Receptor
PDB id Resolution Class Description Source Keywords
4UP5 1.65 Å NON-ENZYME: OTHER CRYSTAL STRUCTURE OF THE PYGO2 PHD FINGER IN COMPLEX WITH THE B9L HD1 DOMAIN AND A CHEMICAL FRAGMENT HOMO SAPIENS TRANSCRIPTION PYGO WNT SIGNALLING HISTONE H3 FRAGMENT SC
Ref.: COMPETITIVE BINDING OF A BENZIMIDAZOLE TO THE HISTO BINDING POCKET OF THE PYGO PHD FINGER. ACS CHEM.BIOL. V. 9 2864 2014
Ligand
Ligand Chain:Residue Validity Ligand Warnings Binding Data NGL Viewer Molecular Weight (Da) Formula SMILES
ZN A:1383;
A:1384;
Part of Protein;
Part of Protein;
none;
none;
submit data
65.409 Zn [Zn+2...
94W A:1385;
Valid;
none;
Kd = 2.5 mM
180.227 C8 H8 N2 O S COc1c...
View in 3D viewer
90% Homology Family
Leader
PDB id Resolution Class Description Source Keywords
4UP5 1.65 Å NON-ENZYME: OTHER CRYSTAL STRUCTURE OF THE PYGO2 PHD FINGER IN COMPLEX WITH THE B9L HD1 DOMAIN AND A CHEMICAL FRAGMENT HOMO SAPIENS TRANSCRIPTION PYGO WNT SIGNALLING HISTONE H3 FRAGMENT SC
Ref.: COMPETITIVE BINDING OF A BENZIMIDAZOLE TO THE HISTO BINDING POCKET OF THE PYGO PHD FINGER. ACS CHEM.BIOL. V. 9 2864 2014
Members (1)
No: PDB id Binding Data Representative ligand Formula Smiles
The Class containing this family consists of a total of 1610 families.
1 4UP5 Kd = 2.5 mM 94W C8 H8 N2 O S COc1ccc2c(....
70% Homology Family (1)
No: PDB id Binding Data Representative ligand Formula Smiles
The Class containing this family consists of a total of 1331 families.
1 4UP5 Kd = 2.5 mM 94W C8 H8 N2 O S COc1ccc2c(....
50% Homology Family (1)
No: PDB id Binding Data Representative ligand Formula Smiles
The Class containing this family consists of a total of 1144 families.
1 4UP5 Kd = 2.5 mM 94W C8 H8 N2 O S COc1ccc2c(....
Polypharmacology
Similar Ligands (2D)
Ligand no: 1; Ligand: 94W; Similar ligands found: 10
No: Ligand ECFP6 Tc MDL keys Tc
1 94W 1 1
2 657 0.591837 0.829268
3 K2T 0.510638 0.805556
4 JBZ 0.490566 0.642857
5 EUB 0.483871 0.809524
6 FBB 0.479167 0.7
7 S0E 0.46 0.7
8 6KT 0.442308 0.707317
9 0NJ 0.433333 0.6
10 EUH 0.418182 0.651163
Similar Ligands (3D)
Ligand no: 1; Ligand: 94W; Similar ligands found: 1145
No: Ligand Similarity coefficient
1 CWJ 0.9974
2 9R5 0.9917
3 A7H 0.9775
4 8ZE 0.9745
5 BCU 0.9729
6 ES2 0.9722
7 VGD 0.9722
8 5XC 0.9702
9 1P8 0.9698
10 36R 0.9675
11 MSR 0.9672
12 MQN 0.9669
13 N2I 0.9661
14 0JD 0.9653
15 ET2 0.9637
16 5OB 0.9636
17 CLW 0.9627
18 5VM 0.9626
19 0TU 0.9621
20 MR1 0.9615
21 KDV 0.9614
22 BZ3 0.9611
23 15N 0.9611
24 2HQ 0.9598
