50 = 2.14 uM QMS C10 H10 N2 O2 S CS(=O)(=O)....
30 2GG2 ic50 = 0.25 uM U12 C10 H7 F3 N6 c1cc(cc(c1....
31 2GGC - MET C5 H11 N O2 S CSCC[C@@H]....
32 2GU4 - NLP C5 H14 N O3 P CCCC[C@H](....
33 2Q93 ic50 = 0.56 uM B21 C12 H10 O4 COc1ccccc1....
34 2GG5 ic50 = 0.25 uM U19 C10 H7 F3 N6 [H]/N=C1/C....
35 3MAT - AHH ALA LEU VAL 0A9 n/a n/a
36 2P9A ic50 = 6.56 uM YE6 C11 H9 Cl N2 O2 c1ccc(c(c1....
50% Homology Family (69)
No: PDB id Binding Data Representative ligand Formula Smiles
The Class containing this family consists of a total of 3 families.
1 2NQ6 ic50 = 1.5 uM HM4 C14 H16 N4 O3 S CC(C)(C)OC....
2 4U69 Ki = 54.8 uM Q07 C6 H16 N O3 P CCC[C@H](C....
3 2G6P ic50 = 0.6 uM HM2 C18 H17 Cl N4 Cc1c(c(nc(....
4 4U73 Ki = 6.6 uM Q02 C7 H10 N O3 P c1ccc(cc1)....
5 4IKT ic50 = 0.67 uM TFV C18 H16 Cl F3 N6 Cc1c(c(nc(....
6 4U6Z Ki = 3.9 uM Q07 C6 H16 N O3 P CCC[C@H](C....
7 4U70 Ki = 9.5 uM Q04 C8 H18 N O3 P C1CCC(CC1)....
8 4FLI ic50 = 3.59 uM Y16 C14 H26 N2 O6 CC(C)(C)/C....
9 4U6C Ki = 9.9 uM Q06 C8 H18 N O3 P C1CCC(C1)C....
10 4IKR ic50 = 0.59 uM PVP C16 H20 Cl N5 O Cc1c(c(nc(....
11 4FLK ic50 = 5.58 uM Y10 C21 H31 N O5 CC(C)(C)/C....
12 4IKU ic50 = 1.79 uM SHX C19 H18 Cl N5 O Cc1c(c(nc(....
13 2NQ7 ic50 = 2.9 uM HM5 C14 H16 N4 O2 S CC(C)(C)C(....
14 4FLL ic50 = 5.14 uM YZ6 C25 H35 N O6 CC(C)(C)/C....
15 4U71 Ki = 6 uM Q03 C7 H16 N O3 P C1CCC(CC1)....
16 4HXX - 1AY C28 H29 Cl2 N5 Cc1c(c(nc(....
17 4IKS ic50 = 7.23 uM TFD C18 H16 Cl F3 N6 Cc1c(c(nc(....
18 4U6E Ki = 111.6 uM Q02 C7 H10 N O3 P c1ccc(cc1)....
19 4U1B Ki = 4.9 uM Q08 C8 H20 N O3 P CCCC(CCC)[....
20 4FLJ ic50 = 7.45 uM Y08 C22 H38 N2 O6 CC(C)(C)/C....
21 2GG0 ic50 = 1.7 uM U11 C16 H20 F3 N3 O5 C[C@@H](C(....
22 1YVM Ki = 0.4 uM TMG C10 H7 N3 S c1ccc2c(c1....
23 2GU6 - NLP C5 H14 N O3 P CCCC[C@H](....
24 2Q95 ic50 = 1.6 uM A05 C11 H6 Cl N O5 c1cc(c(cc1....
25 2GG8 ic50 = 25 uM U15 C20 H31 N3 O5 Cc1ccc(cc1....
26 2GTX - NLP C5 H14 N O3 P CCCC[C@H](....
27 2EVC ic50 = 0.29 uM FC3 C12 H7 F3 O3 c1ccc(c(c1....
28 4A6W ic50 = 1.9 uM 5C1 C10 H7 Cl N2 O3 c1ccc(c(c1....
