Receptor
PDB id Resolution Class Description Source Keywords
1tt1 1.93 Å NON-ENZYME: SIGNAL_HORMONE CRYSTAL STRUCTURE OF THE GLUR6 LIGAND BINDING CORE IN COMPLEX WITH KAINATE 1.93 A RESOLUTION RATTUS NORVEGICUS MEMBRANE PROTEIN
Ref.: CRYSTAL STRUCTURES OF THE GLUR5 AND GLUR6 LIGAND BINDING CORES: MOLECULAR MECHANISMS UNDERLYING KAINATE RECEPTOR SELECTIVITY NEURON V. 45 539 2005
Ligand
Ligand Chain:Residue Validity Ligand Warnings Binding Data Chemaxon Viewer Molecular Weight (Da) Formula SMILES
KAI A:998;
B:999;
Valid;
Valid;
none;
none;
Ki = 64.6 nM 213.23 C10 H15 N O4 CC(=C...
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90% Homology Family
Leader
PDB id Resolution Class Description Source Keywords
3QXM 1.65 Å NON-ENZYME: SIGNAL_HORMONE CRYSTAL STRUCTURE OF HUMAN GLUK2 LIGAND-BINDING CORE IN COMP NOVEL MARINE-DERIVED TOXINS, NEODYSIHERBAINE A HOMO SAPIENS, SYNTHETIC, HOMO SAPIENS TWO DOMAINS LIGAND-BINDING MEMBRANE PROTEIN
Ref.: BINDING AND SELECTIVITY OF THE MARINE TOXIN NEODYSI A AND ITS SYNTHETIC ANALOGUES TO GLUK1 AND GLUK2 KA RECEPTORS. J.MOL.BIOL. V. 413 667 2011
Members (16)
No: PDB id Binding Data Representative ligand Formula Smiles
The Class containing this family consists of a total of 201 families.
1 3QXM Ki = 33 nM NDZ C11 H17 N O8 C1[C@@H]2[....
2 1S9T Ki = 253 nM QUS C5 H7 N3 O5 O1N(C(=O)N....
3 4BDR - KAI C10 H15 N O4 CC(=C)[C@H....
4 2XXT - KAI C10 H15 N O4 CC(=C)[C@H....
5 2XXU - GLU C5 H9 N O4 O=C([O-])C....
6 4BDN - GLU C5 H9 N O4 O=C([O-])C....
7 4BDQ - CYS C3 H7 N O2 S SCC([N+])C....
8 1S50 Ki = 1.4 uM GLU C5 H9 N O4 O=C([O-])C....
9 2XXW - GLU C5 H9 N O4 O=C([O-])C....
10 1SD3 - SYM C6 H10 N O4 C[C@H](C[C....
11 2XXV - KAI C10 H15 N O4 CC(=C)[C@H....
12 4BDL - GLU C5 H9 N O4 O=C([O-])C....
13 2XXX - GLU C5 H9 N O4 O=C([O-])C....
14 2XXR - GLU C5 H9 N O4 O=C([O-])C....
15 1S7Y Ki = 1.4 uM GLU C5 H9 N O4 O=C([O-])C....
16 1TT1 Ki = 64.6 nM KAI C10 H15 N O4 CC(=C)[C@H....