25 J6W 0.9584
26 6NT 0.9581
27 XAZ 0.9579
28 TYL 0.9569
29 2BG 0.9563
30 4YO 0.9562
31 0HO 0.9562
32 H42 0.9557
33 SNO 0.9557
34 E1T 0.9555
35 4JQ 0.9554
36 5LA 0.9554
37 SNU 0.9552
38 1F1 0.9550
39 MS9 0.9548
40 0HN 0.9547
41 JAW 0.9541
42 ODO 0.9533
43 CPZ 0.9531
44 2ZM 0.9525
45 6NI 0.9524
46 KJU 0.9520
47 SLS 0.9517
48 2HU 0.9517
49 5NI 0.9500
50 PNZ 0.9495
51 3A9 0.9494
52 I3E 0.9494
53 2AQ 0.9491
54 4FS 0.9490
55 TGX 0.9489
56 3NY 0.9487
57 F9Y 0.9477
58 ES5 0.9477
59 86J 0.9475
60 OCH 0.9473
61 5JQ 0.9472
62 ANN 0.9469
63 COU 0.9468
64 N8Y 0.9466
65 URC 0.9465
66 HQJ 0.9462
67 03V 0.9460
68 6VD 0.9459
69 5GU 0.9457
70 QX4 0.9454
71 BPN 0.9451
72 GO2 0.9450
73 2FY 0.9449
74 4BZ 0.9445
75 9ZE 0.9442
76 ICB 0.9440
77 BZ2 0.9439
78 1M2 0.9438
79 5JL 0.9434
80 4TU 0.9432
81 DHR 0.9432
82 6RQ 0.9431
83 3BU 0.9430
84 TZF 0.9425
85 75K 0.9424
86 JB8 0.9423
87 AN3 0.9421
88 BZJ 0.9420
89 8TX 0.9418
90 B55 0.9418
91 XIY 0.9417
92 F4E 0.9415
93 2A9 0.9411
94 JDN 0.9411
95 JB5 0.9410
96 JA8 0.9410
97 4FA 0.9409
98 7MU 0.9408
99 TT4 0.9408
100 9FL 0.9407
101 HDH 0.9403
102 4BL 0.9402
103 HHR 0.9401
104 4I8 0.9398
105 8WO 0.9398
106 PH2 0.9396
107 OTR 0.9395
108 XQ0 0.9395
109 CH9 0.9395
110 PHB 0.9394
111 HC4 0.9393
112 RNO 0.9390
113 9CA 0.9389
114 IV2 0.9388
115 8W9 0.9384
116 E5X 0.9384
117 RM1 0.9380
118 3QV 0.9378
119 GJP 0.9378
120 4NM 0.9374
121 X0U 0.9372
122 A29 0.9371
123 HA5 0.9371
124 UNJ 0.9371
125 2F6 0.9366
126 4NB 0.9366
127 I3A 0.9365
128 OW4 0.9364
129 36M 0.9363
130 6ME 0.9363
131 TSS 0.9359
132 AMH 0.9358
133 4BY 0.9354
134 ESX 0.9354
135 5QY 0.9352
136 OW7 0.9351
137 E7S 0.9350
138 30G 0.9349
139 ESP 0.9348
140 HBD 0.9347
141 SYV 0.9346
142 3PF 0.9343
143 PAB 0.9342
144 5TY 0.9341
145 DQU 0.9340
146 B62 0.9340
147 RD4 0.9339
148 JAE 0.9338
149 BTY 0.9335
150 6FZ 0.9335
151 1IT 0.9333
152 G3E 0.9332
153 XHP 0.9331
154 27B 0.9330
155 PZM 0.9329
156 MUA 0.9327
157 0F9 0.9326
158 A7N 0.9324
159 D48 0.9324
160 IAC 0.9320
161 PQ0 0.9318
162 ABI 0.9317
163 OTW 0.9317
164 M2K 0.9316
165 4MA 0.9316
166 IWT 0.9315
167 TTL 0.9314
168 7O4 0.9313
169 0FO 0.9312
170 PRF 0.9309
171 7MX 0.9309
172 069 0.9308
173 11S 0.9308
174 GOJ 0.9307
175 92P 0.9305
176 NPO 0.9304
177 PD2 0.9304
178 FA0 0.9303
179 3ZB 0.9302
180 1P7 0.9302
181 174 0.9302
182 Z82 0.9302
183 44W 0.9301
184 P9E 0.9301
185 4M0 0.9301
186 FK1 0.9300
187 2QC 0.9298
188 M5K 0.9297
189 ES9 0.9297
190 428 0.9297
191 3R4 0.9295
192 1HN 0.9293
193 M6N 0.9292
