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- Biounit PDB : .ZIP | .CSV
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No: | PDB id | Binding Data | Representative ligand | Formula | Smiles |
---|---|---|---|---|---|
The Class containing this family consists of a total of 9 families. | |||||
1 | 3PXF | Kd = 37 uM | 2AN | C16 H13 N O3 S | c1ccc(cc1).... |
2 | 3TI1 | - | B49 | C22 H27 F N4 O2 | CCN(CC)CCN.... |
3 | 2R3G | ic50 = 800 nM | SC9 | C18 H14 F N5 | c1ccc(c(c1.... |
4 | 3PXQ | Kd = 37 uM | 2AN | C16 H13 N O3 S | c1ccc(cc1).... |
5 | 2R3N | ic50 = 70 nM | SCZ | C21 H19 N5 | c1ccc(cc1).... |
6 | 2C69 | ic50 = 26 uM | CT8 | C17 H14 Br N6 | c1cc(cc(c1.... |
7 | 2VTM | ic50 ~ 1 mM | LZM | C7 H4 N4 | c1cnc2c(cn.... |
8 | 1H0V | - | UN4 | C10 H12 N6 O2 | c1[nH]c2c(.... |
9 | 4ERW | - | STU | C28 H26 N4 O3 | CC12C(C(CC.... |
10 | 4NJ3 | Ki = 0.14 uM | 2KD | C27 H21 Cl N2 O6 | COC(=O)C(C.... |
11 | 1JSV | - | U55 | C10 H11 N5 O2 S | c1cc(ccc1N.... |
12 | 1E1V | Ki = 12 uM | CMG | C12 H17 N5 O | c1[nH]c2c(.... |
13 | 1OIQ | ic50 = 2.9 uM | HDU | C14 H13 N5 O | Cc1c(n2ccc.... |
14 | 2VV9 | ic50 = 0.017 uM | IM9 | C23 H29 N7 O2 | Cc1ncc(n1C.... |
15 | 2W17 | ic50 = 0.002 uM | I19 | C24 H30 F N7 O | Cc1ncc(n1C.... |
16 | 2VTP | ic50 = 0.003 uM | LZ9 | C17 H11 F3 N4 O2 | c1cc(c(c(c.... |
17 | 1JVP | ic50 = 1.6 uM | LIG | C15 H11 N3 | c1ccc-2c(c.... |
18 | 1FVT | - | 106 | C14 H9 Br N4 O3 S | c1cc(ccc1N.... |
19 | 4KD1 | - | 1QK | C21 H29 N6 O2 | CCc1cnn2c1.... |
20 | 2BTS | ic50 = 20 nM | U32 | C12 H15 N3 O2 S2 | CC(C)c1cnc.... |
21 | 3LE6 | ic50 = 0.035 uM | 2BZ | C17 H10 Cl N5 O2 | Cc1c-2nc(c.... |
22 | 2VTI | ic50 = 0.66 uM | LZ3 | C14 H12 N4 O3 S | c1ccc2c(c1.... |
23 | 3LFS | Ki = 2.5 uM | A07 | C17 H16 Cl N3 O | CCCC(=O)Nc.... |
24 | 1PXI | - | CK1 | C8 H5 Cl2 N3 S | c1cnc(nc1c.... |
25 | 1URW | ic50 < 0.003 uM | I1P | C21 H24 N8 O2 S | CN(C)CCCNS.... |
26 | 4LYN | - | 1YG | C20 H23 N3 O2 S2 | CC(c1ccccc.... |
27 | 1YKR | ic50 = 0.56 uM | 628 | C20 H14 Cl2 N4 O3 S | c1cc(c(c(c.... |
28 | 1PXN | Ki ~ 0.32 uM | CK6 | C15 H15 N5 O S | Cc1c(sc(n1.... |
29 | 1CKP | - | PVB | C20 H25 Cl N6 O3 | CC(C)C(CO).... |
30 | 1KE6 | ic50 = 5.7 nM | LS2 | C17 H15 N5 O3 S2 | CNS(=O)(=O.... |
31 | 2C6K | ic50 = 0.73 uM | DT2 | C17 H21 N7 O2 S | c1cc(ccc1N.... |
32 | 2R3Q | - | 5SC | C19 H16 Br N5 O | Cc1ccccc1c.... |
33 | 2R3J | ic50 = 10 nM | SCJ | C18 H14 Br N5 | c1ccc(cc1).... |
34 | 3IG7 | ic50 = 9 nM | EFP | C18 H22 N4 O3 | CC(=O)NC1C.... |
35 | 2VTS | ic50 = 0.03 uM | LZC | C16 H23 N7 | CC(C)Nc1cc.... |
36 | 1P2A | ic50 = 12 nM | 5BN | C17 H15 F N4 O | c1cc([nH]c.... |
37 | 2BHE | ic50 = 1 uM | BRY | C16 H9 Br N2 O2 | c1ccc2c(c1.... |
38 | 3UNK | ic50 = 15 uM | 0BY | C17 H13 Cl N4 O2 | c1ccc(c(c1.... |
39 | 1OIT | ic50 < 0.003 uM | HDT | C17 H14 N6 O2 S | c1ccn2c(c1.... |
40 | 2VTQ | ic50 = 0.14 uM | LZA | C16 H17 F2 N5 O2 | c1cc(c(c(c.... |
41 | 3NS9 | ic50 = 0.003 uM | NS9 | C20 H27 N5 O3 | CC(C)c1cnn.... |
42 | 2C68 | ic50 = 1.8 uM | CT6 | C18 H15 Br N5 | c1cc(cc(c1.... |
43 | 3TIZ | - | 3TI | C17 H13 N O2 | c1ccc2c(c1.... |
44 | 3PXY | ic50 = 5.9 uM | JWS | C10 H11 N5 O2 | COc1ccc(c(.... |
45 | 1H01 | ic50 = 22 uM | FAL | C21 H23 Cl2 N5 O2 | CN(C)CC(CO.... |
46 | 2EXM | - | ZIP | C10 H13 N5 | CC(=CCNc1c.... |
47 | 4BGH | ic50 = 4 nM | 3I6 | C13 H16 Br N5 O3 S | CC(CO)Nc1c.... |
48 | 2R3F | ic50 = 500 nM | SC8 | C18 H13 Cl2 N5 | c1cc(c(c(c.... |
49 | 2R3M | ic50 = 10 nM | SCX | C19 H17 F2 N7 | CCc1cnn2c1.... |
50 | 1GII | - | 1PU | C17 H16 N4 O2 | c1ccnc(c1).... |
51 | 2R64 | ic50 = 0.03 uM | 740 | C23 H27 N5 O3 S | c1cc(ccc1C.... |
52 | 2C6O | - | 4SP | C18 H22 N6 O3 S | c1cc(ccc1N.... |
53 | 1V1K | Ki = 35 uM | 3FP | C22 H23 F4 N5 O2 | CN(C)CC(CO.... |
54 | 2VTJ | ic50 = 1.9 uM | LZ4 | C10 H9 Cl N4 O2 S | c1cc(ccc1N.... |
55 | 2C6L | ic50 = 0.27 uM | DT4 | C17 H22 N8 O2 S | c1cc(ccc1N.... |
56 | 2W06 | - | FRV | C18 H20 N6 O2 S | Cc1ncc(n1C.... |
57 | 3EZV | - | EZV | C25 H25 N7 | CN1CCN(CC1.... |
58 | 4EZ7 | - | STU | C28 H26 N4 O3 | CC12C(C(CC.... |
59 | 3PXZ | Kd = 37 uM | 2AN | C16 H13 N O3 S | c1ccc(cc1).... |
60 | 1W0X | - | OLO | C15 H18 N6 O | Cn1cnc2c1n.... |
61 | 2XMY | Ki = 0.11 nM | CDK | C18 H21 N5 O4 S2 | CC1=C(SC(=.... |
62 | 2UZO | ic50 = 18 uM | C62 | C14 H10 N2 O5 S2 | c1cc(ccc1c.... |
63 | 2VTT | ic50 = 0.044 uM | LZD | C16 H17 F2 N5 O2 | c1cc(c(c(c.... |
64 | 1KE7 | ic50 = 8.9 nM | LS3 | C20 H15 N3 O4 S | c1cc2c(cc1.... |
65 | 2VU3 | ic50 = 0.047 uM | LZE | C16 H17 Cl2 N5 O2 | c1cc(c(c(c.... |
66 | 2B54 | - | D05 | C20 H15 Cl3 N4 O3 | CCc1c2c(n(.... |
67 | 1DM2 | - | HMD | C11 H10 Br N5 O2 | C1CNC(=O)C.... |
68 | 1DI8 | ic50 = 1 uM | DTQ | C16 H15 N3 O3 | COc1cc2c(c.... |
69 | 1GZ8 | - | MBP | C10 H13 N5 O2 | CC(C)C(=O).... |
