- Navigate
- Expand All | Collapse All
- Receptor | Ligand | View in 3D
- Family: 90% | 70% | 50% | site
- External Links
-
|
- Download
- Biounit PDB : .ZIP | .CSV
- Family 90% : .ZIP | .CSV
- Class : .ZIP | .CSV
No: | PDB id | Binding Data | Representative ligand | Formula | Smiles |
---|---|---|---|---|---|
The Class containing this family consists of a total of 1 families. | |||||
1 | 3IND | ic50 = 1.53 uM | 593 | C20 H25 N3 O | CN1C(=O)C(.... |
2 | 2HM1 | ic50 = 13 nM | LIQ | C33 H42 F2 N4 O5 S | CCCCCS(=O).... |
3 | 2B8L | ic50 = 15 nM | 5HA | C31 H38 N4 O5 S | CC(c1ccccc.... |
4 | 4LXK | ic50 = 0.004 uM | 1YT | C27 H36 F4 N2 O4 S | CC(C)(C)c1.... |
5 | 4JPE | ic50 = 40 nM | 1M7 | C19 H21 N5 O | CC1(Cc2ccc.... |
6 | 4RCE | ic50 = 2 nM | 3LN | C24 H24 N4 O3 | CC(C)(C)CO.... |
7 | 1TQF | ic50 = 1.4 uM | 32P | C29 H34 F N3 O6 S | CC(c1ccc(c.... |
8 | 3L5E | ic50 = 27 nM | BDW | C32 H49 N5 O2 | CCCC1CN(C(.... |
9 | 2OHN | - | 4FP | C12 H16 F N | c1cc(ccc1C.... |
10 | 4R95 | Ki = 22 nM | 3KW | C28 H39 N5 O | CN1C(=O)C(.... |
11 | 2QMG | Ki = 0.7 nM | SC6 | C34 H39 F2 N3 O5 | Cc1cc(cc(c.... |
12 | 2WJO | - | QUD | C29 H37 N4 O2 | c1ccc(cc1).... |
13 | 4BFD | ic50 = 0.096 uM | 8T3 | C19 H18 Cl F N4 O | CC1(CC2CC2.... |
14 | 2XFK | ic50 = 3 nM | AA9 | C35 H47 N5 O5 S | CCNc1cc(cc.... |
15 | 4D89 | ic50 = 0.002 uM | BXD | C28 H38 F4 N2 O5 S | CCOCC(C(F).... |
16 | 4FM8 | ic50 = 2.4 uM | 0UQ | C24 H32 F N3 O3 S | CC1CC2(CCN.... |
17 | 2IQG | ic50 = 5 nM | F2I | C32 H38 F2 I N3 O3 | CCCN(CCC)C.... |
18 | 3HW1 | ic50 = 0.87 mM | EV2 | C12 H14 N4 | c1ccc2c(c1.... |
19 | 4JOO | ic50 = 36830 nM | 1M4 | C14 H16 Br N3 O2 | CC1(CC2(c3.... |
20 | 4FRI | ic50 = 2.85 uM | DWA | C21 H18 F N3 O2 | COc1ccc(cc.... |
21 | 2ZHR | - | GLU VAL ASN 1OL ALA GLU PHE | n/a | n/a |
22 | 2WF1 | ic50 = 0.002 uM | ZY1 | C32 H38 N4 O5 S | CCc1cn2c3c.... |
23 | 2QP8 | ic50 = 8 nM | SC7 | C31 H43 F2 N3 O4 | CCCN(CCC)C.... |
24 | 3NSH | ic50 = 470 nM | 957 | C24 H32 F2 N2 O2 S | CC(=O)NC(C.... |
25 | 4HZT | ic50 = 0.75 uM | 0ZA | C21 H21 Cl N4 O2 | CC1(Cc2cc(.... |
26 | 4BEK | ic50 = 41.2 uM | XK0 | C12 H16 N2 O S | CC1(CCSC(=.... |
27 | 4J1H | ic50 = 0.776 uM | 1HJ | C19 H15 F4 N5 O2 | CC1(CC(OC(.... |
28 | 4B78 | ic50 = 3.2 uM | KGG | C23 H23 N3 O2 | COc1ccc(cc.... |
29 | 4HA5 | Ki = 56 nM | 13W | C17 H16 N4 O S | CC1(CC(=O).... |
30 | 2P83 | ic50 = 11 nM | MR0 | C33 H40 F2 N4 O5 | CCCN(CCC)C.... |
31 | 4B1C | ic50 = 0.079 uM | 1B1 | C21 H20 N4 | CC#Cc1cc(c.... |
32 | 2OAH | Kd = 2 uM | QIN | C24 H37 N5 O3 S2 | CCCCC(C(Cc.... |
33 | 2B8V | ic50 = 98 nM | 3BN | C29 H33 N3 O5 S | CN(c1cc(cc.... |
34 | 2WF4 | ic50 = 13 nM | ZY4 | C29 H38 N4 O6 S | CCn1cc2c3c.... |
35 | 3IN4 | ic50 = 0.04 uM | BX2 | C23 H24 N6 O | CCc1cc(cc(.... |
36 | 3FKT | ic50 = 2.8 uM | SII | C28 H34 F N5 O2 | CC(=O)Nc1c.... |
37 | 3L5D | ic50 ~ 78000 nM | BDV | C21 H33 N5 O2 | CCCCNC(=O).... |
38 | 2ZE1 | ic50 = 0.6 uM | 411 | C26 H22 Br N5 O2 | [H]N=C(N)N.... |
39 | 2OHS | ic50 = 40 uM | 9IP | C18 H18 N4 O | COc1cc(cnc.... |
40 | 3UDH | ic50 = 1.1 mM | 091 | C11 H12 N2 O | c1ccc2c(c1.... |
41 | 3K5G | ic50 = 0.0025 uM | BJC | C35 H51 N3 O3 | CC(C)c1ccc.... |
42 | 3UDP | ic50 = 6 uM | 09D | C21 H19 Br N2 O3 S | c1ccc2c(c1.... |
43 | 4DH6 | ic50 = 16.8 nM | 0KN | C31 H43 N3 O6 | CC(C(=O)NC.... |
44 | 3RSV | ic50 = 0.0007 uM | 3RS | C27 H33 N3 O2 | Cc1ccccc1c.... |
45 | 3KMX | Kd = 15 uM | G00 | C12 H17 Cl N2 O S | CCCCOc1ccc.... |
46 | 4H3F | Ki = 1 nM | 10O | C24 H22 N6 O2 S | CN1C(=O)C2.... |
47 | 2QK5 | ic50 = 8 nM | CS5 | C33 H41 F2 N3 O4 | CCCN(CCC)C.... |
48 | 3UFL | ic50 = 0.15 uM | 508 | C31 H34 N2 O | c1ccc(cc1).... |
49 | 4I12 | ic50 = 40 uM | 1BC | C27 H29 Cl N6 O S | CCCc1c(c(c.... |
50 | 3LPK | Ki = 0.8 nM | Z76 | C35 H42 F2 N4 O6 S | Cc1cccc(c1.... |
51 | 3CKP | Ki = 5.001 uM | 012 | C31 H39 N5 O4 | CN(C)c1ccc.... |
52 | 4J1K | ic50 = 0.013 uM | 1HG | C19 H14 F5 N5 O2 | CC1(C(C(OC.... |
53 | 3PI5 | ic50 = 0.95 uM | 3P5 | C22 H26 Br N O4 S | c1cc(cc(c1.... |
54 | 1YM2 | - | ACE LEU MET 24O VAL LYT | n/a | n/a |
55 | 4J1C | ic50 = 0.049 uM | 1HO | C18 H13 F4 N5 O2 | c1cc(c(cc1.... |
56 | 3INH | ic50 = 0.02 uM | 569 | C21 H15 F4 N5 O2 | CN1C(=O)C(.... |
57 | 4N00 | ic50 = 9.5 nM | 2EX | C20 H19 F N4 O3 | CN1C(=O)C2.... |
58 | 2HIZ | ic50 = 112 nM | LIJ | C36 H49 N3 O7 S | CCCC(CCC)S.... |
59 | 2P4J | Ki = 1.1 nM | 23I | C36 H55 N5 O7 S | CC(C)CC(C(.... |
60 | 4I0D | ic50 = 0.61 uM | 1B7 | C21 H25 Cl N2 O2 S | CCCc1cscc1.... |
61 | 4R91 | Ki = 430 nM | 3KT | C24 H42 N4 O | CN1C(=O)C(.... |
62 | 4DJX | Ki = 59 nM | 0KQ | C18 H17 Cl N4 O | CN1C(=O)C(.... |
63 | 4ACU | ic50 = 0.00000001 M | QN7 | C24 H20 F3 N5 O | COc1cccc(c.... |
64 | 4H1E | Ki = 3 nM | 10J | C25 H21 N5 O2 S | CN1C(=O)C2.... |
65 | 2IRZ | ic50 = 12 nM | I02 | C28 H30 F N5 O4 S | CC(c1ccc(c.... |
66 | 2VNN | ic50 = 2 nM | CM7 | C32 H35 F3 N4 O4 S | CCc1cn2c3c.... |
67 | 4RRN | ic50 = 48 nM | 3UW | C20 H19 F N4 O3 | CN1C(=O)C2.... |
68 | 4H3I | Ki = 3 nM | 10V | C24 H22 N6 O2 S | CN1C(=O)C2.... |
69 | 2QZK | ic50 = 27 nM | I21 | C34 H27 N3 O3 | CC1(Cc2ccc.... |
70 | 4PZX | ic50 = 0.13 uM | 2X5 | C19 H18 Cl N3 O3 | c1cc2c(cc1.... |
71 | 4RRS | ic50 = 210 nM | 3UY | C20 H20 F N3 O3 | CC12CCCOC1.... |