194 PEY 0.9292
195 259 0.9290
196 OVM 0.9290
197 NAG 0.9290
198 J9Q 0.9289
199 1Y6 0.9286
200 N4E 0.9285
201 L5V 0.9285
202 J5I 0.9284
203 6TZ 0.9284
204 36Y 0.9283
205 CWS 0.9282
206 KTJ 0.9281
207 8NB 0.9280
208 MEW 0.9280
209 DVQ 0.9278
210 4JT 0.9278
211 15E 0.9278
212 4WL 0.9278
213 DE5 0.9277
214 H4N 0.9273
215 AJ2 0.9273
216 CTL 0.9273
217 EUE 0.9272
218 SE2 0.9272
219 LPK 0.9271
220 2AK 0.9270
221 7W1 0.9269
222 KUF 0.9267
223 2K8 0.9267
224 8IG 0.9267
225 AEF 0.9267
226 A5E 0.9267
227 3MB 0.9266
228 GVY 0.9266
229 N1E 0.9265
230 YRL 0.9263
231 Q24 0.9262
232 SN4 0.9262
233 826 0.9262
234 D3G 0.9260
235 DRG 0.9260
236 4VY 0.9254
237 MVN 0.9254
238 TYR 0.9253
239 9FE 0.9252
240 R20 0.9252
241 F60 0.9251
242 DOB 0.9250
243 BHA 0.9250
244 5MB 0.9250
245 ICO 0.9250
246 4RU 0.9249
247 LZM 0.9249
248 PBZ 0.9249
249 R9Y 0.9247
250 6AI 0.9246
251 4HC 0.9245
252 14O 0.9243
253 FDR 0.9241
254 AQO 0.9239
255 BGC 0.9238
256 E3X 0.9238
257 BZX 0.9237
258 5B1 0.9237
259 J9W 0.9234
260 5WV 0.9234
261 2HC 0.9234
262 3DM 0.9232
263 M1Q 0.9231
264 AX7 0.9230
265 ZYR 0.9229
266 4AA 0.9228
267 173 0.9228
268 EN1 0.9226
269 5H1 0.9225
270 44V 0.9224
271 4P5 0.9222
272 8NY 0.9221
273 42A 0.9221
274 EA1 0.9219
275 SKA 0.9219
276 AZ8 0.9218
277 C2Y 0.9217
278 7HQ 0.9217
279 8HC 0.9215
280 F4K 0.9215
281 PDC 0.9214
282 LNR 0.9213
283 5MI 0.9213
284 TSR 0.9212
285 PIM 0.9212
286 5CU 0.9211
287 SRO 0.9209
288 OQC 0.9209
289 ABV 0.9208
290 8XL 0.9208
291 0FN 0.9206
292 5VL 0.9204
293 0FK 0.9201
294 7MW 0.9201
295 SKF 0.9200
296 HNT 0.9200
297 V1T 0.9199
298 4ME 0.9199
299 HIS 0.9198
300 0BP 0.9198
301 FUD 0.9196
302 0P6 0.9195
303 OVP 0.9194
304 HMH 0.9194
305 8WT 0.9194
306 ISZ 0.9191
307 97T 0.9188
308 BNL 0.9188
309 AA 0.9187
310 1KP 0.9186
311 PE0 0.9181
312 M0W 0.9180
313 HHS 0.9180
314 LQ2 0.9179
315 KMY 0.9178
316 1L5 0.9178
317 BK9 0.9177
318 H4E 0.9177
319 GXY 0.9177
320 795 0.9175
321 12Q 0.9174
322 QIV 0.9174
323 PIY 0.9173
324 12T 0.9171
325 TH7 0.9169
326 PPY 0.9169
327 MAJ 0.9168
328 8H8 0.9167
329 2K4 0.9166
330 JG8 0.9166
331 BHO 0.9165
332 LDP 0.9164
333 3VS 0.9162
334 PKU 0.9161
335 NDG 0.9160
336 BEA 0.9159
337 DNF 0.9159
338 HQD 0.9156
339 ESI 0.9156
340 5WZ 0.9154
341 F31 0.9154
342 X0W 0.9153
343 HX4 0.9153
344 ANF 0.9153
345 4LW 0.9153
346 G14 0.9152
347 4MU 0.9151
348 5RN 0.9150
349 7VS 0.9150
350 EYV 0.9149
351 HQT 0.9147
352 BIK 0.9146
353 492 0.9145
354 ISN 0.9145
355 K97 0.9144
356 M4E 0.9144
357 4ZA 0.9143
358 ZZZ 0.9142