70 | 3PY0 | ic50 = 0.13 uM | SU9 | C13 H11 N3 O2 | COc1ccc2c(.... |
71 | 2VTR | ic50 = 1.5 uM | LZB | C10 H10 Cl N5 | CC(C)Nc1cc.... |
72 | 1E1X | Ki = 1.3 uM | NW1 | C11 H17 N5 O2 | C1CCC(CC1).... |
73 | 1GIJ | - | 2PU | C19 H22 N6 O2 | c1cc2c(c(c.... |
74 | 3UNJ | ic50 = 11 uM | 0BX | C17 H14 N4 O2 | c1ccc(cc1).... |
75 | 2A0C | - | CK9 | C19 H26 N6 O2 | CCC(CO)Nc1.... |
76 | 3TIY | - | TIY | C11 H8 O5 | c1c2c(c(c(.... |
77 | 2R3I | ic50 = 1000 nM | SCF | C18 H14 F N5 | c1ccc(c(c1.... |
78 | 2R3P | ic50 = 900 nM | 3SC | C19 H12 Cl2 N6 S | c1cc(c(c(c.... |
79 | 1KE8 | ic50 = 1000 nM | LS4 | C18 H14 N4 O3 S2 | c1ccc2c(c1.... |
80 | 2C6I | ic50 = 11 uM | DT1 | C18 H22 N6 O3 S | c1cc(ccc1N.... |
81 | 1VYZ | ic50 = 290 nM | N5B | C13 H13 N3 O | c1ccc(cc1).... |
82 | 3WBL | ic50 = 23 uM | PDY | C20 H26 N6 O | CCOc1ccc(c.... |
83 | 1PXP | Ki ~ 0.22 uM | CK8 | C17 H19 N5 S | Cc1c(sc(n1.... |
84 | 4RJ3 | ic50 = 93 nM | 3QS | C22 H28 N6 O | COC1CCN(CC.... |
85 | 2VTN | ic50 = 0.85 uM | LZ7 | C12 H11 F N4 O2 | CC(=O)Nc1c.... |
86 | 1AQ1 | - | STU | C28 H26 N4 O3 | CC12C(C(CC.... |
87 | 2UZN | ic50 = 0.03 uM | C96 | C15 H13 N3 O4 S2 | [H]N=C1NC(.... |
88 | 2B55 | ic50 = 96 nM | D31 | C24 H31 N5 O2 | c1cc-2c(c(.... |
89 | 2C6M | ic50 = 0.35 uM | DT5 | C17 H20 N6 O3 S | c1cc(ccc1N.... |
90 | 3PJ8 | - | 404 | C19 H26 N6 O | CCC(CO)Nc1.... |
91 | 3LFQ | - | A28 | C17 H15 F2 N3 O | CCCC(=O)Nc.... |
92 | 2R3L | ic50 = 100 nM | SCW | C18 H14 Br N5 | c1ccc(cc1).... |
93 | 2W05 | ic50 = 0.001 uM | FRT | C20 H26 N6 O3 S | Cc1ncc(n1C.... |
94 | 1H08 | - | BYP BWP | n/a | n/a |
95 | 2XNB | Ki = 149 nM | Y8L | C19 H22 N6 O S | CC1=C(SC(=.... |
96 | 1HCK | - | ATP | C10 H16 N5 O13 P3 | c1nc(c2c(n.... |
97 | 1B38 | Kd = 0.254 uM | ATP | C10 H16 N5 O13 P3 | c1nc(c2c(n.... |
98 | 2B52 | ic50 = 8 nM | D42 | C21 H23 N7 O2 S | Cc1c(sc(n1.... |
99 | 1PXL | - | CK4 | C16 H13 F3 N4 S | Cc1c(sc(n1.... |
100 | 2R3H | ic50 = 20000 nM | SCE | C13 H13 N5 | Cc1cnc2n1c.... |
101 | 3LFN | Ki = 3160 nM | A27 | C23 H21 N3 O2 | CCCC(=O)Nc.... |
102 | 3S2P | ic50 = 0.068 uM | PMU | C17 H22 N4 O3 | CC(C)c1cc(.... |
103 | 2R3O | ic50 = 600 nM | 2SC | C19 H17 N5 O | c1ccc(cc1).... |
104 | 3IGG | ic50 = 95 nM | EFQ | C16 H19 N3 O3 | COc1ccc(cc.... |
105 | 1R78 | ic50 = 3 nM | FMD | C20 H20 F N3 O4 | CC(C(C(C#C.... |
106 | 2FVD | Ki = 0.003 uM | LIA | C18 H21 F2 N5 O4 S | COc1ccc(c(.... |
107 | 2VTL | ic50 = 97 uM | LZ5 | C10 H9 N3 O | c1ccc(cc1).... |
108 | 3PY1 | Kd = 37 uM | 2AN | C16 H13 N O3 S | c1ccc(cc1).... |
109 | 1KE9 | ic50 = 660 nM | LS5 | C16 H15 N5 O3 S | c1ccc2c(c1.... |
110 | 2A4L | ic50 = 0.4 uM | RRC | C19 H26 N6 O | CCC(CO)Nc1.... |
111 | 1Y8Y | ic50 = 2 uM | CT7 | C13 H11 Cl N4 O2 S | CS(=O)(=O).... |
112 | 1OIR | ic50 = 0.032 uM | HDY | C23 H26 N6 O2 | Cc1c(n2ccc.... |
113 | 1PXJ | - | CK2 | C9 H10 N4 S | Cc1c(sc(n1.... |
114 | 2VTO | ic50 = 0.14 uM | LZ8 | C17 H13 F N4 O2 | c1ccc(cc1).... |
115 | 1PYE | ic50 = 0.32 uM | PM1 | C21 H13 F2 N3 O2 | c1ccc(cc1).... |
116 | 2BTR | ic50 = 95 nM | U73 | C13 H15 N3 O S | CC(C)C1=CN.... |
117 | 2VTA | ic50 = 185 uM | LZ1 | C7 H6 N2 | c1ccc2c(c1.... |
118 | 4EZ3 | - | 0S0 | C11 H10 N4 O4 S | c1cc(ccc1N.... |
119 | 3EZR | - | EZR | C26 H27 N7 O | CN1CCN(CC1.... |
120 | 3ULI | ic50 = 0.07 uM | 1N3 | C21 H25 Br N6 O2 | COc1ccc(cc.... |
121 | 2DS1 | ic50 = 6.4 nM | 1CD | C22 H21 N5 O3 | CC1CC2CN1C.... |
122 | 1H07 | ic50 = 3 uM | MFP | C24 H27 Br N6 O2 | Cc1ccc(c(c.... |
123 | 2B53 | ic50 = 0.6 uM | D23 | C19 H19 F3 N4 | CC(C)(C)Nc.... |
124 | 2DUV | ic50 = 0.087 uM | 371 | C19 H17 N O7 S | Cc1cc2c(c(.... |
125 | 2VTH | ic50 = 120 uM | LZ2 | C10 H9 N O3 S | c1cc2c(ccc.... |
126 | 1KE5 | ic50 = 560 nM | LS1 | C16 H15 N3 O3 S | CNS(=O)(=O.... |
127 | 3FZ1 | - | B98 | C13 H15 N3 O2 S | COc1ccc2c(.... |
128 | 1WCC | ic50 = 350 uM | CIG | C4 H4 Cl N3 | c1c(nc(cn1.... |
129 | 4ACM | Ki = 210 nM | 7YG | C20 H23 N7 O3 S | CN(C)CCNS(.... |
130 | 2C5Y | ic50 = 0.25 uM | MTW | C19 H15 N7 O2 | c1cc(cc(c1.... |
131 | 1PXO | Ki = 2 nM | CK7 | C14 H12 N6 O2 S | Cc1c(sc(n1.... |
132 | 1H00 | ic50 = 38 uM | FAP | C21 H23 F2 N5 O2 | CN(C)CC(CO.... |
133 | 2R3R | - | 6SC | C18 H14 Br N5 | c1ccc(cc1).... |
134 | 2R3K | ic50 = 100 nM | SCQ | C18 H14 Br N5 | c1ccc(cc1).... |
135 | 2V0D | - | C53 | C9 H7 N3 O S | [H]N=C1NC(.... |
136 | 1B39 | Kd = 0.12 uM | ATP | C10 H16 N5 O13 P3 | c1nc(c2c(n.... |
137 | 2W1H | ic50 = 0.052 uM | L0F | C17 H13 N5 O | c1ccc(cc1).... |
138 | 1Y91 | ic50 = 0.059 uM | CT9 | C23 H33 N7 O2 S | CC(C)c1cnn.... |
139 | 4AU8 | ic50 = 551 nM | Z3R | C11 H8 N2 O2 S3 | c1ccc2c(c1.... |
140 | 1V0P | ic50 = 0.13 uM | PVB | C20 H25 Cl N6 O3 | CC(C)C(CO).... |
141 | 1V0O | ic50 = 5.5 uM | INR | C16 H10 N2 O5 S | c1ccc2c(c1.... |