72 | 4J0P | ic50 = 0.051 uM | 1H8 | C18 H16 F N5 O2 | CC1(CCOC(=.... |
73 | 2WEZ | ic50 = 0.023 uM | ZYE | C33 H38 N4 O4 | CCn1ccc2c1.... |
74 | 2OHU | ic50 = 4.2 uM | IP7 | C26 H23 N5 O | c1ccnc(c1).... |
75 | 3UDY | ic50 = 2 uM | 09G | C20 H16 Br N3 O3 | c1ccc2c(c1.... |
76 | 4JP9 | ic50 = 24 nM | 1M5 | C20 H20 Cl N3 O2 | CC1(CC2(c3.... |
77 | 3I25 | Ki = 3.1 nM | MV7 | C45 H55 F2 N5 O10 S | CC(C)C(C(=.... |
78 | 2VIZ | ic50 = 605 nM | VG4 | C33 H44 N4 O5 | CCCOc1cc(c.... |
79 | 4RCF | ic50 = 9 nM | 3LO | C25 H19 F2 N3 O3 | c1cc(c(nc1.... |
80 | 3LPJ | ic50 = 120 nM | Z75 | C35 H44 F2 N4 O3 | CCCN(CCC)C.... |
81 | 4EXG | ic50 = 8.5 nM | 916 | C26 H38 N2 O3 S | CC(=O)NC(C.... |
82 | 2XFJ | ic50 = 13 nM | VG5 | C32 H45 N5 O4 | CCNc1cc(cc.... |
83 | 4GID | Ki = 0.017 nM | 0GH | C35 H47 N5 O6 S | CC(C)CNC(=.... |
84 | 2F3E | ic50 = 156 nM | AXQ | C31 H55 N5 O7 S2 | CCCCNC(=O).... |
85 | 2VJ9 | ic50 = 180 nM | VG7 | C29 H40 N4 O3 | CCNc1cc(cc.... |
86 | 2VA7 | ic50 = 640 nM | C27 | C21 H25 N3 O2 | CC1(CC(=O).... |
87 | 3BRA | Kd = 2000 uM | AEF | C8 H11 N O | c1cc(ccc1C.... |
88 | 3KN0 | Kd = 100 uM | 3TO | C20 H23 N3 O | CN(Cc1cccc.... |
89 | 4DPF | ic50 = 400 nM | 0LG | C35 H44 N4 O6 S | CC(C)c1ccc.... |
90 | 4DJY | Ki = 5.4 nM | 0KR | C21 H20 N4 O | CC#Cc1cc(c.... |
91 | 2OHR | ic50 = 100 uM | 8IP | C17 H16 N4 | c1cc(cc(c1.... |
92 | 4D88 | ic50 = 0.049 uM | BXQ | C26 H34 F4 N2 O4 S | CC(C)(C)c1.... |
93 | 3MSL | ic50 = 7 uM | EV5 | C19 H27 Cl N4 O | CCC(CC(=O).... |
94 | 2OHQ | ic50 = 25 uM | 7IP | C20 H20 N2 O | COc1cccc(c.... |
95 | 2WF2 | ic50 = 0.026 uM | ZY2 | C32 H41 N5 O5 S | CCN1CCN2CC.... |
96 | 4I11 | ic50 = 27.2 uM | 1CH | C20 H22 N2 O2 | CC1(Cc2ccc.... |
97 | 3ZMG | ic50 = 0.023 uM | 6Z0 | C18 H14 F3 N5 O2 | CC1(C(COC(.... |
98 | 4I0Z | ic50 = 0.47 uM | 1BB | C24 H22 Cl N5 O | CC1(Cc2cc(.... |
99 | 2VKM | Ki = 1.8 nM | BSD | C36 H42 N4 O6 S | CC(c1ccccc.... |
100 | 4EWO | ic50 = 44 nM | 996 | C26 H40 N4 O2 | CC(=O)NC(C.... |
101 | 4B05 | Ki = 26 nM | 32D | C24 H16 F3 N5 | c1cc(cc(c1.... |
102 | 4J0V | ic50 = 0.028 uM | 1H7 | C18 H15 F2 N5 O2 | CC1(C(COC(.... |
103 | 4DI2 | ic50 = 5.5 nM | 0K9 | C33 H44 N4 O4 S | CC(C(=O)NC.... |
104 | 3OHF | ic50 = 94 nM | 3HF | C36 H46 N4 O4 | CCCCN(CCCC.... |
105 | 3L3A | ic50 = 0.42 uM | 625 | C26 H23 Cl N4 O | c1ccc(c(c1.... |
106 | 2ZDZ | ic50 = 0.7 uM | 310 | C27 H23 Cl N4 O3 | [H]N=C(N)N.... |
107 | 4I0G | - | 1B9 | C18 H18 Br Cl N2 O2 S | CC1(Cc2cc(.... |
108 | 3LNK | ic50 = 1150 nM | 74A | C35 H42 F2 N4 O4 | CCCN(CCC)C.... |
109 | 3IXJ | ic50 = 0.32 nM | 586 | C43 H51 F2 N5 O9 S | CC(C)C(C(=.... |
110 | 3L38 | ic50 = 0.1 uM | 879 | C26 H20 Cl N5 O | c1ccc(c(c1.... |
111 | 2VIY | ic50 = 1.8 uM | VG3 | C31 H45 N3 O5 S | CCCCCS(=O).... |
112 | 3L5C | ic50 = 7000 nM | BDQ | C24 H28 N6 O2 | CC(C)CC1(C.... |
113 | 4J17 | ic50 = 0.054 uM | 1HQ | C18 H14 F3 N5 O2 | c1cc(c(cc1.... |
114 | 3IXK | ic50 = 6.6 nM | 929 | C44 H53 F2 N5 O8 S | CC(C)C(C(=.... |
115 | 4K8S | ic50 = 0.036 uM | 1QT | C32 H44 N2 O3 | CCc1ccc2c(.... |
116 | 2FDP | Ki = 0.026 uM | FRP | C33 H41 F N4 O3 | CCCN(CCC)C.... |
117 | 3BUH | Kd = 220 uM | AED | C14 H21 N O | c1cc(c(cc1.... |
118 | 1YM4 | ic50 = 0.039 uM | GLU VAL ASN 24M ALA | n/a | n/a |
119 | 4FRK | ic50 = 0.008 uM | DWD | C23 H22 N4 O3 | CC(C)COc1c.... |
120 | 4KE0 | ic50 = 0.017 uM | 1R8 | C31 H42 N2 O3 | CCc1ccc2c(.... |
121 | 2G94 | Ki = 0.3 nM | ZPQ | C30 H54 N6 O8 S | Cc1cc(n(n1.... |
122 | 4I0E | - | 1B8 | C21 H20 Br Cl N4 O2 S | CC1(Cc2cc(.... |
123 | 4AZY | ic50 = 125 nM | 7F3 | C24 H14 F5 N5 | c1cc2c(c(c.... |
124 | 4FGX | ic50 = 73 nM | 2OP VAL GNC PSA LEU ALA ZAE | n/a | n/a |
125 | 4I1C | ic50 = 0.4 uM | 1BE | C24 H27 Cl N4 O2 S | CCCc1c(c(c.... |
126 | 4B77 | ic50 = 7.9 uM | 54M | C21 H20 N4 O | COc1ccc(cc.... |
127 | 3VV8 | ic50 = 17.1 uM | B02 | C21 H21 N3 O | Cc1cccc(c1.... |
128 | 3EXO | ic50 = 24 uM | 5MS | C18 H18 N4 O2 S | Cc1ccc(cc1.... |
129 | 3S7L | ic50 = 0.08 uM | 591 | C19 H19 N7 O | CCn1cc(cn1.... |
130 | 2VJ6 | ic50 = 13 nM | VG5 | C32 H45 N5 O4 | CCNc1cc(cc.... |
131 | 3DUY | ic50 = 1.4 uM | AFJ | C25 H49 N3 O4 S | CCCCNC(=O).... |
132 | 3L58 | ic50 = 8 nM | CS5 | C33 H41 F2 N3 O4 | CCCN(CCC)C.... |
133 | 4JPC | ic50 = 94 nM | 1M6 | C21 H20 N4 O2 | CC1(CC2(c3.... |
134 | 4J0T | ic50 = 0.148 uM | 6T9 | C19 H19 F3 N4 O3 | CCOc1ccc(n.... |
135 | 3RU1 | Kd = 14.2 uM | 3RU | C19 H25 N3 O | c1ccc2c(c1.... |
136 | 3K5F | ic50 = 3.7 uM | AYH | C29 H47 N3 O4 | CCCCNC(=O).... |
137 | 4J0Z | ic50 = 0.077 uM | 1H5 | C18 H14 F3 N5 O2 | c1cc(c(cc1.... |
138 | 3RSX | Kd = 38.8 uM | RSV | C13 H10 N2 S | c1cc(nc2c1.... |
139 | 2VA6 | ic50 = 590 nM | H24 | C19 H21 N3 O2 | CC1(CC(=O).... |
140 | 4B00 | ic50 = 2.44 nM | I6X | C30 H25 F N4 O | CCN1C=C(C=.... |
141 | 3VV6 | ic50 = 157 uM | B00 | C14 H15 N3 O | CN1C(=O)C=.... |
142 | 4IVT | ic50 = 1.7 uM | VTI | C20 H19 Cl2 N5 O2 | CC(=O)Nc1c.... |
143 | 3LPI | ic50 = 5 nM | Z74 | C34 H42 F2 N4 O5 S | CCCN(CCC)C.... |
144 | 4J1F | ic50 = 0.012 uM | 1HL | C19 H15 F4 N5 O2 | CC1(CC(OC(.... |
145 | 4DJU | Ki = 3.6 uM | 0KK | C16 H15 N3 O | CN1C(=O)C(.... |
146 | 2OHT | ic50 = 9.1 uM | IP6 | C20 H18 N4 | c1cc(cc(c1.... |