359 DHB 0.9142
360 2AL 0.9141
361 8CM 0.9140
362 4HM 0.9140
363 68A 0.9140
364 HHH 0.9139
365 HMU 0.9137
366 K82 0.9136
367 CFI 0.9134
368 PJW 0.9134
369 363 0.9133
370 KKN 0.9132
371 CLZ 0.9131
372 5NU 0.9131
373 WCE 0.9130
374 GVG 0.9130
375 GCS 0.9129
376 92G 0.9128
377 3NT 0.9127
378 INO 0.9127
379 3VQ 0.9127
380 J9N 0.9126
381 NIZ 0.9125
382 AC6 0.9125
383 K4V 0.9124
384 DIN 0.9124
385 GLC 0.9124
386 YZM 0.9124
387 717 0.9123
388 MO8 0.9121
389 0N7 0.9119
390 PXL 0.9118
391 2LY 0.9115
392 5QX 0.9115
393 3ID 0.9115
394 M1E 0.9115
395 4JC 0.9115
396 52C 0.9114
397 NDH 0.9110
398 7W4 0.9110
399 QWN 0.9109
400 4CS 0.9109
401 HHI 0.9109
402 1A7 0.9108
403 ZZT 0.9108
404 M78 0.9106
405 7VP 0.9105
406 0NX 0.9104
407 PHE 0.9104
408 DRL 0.9103
409 HBA 0.9103
410 FHB 0.9103
411 6FB 0.9103
412 DMD 0.9102
413 XYL 0.9101
414 RB5 0.9101
415 KJH 0.9101
416 KYA 0.9101
417 JND 0.9101
418 ZEC 0.9101
419 YH7 0.9100
420 ES7 0.9099
421 THA 0.9099
422 4HB 0.9099
423 GAB 0.9097
424 M0Q 0.9094
425 XRG 0.9094
426 EWG 0.9094
427 4Z4 0.9092
428 BRT 0.9090
429 OVV 0.9087
430 92K 0.9086
431 W81 0.9086
432 M1H 0.9086
433 AZM 0.9086
434 80G 0.9086
435 344 0.9085
436 NNO 0.9085
437 L14 0.9082
438 NOJ 0.9081
439 VM1 0.9081
440 549 0.9080
441 R8S 0.9080
442 AJ1 0.9080
443 1Z6 0.9080
444 VXX 0.9078
445 ONR 0.9077
446 SHA 0.9077
447 MRW 0.9075
448 9DG 0.9075
449 8NX 0.9074
450 YPN 0.9073
451 JLZ 0.9073
452 3HB 0.9073
453 BPY 0.9072
454 BOA 0.9072
455 2KA 0.9071
456 GNM 0.9071
457 9UL 0.9070
458 PUE 0.9070
459 EOL 0.9069
460 2EC 0.9069
461 TPA 0.9069
462 H8N 0.9069
463 3Z8 0.9068
464 GTQ 0.9068
465 SW7 0.9068
466 BPU 0.9068
467 46P 0.9067
468 NSP 0.9066
469 2MI 0.9063
470 MPV 0.9063
471 4NC 0.9063
472 GF4 0.9062
473 QXW 0.9062
474 4A3 0.9061
475 CHB 0.9060
476 AES 0.9060
477 OGA 0.9060
478 PQK 0.9059
479 270 0.9059
480 2O6 0.9059
481 XAN 0.9058
482 ZZA 0.9058
483 8G0 0.9057
484 3HM 0.9057
485 4V2 0.9056
486 NID 0.9056
487 PH3 0.9056
488 PBA 0.9055
489 FYU 0.9054
490 SOR 0.9054
491 IQ5 0.9054
492 GZL 0.9053
493 G3F 0.9053
494 NCT 0.9053
495 NFM 0.9052
496 M5H 0.9052
497 C1M 0.9051
498 5RO 0.9050
499 BQ2 0.9048
500 A7W 0.9048
501 3R6 0.9046
502 X48 0.9046
503 INE 0.9044
504 KOJ 0.9044
505 3W8 0.9041
506 4VP 0.9040
507 P9P 0.9040
508 TIU 0.9040
509 2FX 0.9040
510 XCG 0.9040
511 KT7 0.9039
512 2FQ 0.9039
513 93K 0.9039
514 4NZ 0.9038
515 P92 0.9036
516 EUG 0.9036
517 67N 0.9034
518 P72 0.9033
519 Y3L 0.9033
520 AKG 0.9033
521 MS0 0.9032
522 LT2 0.9032
523 3F0 0.9029