No: | PDB id | Binding Data | Representative ligand | Formula | Smiles |
---|---|---|---|---|---|
The Class containing this family consists of a total of 68 families. | |||||
1 | 3UOD | Kd = 49 nM | 0C3 | C18 H13 F3 N4 O2 | c1ccc(c(c1.... |
2 | 4UZH | ic50 = 9800 nM | JVE | C15 H13 F N4 O | c1ccc(c(c1.... |
3 | 3EFW | - | AK8 | C25 H21 F3 N6 O2 | Cc1cc(ccc1.... |
4 | 3UO4 | Kd = 299 nM | 0C0 | C23 H18 N4 O2 | c1ccc(cc1).... |
5 | 3UP2 | Kd = 40 nM | 0C8 | C18 H13 F3 N4 O3 | c1ccc(c(c1.... |
6 | 2C6E | - | HPM | C28 H31 N7 O4 | COc1cc2c(c.... |
7 | 3H0Y | ic50 = 0.006 uM | 48B | C23 H17 Cl F N5 O2 | c1ccc(c(c1.... |
8 | 4B0G | ic50 = 0.015 uM | VEK | C19 H21 Br N8 O | Cc1cc(no1).... |
9 | 4JBP | ic50 = 41 nM | YPH | C34 H36 N6 O4 | c1ccc(cc1).... |
10 | 3H10 | - | 97B | C30 H25 Cl F2 N6 O | CN1CCN(CC1.... |
11 | 3DJ5 | - | AK5 | C21 H20 Br N5 O3 S | COc1ccc(cc.... |
12 | 3UOL | ic50 = 3.1 nM | 0C7 | C17 H13 Cl N8 | c1ccc(c(c1.... |
13 | 3D14 | ic50 = 22 nM | AK1 | C19 H15 F3 N6 O S2 | c1cc(cc(c1.... |
14 | 1MQ4 | - | ADP | C10 H15 N5 O10 P2 | c1nc(c2c(n.... |
15 | 4BN1 | - | ADP | C10 H15 N5 O10 P2 | c1nc(c2c(n.... |
16 | 2NP8 | ic50 = 42 nM | CC3 | C21 H18 F3 N5 O | c1cc(cc(c1.... |
17 | 4JBQ | - | VX6 | C23 H28 N8 O S | Cc1cc([nH].... |
18 | 3DJ6 | - | AK6 | C25 H24 N4 O3 S | COc1ccc(cc.... |
19 | 2WQE | - | ADP | C10 H15 N5 O10 P2 | c1nc(c2c(n.... |
20 | 4UYN | ic50 = 2 nM | Y3M | C25 H22 N4 O4 S | CCOC(=O)c1.... |
21 | 2WTV | Ki = 1.8 nM | ZZL | C25 H15 Cl F2 N4 O2 | c1cc(c(c(c.... |
22 | 3FDN | ic50 = 0.033 uM | MMH | C21 H22 N6 O3 | Cc1c(c([nH.... |
23 | 4J8M | ic50 = 48 nM | CJ5 | C26 H25 F3 N8 O | c1cc(cc(c1.... |
24 | 3O50 | - | LJE | C24 H17 F3 N4 O2 | Cc1cc(ccc1.... |
25 | 2J4Z | ic50 = 65 nM | 626 | C23 H24 N6 O2 S | CN1CCN(CC1.... |
26 | 3LAU | ic50 = 0.044 uM | OFI | C17 H17 N3 O2 | CCCC(=O)Nc.... |
27 | 4DEA | ic50 = 256 nM | NHI | C18 H14 N4 O4 | c1cc(ccc1C.... |
28 | 3DAJ | ic50 = 2.9 uM | FXG | C22 H29 N7 O2 | CCCCNC(=O).... |
29 | 4JBO | ic50 = 24 nM | WPH | C31 H32 N6 O3 | CN(C)CCOc1.... |
30 | 2C6D | - | ANP | C10 H17 N6 O12 P3 | c1nc(c2c(n.... |
31 | 4DEE | - | ADP | C10 H15 N5 O10 P2 | c1nc(c2c(n.... |
32 | 3K5U | ic50 = 309 nM | PFQ | C20 H17 N3 O2 | c1ccc(cc1).... |
33 | 1JSV | - | U55 | C10 H11 N5 O2 S | c1cc(ccc1N.... |
34 | 1E1V | Ki = 12 uM | CMG | C12 H17 N5 O | c1[nH]c2c(.... |
35 | 1OIQ | ic50 = 2.9 uM | HDU | C14 H13 N5 O | Cc1c(n2ccc.... |
36 | 2VV9 | ic50 = 0.017 uM | IM9 | C23 H29 N7 O2 | Cc1ncc(n1C.... |
37 | 2W17 | ic50 = 0.002 uM | I19 | C24 H30 F N7 O | Cc1ncc(n1C.... |
38 | 2VTP | ic50 = 0.003 uM | LZ9 | C17 H11 F3 N4 O2 | c1cc(c(c(c.... |
39 | 1JVP | ic50 = 1.6 uM | LIG | C15 H11 N3 | c1ccc-2c(c.... |
40 | 1FVT | - | 106 | C14 H9 Br N4 O3 S | c1cc(ccc1N.... |
41 | 4KD1 | - | 1QK | C21 H29 N6 O2 | CCc1cnn2c1.... |
42 | 2BTS | ic50 = 20 nM | U32 | C12 H15 N3 O2 S2 | CC(C)c1cnc.... |
43 | 3LE6 | ic50 = 0.035 uM | 2BZ | C17 H10 Cl N5 O2 | Cc1c-2nc(c.... |
44 | 2VTI | ic50 = 0.66 uM | LZ3 | C14 H12 N4 O3 S | c1ccc2c(c1.... |
45 | 3LFS | Ki = 2.5 uM | A07 | C17 H16 Cl N3 O | CCCC(=O)Nc.... |
46 | 1PXI | - | CK1 | C8 H5 Cl2 N3 S | c1cnc(nc1c.... |
47 | 1URW | ic50 < 0.003 uM | I1P | C21 H24 N8 O2 S | CN(C)CCCNS.... |
48 | 4LYN | - | 1YG | C20 H23 N3 O2 S2 | CC(c1ccccc.... |
49 | 1YKR | ic50 = 0.56 uM | 628 | C20 H14 Cl2 N4 O3 S | c1cc(c(c(c.... |
50 | 1PXN | Ki ~ 0.32 uM | CK6 | C15 H15 N5 O S | Cc1c(sc(n1.... |
51 | 1CKP | - | PVB | C20 H25 Cl N6 O3 | CC(C)C(CO).... |
52 | 1KE6 | ic50 = 5.7 nM | LS2 | C17 H15 N5 O3 S2 | CNS(=O)(=O.... |
53 | 2C6K | ic50 = 0.73 uM | DT2 | C17 H21 N7 O2 S | c1cc(ccc1N.... |
54 | 2R3Q | - | 5SC | C19 H16 Br N5 O | Cc1ccccc1c.... |
55 | 2R3J | ic50 = 10 nM | SCJ | C18 H14 Br N5 | c1ccc(cc1).... |
56 | 3IG7 | ic50 = 9 nM | EFP | C18 H22 N4 O3 | CC(=O)NC1C.... |
57 | 2VTS | ic50 = 0.03 uM | LZC | C16 H23 N7 | CC(C)Nc1cc.... |
58 | 1P2A | ic50 = 12 nM | 5BN | C17 H15 F N4 O | c1cc([nH]c.... |
59 | 2BHE | ic50 = 1 uM | BRY | C16 H9 Br N2 O2 | c1ccc2c(c1.... |
60 | 3UNK | ic50 = 15 uM | 0BY | C17 H13 Cl N4 O2 | c1ccc(c(c1.... |
61 | 1OIT | ic50 < 0.003 uM | HDT | C17 H14 N6 O2 S | c1ccn2c(c1.... |
62 | 2VTQ | ic50 = 0.14 uM | LZA | C16 H17 F2 N5 O2 | c1cc(c(c(c.... |
63 | 3NS9 | ic50 = 0.003 uM | NS9 | C20 H27 N5 O3 | CC(C)c1cnn.... |
64 | 2C68 | ic50 = 1.8 uM | CT6 | C18 H15 Br N5 | c1cc(cc(c1.... |
65 | 3TIZ | - | 3TI | C17 H13 N O2 | c1ccc2c(c1.... |
66 | 3PXY | ic50 = 5.9 uM | JWS | C10 H11 N5 O2 | COc1ccc(c(.... |
67 | 1H01 | ic50 = 22 uM | FAL | C21 H23 Cl2 N5 O2 | CN(C)CC(CO.... |
68 | 2EXM | - | ZIP | C10 H13 N5 | CC(=CCNc1c.... |
69 | 4BGH | ic50 = 4 nM | 3I6 | C13 H16 Br N5 O3 S | CC(CO)Nc1c.... |
70 | 2R3F | ic50 = 500 nM | SC8 | C18 H13 Cl2 N5 | c1cc(c(c(c.... |