29 2GG3 ic50 = 0.58 uM U13 C9 H7 F N6 [H]/N=C/1C....
30 3D27 ic50 = 55.7 uM W29 C12 H12 O2 S CCc1ccsc1c....
31 2GG7 ic50 = 1.75 uM U14 C10 H8 N6 O2 [H]/N=C1/C....
32 2GU5 - NLP C5 H14 N O3 P CCCC[C@H](....
33 1XNZ ic50 = 0.24 uM FCD C11 H7 Cl O3 c1ccc(c(c1....
34 4A6V ic50 = 1.9 uM IKY C11 H7 F3 N2 O3 c1ccc(c(c1....
35 1C21 - MET C5 H11 N O2 S CSCC[C@@H]....
36 2Q92 ic50 = 1.1 uM B23 C11 H7 N O5 c1ccc(c(c1....
37 1C27 - NLP C5 H14 N O3 P CCCC[C@H](....
38 1C24 - MPJ C4 H12 N O2 P S CSCC[C@H](....
39 2EVO ic50 = 0.067 uM CT0 C10 H13 N3 O2 S c1csc(n1)N....
40 2P99 ic50 = 1.16 uM YE6 C11 H9 Cl N2 O2 c1ccc(c(c1....
41 2GG9 ic50 = 3.5 uM U16 C22 H35 N3 O5 CC(C)C[C@H....
42 2Q94 ic50 = 0.37 uM A04 C12 H7 F3 O4 c1ccc(c(c1....
43 2P98 ic50 = 0.64 uM YE7 C12 H10 N4 O c1ccc2c(c1....
44 2GGB ic50 = 12 uM U17 C17 H33 N3 O6 CCCC[C@H](....
45 2EVM ic50 = 0.693 uM FC2 C11 H6 Cl2 O3 c1cc(c(cc1....
46 1C22 - MF3 C5 H8 F3 N O2 S C(CSC(F)(F....
47 1C23 - MPH C4 H12 N O3 P S CSCC[C@H](....
48 2Q96 ic50 = 1.2 uM A18 C12 H9 Cl O3 c1ccc(c(c1....
49 2BB7 ic50 = 2.14 uM QMS C10 H10 N2 O2 S CS(=O)(=O)....
50 2GG2 ic50 = 0.25 uM U12 C10 H7 F3 N6 c1cc(cc(c1....
51 2GGC - MET C5 H11 N O2 S CSCC[C@@H]....
52 2GU4 - NLP C5 H14 N O3 P CCCC[C@H](....
53 2Q93 ic50 = 0.56 uM B21 C12 H10 O4 COc1ccccc1....
54 2GG5 ic50 = 0.25 uM U19 C10 H7 F3 N6 [H]/N=C1/C....
55 3MAT - AHH ALA LEU VAL 0A9 n/a n/a
56 2P9A ic50 = 6.56 uM YE6 C11 H9 Cl N2 O2 c1ccc(c(c1....
57 4IU6 - FZ1 C24 H23 N5 O COc1ccc(cc....
58 1QXZ ic50 = 19 uM M3C C8 H14 N2 O2 S2 CSCC[C@@H]....
59 1QXY ic50 = 16 uM M2C C10 H16 N2 O2 S CSCC[C@@H]....
60 1QXW ic50 = 7 uM M1C C10 H22 N2 O2 CCCC[C@@H]....
61 3IU9 ic50 = 0.24 uM T07 C9 H8 Cl2 N4 S c1cc(c(cc1....
62 3IU7 ic50 = 16 uM FCD C11 H7 Cl O3 c1ccc(c(c1....
63 3PKE - Y10 C21 H31 N O5 CC(C)(C)/C....
64 3PKB ic50 = 0.62 uM Y16 C14 H26 N2 O6 CC(C)(C)/C....
65 3PKA ic50 = 0.54 uM Y02 C23 H37 N O6 Cc1cc(c(c(....
66 3PKC ic50 = 0.96 uM Y08 C22 H38 N2 O6 CC(C)(C)/C....