524 B1J 0.9029
525 BSX 0.9028
526 3HA 0.9028
527 GUN 0.9027
528 M6Z 0.9026
529 2HO 0.9025
530 TMG 0.9025
531 8GC 0.9024
532 BP7 0.9024
533 HX3 0.9023
534 DBJ 0.9023
535 I1E 0.9022
536 54G 0.9022
537 CKA 0.9022
538 ST2 0.9021
539 3VX 0.9021
540 6QF 0.9019
541 TAG 0.9018
542 FBM 0.9018
543 EE8 0.9016
544 AL0 0.9016
545 3DO 0.9016
546 FBF 0.9016
547 ASC 0.9013
548 9NB 0.9013
549 DIE 0.9011
550 GLO 0.9011
551 MYJ 0.9011
552 3AE 0.9011
553 1XM 0.9010
554 AJY 0.9010
555 ALE 0.9010
556 M4S 0.9008
557 TWO 0.9008
558 6AP 0.9007
559 EVF 0.9006
560 CXH 0.9006
561 RNS 0.9005
562 XDK 0.9005
563 XM0 0.9005
564 UA5 0.9004
565 E7Z 0.9003
566 ENO 0.9003
567 L99 0.9002
568 HBO 0.9002
569 61M 0.9002
570 AZA 0.9002
571 UFO 0.9001
572 8OZ 0.9000
573 6M9 0.9000
574 AZ9 0.8999
575 A2F 0.8998
576 TCA 0.8998
577 20J 0.8998
578 DA4 0.8996
579 VNL 0.8995
580 ODK 0.8995
581 3BZ 0.8993
582 IHB 0.8993
583 0LH 0.8992
584 3AB 0.8992
585 UAN 0.8992
586 NMJ 0.8992
587 4MB 0.8992
588 HSO 0.8991
589 4NP 0.8991
590 M1A 0.8989
591 1DW 0.8989
592 AJV 0.8987
593 5RG 0.8987
594 39O 0.8986
595 53C 0.8986
596 QBM 0.8986
597 4KL 0.8985
598 5HN 0.8983
599 DEW 0.8982
600 FHC 0.8982
601 DBH 0.8982
602 H5B 0.8982
603 42J 0.8981
604 NOY 0.8980
605 3M0 0.8980
606 SAN 0.8980
607 P81 0.8979
608 HHA 0.8977
609 8S0 0.8977
610 5XB 0.8976
611 FK8 0.8975
612 LEL 0.8975
613 Z5P 0.8975
614 DJN 0.8974
615 NLA 0.8974
616 BDP 0.8973
617 4XR 0.8970
618 7ME 0.8968
619 ANC 0.8968
620 TTY 0.8967
621 APS 0.8964
622 FDB 0.8964
623 6CS 0.8964
624 4NS 0.8964
625 L22 0.8962
626 IGA 0.8962
627 R8V 0.8961
628 AZG 0.8960
629 4JM 0.8960
630 4J8 0.8960
631 9TW 0.8958
632 LDR 0.8958
633 PRZ 0.8958
634 86L 0.8957
635 141 0.8957
636 268 0.8956
637 3XR 0.8956
638 2D0 0.8956
639 SSC 0.8955
640 IOS 0.8955
641 TSU 0.8955
642 27K 0.8955
643 M45 0.8954
644 B53 0.8954
645 B60 0.8954
646 DNA 0.8954
647 NGA 0.8954
648 RKV 0.8953
649 7FU 0.8953
650 4AV 0.8952
651 K34 0.8952
652 A98 0.8950
653 S7J 0.8949
654 OAA 0.8949
655 28N 0.8949
656 QUS 0.8948
657 RBL 0.8947
658 XBT 0.8947
659 L03 0.8945
660 5M0 0.8945
661 BCP 0.8944
662 F9P 0.8942
663 GDL 0.8942
664 VOH 0.8941
665 TXW 0.8940
666 XDE 0.8939
667 82I 0.8939
668 QBK 0.8938
669 N91 0.8938
670 FBS 0.8937
671 AEG 0.8935
672 0CU 0.8934
673 IPB 0.8934
674 ST3 0.8934
675 36E 0.8933
676 ARP 0.8932
677 5F5 0.8932
678 MAQ 0.8932
679 258 0.8931
680 PFL 0.8931
681 VK3 0.8929
682 2BX 0.8928
683 5GT 0.8927
684 QSB 0.8927
685 9AP 0.8927
686 0RW 0.8927
687 GAL 0.8927