71 | 2R3M | ic50 = 10 nM | SCX | C19 H17 F2 N7 | CCc1cnn2c1.... |
72 | 1GII | - | 1PU | C17 H16 N4 O2 | c1ccnc(c1).... |
73 | 2R64 | ic50 = 0.03 uM | 740 | C23 H27 N5 O3 S | c1cc(ccc1C.... |
74 | 2C6O | - | 4SP | C18 H22 N6 O3 S | c1cc(ccc1N.... |
75 | 1V1K | Ki = 35 uM | 3FP | C22 H23 F4 N5 O2 | CN(C)CC(CO.... |
76 | 2VTJ | ic50 = 1.9 uM | LZ4 | C10 H9 Cl N4 O2 S | c1cc(ccc1N.... |
77 | 2C6L | ic50 = 0.27 uM | DT4 | C17 H22 N8 O2 S | c1cc(ccc1N.... |
78 | 2W06 | - | FRV | C18 H20 N6 O2 S | Cc1ncc(n1C.... |
79 | 3EZV | - | EZV | C25 H25 N7 | CN1CCN(CC1.... |
80 | 4EZ7 | - | STU | C28 H26 N4 O3 | CC12C(C(CC.... |
81 | 3PXZ | Kd = 37 uM | 2AN | C16 H13 N O3 S | c1ccc(cc1).... |
82 | 1W0X | - | OLO | C15 H18 N6 O | Cn1cnc2c1n.... |
83 | 2XMY | Ki = 0.11 nM | CDK | C18 H21 N5 O4 S2 | CC1=C(SC(=.... |
84 | 2UZO | ic50 = 18 uM | C62 | C14 H10 N2 O5 S2 | c1cc(ccc1c.... |
85 | 2VTT | ic50 = 0.044 uM | LZD | C16 H17 F2 N5 O2 | c1cc(c(c(c.... |
86 | 1KE7 | ic50 = 8.9 nM | LS3 | C20 H15 N3 O4 S | c1cc2c(cc1.... |
87 | 2VU3 | ic50 = 0.047 uM | LZE | C16 H17 Cl2 N5 O2 | c1cc(c(c(c.... |
88 | 2B54 | - | D05 | C20 H15 Cl3 N4 O3 | CCc1c2c(n(.... |
89 | 1DM2 | - | HMD | C11 H10 Br N5 O2 | C1CNC(=O)C.... |
90 | 1DI8 | ic50 = 1 uM | DTQ | C16 H15 N3 O3 | COc1cc2c(c.... |
91 | 1GZ8 | - | MBP | C10 H13 N5 O2 | CC(C)C(=O).... |
92 | 3PY0 | ic50 = 0.13 uM | SU9 | C13 H11 N3 O2 | COc1ccc2c(.... |
93 | 2VTR | ic50 = 1.5 uM | LZB | C10 H10 Cl N5 | CC(C)Nc1cc.... |
94 | 1E1X | Ki = 1.3 uM | NW1 | C11 H17 N5 O2 | C1CCC(CC1).... |
95 | 1GIJ | - | 2PU | C19 H22 N6 O2 | c1cc2c(c(c.... |
96 | 3UNJ | ic50 = 11 uM | 0BX | C17 H14 N4 O2 | c1ccc(cc1).... |
97 | 2A0C | - | CK9 | C19 H26 N6 O2 | CCC(CO)Nc1.... |
98 | 3TIY | - | TIY | C11 H8 O5 | c1c2c(c(c(.... |
99 | 2R3I | ic50 = 1000 nM | SCF | C18 H14 F N5 | c1ccc(c(c1.... |
100 | 2R3P | ic50 = 900 nM | 3SC | C19 H12 Cl2 N6 S | c1cc(c(c(c.... |
101 | 1KE8 | ic50 = 1000 nM | LS4 | C18 H14 N4 O3 S2 | c1ccc2c(c1.... |
102 | 2C6I | ic50 = 11 uM | DT1 | C18 H22 N6 O3 S | c1cc(ccc1N.... |
103 | 1VYZ | ic50 = 290 nM | N5B | C13 H13 N3 O | c1ccc(cc1).... |
104 | 3WBL | ic50 = 23 uM | PDY | C20 H26 N6 O | CCOc1ccc(c.... |
105 | 1PXP | Ki ~ 0.22 uM | CK8 | C17 H19 N5 S | Cc1c(sc(n1.... |
106 | 4RJ3 | ic50 = 93 nM | 3QS | C22 H28 N6 O | COC1CCN(CC.... |
107 | 2VTN | ic50 = 0.85 uM | LZ7 | C12 H11 F N4 O2 | CC(=O)Nc1c.... |
108 | 1AQ1 | - | STU | C28 H26 N4 O3 | CC12C(C(CC.... |
109 | 2UZN | ic50 = 0.03 uM | C96 | C15 H13 N3 O4 S2 | [H]N=C1NC(.... |
110 | 2B55 | ic50 = 96 nM | D31 | C24 H31 N5 O2 | c1cc-2c(c(.... |
111 | 2C6M | ic50 = 0.35 uM | DT5 | C17 H20 N6 O3 S | c1cc(ccc1N.... |
112 | 3PJ8 | - | 404 | C19 H26 N6 O | CCC(CO)Nc1.... |
113 | 3LFQ | - | A28 | C17 H15 F2 N3 O | CCCC(=O)Nc.... |
114 | 2R3L | ic50 = 100 nM | SCW | C18 H14 Br N5 | c1ccc(cc1).... |
115 | 2W05 | ic50 = 0.001 uM | FRT | C20 H26 N6 O3 S | Cc1ncc(n1C.... |
116 | 1H08 | - | BYP BWP | n/a | n/a |
117 | 2XNB | Ki = 149 nM | Y8L | C19 H22 N6 O S | CC1=C(SC(=.... |
118 | 1HCK | - | ATP | C10 H16 N5 O13 P3 | c1nc(c2c(n.... |
119 | 1B38 | Kd = 0.254 uM | ATP | C10 H16 N5 O13 P3 | c1nc(c2c(n.... |
120 | 2B52 | ic50 = 8 nM | D42 | C21 H23 N7 O2 S | Cc1c(sc(n1.... |
121 | 1PXL | - | CK4 | C16 H13 F3 N4 S | Cc1c(sc(n1.... |
122 | 2R3H | ic50 = 20000 nM | SCE | C13 H13 N5 | Cc1cnc2n1c.... |
123 | 3LFN | Ki = 3160 nM | A27 | C23 H21 N3 O2 | CCCC(=O)Nc.... |
124 | 3S2P | ic50 = 0.068 uM | PMU | C17 H22 N4 O3 | CC(C)c1cc(.... |
125 | 2R3O | ic50 = 600 nM | 2SC | C19 H17 N5 O | c1ccc(cc1).... |
126 | 3IGG | ic50 = 95 nM | EFQ | C16 H19 N3 O3 | COc1ccc(cc.... |
127 | 1R78 | ic50 = 3 nM | FMD | C20 H20 F N3 O4 | CC(C(C(C#C.... |
128 | 2FVD | Ki = 0.003 uM | LIA | C18 H21 F2 N5 O4 S | COc1ccc(c(.... |
129 | 2VTL | ic50 = 97 uM | LZ5 | C10 H9 N3 O | c1ccc(cc1).... |
130 | 3PY1 | Kd = 37 uM | 2AN | C16 H13 N O3 S | c1ccc(cc1).... |
131 | 1KE9 | ic50 = 660 nM | LS5 | C16 H15 N5 O3 S | c1ccc2c(c1.... |
132 | 2A4L | ic50 = 0.4 uM | RRC | C19 H26 N6 O | CCC(CO)Nc1.... |
133 | 1Y8Y | ic50 = 2 uM | CT7 | C13 H11 Cl N4 O2 S | CS(=O)(=O).... |
134 | 1OIR | ic50 = 0.032 uM | HDY | C23 H26 N6 O2 | Cc1c(n2ccc.... |
135 | 1PXJ | - | CK2 | C9 H10 N4 S | Cc1c(sc(n1.... |
136 | 2VTO | ic50 = 0.14 uM | LZ8 | C17 H13 F N4 O2 | c1ccc(cc1).... |
137 | 1PYE | ic50 = 0.32 uM | PM1 | C21 H13 F2 N3 O2 | c1ccc(cc1).... |
138 | 2BTR | ic50 = 95 nM | U73 | C13 H15 N3 O S | CC(C)C1=CN.... |
139 | 2VTA | ic50 = 185 uM | LZ1 | C7 H6 N2 | c1ccc2c(c1.... |
140 | 4EZ3 | - | 0S0 | C11 H10 N4 O4 S | c1cc(ccc1N.... |
141 | 3EZR | - | EZR | C26 H27 N7 O | CN1CCN(CC1.... |
142 | 3ULI | ic50 = 0.07 uM | 1N3 | C21 H25 Br N6 O2 | COc1ccc(cc.... |
143 | 2DS1 | ic50 = 6.4 nM | 1CD | C22 H21 N5 O3 | CC1CC2CN1C.... |