147 | 2OHK | - | 1SQ | C9 H8 N2 | c1ccc2c(c1.... |
148 | 3UDN | ic50 = 7 uM | 09B | C20 H17 N3 O3 | c1ccc2c(c1.... |
149 | 4J1I | ic50 = 0.04 uM | 1HH | C19 H14 F5 N5 O2 | CC1(C(C(OC.... |
150 | 2QMF | ic50 = 3 nM | CS9 | C34 H41 F2 N3 O4 | CCCN(CCC)C.... |
151 | 3CIC | ic50 = 3 nM | 316 | C35 H42 F2 N4 O4 | CCCN(CCC)C.... |
152 | 4I10 | ic50 = 0.17 uM | 1BS | C26 H24 Cl N5 O | CC1(Cc2cc(.... |
153 | 3IGB | ic50 = 38 uM | 454 | C18 H18 N4 | c1ccc(cc1).... |
154 | 1M4H | - | GLU LEU ASP 1OL VAL GLU PHE | n/a | n/a |
155 | 2F3F | ic50 = 190 nM | AXF | C24 H42 N4 O4 S2 | CCCCNC(=O).... |
156 | 3INF | ic50 = 0.04 uM | X45 | C23 H22 N4 O2 | Cc1cc(ccc1.... |
157 | 3MSK | ic50 = 26 uM | EV4 | C18 H25 Cl N4 O | CN(C1CCCCC.... |
158 | 4R93 | Ki = 16 nM | 779 | C26 H39 N5 O2 | CN1C(=O)C(.... |
159 | 3IVI | ic50 = 12 nM | 2LI | C29 H36 F2 N4 O2 | CC(=O)NC(C.... |
160 | 4B72 | ic50 = 0.63 uM | 2FB | C23 H19 N5 O S | Cc1nc2c(s1.... |
161 | 4R5N | ic50 = 76 nM | 3J9 | C20 H20 F N3 O3 | CC12CCCOC1.... |
162 | 2PH6 | ic50 = 27 nM | 712 | C28 H32 F N3 O5 S | CC(c1ccc(c.... |
163 | 4I0F | ic50 = 0.45 uM | 1BF | C21 H21 Cl N4 O2 S | CC1(Cc2cc(.... |
164 | 4H3G | Ki = 6 nM | 10Q | C24 H19 N7 O S | CN1C(=O)C2.... |
165 | 2QU3 | ic50 = 0.59 uM | 462 | C22 H22 Cl N3 O2 S | [H]N=C(N)N.... |
166 | 4B1E | - | 6T6 | C21 H20 N4 | CC1(NC(=C(.... |
167 | 4DVF | ic50 = 128 nM | QSC USC PSA LEU ALA ZAE PLJ | n/a | n/a |
168 | 4DV9 | ic50 = 189 nM | 2OP VAL GNC PSA LEU ALA ZAE PLJ | n/a | n/a |
169 | 3L5F | ic50 = 605 nM | BDX | C19 H33 N3 O | CN1C(=O)C(.... |
170 | 4LXM | ic50 = 0.088 uM | 1YU | C26 H31 F7 N2 O3 S | CC(C)(C)c1.... |
171 | 2OHP | ic50 = 94 uM | 6IP | C15 H15 N3 | c1cc(nc(c1.... |
172 | 3UDJ | ic50 = 242 uM | 092 | C13 H14 N2 O3 | COC(=O)C1C.... |
173 | 2XFI | ic50 = 15 nM | XFI | C33 H42 N4 O5 S | CC(C(=O)NC.... |
174 | 2OF0 | - | CMZ | C15 H23 N O3 | Cc1ccc(c(c.... |
175 | 4LXA | ic50 = 0.002 uM | 1YS | C26 H31 F7 N2 O3 S | CC(C)(C)c1.... |
176 | 3UDR | ic50 = 11 uM | 09F | C19 H21 N3 O3 | c1ccc2c(c1.... |
177 | 3TPP | ic50 = 15 nM | 5HA | C31 H38 N4 O5 S | CC(c1ccccc.... |
178 | 2IS0 | ic50 = 200 nM | I03 | C28 H32 F N3 O6 S | CC(c1ccc(c.... |
179 | 3K5C | ic50 = 17 nM | 0BI | C35 H45 N3 O4 | CC(C)c1ccc.... |
180 | 3LHG | ic50 = 0.02 uM | Z81 | C21 H16 F2 N4 O | CN1C(=O)C(.... |
181 | 3L5B | Kd = 123 uM | BDO | C15 H20 Cl N3 O | CC(C)CC1(C.... |
182 | 3S7M | ic50 = 0.06 uM | 532 | C19 H16 N4 O S | CN1C(=O)C(.... |
183 | 4B70 | ic50 = 6.3 uM | WM9 | C17 H17 Cl N2 O | CC1(N=C(CC.... |
184 | 3VEU | ic50 = 55 nM | 0GO | C33 H48 N4 O3 | CCCN1CCCC1.... |
185 | 4DJV | Ki = 0.19 uM | 0KM | C23 H21 N3 O2 | CN1C(=O)C(.... |
186 | 4R8Y | Ki = 0.64 uM | 3KO | C24 H40 N4 O2 | CN1C(=O)C(.... |
187 | 2VJ7 | ic50 = 40 nM | VG6 | C31 H35 F3 N4 O3 | CCNc1cc(cc.... |
188 | 3ZOV | - | WZV | C20 H20 F3 N5 O3 | CC1(CC(=O).... |
189 | 3INE | ic50 = 0.17 uM | X17 | C22 H29 N3 O2 | Cc1cc(ccc1.... |
190 | 4J0Y | ic50 = 0.435 uM | 1H6 | C18 H15 F2 N5 O2 | CC1(C(COC(.... |
191 | 2Q15 | Ki = 11 nM | 3MR | C31 H42 N4 O2 | CN(C1CCCCC.... |
192 | 4J1E | ic50 = 0.019 uM | 1HM | C19 H14 F5 N5 O2 | c1cc(c(cc1.... |
193 | 4D8C | ic50 = 0.002 uM | BXD | C28 H38 F4 N2 O5 S | CCOCC(C(F).... |
194 | 2VIE | ic50 = 33 nM | VG0 | C32 H48 N4 O3 | CCNc1cc(cc.... |
195 | 2NTR | - | L00 | C26 H35 Cl N6 O4 S | CC1CC1CN(C.... |
196 | 3VV7 | ic50 = 4.6 uM | 0B1 | C21 H21 N3 O2 | CN1C(=O)C=.... |
197 | 3DV5 | ic50 = 0.027 uM | BAV | C29 H49 N3 O3 | CC1CCCCCCC.... |
198 | 3L59 | Kd = 200 uM | BDJ | C12 H14 Cl N3 O | CC1(C(=O)N.... |
199 | 2VIJ | - | C44 | C33 H42 N4 O4 S | CCNc1cc(cc.... |
200 | 4FM7 | ic50 = 0.1 uM | 0UP | C24 H32 F N3 O4 S | CC1CC2(CCN.... |
201 | 3UDM | ic50 = 33 uM | 09A | C19 H18 N2 O3 | c1ccc(cc1).... |
202 | 1FKN | - | GLU VAL ASN 1OL ALA GLU PHE | n/a | n/a |
203 | 4D83 | ic50 = 0.055 uM | 0GT | C27 H34 F2 N2 O3 S | CC(C)(C)c1.... |
204 | 4DPI | ic50 = 78 nM | 0N1 | C34 H41 N3 O4 | Cc1cc2cc(c.... |
205 | 4B1D | ic50 = 0.012 uM | 6TG | C23 H23 N5 O | Cc1cc(cc(c.... |
206 | 4ACX | ic50 = 0.00000001 M | S8Z | C23 H20 F4 N4 O2 | COCC#Cc1cc.... |
207 | 3VG1 | ic50 = 0.055 uM | 0GT | C27 H34 F2 N2 O3 S | CC(C)(C)c1.... |
208 | 2P8H | ic50 = 71 nM | MY9 | C33 H40 F N5 O6 S | CC(c1ccc(c.... |
209 | 3BUG | Kd = 660 uM | AEH | C10 H15 N O | CCc1cc(ccc.... |
210 | 2QMD | ic50 = 5 nM | CS7 | C35 H43 F2 N3 O4 | CCCN(CCC)C.... |
211 | 4KE1 | ic50 = 0.0025 uM | 1R6 | C34 H41 N3 O4 | CCc1ccc2c(.... |
212 | 2WF0 | ic50 = 0.21 uM | ZY0 | C34 H35 F3 N4 O3 | CCc1ccnc2c.... |
213 | 3IN3 | ic50 = 0.06 uM | 472 | C20 H17 N5 O | CN1C(=O)C(.... |
214 | 3HVG | ic50 ~ 2 mM | EV0 | C7 H11 N3 O | CCCC1=CC(=.... |
215 | 3CIB | ic50 = 14 nM | 314 | C36 H45 F2 N3 O3 | CCCN(CCC)C.... |
216 | 3OHH | ic50 = 18 nM | 3HH | C34 H37 F2 N5 O4 | CCCCN(C)C(.... |
217 | 2WF3 | ic50 = 0.019 uM | ZY3 | C31 H40 N4 O5 S | CCNc1cc(cc.... |
218 | 3WB5 | ic50 = 18 uM | 0B4 | C15 H19 N3 O | CC1(CC(=O).... |
219 | 4RRO | ic50 = 26 nM | 3UX | C21 H21 F N4 O3 | CC12CCCOC1.... |
220 | 3VF3 | ic50 = 1.37 uM | 0GS | C21 H24 Br F3 N2 O3 S | CC(c1cccc(.... |
221 | 4FRJ | ic50 = 0.28 uM | DWB | C22 H16 Cl F N2 O3 | COc1ccc2c(.... |
222 | 2VNM | ic50 = 3 nM | CM8 | C31 H37 F3 N4 O4 S | CCNc1cc(cc.... |