688 SKM 0.8927
689 S2G 0.8927
690 OHJ 0.8925
691 CSN 0.8925
692 B57 0.8924
693 PHU 0.8924
694 NQ 0.8923
695 DX4 0.8922
696 AOT 0.8920
697 ES0 0.8920
698 1QP 0.8919
699 88L 0.8918
700 GCU 0.8917
701 IFL 0.8915
702 AMR 0.8915
703 209 0.8915
704 9MG 0.8913
705 2H5 0.8913
706 C2B 0.8912
707 XX2 0.8911
708 2CK 0.8911
709 AHR 0.8910
710 D2G 0.8908
711 FE DB1 0.8908
712 JU2 0.8908
713 CWM 0.8907
714 NVU 0.8907
715 BNF 0.8907
716 4XF 0.8906
717 SOE 0.8903
718 6SD 0.8902
719 KBZ 0.8900
720 F05 0.8899
721 PO6 0.8898
722 MD6 0.8898
723 FP1 0.8898
724 MLT 0.8898
725 FCR 0.8895
726 S7S 0.8894
727 B5D 0.8893
728 0W1 0.8893
729 Q88 0.8892
730 TCR 0.8892
731 ALL 0.8891
732 14J 0.8891
733 3TC 0.8889
734 XQG 0.8889
735 F2W 0.8888
736 HJ7 0.8888
737 B56 0.8888
738 JF2 0.8887
739 JYB 0.8887
740 24B 0.8884
741 5WY 0.8884
742 Q71 0.8883
743 SX1 0.8883
744 N0Z 0.8882
745 1AL 0.8879
746 JF1 0.8877
747 9TZ 0.8877
748 4JL 0.8877
749 1VK 0.8876
750 GWM 0.8874
751 KJY 0.8874
752 Q02 0.8873
753 RXA 0.8872
754 TYE 0.8871
755 5MK 0.8871
756 MZM 0.8870
757 RMN 0.8869
758 DIU 0.8869
759 AX3 0.8869
760 2GS 0.8868
761 4CM 0.8868
762 DHY 0.8867
763 HH5 0.8867
764 N3W 0.8866
765 XUL 0.8866
766 GDE 0.8866
767 DHC 0.8866
768 6M4 0.8865
769 Q6T 0.8865
770 4VS 0.8864
771 DZA 0.8864
772 S60 0.8864
773 MWP 0.8863
774 54Z 0.8862
775 CIT 0.8862
776 X0V 0.8862
777 QUZ 0.8862
778 C53 0.8861
779 60L 0.8861
780 RAT 0.8858
781 JBK 0.8857
782 DBX 0.8857
783 9LI 0.8856
784 091 0.8855
785 JP2 0.8855
786 PPT 0.8854
787 V55 0.8852
788 EV3 0.8849
789 ITE 0.8849
790 AEH 0.8848
791 ASO 0.8847
792 FIX 0.8847
793 FCD 0.8846
794 4FH 0.8845
795 DEE 0.8845
796 AAS 0.8844
797 FQI 0.8842
798 4XV 0.8841
799 NPY 0.8840
800 7B4 0.8838
801 AHN 0.8837
802 CFA 0.8837
803 4XS 0.8835
804 EGR 0.8834
805 AY4 0.8834
806 PAC 0.8834
807 G2F 0.8832
808 56D 0.8832
809 7B3 0.8831
810 D07 0.8829
811 MTL 0.8829
812 4LV 0.8829
813 OKG 0.8829
814 1PT 0.8829
815 A2G 0.8827
816 ZBT 0.8827
817 ZYX 0.8825
818 LR5 0.8824
819 4JE 0.8822
820 K32 0.8818
821 H33 0.8817
822 PQZ 0.8817
823 3YP 0.8816
824 PRL 0.8815
825 CS2 0.8813
826 5NE 0.8813
827 261 0.8813
828 ZXD 0.8811
829 M3H 0.8811
830 3OC 0.8810
831 SYE 0.8810
832 CN0 0.8809
833 FF2 0.8809
834 NGW 0.8808
835 NGT 0.8808
836 CK2 0.8808
837 9EW 0.8808
838 JAH 0.8808
839 GNL 0.8807
840 NSG 0.8807
841 KTW 0.8805
842 0XT 0.8805
843 DGJ 0.8803
844 1FE 0.8802
845 M1Z 0.8802
846 HA7 0.8801
847 DHK 0.8801
848 JA5 0.8800
849 45L 0.8799
850 F12 0.8799
851 QWW 0.8798