144 | 1H07 | ic50 = 3 uM | MFP | C24 H27 Br N6 O2 | Cc1ccc(c(c.... |
145 | 2B53 | ic50 = 0.6 uM | D23 | C19 H19 F3 N4 | CC(C)(C)Nc.... |
146 | 2DUV | ic50 = 0.087 uM | 371 | C19 H17 N O7 S | Cc1cc2c(c(.... |
147 | 2VTH | ic50 = 120 uM | LZ2 | C10 H9 N O3 S | c1cc2c(ccc.... |
148 | 1KE5 | ic50 = 560 nM | LS1 | C16 H15 N3 O3 S | CNS(=O)(=O.... |
149 | 3FZ1 | - | B98 | C13 H15 N3 O2 S | COc1ccc2c(.... |
150 | 1WCC | ic50 = 350 uM | CIG | C4 H4 Cl N3 | c1c(nc(cn1.... |
151 | 4ACM | Ki = 210 nM | 7YG | C20 H23 N7 O3 S | CN(C)CCNS(.... |
152 | 2C5Y | ic50 = 0.25 uM | MTW | C19 H15 N7 O2 | c1cc(cc(c1.... |
153 | 1PXO | Ki = 2 nM | CK7 | C14 H12 N6 O2 S | Cc1c(sc(n1.... |
154 | 1H00 | ic50 = 38 uM | FAP | C21 H23 F2 N5 O2 | CN(C)CC(CO.... |
155 | 2R3R | - | 6SC | C18 H14 Br N5 | c1ccc(cc1).... |
156 | 2R3K | ic50 = 100 nM | SCQ | C18 H14 Br N5 | c1ccc(cc1).... |
157 | 2V0D | - | C53 | C9 H7 N3 O S | [H]N=C1NC(.... |
158 | 1B39 | Kd = 0.12 uM | ATP | C10 H16 N5 O13 P3 | c1nc(c2c(n.... |
159 | 2W1H | ic50 = 0.052 uM | L0F | C17 H13 N5 O | c1ccc(cc1).... |
160 | 1Y91 | ic50 = 0.059 uM | CT9 | C23 H33 N7 O2 S | CC(C)c1cnn.... |
161 | 2ZJW | ic50 = 0.04 uM | REF | C14 H6 O8 | c1c2c-3c(c.... |
162 | 3AT4 | Kd = 2.26 nM | CCK | C20 H20 N6 O2 | CC(C)Nc1cc.... |
163 | 3OWJ | Ki = 0.86 uM | 1EL | C17 H14 N2 O2 | Cc1c2c(c(c.... |
164 | 3MB7 | ic50 = 200 nM | 14I | C16 H8 O6 | c1cc2c(cc(.... |
165 | 2E9O | ic50 = 20 nM | A58 | C25 H27 N3 O2 | CC1CCC(CC1.... |
166 | 2WMQ | - | ZYQ | C9 H11 N3 O2 S | CC(=O)Nc1n.... |
167 | 2C3J | Ki = 0.659 uM | DBQ | C11 H11 N5 O2 | c1c[nH]c2c.... |
168 | 2YM7 | ic50 = 0.13 uM | YM7 | C15 H18 N8 | c1c(ncnc1N.... |
169 | 2X8I | ic50 = 0.19 uM | X8I | C17 H13 N3 O2 | CC1=CC2=NN.... |
170 | 2YDJ | ic50 = 0.005 uM | YDJ | C17 H19 F N4 O2 S | c1cc(cc(c1.... |
171 | 4QYE | ic50 = 1.2 uM | 3DL | C17 H12 N2 O3 | c1cc(cc(c1.... |
172 | 2BRO | ic50 = 1.4 uM | DF2 | C21 H20 N4 O2 | c1ccc(cc1).... |
173 | 2BRG | ic50 = 6.1 uM | DFY | C21 H19 N3 O2 | CN(CCO)c1c.... |
174 | 2YM5 | ic50 = 0.43 uM | YM5 | C18 H21 N5 O2 | c1cc(cc(c1.... |
175 | 4HYH | ic50 = 1 nM | 1AM | C22 H22 N6 O3 S | COc1ccc2c(.... |
176 | 2CGU | ic50 = 13.4 uM | 3A3 | C17 H13 N O7 | c1cc-2c(cc.... |
177 | 1NVS | Ki = 15 nM | UCM | C24 H15 N3 O3 | c1ccc2c(c1.... |
178 | 2YDK | ic50 = 0.007 uM | YDK | C17 H20 N4 O2 S | c1ccc(cc1).... |
179 | 3OT3 | ic50 = 0.005 uM | 22K | C16 H20 Br N7 | Cn1cc(cn1).... |
180 | 2WMR | ic50 = 52 uM | ZYR | C10 H10 N2 O S | C1CCc2c(c3.... |
181 | 3PA5 | ic50 = 2 nM | C73 | C17 H19 Cl N4 O2 S | c1cc(ccc1c.... |
182 | 2WMV | ic50 = 9.2 uM | ZYV | C10 H14 N6 O | c1[nH]c2c(.... |
183 | 2BRH | ic50 = 22 uM | DFW | C20 H15 N3 O3 | c1ccc(cc1).... |
184 | 1NVR | Ki = 7.8 nM | STU | C28 H26 N4 O3 | CC12C(C(CC.... |
185 | 2CGX | ic50 = 15.6 uM | 3D3 | C7 H8 N6 O S | c1nc(c2c(n.... |
186 | 3OT8 | ic50 = 0.009 uM | MI5 | C19 H22 N8 S | Cc1cc(sn1).... |
187 | 2YM4 | ic50 = 1.5 uM | 4YM | C21 H22 N6 O3 | CCOC(=O)c1.... |
188 | 4HYI | ic50 = 2 nM | 1AO | C21 H20 N6 O S | c1ccc2c(c1.... |
189 | 4QYF | - | 3DV | C17 H13 N3 O3 | c1cc(cc(c1.... |
190 | 3JVS | Ki = 0.146 uM | AGY | C22 H22 N4 O4 | CC(C)(C)c1.... |
191 | 2WMW | ic50 = 0.39 uM | ZYW | C11 H14 Br N5 O | c1c2c(c(cn.... |
192 | 2BR1 | Ki = 7.2 uM | PFP | C22 H21 N3 O4 | COc1ccc(cc.... |
193 | 2XF0 | ic50 = 30 uM | 4UB | C15 H11 N5 | c1ccc(cc1).... |
194 | 2C3L | Ki = 0.026 uM | IDZ | C14 H10 N4 | c1ccc2c(c1.... |
195 | 2YM6 | ic50 = 0.88 uM | YM6 | C14 H16 N6 O | c1cncc2c1c.... |
196 | 2X8E | ic50 = 0.014 uM | X8E | C16 H12 N4 O | CC1=CC2=NN.... |
197 | 4QYG | ic50 = 0.0041 uM | 3DW | C22 H21 N5 O2 | CN1CCN(CC1.... |
198 | 2X8D | ic50 = 0.8 uM | X8D | C11 H9 N3 O | CC1=CC2=NN.... |
199 | 2YEX | ic50 = 0.0001 uM | YEX | C15 H12 N4 O | CC1=CC2=NN.... |
200 | 2BRM | Ki = 1.3 uM | DFZ | C20 H18 N4 O | c1ccc(cc1).... |
201 | 2XEZ | ic50 = 1.5 uM | XEZ | C12 H9 N7 | c1c[nH]nc1.... |
202 | 1NVQ | Ki = 5.6 nM | UCN | C28 H26 N4 O4 | CC12C(C(CC.... |
203 | 3PA4 | ic50 = 3 nM | C72 | C19 H19 Cl N4 O S | c1cc(ccc1c.... |
204 | 2E9N | ic50 = 6.2 nM | 76A | C29 H27 N3 O3 | c1cc(ccc1c.... |
205 | 2YM3 | ic50 = 1.2 uM | YM3 | C14 H19 N5 O3 | CCOC(=O)c1.... |
206 | 2YDI | - | YDI | C16 H20 N4 O3 S | CN(C)CCOc1.... |
207 | 3EHA | - | ANP | C10 H17 N6 O12 P3 | c1nc(c2c(n.... |
208 | 1JKL | - | ANP | C10 H17 N6 O12 P3 | c1nc(c2c(n.... |
209 | 1JKK | - | ANP | C10 H17 N6 O12 P3 | c1nc(c2c(n.... |
210 | 3F5G | - | ADP | C10 H15 N5 O10 P2 | c1nc(c2c(n.... |
211 | 3F5U | - | ANP | C10 H17 N6 O12 P3 | c1nc(c2c(n.... |
212 | 1P4F | - | DRG | C12 H11 N3 | c1ccc-2c(c.... |
213 | 4TXC | Kd = 0.24 uM | 38G | C24 H27 N5 O3 | CN(C)CCNC(.... |
214 | 2YAK | ic50 = 2 nM | OSV | C27 H31 F N4 O3 Ru S4 | CC(C)Oc1cc.... |