223 | 2Q11 | Ki = 900 nM | XX4 | C25 H30 N4 O2 | CN(C1CCCCC.... |
224 | 3CID | ic50 = 5 nM | 318 | C34 H40 F2 N4 O4 | CCCN(CCC)C.... |
225 | 3QBH | ic50 = 0.15 uM | QBH | C29 H40 N2 O6 S | CCCN1C(COC.... |
226 | 3KMY | Kd = 32 uM | D8Y | C13 H13 Cl N2 | c1cc(cc(c1.... |
227 | 4R92 | Ki = 39 nM | 3KU | C25 H37 N5 O2 | CN1C(=O)C(.... |
228 | 4DJW | Ki = 0.53 uM | 0KP | C21 H18 N4 O | CN1C(=O)C(.... |
229 | 3IVH | ic50 = 47 nM | 1LI | C28 H38 F2 N2 O2 | CC(=O)NC(C.... |
230 | 3MSJ | ic50 = 770 uM | EV3 | C10 H12 Cl N3 O | c1cc2c(cc1.... |
231 | 3DV1 | ic50 = 0.59 uM | AR9 | C24 H45 N3 O4 | CCCCNC(=O).... |
232 | 3BUF | Kd = 800 uM | AEG | C9 H13 N O | CC(Cc1ccc(.... |
233 | 4H3J | Ki = 90 nM | 10W | C24 H20 F N5 O S | CN1C(=O)C2.... |
234 | 4PZW | ic50 = 0.11 uM | 2X4 | C19 H18 Cl N3 O3 | c1cc2c(cc1.... |
235 | 2QZL | ic50 = 8 nM | IXS | C34 H44 F N5 O5 S | CC(C)CNC(=.... |
236 | 3WB4 | ic50 = 220 uM | 0B3 | C14 H19 N3 O | CC1(CC(=O).... |
237 | 3OOZ | ic50 = 0.014 uM | ZOO | C22 H19 F4 N3 O2 | CN1C(=O)C(.... |
238 | 2PH8 | ic50 = 1800 nM | 35A | C24 H33 N3 O4 S | CC1CCc2ccc.... |
239 | 4K9H | ic50 = 0.076 uM | 1QU | C33 H37 F3 N4 O4 | c1ccc(cc1).... |
240 | 3ZKI | - | WZV | C20 H20 F3 N5 O3 | CC1(CC(=O).... |
No: | PDB id | Binding Data | Representative ligand | Formula | Smiles |
---|---|---|---|---|---|
The Class containing this family consists of a total of 1 families. | |||||
1 | 3IND | ic50 = 1.53 uM | 593 | C20 H25 N3 O | CN1C(=O)C(.... |
2 | 2HM1 | ic50 = 13 nM | LIQ | C33 H42 F2 N4 O5 S | CCCCCS(=O).... |
3 | 2B8L | ic50 = 15 nM | 5HA | C31 H38 N4 O5 S | CC(c1ccccc.... |
4 | 4LXK | ic50 = 0.004 uM | 1YT | C27 H36 F4 N2 O4 S | CC(C)(C)c1.... |
5 | 4JPE | ic50 = 40 nM | 1M7 | C19 H21 N5 O | CC1(Cc2ccc.... |
6 | 4RCE | ic50 = 2 nM | 3LN | C24 H24 N4 O3 | CC(C)(C)CO.... |
7 | 1TQF | ic50 = 1.4 uM | 32P | C29 H34 F N3 O6 S | CC(c1ccc(c.... |
8 | 3L5E | ic50 = 27 nM | BDW | C32 H49 N5 O2 | CCCC1CN(C(.... |
9 | 2OHN | - | 4FP | C12 H16 F N | c1cc(ccc1C.... |
10 | 4R95 | Ki = 22 nM | 3KW | C28 H39 N5 O | CN1C(=O)C(.... |
11 | 2QMG | Ki = 0.7 nM | SC6 | C34 H39 F2 N3 O5 | Cc1cc(cc(c.... |
12 | 2WJO | - | QUD | C29 H37 N4 O2 | c1ccc(cc1).... |
13 | 4BFD | ic50 = 0.096 uM | 8T3 | C19 H18 Cl F N4 O | CC1(CC2CC2.... |
14 | 2XFK | ic50 = 3 nM | AA9 | C35 H47 N5 O5 S | CCNc1cc(cc.... |
15 | 4D89 | ic50 = 0.002 uM | BXD | C28 H38 F4 N2 O5 S | CCOCC(C(F).... |
16 | 4FM8 | ic50 = 2.4 uM | 0UQ | C24 H32 F N3 O3 S | CC1CC2(CCN.... |
17 | 2IQG | ic50 = 5 nM | F2I | C32 H38 F2 I N3 O3 | CCCN(CCC)C.... |
18 | 3HW1 | ic50 = 0.87 mM | EV2 | C12 H14 N4 | c1ccc2c(c1.... |
19 | 4JOO | ic50 = 36830 nM | 1M4 | C14 H16 Br N3 O2 | CC1(CC2(c3.... |
20 | 4FRI | ic50 = 2.85 uM | DWA | C21 H18 F N3 O2 | COc1ccc(cc.... |
21 | 2ZHR | - | GLU VAL ASN 1OL ALA GLU PHE | n/a | n/a |
22 | 2WF1 | ic50 = 0.002 uM | ZY1 | C32 H38 N4 O5 S | CCc1cn2c3c.... |
23 | 2QP8 | ic50 = 8 nM | SC7 | C31 H43 F2 N3 O4 | CCCN(CCC)C.... |
24 | 3NSH | ic50 = 470 nM | 957 | C24 H32 F2 N2 O2 S | CC(=O)NC(C.... |
25 | 4HZT | ic50 = 0.75 uM | 0ZA | C21 H21 Cl N4 O2 | CC1(Cc2cc(.... |
26 | 4BEK | ic50 = 41.2 uM | XK0 | C12 H16 N2 O S | CC1(CCSC(=.... |
27 | 4J1H | ic50 = 0.776 uM | 1HJ | C19 H15 F4 N5 O2 | CC1(CC(OC(.... |
28 | 4B78 | ic50 = 3.2 uM | KGG | C23 H23 N3 O2 | COc1ccc(cc.... |
29 | 4HA5 | Ki = 56 nM | 13W | C17 H16 N4 O S | CC1(CC(=O).... |
30 | 2P83 | ic50 = 11 nM | MR0 | C33 H40 F2 N4 O5 | CCCN(CCC)C.... |
31 | 4B1C | ic50 = 0.079 uM | 1B1 | C21 H20 N4 | CC#Cc1cc(c.... |
32 | 2OAH | Kd = 2 uM | QIN | C24 H37 N5 O3 S2 | CCCCC(C(Cc.... |
33 | 2B8V | ic50 = 98 nM | 3BN | C29 H33 N3 O5 S | CN(c1cc(cc.... |
34 | 2WF4 | ic50 = 13 nM | ZY4 | C29 H38 N4 O6 S | CCn1cc2c3c.... |
35 | 3IN4 | ic50 = 0.04 uM | BX2 | C23 H24 N6 O | CCc1cc(cc(.... |
36 | 3FKT | ic50 = 2.8 uM | SII | C28 H34 F N5 O2 | CC(=O)Nc1c.... |
37 | 3L5D | ic50 ~ 78000 nM | BDV | C21 H33 N5 O2 | CCCCNC(=O).... |
38 | 2ZE1 | ic50 = 0.6 uM | 411 | C26 H22 Br N5 O2 | [H]N=C(N)N.... |
39 | 2OHS | ic50 = 40 uM | 9IP | C18 H18 N4 O | COc1cc(cnc.... |
40 | 3UDH | ic50 = 1.1 mM | 091 | C11 H12 N2 O | c1ccc2c(c1.... |
41 | 3K5G | ic50 = 0.0025 uM | BJC | C35 H51 N3 O3 | CC(C)c1ccc.... |
42 | 3UDP | ic50 = 6 uM | 09D | C21 H19 Br N2 O3 S | c1ccc2c(c1.... |
43 | 4DH6 | ic50 = 16.8 nM | 0KN | C31 H43 N3 O6 | CC(C(=O)NC.... |
44 | 3RSV | ic50 = 0.0007 uM | 3RS | C27 H33 N3 O2 | Cc1ccccc1c.... |
45 | 3KMX | Kd = 15 uM | G00 | C12 H17 Cl N2 O S | CCCCOc1ccc.... |
46 | 4H3F | Ki = 1 nM | 10O | C24 H22 N6 O2 S | CN1C(=O)C2.... |
47 | 2QK5 | ic50 = 8 nM | CS5 | C33 H41 F2 N3 O4 | CCCN(CCC)C.... |
48 | 3UFL | ic50 = 0.15 uM | 508 | C31 H34 N2 O | c1ccc(cc1).... |
49 | 4I12 | ic50 = 40 uM | 1BC | C27 H29 Cl N6 O S | CCCc1c(c(c.... |
50 | 3LPK | Ki = 0.8 nM | Z76 | C35 H42 F2 N4 O6 S | Cc1cccc(c1.... |
51 | 3CKP | Ki = 5.001 uM | 012 | C31 H39 N5 O4 | CN(C)c1ccc.... |
52 | 4J1K | ic50 = 0.013 uM | 1HG | C19 H14 F5 N5 O2 | CC1(C(C(OC.... |
53 | 3PI5 | ic50 = 0.95 uM | 3P5 | C22 H26 Br N O4 S | c1cc(cc(c1.... |
54 | 1YM2 | - | ACE LEU MET 24O VAL LYT | n/a | n/a |
55 | 4J1C | ic50 = 0.049 uM | 1HO | C18 H13 F4 N5 O2 | c1cc(c(cc1.... |
56 | 3INH | ic50 = 0.02 uM | 569 | C21 H15 F4 N5 O2 | CN1C(=O)C(.... |