67 3IU8 ic50 = 0.58 uM T03 C9 H8 F N3 S c1cc(ccc1C....
68 3PKD ic50 = 0.76 uM Y10 C21 H31 N O5 CC(C)(C)/C....
69 1YJ3 - MET C5 H11 N O2 S CSCC[C@@H]....
Polypharmacology
Similar Ligands (2D)
Ligand no: 1; Ligand: 5C1; Similar ligands found: 2
No: Ligand ECFP6 Tc MDL keys Tc
1 5C1 1 1
2 YE6 0.403226 0.74
Similar Ligands (3D)
Ligand no: 1; Ligand: 5C1; Similar ligands found: 541
No: Ligand Similarity coefficient
1 G14 0.9606
2 FCD 0.9572
3 TI7 0.9572
4 ZZA 0.9563
5 B21 0.9559
6 KW7 0.9510
7 WVV 0.9510
8 M4N 0.9497
9 AUV 0.9488
10 NK5 0.9488
11 3VQ 0.9467
12 8CC 0.9462
13 LVP 0.9461
14 A9B 0.9461
15 5VU 0.9435
16 0UL 0.9426
17 3GV 0.9416
18 TJM 0.9410
19 ODK 0.9402
20 D9Z 0.9383
21 5F8 0.9378
22 II4 0.9378
23 5WK 0.9372
24 4AU 0.9360
25 PIQ 0.9356
26 RGK 0.9353
27 H7S 0.9353
28 MD6 0.9348
29 Q4G 0.9343
30 EQA 0.9340
31 P7V 0.9339
32 A7Q 0.9331
33 6MW 0.9323
34 272 0.9321
35 NKI 0.9320
36 FC2 0.9317
37 4FF 0.9317
38 47V 0.9314
39 JMG 0.9311
40 A6W 0.9308
41 LR2 0.9308
42 9JT 0.9304
43 KLE 0.9292
44 IDZ 0.9291
45 78Y 0.9282
46 0NX 0.9277
47 1XS 0.9275
48 IQQ 0.9272
49 1SF 0.9268
50 0K7 0.9260
51 ZSP 0.9258
52 9FH 0.9256
53 IKY 0.9254
54 1ER 0.9253
55 PUE 0.9252
56 K48 0.9251
57 8D6 0.9251
58 JF8 0.9250
59 CBE 0.9245
60 3C5 0.9245
61 1AJ 0.9242
62 EAJ 0.9242
63 D1Y 0.9241
64 LL1 0.9240
65 BIO 0.9238
66 XI7 0.9237
67 YZ9 0.9234
68 A7K 0.9231
69 J38 0.9227
70 WLH 0.9222
71 L5D 0.9220
72 FHV 0.9219
73 1FL 0.9216
74 20D 0.9215
75 KYN 0.9214
76 DFL 0.9211
77 5FL 0.9209
78 L1T 0.9209
79 GNR 0.9206
80 7O4 0.9206
81 5E5 0.9205
82 D25 0.9203
83 J84 0.9203
84 1V1 0.9202
85 4EU 0.9202
86 6DE 0.9202
87 KCH 0.9200
88 Q0K 0.9199
89 VM1 0.9193
90 H4B 0.9192
91 A73 0.9189
92 ENG 0.9187
93 2D2 0.9186
94 6FG 0.9184
95 MIL 0.9183
96 9UL 0.9175
97 LR8 0.9175
98 F40 0.9175
99 0LO 0.9171
100 J1K 0.9170
101 27M 0.9168
102 LFQ 0.9168
103 9CE 0.9167
104 3SU 0.9166
105 5B2 0.9161
106 D2G 0.9158
107 5H6 0.9150
108 JWS 0.9150
109 AVA 0.9149
110 D3G 0.9145
111 JCZ 0.9142
112 X6P 0.9141
113 TRP 0.9140
114 FCW 0.9135
115 0FR 0.9132
116 39Z 0.9131
117 EV2 0.9129
118 D1G 0.9125
119 2QU 0.9124
120 AJ4 0.9124
121 7EH 0.9123
122 7G2 0.9121
123 1Q1 0.9112
124 ZEA 0.9110
125 ERZ 0.9110
126 EQW 0.9110
127 0DF 0.9108
128 ZRK 0.9106