215 | 3EH9 | - | ADP | C10 H15 N5 O10 P2 | c1nc(c2c(n.... |
216 | 1IG1 | - | ANP | C10 H17 N6 O12 P3 | c1nc(c2c(n.... |
217 | 3SHE | - | I85 | C24 H22 F3 N5 O2 | c1cc(cc(c1.... |
218 | 3R1N | - | 05B | C22 H21 N5 O3 | c1cc2c(cc1.... |
219 | 4AU8 | ic50 = 551 nM | Z3R | C11 H8 N2 O2 S3 | c1ccc2c(c1.... |
220 | 1REJ | Ki = 5 nM | B1L | C20 H22 N2 O5 | c1cc(ccc1C.... |
221 | 3BWJ | ic50 = 2.6 uM | ARX | C28 H47 N15 O7 | c1nc(c2c(n.... |
222 | 3AG9 | Ki = 9 nM | A02 | C40 H70 N18 O9 | c1nc(c2c(n.... |
223 | 3AGL | Ki = 16 nM | A03 | C37 H63 N17 O9 | CC(C(=O)NC.... |
224 | 1RE8 | Ki = 0.3 nM | BD2 | C27 H26 N2 O6 | c1ccc(c(c1.... |
225 | 2VZ6 | - | FEF | C20 H19 N3 O4 | c1ccc2c(c1.... |
226 | 2Z7Q | - | ACP | C11 H18 N5 O12 P3 | c1nc(c2c(n.... |
227 | 2Z7R | ic50 = 3 nM | STU | C28 H26 N4 O3 | CC12C(C(CC.... |
228 | 3QD4 | ic50 = 0.00000001 M | 3Q6 | C22 H30 N8 O2 | CC1CC(CN(C.... |
229 | 1Z5M | ic50 = 30 nM | LI8 | C23 H31 Br N8 O3 | CC(C)(C(=O.... |
230 | 3RCJ | ic50 = 0.8 uM | 3RC | C16 H13 N5 | c1ccc(cc1).... |
231 | 2PE0 | - | 39Z | C14 H12 N2 O2 | CC(c1ccc[n.... |
232 | 4CT2 | - | ATP | C10 H16 N5 O13 P3 | c1nc(c2c(n.... |
233 | 3QD0 | ic50 = 0.00000001 M | 3Q4 | C24 H26 N8 O | CC1CCC(CN1.... |
234 | 3ORZ | - | BI4 | C27 H26 N4 O2 | CN1CCCC1CC.... |
235 | 3HRC | - | ATP | C10 H16 N5 O13 P3 | c1nc(c2c(n.... |
236 | 3ION | ic50 = 8 nM | 8H1 | C28 H27 N5 O3 | COc1cc2c3c.... |
237 | 2XCH | ic50 = 374 nM | CKG | C22 H25 N7 O | c1c2c(nc(n.... |
238 | 4AW0 | - | MJF | C18 H15 Cl O5 | c1ccc(cc1).... |
239 | 1UU7 | ic50 = 14 uM | BI2 | C27 H26 N4 O2 | CN1CCCC1CC.... |
240 | 3OTU | - | BI4 | C27 H26 N4 O2 | CN1CCCC1CC.... |
241 | 3HRF | Kd = 10.3 uM | P47 | C17 H15 Cl O2 | c1ccc(cc1).... |
242 | 3QCS | ic50 = 0.00000001 M | 3Q1 | C15 H17 N7 O | c1cc2c(cc1.... |
243 | 3QCX | ic50 = 0.00000001 M | 3Q2 | C16 H19 N7 O | CC1COCCN1c.... |
244 | 1UU3 | ic50 = 0.75 uM | LY4 | C28 H28 N4 O3 | CN(C)CC1CC.... |
245 | 1H1W | - | ATP | C10 H16 N5 O13 P3 | c1nc(c2c(n.... |
246 | 3QC4 | ic50 = 0.002 uM | MP7 | C28 H22 F2 N4 O4 | c1ccc(cc1).... |
247 | 4AW1 | - | ATP | C10 H16 N5 O13 P3 | c1nc(c2c(n.... |
248 | 3QCY | ic50 = 0.00000001 M | 3Q3 | C22 H22 N8 O2 | c1ccc(cc1).... |
249 | 1UU8 | ic50 = 9 uM | BI1 | C25 H24 N4 O2 | CN(C)CCCn1.... |
250 | 4CT1 | - | ATP | C10 H16 N5 O13 P3 | c1nc(c2c(n.... |
251 | 2PE2 | - | 464 | C28 H30 N6 O3 | c1cc(cc(c1.... |
252 | 3H9O | ic50 = 70 nM | 9BD | C19 H19 N5 O3 | COCCOc1cc2.... |
253 | 4A07 | - | AZ7 | C17 H13 Cl3 N2 O2 | c1cc(ccc1C.... |
254 | 4KS7 | - | X4Z | C25 H28 N8 O S | Cc1nc2ccsc.... |
255 | 4KS8 | - | B49 | C22 H27 F N4 O2 | CCN(CC)CCN.... |
256 | 4DGO | ic50 = 0.57 uM | 0JW | C10 H10 N2 O3 | c1cc(c(cc1.... |
257 | 4DGM | ic50 = 1.2 uM | AGI | C15 H10 O5 | c1cc(ccc1C.... |
258 | 2PVJ | Ki = 0.005 uM | P44 | C19 H21 N7 | c1ccc(cc1).... |
259 | 4DGN | ic50 = 0.35 uM | LU2 | C15 H10 O6 | c1cc(c(cc1.... |
260 | 1M2Q | - | MNX | C13 H7 N O6 | c1cc(c2c(c.... |
261 | 1OM1 | Ki = 0.17 uM | IQA | C17 H12 N2 O3 | c1ccc2c(c1.... |
262 | 1ZOH | Ki = 0.1 uM | K44 | C10 H7 Br4 N3 | CN1CCn2c1n.... |
263 | 1M2R | - | MNY | C14 H10 N2 O4 | c1cc(c2c(c.... |
264 | 3KXN | - | K8X | C7 H2 I4 N2 | c1[nH]c2c(.... |
265 | 2PVK | Ki = 0.008 uM | P45 | C19 H14 Cl N7 | c1ccc(cc1).... |
266 | 1DAY | - | GNP | C10 H17 N6 O13 P3 | c1nc2c(n1C.... |
267 | 3SLS | - | ANP | C10 H17 N6 O12 P3 | c1nc(c2c(n.... |
268 | 4AUA | ic50 = 7.2 uM | 4AU | C12 H9 N3 O | c1ccc2c(c1.... |
269 | 2QHN | ic50 = 980 nM | 582 | C13 H13 N3 O | CCN1c2cccc.... |
270 | 3TKI | ic50 = 0.05 nM | S25 | C20 H23 N7 O2 S | c1cnc(cc1N.... |
271 | 2HXQ | ic50 = 144 nM | 373 | C24 H26 N4 O | c1ccc2c(c1.... |
272 | 2QHM | ic50 = 660 nM | 7CS | C16 H19 N3 O2 | CN1C2CCC1C.... |
273 | 2R0U | ic50 = 1 nM | M54 | C25 H22 N4 O2 | c1cc(cc(c1.... |
274 | 3TKH | ic50 = 47 nM | 07S | C23 H27 N7 O2 S | c1cc(cnc1).... |
275 | 2HXL | ic50 = 12 nM | 422 | C23 H24 N6 | c1cc2c(cc1.... |
276 | 2HOG | ic50 = 0.3 nM | 710 | C24 H25 N7 O | c1cc2c(cc1.... |
277 | 2XK6 | - | EQH | C18 H21 N3 O2 S | c1csc(c1C2.... |
278 | 2WQO | - | VGK | C21 H20 N2 O5 | COc1cc(cc(.... |
279 | 2XKE | ic50 = 4.2 uM | WI2 | C17 H20 N4 O3 | COc1cccc(c.... |
280 | 2XNN | - | 430 | C21 H16 F3 N3 O2 S | CC(c1ccccc.... |
281 | 2XK7 | ic50 = 1.5 uM | 30E | C21 H28 N4 O5 | CCC1CN(CCC.... |
282 | 4EQU | - | G6I | C30 H24 F3 N7 O2 | Cc1ccc(cc1.... |
283 | 2J7T | - | 274 | C28 H30 Cl N5 O4 S | Cc1c([nH]c.... |
284 | 3GGF | - | GVD | C22 H19 N7 | c1ccc2c(c1.... |
285 | 3D0E | ic50 = 13 nM | G93 | C21 H27 N7 O3 | CCn1c2c(cn.... |
286 | 2JDO | ic50 = 0.23 uM | I5S | C20 H22 Cl N3 O3 S | c1cc2cnccc.... |
287 | 2X39 | ic50 = 30 nM | X39 | C19 H21 Cl N6 O | c1cc(ccc1C.... |
288 | 3E87 | - | GLY ARG PRO ARG THR THR SER PHE ALA GLU | n/a | n/a |