57 | 4N00 | ic50 = 9.5 nM | 2EX | C20 H19 F N4 O3 | CN1C(=O)C2.... |
58 | 2HIZ | ic50 = 112 nM | LIJ | C36 H49 N3 O7 S | CCCC(CCC)S.... |
59 | 2P4J | Ki = 1.1 nM | 23I | C36 H55 N5 O7 S | CC(C)CC(C(.... |
60 | 4I0D | ic50 = 0.61 uM | 1B7 | C21 H25 Cl N2 O2 S | CCCc1cscc1.... |
61 | 4R91 | Ki = 430 nM | 3KT | C24 H42 N4 O | CN1C(=O)C(.... |
62 | 4DJX | Ki = 59 nM | 0KQ | C18 H17 Cl N4 O | CN1C(=O)C(.... |
63 | 4ACU | ic50 = 0.00000001 M | QN7 | C24 H20 F3 N5 O | COc1cccc(c.... |
64 | 4H1E | Ki = 3 nM | 10J | C25 H21 N5 O2 S | CN1C(=O)C2.... |
65 | 2IRZ | ic50 = 12 nM | I02 | C28 H30 F N5 O4 S | CC(c1ccc(c.... |
66 | 2VNN | ic50 = 2 nM | CM7 | C32 H35 F3 N4 O4 S | CCc1cn2c3c.... |
67 | 4RRN | ic50 = 48 nM | 3UW | C20 H19 F N4 O3 | CN1C(=O)C2.... |
68 | 4H3I | Ki = 3 nM | 10V | C24 H22 N6 O2 S | CN1C(=O)C2.... |
69 | 2QZK | ic50 = 27 nM | I21 | C34 H27 N3 O3 | CC1(Cc2ccc.... |
70 | 4PZX | ic50 = 0.13 uM | 2X5 | C19 H18 Cl N3 O3 | c1cc2c(cc1.... |
71 | 4RRS | ic50 = 210 nM | 3UY | C20 H20 F N3 O3 | CC12CCCOC1.... |
72 | 4J0P | ic50 = 0.051 uM | 1H8 | C18 H16 F N5 O2 | CC1(CCOC(=.... |
73 | 2WEZ | ic50 = 0.023 uM | ZYE | C33 H38 N4 O4 | CCn1ccc2c1.... |
74 | 2OHU | ic50 = 4.2 uM | IP7 | C26 H23 N5 O | c1ccnc(c1).... |
75 | 3UDY | ic50 = 2 uM | 09G | C20 H16 Br N3 O3 | c1ccc2c(c1.... |
76 | 4JP9 | ic50 = 24 nM | 1M5 | C20 H20 Cl N3 O2 | CC1(CC2(c3.... |
77 | 3I25 | Ki = 3.1 nM | MV7 | C45 H55 F2 N5 O10 S | CC(C)C(C(=.... |
78 | 2VIZ | ic50 = 605 nM | VG4 | C33 H44 N4 O5 | CCCOc1cc(c.... |
79 | 4RCF | ic50 = 9 nM | 3LO | C25 H19 F2 N3 O3 | c1cc(c(nc1.... |
80 | 3LPJ | ic50 = 120 nM | Z75 | C35 H44 F2 N4 O3 | CCCN(CCC)C.... |
81 | 4EXG | ic50 = 8.5 nM | 916 | C26 H38 N2 O3 S | CC(=O)NC(C.... |
82 | 2XFJ | ic50 = 13 nM | VG5 | C32 H45 N5 O4 | CCNc1cc(cc.... |
83 | 4GID | Ki = 0.017 nM | 0GH | C35 H47 N5 O6 S | CC(C)CNC(=.... |
84 | 2F3E | ic50 = 156 nM | AXQ | C31 H55 N5 O7 S2 | CCCCNC(=O).... |
85 | 2VJ9 | ic50 = 180 nM | VG7 | C29 H40 N4 O3 | CCNc1cc(cc.... |
86 | 2VA7 | ic50 = 640 nM | C27 | C21 H25 N3 O2 | CC1(CC(=O).... |
87 | 3BRA | Kd = 2000 uM | AEF | C8 H11 N O | c1cc(ccc1C.... |
88 | 3KN0 | Kd = 100 uM | 3TO | C20 H23 N3 O | CN(Cc1cccc.... |
89 | 4DPF | ic50 = 400 nM | 0LG | C35 H44 N4 O6 S | CC(C)c1ccc.... |
90 | 4DJY | Ki = 5.4 nM | 0KR | C21 H20 N4 O | CC#Cc1cc(c.... |
91 | 2OHR | ic50 = 100 uM | 8IP | C17 H16 N4 | c1cc(cc(c1.... |
92 | 4D88 | ic50 = 0.049 uM | BXQ | C26 H34 F4 N2 O4 S | CC(C)(C)c1.... |
93 | 3MSL | ic50 = 7 uM | EV5 | C19 H27 Cl N4 O | CCC(CC(=O).... |
94 | 2OHQ | ic50 = 25 uM | 7IP | C20 H20 N2 O | COc1cccc(c.... |
95 | 2WF2 | ic50 = 0.026 uM | ZY2 | C32 H41 N5 O5 S | CCN1CCN2CC.... |
96 | 4I11 | ic50 = 27.2 uM | 1CH | C20 H22 N2 O2 | CC1(Cc2ccc.... |
97 | 3ZMG | ic50 = 0.023 uM | 6Z0 | C18 H14 F3 N5 O2 | CC1(C(COC(.... |
98 | 4I0Z | ic50 = 0.47 uM | 1BB | C24 H22 Cl N5 O | CC1(Cc2cc(.... |
99 | 2VKM | Ki = 1.8 nM | BSD | C36 H42 N4 O6 S | CC(c1ccccc.... |
100 | 4EWO | ic50 = 44 nM | 996 | C26 H40 N4 O2 | CC(=O)NC(C.... |
101 | 4B05 | Ki = 26 nM | 32D | C24 H16 F3 N5 | c1cc(cc(c1.... |
102 | 4J0V | ic50 = 0.028 uM | 1H7 | C18 H15 F2 N5 O2 | CC1(C(COC(.... |
103 | 4DI2 | ic50 = 5.5 nM | 0K9 | C33 H44 N4 O4 S | CC(C(=O)NC.... |
104 | 3OHF | ic50 = 94 nM | 3HF | C36 H46 N4 O4 | CCCCN(CCCC.... |
105 | 3L3A | ic50 = 0.42 uM | 625 | C26 H23 Cl N4 O | c1ccc(c(c1.... |
106 | 2ZDZ | ic50 = 0.7 uM | 310 | C27 H23 Cl N4 O3 | [H]N=C(N)N.... |
107 | 4I0G | - | 1B9 | C18 H18 Br Cl N2 O2 S | CC1(Cc2cc(.... |
108 | 3LNK | ic50 = 1150 nM | 74A | C35 H42 F2 N4 O4 | CCCN(CCC)C.... |
109 | 3IXJ | ic50 = 0.32 nM | 586 | C43 H51 F2 N5 O9 S | CC(C)C(C(=.... |
110 | 3L38 | ic50 = 0.1 uM | 879 | C26 H20 Cl N5 O | c1ccc(c(c1.... |
111 | 2VIY | ic50 = 1.8 uM | VG3 | C31 H45 N3 O5 S | CCCCCS(=O).... |
112 | 3L5C | ic50 = 7000 nM | BDQ | C24 H28 N6 O2 | CC(C)CC1(C.... |
113 | 4J17 | ic50 = 0.054 uM | 1HQ | C18 H14 F3 N5 O2 | c1cc(c(cc1.... |
114 | 3IXK | ic50 = 6.6 nM | 929 | C44 H53 F2 N5 O8 S | CC(C)C(C(=.... |
115 | 4K8S | ic50 = 0.036 uM | 1QT | C32 H44 N2 O3 | CCc1ccc2c(.... |
116 | 2FDP | Ki = 0.026 uM | FRP | C33 H41 F N4 O3 | CCCN(CCC)C.... |
117 | 3BUH | Kd = 220 uM | AED | C14 H21 N O | c1cc(c(cc1.... |
118 | 1YM4 | ic50 = 0.039 uM | GLU VAL ASN 24M ALA | n/a | n/a |
119 | 4FRK | ic50 = 0.008 uM | DWD | C23 H22 N4 O3 | CC(C)COc1c.... |
120 | 4KE0 | ic50 = 0.017 uM | 1R8 | C31 H42 N2 O3 | CCc1ccc2c(.... |
121 | 2G94 | Ki = 0.3 nM | ZPQ | C30 H54 N6 O8 S | Cc1cc(n(n1.... |
122 | 4I0E | - | 1B8 | C21 H20 Br Cl N4 O2 S | CC1(Cc2cc(.... |
123 | 4AZY | ic50 = 125 nM | 7F3 | C24 H14 F5 N5 | c1cc2c(c(c.... |
124 | 4FGX | ic50 = 73 nM | 2OP VAL GNC PSA LEU ALA ZAE | n/a | n/a |
125 | 4I1C | ic50 = 0.4 uM | 1BE | C24 H27 Cl N4 O2 S | CCCc1c(c(c.... |
126 | 4B77 | ic50 = 7.9 uM | 54M | C21 H20 N4 O | COc1ccc(cc.... |
127 | 3VV8 | ic50 = 17.1 uM | B02 | C21 H21 N3 O | Cc1cccc(c1.... |
128 | 3EXO | ic50 = 24 uM | 5MS | C18 H18 N4 O2 S | Cc1ccc(cc1.... |
129 | 3S7L | ic50 = 0.08 uM | 591 | C19 H19 N7 O | CCn1cc(cn1.... |
130 | 2VJ6 | ic50 = 13 nM | VG5 | C32 H45 N5 O4 | CCNc1cc(cc.... |
131 | 3DUY | ic50 = 1.4 uM | AFJ | C25 H49 N3 O4 S | CCCCNC(=O).... |