129 KLS 0.9105
130 D8Q 0.9105
131 RKV 0.9100
132 S1D 0.9099
133 1FE 0.9099
134 6C8 0.9098
135 EWG 0.9097
136 GZV 0.9095
137 EAT 0.9090
138 6HO 0.9089
139 BVS 0.9087
140 363 0.9087
141 0OL 0.9080
142 JSX 0.9079
143 AMR 0.9075
144 28A 0.9075
145 WCU 0.9075
146 25F 0.9074
147 KWV 0.9066
148 68B 0.9065
149 SZ5 0.9057
150 5F5 0.9053
151 LVY 0.9050
152 HNT 0.9049
153 DXK 0.9047
154 CUQ 0.9046
155 P4L 0.9041
156 5TO 0.9041
157 0SY 0.9037
158 XYP XIF 0.9035
159 XIF XYP 0.9035
160 795 0.9032
161 RA7 0.9031
162 RSV 0.9030
163 SNV 0.9030
164 1V3 0.9026
165 9FG 0.9025
166 JF5 0.9023
167 3N0 0.9020
168 DDC 0.9018
169 3F4 0.9018
170 2GQ 0.9017
171 U14 0.9017
172 8YH 0.9015
173 3VW 0.9015
174 HA6 0.9013
175 7KE 0.9012
176 3DE 0.9011
177 P93 0.9010
178 X48 0.9009
179 27K 0.9007
180 C4E 0.9006
181 U2Z 0.9006
182 7MW 0.9003
183 1HP 0.9003
184 DBE 0.9003
185 4G2 0.9002
186 5AD 0.9001
187 KP2 0.9000
188 X6W 0.9000
189 HH6 0.8999
190 UN9 0.8999
191 M83 0.8998
192 UN3 0.8997
193 BP7 0.8997
194 6C4 0.8996
195 VBC 0.8995
196 848 0.8994
197 PZX 0.8991
198 NIR 0.8991
199 BXZ 0.8991
200 2GD 0.8991
201 B23 0.8991
202 JGB 0.8990
203 1V4 0.8990
204 22F 0.8990
205 2JX 0.8990
206 ONZ 0.8985
207 HL6 0.8984
208 NAL 0.8980
209 28B 0.8979
210 H35 0.8978
211 TPM 0.8974
212 49P 0.8973
213 3IP 0.8973
214 C0H 0.8971
215 4GU 0.8971
216 GXD 0.8971
217 6C9 0.8970
218 P4T 0.8969
219 6C5 0.8968
220 LIG 0.8964
221 2P3 0.8962
222 B1J 0.8962
223 7L4 0.8961
224 EF2 0.8961
225 N9M 0.8960
226 7XX 0.8959
227 HBI 0.8959
228 0QV 0.8956
229 E9S 0.8954
230 0OY 0.8954
231 AWE 0.8954
232 D26 0.8953
233 5ER 0.8951
234 SB7 0.8944
235 XEV 0.8942
236 1HR 0.8942
237 QME 0.8942
238 L2K 0.8940
239 OA1 0.8939
240 JVD 0.8939
241 Q11 0.8938
242 TCC 0.8938
243 68C 0.8938
244 TB8 0.8937
245 FHI 0.8935
246 GOE 0.8934
247 833 0.8933
248 A98 0.8933
249 EMU 0.8931
250 1A7 0.8931
251 3XH 0.8930
252 4Z1 0.8927
253 4CN 0.8926
254 FC3 0.8925
255 X29 0.8925
256 TYR 0.8924
257 5SJ 0.8922
258 36Z 0.8919
259 NFZ 0.8917
260 36M 0.8917
261 MKN 0.8917
262 MEX 0.8917
263 IOP 0.8915
264 H2B 0.8915
265 CK2 0.8915
266 B41 0.8914
267 5GV 0.8913
268 NQ7 0.8910
269 SOJ 0.8908
270 BZM 0.8907
271 PFT 0.8907
272 C0W 0.8906
273 26C 0.8906
274 XDL XYP 0.8905
275 XIL 0.8905