852 3J8 0.8798
853 EXD 0.8798
854 SMN 0.8797
855 GCO 0.8797
856 FBA 0.8796
857 XIZ 0.8796
858 DYA 0.8796
859 CUW 0.8795
860 KIB 0.8794
861 CFP 0.8793
862 BZE 0.8793
863 5F8 0.8793
864 290 0.8792
865 EYJ 0.8792
866 AMS 0.8792
867 152 0.8792
868 FLC 0.8791
869 DHI 0.8789
870 SAL 0.8788
871 K22 0.8787
872 2LP 0.8787
873 4M4 0.8785
874 8MO 0.8785
875 BVA 0.8784
876 KDG 0.8783
877 M4T 0.8783
878 GO8 0.8782
879 APG 0.8781
880 XLS 0.8780
881 IFP 0.8779
882 AM4 0.8779
883 K7H 0.8779
884 5OO 0.8778
885 N7I 0.8778
886 N2M 0.8777
887 RA7 0.8777
888 EV2 0.8776
889 JXW 0.8775
890 37T 0.8775
891 ZHA 0.8774
892 F81 0.8774
893 S24 0.8773
894 EVA 0.8773
895 MQB 0.8771
896 II6 0.8771
897 KMH 0.8771
898 LGC 0.8770
899 R2P 0.8770
900 78Y 0.8769
901 NYL 0.8769
902 5TZ 0.8769
903 HNK 0.8768
904 HNL 0.8768
905 BBK 0.8768
906 4SX 0.8767
907 CTS 0.8766
908 DNC 0.8766
909 3W3 0.8765
910 3W6 0.8765
911 MNM 0.8764
912 SHG 0.8762
913 C9E 0.8761
914 42C 0.8761
915 OMD 0.8760
916 QBS 0.8758
917 R9S 0.8758
918 Z13 0.8757
919 0W8 0.8757
920 EKZ 0.8757
921 ROI 0.8757
922 BGU 0.8756
923 6BL 0.8756
924 7ZE 0.8755
925 I6G 0.8755
926 QPR 0.8754
927 6E8 0.8752
928 QMS 0.8751
929 7NI 0.8751
930 FLV 0.8751
931 51R 0.8751
932 1SQ 0.8750
933 6R8 0.8750
934 QX2 0.8749
935 SYA 0.8746
936 OA3 0.8745
937 S7G 0.8745
938 23A 0.8745
939 226 0.8745
940 1NP 0.8744
941 ADZ 0.8741
942 FZM 0.8741
943 APZ 0.8739
944 3AL 0.8737
945 JXN 0.8737
946 URO 0.8736
947 F0J 0.8735
948 LYL 0.8735
949 BE2 0.8734
950 FBW 0.8733
951 DX3 0.8732
952 OK7 0.8731
953 C2U 0.8731
954 1LQ 0.8731
955 6MW 0.8731
956 FAN 0.8730
957 5SG 0.8730
958 5IQ 0.8730
959 54X 0.8730
960 J9T 0.8727
961 I2E 0.8723
962 4FF 0.8723
963 EV0 0.8722
964 TOF 0.8722
965 PYQ 0.8722
966 G12 0.8722
967 5GV 0.8721
968 K3D 0.8721
969 GZ2 0.8721
970 24W 0.8720
971 C82 0.8716
972 5Q0 0.8716
973 UNC 0.8716
974 0GZ 0.8713
975 BL0 0.8711
976 SVN 0.8711
977 5H6 0.8711
978 AC0 0.8711
979 P7Y 0.8710
980 4YS 0.8710
981 AKH 0.8710
982 LMR 0.8710
983 TH0 0.8710
984 5FL 0.8709
985 SWX 0.8709
986 YIE 0.8708
987 6GU 0.8707
988 BHQ 0.8706
989 39U 0.8706
990 HKD 0.8704
991 3FH 0.8704
992 X05 0.8703
993 0LO 0.8703
994 WOO 0.8702
995 FGZ 0.8702
996 Q77 0.8701
997 PNP 0.8700
998 DHQ 0.8700
999 1P3 0.8697
1000 HCI 0.8697
1001 32X 0.8696
1002 9KT 0.8696
1003 U7E 0.8695
1004 EYK 0.8694
1005 PXM 0.8694
1006 3U4 0.8694
1007 PRY 0.8693
1008 2UZ 0.8693
1009 HLD 0.8693
1010 ZSP 0.8693
1011 4SV 0.8691
1012 Q7A 0.8690
1013 N9J 0.8687
1014 23J 0.8686
1015 IF7 0.8685