132 | 3L58 | ic50 = 8 nM | CS5 | C33 H41 F2 N3 O4 | CCCN(CCC)C.... |
133 | 4JPC | ic50 = 94 nM | 1M6 | C21 H20 N4 O2 | CC1(CC2(c3.... |
134 | 4J0T | ic50 = 0.148 uM | 6T9 | C19 H19 F3 N4 O3 | CCOc1ccc(n.... |
135 | 3RU1 | Kd = 14.2 uM | 3RU | C19 H25 N3 O | c1ccc2c(c1.... |
136 | 3K5F | ic50 = 3.7 uM | AYH | C29 H47 N3 O4 | CCCCNC(=O).... |
137 | 4J0Z | ic50 = 0.077 uM | 1H5 | C18 H14 F3 N5 O2 | c1cc(c(cc1.... |
138 | 3RSX | Kd = 38.8 uM | RSV | C13 H10 N2 S | c1cc(nc2c1.... |
139 | 2VA6 | ic50 = 590 nM | H24 | C19 H21 N3 O2 | CC1(CC(=O).... |
140 | 4B00 | ic50 = 2.44 nM | I6X | C30 H25 F N4 O | CCN1C=C(C=.... |
141 | 3VV6 | ic50 = 157 uM | B00 | C14 H15 N3 O | CN1C(=O)C=.... |
142 | 4IVT | ic50 = 1.7 uM | VTI | C20 H19 Cl2 N5 O2 | CC(=O)Nc1c.... |
143 | 3LPI | ic50 = 5 nM | Z74 | C34 H42 F2 N4 O5 S | CCCN(CCC)C.... |
144 | 4J1F | ic50 = 0.012 uM | 1HL | C19 H15 F4 N5 O2 | CC1(CC(OC(.... |
145 | 4DJU | Ki = 3.6 uM | 0KK | C16 H15 N3 O | CN1C(=O)C(.... |
146 | 2OHT | ic50 = 9.1 uM | IP6 | C20 H18 N4 | c1cc(cc(c1.... |
147 | 2OHK | - | 1SQ | C9 H8 N2 | c1ccc2c(c1.... |
148 | 3UDN | ic50 = 7 uM | 09B | C20 H17 N3 O3 | c1ccc2c(c1.... |
149 | 4J1I | ic50 = 0.04 uM | 1HH | C19 H14 F5 N5 O2 | CC1(C(C(OC.... |
150 | 2QMF | ic50 = 3 nM | CS9 | C34 H41 F2 N3 O4 | CCCN(CCC)C.... |
151 | 3CIC | ic50 = 3 nM | 316 | C35 H42 F2 N4 O4 | CCCN(CCC)C.... |
152 | 4I10 | ic50 = 0.17 uM | 1BS | C26 H24 Cl N5 O | CC1(Cc2cc(.... |
153 | 3IGB | ic50 = 38 uM | 454 | C18 H18 N4 | c1ccc(cc1).... |
154 | 1M4H | - | GLU LEU ASP 1OL VAL GLU PHE | n/a | n/a |
155 | 2F3F | ic50 = 190 nM | AXF | C24 H42 N4 O4 S2 | CCCCNC(=O).... |
156 | 3INF | ic50 = 0.04 uM | X45 | C23 H22 N4 O2 | Cc1cc(ccc1.... |
157 | 3MSK | ic50 = 26 uM | EV4 | C18 H25 Cl N4 O | CN(C1CCCCC.... |
158 | 4R93 | Ki = 16 nM | 779 | C26 H39 N5 O2 | CN1C(=O)C(.... |
159 | 3IVI | ic50 = 12 nM | 2LI | C29 H36 F2 N4 O2 | CC(=O)NC(C.... |
160 | 4B72 | ic50 = 0.63 uM | 2FB | C23 H19 N5 O S | Cc1nc2c(s1.... |
161 | 4R5N | ic50 = 76 nM | 3J9 | C20 H20 F N3 O3 | CC12CCCOC1.... |
162 | 2PH6 | ic50 = 27 nM | 712 | C28 H32 F N3 O5 S | CC(c1ccc(c.... |
163 | 4I0F | ic50 = 0.45 uM | 1BF | C21 H21 Cl N4 O2 S | CC1(Cc2cc(.... |
164 | 4H3G | Ki = 6 nM | 10Q | C24 H19 N7 O S | CN1C(=O)C2.... |
165 | 2QU3 | ic50 = 0.59 uM | 462 | C22 H22 Cl N3 O2 S | [H]N=C(N)N.... |
166 | 4B1E | - | 6T6 | C21 H20 N4 | CC1(NC(=C(.... |
167 | 4DVF | ic50 = 128 nM | QSC USC PSA LEU ALA ZAE PLJ | n/a | n/a |
168 | 4DV9 | ic50 = 189 nM | 2OP VAL GNC PSA LEU ALA ZAE PLJ | n/a | n/a |
169 | 3L5F | ic50 = 605 nM | BDX | C19 H33 N3 O | CN1C(=O)C(.... |
170 | 4LXM | ic50 = 0.088 uM | 1YU | C26 H31 F7 N2 O3 S | CC(C)(C)c1.... |
171 | 2OHP | ic50 = 94 uM | 6IP | C15 H15 N3 | c1cc(nc(c1.... |
172 | 3UDJ | ic50 = 242 uM | 092 | C13 H14 N2 O3 | COC(=O)C1C.... |
173 | 2XFI | ic50 = 15 nM | XFI | C33 H42 N4 O5 S | CC(C(=O)NC.... |
174 | 2OF0 | - | CMZ | C15 H23 N O3 | Cc1ccc(c(c.... |
175 | 4LXA | ic50 = 0.002 uM | 1YS | C26 H31 F7 N2 O3 S | CC(C)(C)c1.... |
176 | 3UDR | ic50 = 11 uM | 09F | C19 H21 N3 O3 | c1ccc2c(c1.... |
177 | 3TPP | ic50 = 15 nM | 5HA | C31 H38 N4 O5 S | CC(c1ccccc.... |
178 | 2IS0 | ic50 = 200 nM | I03 | C28 H32 F N3 O6 S | CC(c1ccc(c.... |
179 | 3K5C | ic50 = 17 nM | 0BI | C35 H45 N3 O4 | CC(C)c1ccc.... |
180 | 3LHG | ic50 = 0.02 uM | Z81 | C21 H16 F2 N4 O | CN1C(=O)C(.... |
181 | 3L5B | Kd = 123 uM | BDO | C15 H20 Cl N3 O | CC(C)CC1(C.... |
182 | 3S7M | ic50 = 0.06 uM | 532 | C19 H16 N4 O S | CN1C(=O)C(.... |
183 | 4B70 | ic50 = 6.3 uM | WM9 | C17 H17 Cl N2 O | CC1(N=C(CC.... |
184 | 3VEU | ic50 = 55 nM | 0GO | C33 H48 N4 O3 | CCCN1CCCC1.... |
185 | 4DJV | Ki = 0.19 uM | 0KM | C23 H21 N3 O2 | CN1C(=O)C(.... |
186 | 4R8Y | Ki = 0.64 uM | 3KO | C24 H40 N4 O2 | CN1C(=O)C(.... |
187 | 2VJ7 | ic50 = 40 nM | VG6 | C31 H35 F3 N4 O3 | CCNc1cc(cc.... |
188 | 3ZOV | - | WZV | C20 H20 F3 N5 O3 | CC1(CC(=O).... |
189 | 3INE | ic50 = 0.17 uM | X17 | C22 H29 N3 O2 | Cc1cc(ccc1.... |
190 | 4J0Y | ic50 = 0.435 uM | 1H6 | C18 H15 F2 N5 O2 | CC1(C(COC(.... |
191 | 2Q15 | Ki = 11 nM | 3MR | C31 H42 N4 O2 | CN(C1CCCCC.... |
192 | 4J1E | ic50 = 0.019 uM | 1HM | C19 H14 F5 N5 O2 | c1cc(c(cc1.... |
193 | 4D8C | ic50 = 0.002 uM | BXD | C28 H38 F4 N2 O5 S | CCOCC(C(F).... |
194 | 2VIE | ic50 = 33 nM | VG0 | C32 H48 N4 O3 | CCNc1cc(cc.... |
195 | 2NTR | - | L00 | C26 H35 Cl N6 O4 S | CC1CC1CN(C.... |
196 | 3VV7 | ic50 = 4.6 uM | 0B1 | C21 H21 N3 O2 | CN1C(=O)C=.... |
197 | 3DV5 | ic50 = 0.027 uM | BAV | C29 H49 N3 O3 | CC1CCCCCCC.... |
198 | 3L59 | Kd = 200 uM | BDJ | C12 H14 Cl N3 O | CC1(C(=O)N.... |
199 | 2VIJ | - | C44 | C33 H42 N4 O4 S | CCNc1cc(cc.... |
200 | 4FM7 | ic50 = 0.1 uM | 0UP | C24 H32 F N3 O4 S | CC1CC2(CCN.... |
201 | 3UDM | ic50 = 33 uM | 09A | C19 H18 N2 O3 | c1ccc(cc1).... |
202 | 1FKN | - | GLU VAL ASN 1OL ALA GLU PHE | n/a | n/a |
203 | 4D83 | ic50 = 0.055 uM | 0GT | C27 H34 F2 N2 O3 S | CC(C)(C)c1.... |
204 | 4DPI | ic50 = 78 nM | 0N1 | C34 H41 N3 O4 | Cc1cc2cc(c.... |
205 | 4B1D | ic50 = 0.012 uM | 6TG | C23 H23 N5 O | Cc1cc(cc(c.... |
206 | 4ACX | ic50 = 0.00000001 M | S8Z | C23 H20 F4 N4 O2 | COCC#Cc1cc.... |
207 | 3VG1 | ic50 = 0.055 uM | 0GT | C27 H34 F2 N2 O3 S | CC(C)(C)c1.... |