276 5NN 0.8905
277 FT6 0.8904
278 5V7 0.8903
279 4I8 0.8903
280 6DQ 0.8903
281 TIA 0.8901
282 B2T 0.8899
283 LWS 0.8899
284 4ZF 0.8897
285 EEK 0.8896
286 HDI 0.8893
287 XDK 0.8890
288 6H2 0.8889
289 SQV 0.8888
290 ZMG 0.8885
291 60L 0.8884
292 S8P 0.8883
293 BBY 0.8879
294 G30 0.8878
295 TIZ 0.8878
296 FMQ 0.8877
297 38B 0.8877
298 V2Z 0.8876
299 Q9T 0.8876
300 90G 0.8875
301 1ZC 0.8873
302 KWB 0.8872
303 S46 0.8868
304 79W 0.8867
305 MQS 0.8858
306 XYP XDN 0.8857
307 XDN XYP 0.8857
308 CX5 0.8856
309 VAO 0.8855
310 GJG 0.8855
311 11X 0.8855
312 S8G 0.8854
313 Q5M 0.8852
314 7ZO 0.8852
315 3IL 0.8851
316 MQR 0.8847
317 I2E 0.8847
318 GXG 0.8846
319 LJ4 0.8844
320 FZM 0.8844
321 JFS 0.8843
322 CC5 0.8842
323 XYP XYP 0.8842
324 3D8 0.8842
325 ELH 0.8841
326 SOV 0.8840
327 SNJ 0.8840
328 0OK 0.8839
329 0ON 0.8837
330 FER 0.8837
331 WDW 0.8836
332 A18 0.8836
333 BQ2 0.8835
334 492 0.8835
335 92G 0.8834
336 4NR 0.8832
337 0OO 0.8832
338 0MB 0.8831
339 PZ8 0.8830
340 AED 0.8827
341 U4J 0.8826
342 A4G 0.8826
343 0X2 0.8825
344 39R 0.8824
345 BDI 0.8824
346 SU9 0.8822
347 K4T 0.8817
348 QKU 0.8816
349 KF5 0.8815
350 7AP 0.8813
351 CU8 0.8812
352 F63 0.8811
353 1VK 0.8811
354 4AB 0.8811
355 WSD 0.8810
356 KU1 0.8810
357 7VF 0.8808
358 3RP 0.8808
359 AX4 0.8807
360 EMF 0.8803
361 DTR 0.8802
362 RFZ 0.8802
363 4FP 0.8800
364 657 0.8798
365 PTB 0.8798
366 RF2 0.8795
367 FY8 0.8794
368 4BX 0.8793
369 NIF 0.8793
370 EGV 0.8792
371 2L1 0.8792
372 2GE 0.8791
373 C53 0.8787
374 AVX 0.8786
375 WOE 0.8785
376 7VP 0.8785
377 5I5 0.8782
378 FNT 0.8778
379 5ZM 0.8775
380 96Z 0.8774
381 3D3 0.8774
382 JPQ 0.8773
383 S7D 0.8771
384 ATX 0.8771
385 EN1 0.8769
386 VFM 0.8769
387 ZIP 0.8769
388 5O6 0.8769
389 TOH 0.8769
390 L02 0.8768
391 6ZX 0.8768
392 7FZ 0.8766
393 EYJ 0.8766
394 LJ3 0.8765
395 ADN 0.8765
396 7N8 0.8764
397 F4U 0.8763
398 3AD 0.8763
399 IQW 0.8763
400 3TC 0.8763
401 3GX 0.8761
402 B4O 0.8759
403 X11 0.8758
404 DBS 0.8757
405 2LW 0.8755
406 BHS 0.8753
407 Y70 0.8752
408 7MX 0.8751
409 H4E 0.8751
410 38E 0.8751
411 VJJ 0.8750
412 LI7 0.8749
413 51Y 0.8748
414 P2L 0.8746
415 3JC 0.8743
416 C82 0.8742
417 4AF 0.8741
418 2OH 0.8741
419 ALE 0.8741
420 NEU 0.8737
421 B2E 0.8737
422 5NR 0.8735