1016 2ZQ 0.8685
1017 FQX 0.8685
1018 OXC 0.8684
1019 8U3 0.8682
1020 GLT 0.8682
1021 TRP 0.8682
1022 NDM 0.8680
1023 PZI 0.8680
1024 6ZX 0.8679
1025 1LM 0.8679
1026 GLU 0.8676
1027 PRO GLY 0.8675
1028 5NS 0.8675
1029 SSB 0.8674
1030 UEG 0.8673
1031 QSH 0.8673
1032 LI6 0.8672
1033 NGO 0.8671
1034 N5J 0.8666
1035 P3K 0.8666
1036 JTH 0.8665
1037 EPR 0.8662
1038 ES1 0.8662
1039 T9G 0.8662
1040 FRU 0.8662
1041 8GK 0.8661
1042 XI7 0.8661
1043 X8D 0.8661
1044 3VW 0.8660
1045 67X 0.8657
1046 ES6 0.8656
1047 HBI 0.8653
1048 3HG 0.8651
1049 RUY 0.8650
1050 GYE 0.8650
1051 D1G 0.8649
1052 YE6 0.8649
1053 O72 0.8649
1054 WSD 0.8648
1055 GLA 0.8645
1056 CXP 0.8644
1057 SG2 0.8642
1058 AJG 0.8642
1059 HNE 0.8642
1060 7WR 0.8641
1061 E1K 0.8641
1062 JPZ 0.8640
1063 2JK 0.8639
1064 X6X 0.8638
1065 SR1 0.8637
1066 K5W 0.8636
1067 BIO 0.8636
1068 PRA 0.8636
1069 K7M 0.8635
1070 RBJ 0.8630
1071 AAN 0.8630
1072 BA5 0.8630
1073 3XX 0.8630
1074 HQY 0.8629
1075 DK1 0.8629
1076 4BF 0.8623
1077 SWA 0.8622
1078 149 0.8622
1079 E79 0.8620
1080 P80 0.8620
1081 0FR 0.8619
1082 5JC 0.8617
1083 6X9 0.8616
1084 HHT 0.8614
1085 EMZ 0.8614
1086 3MG 0.8614
1087 SQ7 0.8611
1088 HPP 0.8610
1089 GXL 0.8608
1090 TEP 0.8607
1091 GCB 0.8606
1092 P84 0.8602
1093 FTV 0.8602
1094 JBH 0.8602
1095 HL4 0.8600
1096 PFF 0.8599
1097 L1O 0.8597
1098 B85 0.8596
1099 RHU 0.8594
1100 1GN 0.8592
1101 QMP 0.8591
1102 4XH 0.8591
1103 RSV 0.8590
1104 GAF 0.8590
1105 JRB 0.8589
1106 GNY 0.8588
1107 AW5 0.8588
1108 2D2 0.8587
1109 E3D 0.8585
1110 9KZ 0.8583
1111 K37 0.8583
1112 GIF 0.8582
1113 JVN 0.8580
1114 R1P 0.8578
1115 TZM 0.8577
1116 XCZ 0.8576
1117 2CQ 0.8575
1118 DPZ 0.8574
1119 PCS 0.8573
1120 CIY 0.8572
1121 7WG 0.8572
1122 ZZ8 0.8572
1123 FDK 0.8570
1124 4HP 0.8567
1125 DGN 0.8567
1126 SME 0.8566
1127 9BF 0.8565
1128 JBE 0.8564
1129 1WG 0.8564
1130 TBS 0.8563
1131 PYD 0.8561
1132 49O 0.8559
1133 5O6 0.8559
1134 F1A 0.8558
1135 ADA 0.8555
1136 HH8 0.8553
1137 41K 0.8547
1138 LZ2 0.8545
1139 AGK 0.8542
1140 IND 0.8535
1141 X11 0.8535
1142 FOT 0.8531
1143 M44 0.8529
1144 HJP 0.8525
1145 SXS 0.8514
Similar Binding Sites (Proteins are less than 50% similar to leader)
Pocket No.: 1; Query (leader) PDB : 4UP5; Ligand: 94W; Similar sites found with APoc: No similar binding sites found, or similarity not calculated due to duplicate pocket.
This union binding pocket(no: 1) in the query (biounit: 4up5.bio1) has 10 residues
No: Leader PDB Ligand Sequence Similarity
APoc FAQ
Feedback