208 | 2P8H | ic50 = 71 nM | MY9 | C33 H40 F N5 O6 S | CC(c1ccc(c.... |
209 | 3BUG | Kd = 660 uM | AEH | C10 H15 N O | CCc1cc(ccc.... |
210 | 2QMD | ic50 = 5 nM | CS7 | C35 H43 F2 N3 O4 | CCCN(CCC)C.... |
211 | 4KE1 | ic50 = 0.0025 uM | 1R6 | C34 H41 N3 O4 | CCc1ccc2c(.... |
212 | 2WF0 | ic50 = 0.21 uM | ZY0 | C34 H35 F3 N4 O3 | CCc1ccnc2c.... |
213 | 3IN3 | ic50 = 0.06 uM | 472 | C20 H17 N5 O | CN1C(=O)C(.... |
214 | 3HVG | ic50 ~ 2 mM | EV0 | C7 H11 N3 O | CCCC1=CC(=.... |
215 | 3CIB | ic50 = 14 nM | 314 | C36 H45 F2 N3 O3 | CCCN(CCC)C.... |
216 | 3OHH | ic50 = 18 nM | 3HH | C34 H37 F2 N5 O4 | CCCCN(C)C(.... |
217 | 2WF3 | ic50 = 0.019 uM | ZY3 | C31 H40 N4 O5 S | CCNc1cc(cc.... |
218 | 3WB5 | ic50 = 18 uM | 0B4 | C15 H19 N3 O | CC1(CC(=O).... |
219 | 4RRO | ic50 = 26 nM | 3UX | C21 H21 F N4 O3 | CC12CCCOC1.... |
220 | 3VF3 | ic50 = 1.37 uM | 0GS | C21 H24 Br F3 N2 O3 S | CC(c1cccc(.... |
221 | 4FRJ | ic50 = 0.28 uM | DWB | C22 H16 Cl F N2 O3 | COc1ccc2c(.... |
222 | 2VNM | ic50 = 3 nM | CM8 | C31 H37 F3 N4 O4 S | CCNc1cc(cc.... |
223 | 2Q11 | Ki = 900 nM | XX4 | C25 H30 N4 O2 | CN(C1CCCCC.... |
224 | 3CID | ic50 = 5 nM | 318 | C34 H40 F2 N4 O4 | CCCN(CCC)C.... |
225 | 3QBH | ic50 = 0.15 uM | QBH | C29 H40 N2 O6 S | CCCN1C(COC.... |
226 | 3KMY | Kd = 32 uM | D8Y | C13 H13 Cl N2 | c1cc(cc(c1.... |
227 | 4R92 | Ki = 39 nM | 3KU | C25 H37 N5 O2 | CN1C(=O)C(.... |
228 | 4DJW | Ki = 0.53 uM | 0KP | C21 H18 N4 O | CN1C(=O)C(.... |
229 | 3IVH | ic50 = 47 nM | 1LI | C28 H38 F2 N2 O2 | CC(=O)NC(C.... |
230 | 3MSJ | ic50 = 770 uM | EV3 | C10 H12 Cl N3 O | c1cc2c(cc1.... |
231 | 3DV1 | ic50 = 0.59 uM | AR9 | C24 H45 N3 O4 | CCCCNC(=O).... |
232 | 3BUF | Kd = 800 uM | AEG | C9 H13 N O | CC(Cc1ccc(.... |
233 | 4H3J | Ki = 90 nM | 10W | C24 H20 F N5 O S | CN1C(=O)C2.... |
234 | 4PZW | ic50 = 0.11 uM | 2X4 | C19 H18 Cl N3 O3 | c1cc2c(cc1.... |
235 | 2QZL | ic50 = 8 nM | IXS | C34 H44 F N5 O5 S | CC(C)CNC(=.... |
236 | 3WB4 | ic50 = 220 uM | 0B3 | C14 H19 N3 O | CC1(CC(=O).... |
237 | 3OOZ | ic50 = 0.014 uM | ZOO | C22 H19 F4 N3 O2 | CN1C(=O)C(.... |
238 | 2PH8 | ic50 = 1800 nM | 35A | C24 H33 N3 O4 S | CC1CCc2ccc.... |
239 | 4K9H | ic50 = 0.076 uM | 1QU | C33 H37 F3 N4 O4 | c1ccc(cc1).... |
240 | 3ZKI | - | WZV | C20 H20 F3 N5 O3 | CC1(CC(=O).... |
This union binding pocket(no: 1) in the query (biounit: 4gid.bio2) has 98 residues | ||||
---|---|---|---|---|
No: | Leader PDB | Ligand | P-value (APoc) | PS_Score (APoc) |
1 | 3EMY | IVA VAL VAL STA ALA STA | 0.000000005367 | 0.76615 |
2 | 1WKR | IVA VAL VAL STA ALA STA | 0.000000003481 | 0.74998 |
3 | 1J71 | THR ILE THR SER | 0.000000283 | 0.74888 |
4 | 2H6T | IVA VAL VAL STA ALA STA | 0.00000003002 | 0.73666 |
5 | 1BXO | PP7 | 0.00000005976 | 0.63166 |
6 | 4L1A | AB1 | 0.0002198 | 0.53173 |
7 | 5UPJ | UIN | 0.000777 | 0.51759 |
8 | 2R5P | MK1 | 0.0000656 | 0.51561 |
9 | 3MWS | 017 | 0.00005529 | 0.51529 |
10 | 2R5P | MK1 | 0.00007462 | 0.51319 |
11 | 3WSJ | MK1 | 0.00007852 | 0.50879 |
12 | 3WSJ | MK1 | 0.00007852 | 0.50879 |
13 | 1SIV | PSI | 0.00009072 | 0.50281 |
14 | 8HVP | VAL SER GLN ASN LOV ILE VAL | 0.0001155 | 0.50164 |
15 | 5FIV | 3TL | 0.002223 | 0.49301 |
16 | 6FIV | 3TL | 0.002836 | 0.48731 |
17 | 7HVP | ACE SER LEU ASN JG3 ILE VME | 0.0001982 | 0.48553 |
18 | 2P3C | 3TL | 0.0001117 | 0.48413 |
19 | 6UPJ | NIU | 0.004034 | 0.47906 |
20 | 3KYG | 5GP 5GP | 0.00351 | 0.47819 |
21 | 3KYG | 5GP 5GP | 0.003633 | 0.46977 |
22 | 1GOJ | ADP | 0.0171 | 0.46596 |
23 | 4DS0 | A2G GAL NAG FUC | 0.02526 | 0.46337 |
24 | 3QSB | 743 | 0.01389 | 0.4577 |
25 | 4M8X | KGQ | 0.0006965 | 0.45285 |
26 | 3KYF | 5GP 5GP | 0.0179 | 0.45146 |
27 | 3LRE | ADP | 0.0277 | 0.44829 |
28 | 3QRC | SCR | 0.02732 | 0.44649 |
29 | 3QRC | SCR | 0.02767 | 0.44593 |
30 | 3LRE | ADP | 0.03167 | 0.44487 |
31 | 3LRE | ADP | 0.03167 | 0.44487 |
32 | 3D91 | REM | 0.00000008972 | 0.44284 |
33 | 1K0E | TRP | 0.02059 | 0.44078 |
34 | 3D91 | REM | 0.00001768 | 0.44055 |
35 | 3D91 | REM | 0.000000107 | 0.44048 |
36 | 3ZJX | BOG | 0.03565 | 0.44028 |
37 | 2PL3 | ADP | 0.03702 | 0.43717 |
38 | 1Y8E | SVR | 0.04196 | 0.43253 |
39 | 1MUU | SUC | 0.04355 | 0.42466 |
40 | 1HMU | ASG GCD | 0.04272 | 0.42345 |
41 | 4KBA | 1QM | 0.04008 | 0.41909 |
42 | 1GRN | GDP | 0.04625 | 0.4158 |
43 | 3UZP | 0CK | 0.04607 | 0.41322 |
44 | 3UZP | 0CK | 0.04607 | 0.41322 |
45 | 3NHT | U46 | 0.03474 | 0.40739 |
46 | 2VZZ | SCA | 0.02544 | 0.40527 |
47 | 4CKU | P2F | 0.00000124 | 0.40024 |
This union binding pocket(no: 2) in the query (biounit: 4gid.bio1) has 102 residues | ||||
---|---|---|---|---|
No: | Leader PDB | Ligand | P-value (APoc) | PS_Score (APoc) |
1 | 3EMY | IVA VAL VAL STA ALA STA | 0.000000007392 | 0.76344 |
2 | 1J71 | THR ILE THR SER | 0.0000002159 | 0.76007 |
3 | 1WKR | IVA VAL VAL STA ALA STA | 0.000000004628 | 0.74845 |
4 | 2H6T | IVA VAL VAL STA ALA STA | 0.00000003995 | 0.73435 |
5 | 1BXO | PP7 | 0.0000000434 | 0.64152 |
6 | 4L1A | AB1 | 0.0002456 | 0.53211 |
7 | 2R5P | MK1 | 0.00008287 | 0.51421 |
8 | 3MWS | 017 | 0.00007172 | 0.51348 |
9 | 5UPJ | UIN | 0.001081 | 0.51249 |
10 | 2R5P | MK1 | 0.00009399 | 0.51183 |
11 | 3WSJ | MK1 | 0.00009994 | 0.50729 |
12 | 3WSJ | MK1 | 0.00009994 | 0.50729 |