423 NU3 0.8733
424 7PJ 0.8733
425 XYS XYS 0.8728
426 H75 0.8727
427 22T 0.8725
428 HKK 0.8725
429 YZM 0.8724
430 CK1 0.8722
431 6WR 0.8721
432 57D 0.8721
433 2QV 0.8721
434 EYY 0.8718
435 7PS 0.8715
436 78U 0.8715
437 22L 0.8714
438 MS0 0.8713
439 M01 0.8713
440 4MB 0.8709
441 PMM 0.8707
442 LNN 0.8707
443 1Q2 0.8707
444 AJ6 0.8704
445 37E 0.8703
446 Q2S 0.8702
447 PQM 0.8702
448 NPS 0.8700
449 8V8 0.8700
450 092 0.8696
451 RBV 0.8696
452 C1E 0.8694
453 9XZ 0.8694
454 MMJ 0.8692
455 46P 0.8692
456 6NZ 0.8691
457 NIY 0.8689
458 ASE 0.8684
459 ET0 0.8683
460 S7S 0.8682
461 CWD 0.8680
462 Q2R 0.8679
463 TT4 0.8679
464 5S9 0.8678
465 2OX 0.8676
466 STV 0.8675
467 NNR 0.8675
468 NE1 0.8675
469 2L2 0.8671
470 A05 0.8668
471 HX8 0.8665
472 0XR 0.8665
473 EZN 0.8664
474 5P3 0.8664
475 4HG 0.8663
476 AOY 0.8661
477 RUG 0.8657
478 BWD 0.8655
479 PRH 0.8654
480 5M2 0.8654
481 90M 0.8654
482 4RV 0.8653
483 1QP 0.8649
484 3CX 0.8648
485 5DE 0.8648
486 DFV 0.8647
487 AZY 0.8646
488 9BF 0.8645
489 XRS 0.8641
490 XYS XYP 0.8634
491 Q8G 0.8633
492 IWD 0.8631
493 GNW 0.8625
494 531 0.8625
495 GHQ 0.8624
496 69W 0.8624
497 7ZL 0.8623
498 4L2 0.8619
499 GZ2 0.8618
500 HHV 0.8613
501 6N4 0.8612
502 CJB 0.8611
503 A51 0.8606
504 S45 0.8605
505 DKZ 0.8601
506 G2V 0.8599
507 Z25 0.8596
508 0OP 0.8594
509 RPN 0.8594
510 JOT 0.8592
511 4KN 0.8591
512 B5A 0.8591
513 S0B 0.8590
514 MBP 0.8588
515 GGB 0.8582
516 40N 0.8579
517 GPK 0.8578
518 4YE 0.8577
519 NE2 0.8569
520 BRY 0.8567
521 A4V 0.8566
522 6DH 0.8565
523 1Q4 0.8565
524 ZYW 0.8565
525 N9J 0.8563
526 FWD 0.8563
527 SSC 0.8557
528 88X 0.8548
529 KPV 0.8547
530 0LA 0.8542
531 15Q 0.8541
532 3G3 0.8541
533 50Q 0.8534
534 AV4 0.8534
535 5RP 0.8526
536 8Y7 0.8523
537 M77 0.8521
538 NFL 0.8521
539 LAH 0.8517
540 PRO GLY 0.8513
541 SCE 0.8505
Similar Binding Sites (Proteins are less than 50% similar to leader)
Pocket No.: 1; Query (leader) PDB : 1YVM; Ligand: TMG; Similar sites found with APoc: No similar binding sites found, or similarity not calculated due to duplicate pocket.
This union binding pocket(no: 1) in the query (biounit: 1yvm.bio1) has 18 residues
No: Leader PDB Ligand Sequence Similarity
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