Receptor
PDB id Resolution Class Description Source Keywords
3MEV 1.83 Å NON-ENZYME: OTHER CRYSTAL STRUCTURE OF SGF29 IN COMPLEX WITH R2AK4ME3 HOMO SAPIENS STRUCTURAL GENOMICS CONSORTIUM SGC NUCLEUS TRANSCRIPTIONTRANSCRIPTION REGULATION CHROMOSOMAL PROTEIN DNA-BINDINGNUCLEOSOME CORE
Ref.: SGF29 BINDS HISTONE H3K4ME2/3 AND IS REQUIRED FOR S COMPLEX RECRUITMENT AND HISTONE H3 ACETYLATION. EMBO J. V. 30 2829 2011
Ligand
Ligand Chain:Residue Validity Ligand Warnings Binding Data NGL Viewer Molecular Weight (Da) Formula SMILES
ALA ALA THR M3L GLN THR ALA ARG C:1;
D:1;
Valid;
Valid;
none;
none;
submit data
n/a n/a
GOL B:1;
Invalid;
none;
submit data
92.094 C3 H8 O3 C(C(C...
SO4 A:1;
B:2;
Invalid;
Invalid;
none;
none;
submit data
96.063 O4 S [O-]S...
View in 3D viewer
90% Homology Family
Leader
PDB id Resolution Class Description Source Keywords
5C0M 1.6 Å NON-ENZYME: OTHER CRYSTAL STRUCTURE OF SGF29 TANDEM TUDOR DOMAIN IN COMPLEX WI CONTAINING PEPTIDE HOMO SAPIENS SGF29 TANDEM TUDOR DOMAIN CARBA CONTAINING PEPTIDE STRUCTGENOMICS STRUCTURAL GENOMICS CONSORTIUM SGC TRANSCRIPTIO
Ref.: CHEMICAL BASIS FOR THE RECOGNITION OF TRIMETHYLLYSI EPIGENETIC READER PROTEINS. NAT COMMUN V. 6 8911 2015
Members (2)
No: PDB id Binding Data Representative ligand Formula Smiles
The Class containing this family consists of a total of 1610 families.
1 3MEV - ALA ALA THR M3L GLN THR ALA ARG n/a n/a
2 5C0M Kd = 1.4 uM ALA ARG THR 4WQ GLN THR ALA ARG LYS SER n/a n/a
70% Homology Family (2)
No: PDB id Binding Data Representative ligand Formula Smiles
The Class containing this family consists of a total of 1331 families.
1 3MEV - ALA ALA THR M3L GLN THR ALA ARG n/a n/a
2 5C0M Kd = 1.4 uM ALA ARG THR 4WQ GLN THR ALA ARG LYS SER n/a n/a
50% Homology Family (2)
No: PDB id Binding Data Representative ligand Formula Smiles
The Class containing this family consists of a total of 1144 families.
1 3MEV - ALA ALA THR M3L GLN THR ALA ARG n/a n/a
2 5C0M Kd = 1.4 uM ALA ARG THR 4WQ GLN THR ALA ARG LYS SER n/a n/a
Polypharmacology
Similar Ligands (2D)
Ligand no: 1; Ligand: ALA ALA THR M3L GLN THR ALA ARG; Similar ligands found: 0
No: Ligand ECFP6 Tc MDL keys Tc
Similar Ligands (3D)
Ligand no: 1; Ligand: ALA ALA THR M3L GLN THR ALA ARG; Similar ligands found: 0
No: Ligand Similarity coefficient
Similar Binding Sites (Proteins are less than 50% similar to leader) APoc FAQ
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