13 | 6FIV | 3TL | 0.001447 | 0.50562 |
14 | 8HVP | VAL SER GLN ASN LOV ILE VAL | 0.0001301 | 0.50236 |
15 | 5FIV | 3TL | 0.00172 | 0.50155 |
16 | 1SIV | PSI | 0.0001144 | 0.50152 |
17 | 2P3C | 3TL | 0.00005989 | 0.49783 |
18 | 7HVP | ACE SER LEU ASN JG3 ILE VME | 0.0001508 | 0.49336 |
19 | 1GOJ | ADP | 0.01498 | 0.47473 |
20 | 3QSB | 743 | 0.008799 | 0.47119 |
21 | 6UPJ | NIU | 0.006442 | 0.47045 |
22 | 2VDF | OCT | 0.0007752 | 0.46291 |
23 | 3KYG | 5GP 5GP | 0.009221 | 0.45829 |
24 | 3LRE | ADP | 0.02625 | 0.45444 |
25 | 2CJU | PHX | 0.02582 | 0.45345 |
26 | 3KYG | 5GP 5GP | 0.008486 | 0.45331 |
27 | 4M8X | KGQ | 0.0007961 | 0.45323 |
28 | 2ZTG | A5A | 0.01086 | 0.45107 |
29 | 1OFL | NGK GCD | 0.01731 | 0.44992 |
30 | 3LRE | ADP | 0.03412 | 0.44654 |
31 | 3LRE | ADP | 0.03412 | 0.44654 |
32 | 3D91 | REM | 0.00000002548 | 0.44559 |
33 | 3D91 | REM | 0.00000003259 | 0.44266 |
34 | 3ZJX | BOG | 0.03528 | 0.44254 |
35 | 2PL3 | ADP | 0.03288 | 0.4423 |
36 | 3D91 | REM | 0.000007919 | 0.44224 |
37 | 2IU8 | PLM | 0.01098 | 0.44148 |
38 | 2PKA | BEN | 0.04355 | 0.44125 |
39 | 2PKA | BEN | 0.04355 | 0.44125 |
40 | 4NPT | 017 | 0.03357 | 0.43807 |
41 | 1W6P | NDG GAL | 0.04209 | 0.43337 |
42 | 3HXU | A5A | 0.02371 | 0.42225 |
43 | 1MUU | SUC | 0.04799 | 0.42176 |
44 | 3UZP | 0CK | 0.04093 | 0.41798 |
45 | 3UZP | 0CK | 0.04093 | 0.41798 |
This union binding pocket(no: 3) in the query (biounit: 4gid.bio3) has 86 residues | ||||
---|---|---|---|---|
No: | Leader PDB | Ligand | P-value (APoc) | PS_Score (APoc) |
1 | 3EMY | IVA VAL VAL STA ALA STA | 0.000000004326 | 0.76423 |
2 | 1J71 | THR ILE THR SER | 0.0000001911 | 0.75356 |
3 | 2H6T | IVA VAL VAL STA ALA STA | 0.00000001658 | 0.74362 |
4 | 1WKR | IVA VAL VAL STA ALA STA | 0.000000004268 | 0.73903 |
5 | 1BXO | PP7 | 0.00000004499 | 0.63061 |
6 | 4L1A | AB1 | 0.0003321 | 0.51841 |
7 | 5UPJ | UIN | 0.0006967 | 0.5161 |
8 | 3MWS | 017 | 0.0001045 | 0.49903 |
9 | 3WSJ | MK1 | 0.0001284 | 0.49526 |
10 | 3WSJ | MK1 | 0.0001284 | 0.49526 |
11 | 2R5P | MK1 | 0.0001673 | 0.49366 |
12 | 2R5P | MK1 | 0.0001914 | 0.49115 |
13 | 5FIV | 3TL | 0.002277 | 0.48866 |
14 | 2VDF | OCT | 0.001082 | 0.48803 |
15 | 1SIV | PSI | 0.0001767 | 0.48628 |
16 | 8HVP | VAL SER GLN ASN LOV ILE VAL | 0.000215 | 0.48582 |
17 | 6FIV | 3TL | 0.002792 | 0.48394 |
18 | 3KYG | 5GP 5GP | 0.002547 | 0.48179 |
19 | 6UPJ | NIU | 0.004149 | 0.47475 |
20 | 3KYG | 5GP 5GP | 0.003222 | 0.46872 |
21 | 2P3C | 3TL | 0.0003484 | 0.4605 |
22 | 1GOJ | ADP | 0.01905 | 0.45951 |
23 | 7HVP | ACE SER LEU ASN JG3 ILE VME | 0.0006843 | 0.45914 |
24 | 3D91 | REM | 0.0000001292 | 0.45461 |
25 | 3QSB | 743 | 0.01375 | 0.45455 |
26 | 3D91 | REM | 0.0000163 | 0.45219 |
27 | 3KYF | 5GP 5GP | 0.01573 | 0.45129 |
28 | 3D91 | REM | 0.0000001663 | 0.45086 |
29 | 3QRC | SCR | 0.009329 | 0.44693 |
30 | 3QRC | SCR | 0.009487 | 0.44597 |
31 | 2W58 | ADP | 0.03565 | 0.43828 |
32 | 3LRE | ADP | 0.03645 | 0.43717 |
33 | 4M8X | KGQ | 0.001628 | 0.43447 |
34 | 1RYD | GLC | 0.04474 | 0.43438 |
35 | 1K0E | TRP | 0.02814 | 0.43016 |
36 | 2OID | ANP | 0.04035 | 0.41866 |
37 | 2G30 | ALA ALA PHE | 0.02686 | 0.41725 |
38 | 3LKF | PC | 0.04859 | 0.4169 |
39 | 4ER2 | IVA VAL VAL STA ALA STA | 0.00000007533 | 0.4144 |
40 | 4CKU | P2F | 0.000002494 | 0.40544 |
This union binding pocket(no: 4) in the query (biounit: 4gid.bio4) has 33 residues | ||||
---|---|---|---|---|
No: | Leader PDB | Ligand | P-value (APoc) | PS_Score (APoc) |
1 | 3EMY | IVA VAL VAL STA ALA STA | 0.0000000003827 | 0.74889 |
2 | 1J71 | THR ILE THR SER | 0.0000001409 | 0.70585 |
3 | 1WKR | IVA VAL VAL STA ALA STA | 0.000000001462 | 0.69571 |
4 | 2H6T | IVA VAL VAL STA ALA STA | 0.00000001619 | 0.68363 |
5 | 3D91 | REM | 0.000000004349 | 0.6587 |
6 | 3D91 | REM | 0.00000006762 | 0.6587 |
7 | 3D91 | REM | 0.000000004544 | 0.65664 |
8 | 4ER2 | IVA VAL VAL STA ALA STA | 0.000000006524 | 0.62066 |
9 | 1QRP | HH0 | 0.000000001657 | 0.58985 |
10 | 3ZLQ | 6T9 | 0.00000000005621 | 0.58952 |
11 | 1BXO | PP7 | 0.00000001969 | 0.58171 |
12 | 1FQ5 | 0GM | 0.00000001801 | 0.56964 |
13 | 4CKU | P2F | 0.0000004451 | 0.5648 |
14 | 1LYB | IVA VAL VAL STA ALA STA | 0.00000002348 | 0.56435 |
15 | 4CKU | P2F | 0.0000001572 | 0.55734 |
16 | 1ZAP | A70 | 0.00000009101 | 0.55045 |
17 | 1CZI | PRO PHI SMC NOR | 0.000000007975 | 0.54638 |
18 | 1IZE | IVA VAL VAL STA ALA STA | 0.00000001269 | 0.54491 |
19 | 3FV3 | IVA VAL VAL STA ALA STA | 0.00000001617 | 0.53683 |
20 | 2QZX | IVA VAL VAL STA ALA STA | 0.00000002628 | 0.5333 |
21 | 1QS8 | IVA VAL VAL STA ALA STA | 0.00000000964 | 0.51229 |
22 | 4L1A | AB1 | 0.0001264 | 0.49769 |
23 | 5UPJ | UIN | 0.0005722 | 0.48198 |
24 | 3O9L | LPN | 0.00005216 | 0.47601 |
25 | 3UCB | 017 | 0.00003409 | 0.47303 |
26 | 1GOJ | ADP | 0.003832 | 0.47105 |
27 | 3MWS | 017 | 0.00005942 | 0.46597 |
28 | 3O9L | LPN | 0.00009018 | 0.46571 |
29 | 3SM2 | 478 | 0.00008928 | 0.46326 |
30 | 3FSM | 2NC | 0.00006931 | 0.46314 |
31 | 6UPJ | NIU | 0.001427 | 0.46272 |
32 | 2R5P | MK1 | 0.00009955 | 0.46097 |
33 | 2R5P | MK1 | 0.0001134 | 0.45883 |
34 | 1IDA | 0PO | 0.00009796 | 0.45756 |
35 | 8HVP | VAL SER GLN ASN LOV ILE VAL | 0.0001021 | 0.45719 |
36 | 2BJU |