289 | 1O6K | - | GLY ARG PRO ARG THR THR SER PHE ALA GLU | n/a | n/a |
290 | 3E88 | Ki = 2 nM | G96 | C24 H27 N7 O3 | CCn1c2cc(n.... |
291 | 4OBQ | ic50 = 0.065 uM | 2QT | C20 H20 F N5 O | c1cc2c(cc1.... |
292 | 4U43 | Kd = 48 uM | 3D8 | C11 H9 N5 | c1cc(cnc1).... |
293 | 4OBP | ic50 = 0.017 uM | 2QU | C12 H8 F N5 | c1cc(nc2c1.... |
294 | 4OBO | ic50 = 0.077 uM | 2QV | C14 H10 Cl N3 | c1cc(cc(c1.... |
295 | 4U44 | ic50 = 0.008 uM | 3D9 | C17 H13 N5 | c1ccc(cc1).... |
296 | 3DAK | - | ANP | C10 H17 N6 O12 P3 | c1nc(c2c(n.... |
297 | 4NW5 | ic50 = 0.02 uM | 2NR | C23 H21 F N2 O5 | COc1cccc(c.... |
298 | 4EL9 | - | AFE | C21 H20 O10 | CC1C(C(C(C.... |
299 | 4NUS | ic50 = 0.005 uM | 2NK | C22 H21 F2 N3 O | CN1CCN(CC1.... |
300 | 4NW6 | ic50 = 0.004 uM | 2NS | C23 H20 N4 O4 | COc1cc(cc(.... |
301 | 4GRB | ic50 = 17 nM | 0XG | C19 H18 N4 O4 S | CN(C)C(=O).... |
302 | 2YIT | ic50 = 0.29 nM | YIT | C21 H24 N6 O2 | CCCC(=NNC(.... |
303 | 2W0J | ic50 = 240 nM | ZAT | C19 H24 N10 O | [H]N=C(N)N.... |
304 | 2W7X | ic50 = 138 nM | D1A | C18 H17 N7 O3 | CC(=NNC(=N.... |
305 | 4A9U | - | A9U | C27 H28 N4 O2 | c1ccc(cc1).... |
306 | 2XK9 | ic50 = 0.03 nM | XK9 | C18 H17 N7 O4 | CC(=NNC(=N.... |
307 | 2YCS | ic50 = 1.36 nM | NXP | C18 H18 N6 O | CC(=NNC(=N.... |
308 | 2YCF | ic50 = 0.7 nM | YCF | C19 H24 N10 O3 | CC(=NNC(=N.... |
309 | 2WTI | ic50 = 0.092 uM | WTI | C18 H15 N3 O3 S | c1cc(ccc1c.... |
310 | 2YIR | ic50 = 0.17 nM | YIR | C20 H19 N7 O3 | c1cc2cc([n.... |
311 | 2XBJ | ic50 = 0.86 uM | XBJ | C23 H27 F N4 O4 | CC(C)(C1CN.... |
312 | 4BDI | ic50 = 227.7 uM | HAU | C14 H19 N3 O2 | Cc1ccc(nc1.... |
313 | 2XM9 | ic50 = 0.009 uM | LWH | C21 H20 N6 O | c1ccc2c(c1.... |
314 | 2YCR | ic50 = 69.6 nM | HCW | C23 H28 N10 O | CC(=NNC1=N.... |
315 | 2YIQ | ic50 = 12.67 nM | YIQ | C20 H19 N7 O | CC(=NNC(=N.... |
316 | 2WTJ | ic50 = 0.7 uM | WTJ | C16 H20 N4 O3 S | CN(C)CCNC(.... |
317 | 2CN5 | - | ADP | C10 H15 N5 O10 P2 | c1nc(c2c(n.... |
318 | 4FII | - | ARG PRO LYS PRO LEU VAL ASP PRO | n/a | n/a |
319 | 4JDK | - | ARG ARG ARG ARG SER TRP TYR | n/a | n/a |
320 | 4JDI | - | ARG ARG ARG ARG SER TRP TYR | n/a | n/a |
321 | 3A7H | - | ATP | C10 H16 N5 O13 P3 | c1nc(c2c(n.... |
322 | 3A7J | - | ADP | C10 H15 N5 O10 P2 | c1nc(c2c(n.... |
323 | 3A7I | - | ADE | C5 H5 N5 | c1[nH]c2c(.... |
324 | 1U5R | - | ATP | C10 H16 N5 O13 P3 | c1nc(c2c(n.... |
325 | 3EQC | - | AGS | C10 H16 N5 O12 P3 S | c1nc(c2c(n.... |
326 | 3EQH | - | ADP | C10 H15 N5 O10 P2 | c1nc(c2c(n.... |
327 | 3EQI | - | ADP | C10 H15 N5 O10 P2 | c1nc(c2c(n.... |
328 | 2J51 | - | DKI | C15 H13 F2 N7 O2 S2 | c1cc(c(c(c.... |
329 | 2UV2 | - | GVD | C22 H19 N7 | c1ccc2c(c1.... |
330 | 2JFL | - | DKI | C15 H13 F2 N7 O2 S2 | c1cc(c(c(c.... |
331 | 4FG9 | - | ATP | C10 H16 N5 O13 P3 | c1nc(c2c(n.... |
332 | 4FG8 | - | ATP | C10 H16 N5 O13 P3 | c1nc(c2c(n.... |
333 | 4JQE | - | ANP | C10 H17 N6 O12 P3 | c1nc(c2c(n.... |
334 | 1QL6 | - | ATP | C10 H16 N5 O13 P3 | c1nc(c2c(n.... |
335 | 1PHK | - | ATP | C10 H16 N5 O13 P3 | c1nc(c2c(n.... |
336 | 2F57 | - | 23D | C19 H24 Cl N7 | CCn1cnc2c1.... |
337 | 1XJD | Ki = 0.33 nM | STU | C28 H26 N4 O3 | CC12C(C(CC.... |
338 | 3A62 | - | STU | C28 H26 N4 O3 | CC12C(C(CC.... |
339 | 3WF9 | ic50 = 567 nM | FS7 | C24 H25 N3 O5 S | CC1CCc2c(c.... |
340 | 3WF8 | ic50 = 232 nM | F76 | C23 H23 N3 O5 S | c1ccc2c(c1.... |
341 | 4L3L | - | 5FI | C19 H21 F3 N6 | CCc1cncnc1.... |
342 | 3WE4 | ic50 = 15 nM | 5FI | C19 H21 F3 N6 | CCc1cncnc1.... |
343 | 3WF7 | ic50 = 206 nM | FS9 | C18 H17 F3 N6 O | c1cc(cc(c1.... |
344 | 4L3J | - | 5FI | C19 H21 F3 N6 | CCc1cncnc1.... |
345 | 3WF6 | ic50 = 33 nM | FZ9 | C18 H16 N6 | c1ccc2c(c1.... |
346 | 4OTI | ic50 = 43 nM | MI1 | C16 H20 N6 O | CC1CCN(CC1.... |
347 | 2VN9 | - | GVD | C22 H19 N7 | c1ccc2c(c1.... |
348 | 4EJN | ic50 = 0.005 uM | 0R4 | C33 H26 F N7 O2 | CC(=O)Nc1c.... |
349 | 2V7O | - | DRN | C25 H23 N5 O2 S | [H]N=C(N)S.... |
350 | 2WEI | ic50 = 3.4 nM | VGG | C17 H21 N5 | Cc1cccc(c1.... |
351 | 3CQW | ic50 = 42 nM | CQW | C12 H11 Cl N6 | c1c(c2c([n.... |
352 | 3MV5 | ic50 = 180 nM | XFE | C11 H15 N5 | Cc1c[nH]c2.... |
353 | 3QKL | - | SMR | C29 H40 N4 O5 S | CCOCCN(CC(.... |
354 | 4GV1 | ic50 = 3 nM | 0XZ | C21 H25 Cl N6 O2 | c1cc(ccc1C.... |
355 | 3QKM | ic50 = 0.038 uM | SM9 | C31 H43 N5 O4 S | CCOCCN(CC(.... |
356 | 3MVH | ic50 = 0.5 nM | WFE | C20 H22 F2 N6 O | CCc1c[nH]c.... |
357 | 3CQU | ic50 = 151 nM | CQU | C15 H13 N7 | Cc1[nH]c(n.... |
358 | 3Q53 | - | ATP | C10 H16 N5 O13 P3 | c1nc(c2c(n.... |
359 | 4O0R | Ki = 0.036 uM | X4Z | C25 H28 N8 O S | Cc1nc2ccsc.... |
360 | 4EQC | ic50 = 0.008 uM | XR1 | C29 H28 Cl N7 O S | CCN1c2c(cn.... |
361 | 3FY0 | ic50 = 1090 nM | DW1 | C23 H13 N3 O4 Ru | C1=CC(C=C1.... |
362 | 3FXZ | ic50 = 130 nM | FLL | C30 H18 Cl F N5 O4 Ru | c1ccc(cc1).... |
363 | 3Q4Z | - | ANP | C10 H17 N6 O12 P3 | c1nc(c2c(n.... |
364 | 3GC0 | - | AMP | C10 H14 N5 O7 P | c1nc(c2c(n.... |
365 | 3MFU | - | ANP | C10 H17 N6 O12 P3 | c1nc(c2c(n.... |
366 | 3C0I | - | 3AM | C10 H14 N5 O7 P | c1nc(c2c(n.... |
367 | 3MFS | - | ANP | C10 H17 N6 O12 P3 | c1nc(c2c(n.... |
368 | 3MFR | - | ANP | C10 H17 N6 O12 P3 | c1nc(c2c(n.... |
369 | 3TXO | ic50 = 9 nM | 07U | C17 H19 N5 | CC(C)(CNc1.... |
370 | 4OTH | ic50 = 9 nM | DRN | C25 H23 N5 O2 S | [H]N=C(N)S.... |
371 | 2J90 | - | IZA | C18 H16 F N3 O | CC(C)(C)c1.... |
372 | 3BHY | - | 7CP | C18 H18 Cl2 N4 O | Cn1c2c(ccc.... |
373 | 1V0P | ic50 = 0.13 uM | PVB | C20 H25 Cl N6 O3 | CC(C)C(CO).... |
374 | 1V0O | ic50 = 5.5 uM | INR | C16 H10 N2 O5 S | c1ccc2c(c1.... |
375 | 4NJD | ic50 = 0.79 uM | NJD | C21 H20 N8 O | COc1nc(nc(.... |
376 | 4APP | Ki = 0.064 uM | N53 | C33 H36 N6 O3 | CC1(c2c(c(.... |
377 | 4O0X | Ki = 0.068 uM | 2OQ | C19 H20 N6 O | Cc1nc2ccc(.... |
378 | 2X4Z | Ki = 18.7 nM | X4Z | C25 H28 N8 O S | Cc1nc2ccsc.... |
379 | 4O0Y | Ki = 0.06 uM | 2OO | C17 H19 N7 O | CCNc1nc2cc.... |
380 | 2CDZ | - | 23D | C19 H24 Cl N7 | CCn1cnc2c1.... |
381 | 3A8W | - | ATP | C10 H16 N5 O13 P3 | c1nc(c2c(n.... |
382 | 3AQV | - | TAK | C24 H25 N5 O | c1cc(ccc1c.... |
383 | 3WAR | - | NIO | C6 H5 N O2 | c1cc(cnc1).... |
384 | 2YAB | - | AMP | C10 H14 N5 O7 P | c1nc(c2c(n.... |
385 | 2YAA | - | ATP | C10 H16 N5 O13 P3 | c1nc(c2c(n.... |
This union binding pocket(no: 1) in the query (biounit: 2xmy.bio1) has 51 residues | ||||
---|---|---|---|---|
No: | Leader PDB | Ligand | P-value (APoc) | PS_Score (APoc) |
1 | 4K77 | 1Q4 | 0.000000008642 | 0.78177 |
2 | 2OIC | STU | 0.000000004078 | 0.77562 |
3 | 2OIC | STU | 0.000000004306 | 0.77439 |
4 | 2OIC | STU | 0.000000003673 | 0.767 |
5 | 4IVB | 1J5 | 0.000000006492 | 0.75438 |
6 | 4IVC | 1J6 | 0.000000001688 | 0.7536 |
7 | 4C4F | 7CE | 0.000000001111 | 0.75291 |
8 | 2NRY | STU | 0.000000004389 | 0.75275 |
9 | 4IVB | 1J5 | 0.000000005006 | 0.74989 |
10 | 4EHZ | JAK | 0.00000001335 | 0.74877 |
11 | 4EHZ | JAK | 0.00000001349 | 0.74855 |
12 | 4EHZ | JAK | 0.00000001383 | 0.74799 |
13 | 4K77 | 1Q4 | 0.0000000224 | 0.74779 |
14 | 4EI4 | 0Q2 | 0.00000001404 | 0.74763 |
15 | 4EI4 | 0Q2 | 0.00000001418 | 0.74742 |
16 | 4IVC | 1J6 | 0.000000002339 | 0.74679 |
17 | 4E4L | 0NH | 0.000000009809 | 0.74524 |
18 | 4C58 | 824 | 0.000000006763 | 0.74337 |
19 | 4E4L | 0NH | 0.00000001068 | 0.74336 |
20 | 4EHZ | JAK | 0.00000001965 | 0.74003 |
21 | 3HMO | STU | 0.000000008125 | 0.73939 |
22 | 3V8S | 0HD | 0.000000008214 | 0.73915 |
23 | 4JR7 | GNP | 0.00000001323 | 0.73862 |
24 | 3V8S | 0HD | 0.000000008439 | 0.73857 |
25 | 4IVD | 15T | 0.000000002361 | 0.73749 |
26 | 4E4L | 0NH | 0.00000000897 | 0.73724 |
27 | 3LXN | MI1 | 0.000000002483 | 0.73645 |
28 | 4IVD | 15T | 0.00000000256 | 0.73583 |
29 | 3OFM | 4B0 | 0.0000001483 | 0.73529 |
30 | 2OIC | STU | 0.00000002605 | 0.73365 |
31 | 2R5T | ANP | 0.000000001862 | 0.73355 |
32 | 2R5T | ANP | 0.000000001862 | 0.73355 |
33 | 2OID | ANP | 0.000000007709 | 0.73099 |
34 | 4C2W | ANP | 0.00000006403 | 0.72349 |
35 | 1U59 | STU | 0.00000001117 | 0.7231 |
36 | 2F2U | M77 | 0.00000006693 | 0.72247 |
37 | 4E4N | 0NL | 0.000000007792 | 0.7217 |
38 | 4E6Q | 0NV | 0.000000007985 | 0.72119 |
39 | 4E6Q | 0NV | 0.000000005634 | 0.71969 |
40 | 2NRY | STU | 0.00000002093 | 0.71886 |
41 | 2NRY | STU | 0.00000003512 | 0.71699 |
42 | 2OID | ANP | 0.00000002291 | 0.71689 |
43 | 3EYH | IZA | 0.00000001518 | 0.71658 |
44 | 4FK6 | 0UJ | 0.00000002403 | 0.71586 |
45 | 4E6D | 0NU | 0.00000001066 | 0.71517 |
46 | 2R5T | ANP | 0.000000003173 | 0.71461 |
47 | 3EYG | MI1 | 0.00000001133 | 0.71389 |
48 | 2ZV2 | 609 | 0.0000001003 | 0.7131 |
49 | 4FK6 | 0UJ | 0.00000002736 | 0.71305 |
50 | 1O9U | ADZ | 0.0000005691 | 0.71281 |
51 | 4E4N | 0NL | 0.00000001899 | 0.71182 |
52 | 2NRY | STU | 0.00000002931 | 0.71155 |
53 | 2F2U | M77 | 0.0000001105 | 0.71086 |
54 | 4G31 | 0WH | 0.00000002408 | 0.70677 |
55 | 3UIM | ANP | 0.00000002523 | 0.70578 |
56 | 2PVN | P63 | 0.0000000006883 | 0.70575 |
57 | 3OWL | 19E | 0.0000004353 | 0.70477 |
58 | 3HZT | J60 | 0.0000001467 | 0.7043 |
59 | 4KWP | EXX | 0.0000005084 | 0.70193 |
60 | 3SRV | S19 | 0.00000004779 | 0.70094 |
61 | 2B9F | ADP | 0.00000003364 | 0.69966 |
62 | 3F7Z | 34O | 0.00000005134 | 0.69939 |
63 | 4E1Z | 0MX | 0.000000006907 | 0.69926 |
64 | 4GJ3 | 0XP | 0.0000000004638 | 0.69894 |
65 | 4N6Z | 2HW | 0.0000001266 | 0.69787 |
66 | 3LXK | MI1 | 0.000000001612 | 0.69729 |
67 | 4OH4 | ANP | 0.00000004109 | 0.69541 |
68 | 3OWK | 18E | 0.0000006425 | 0.69436 |
69 | 4F9C | 0SX | 0.00000006635 | 0.69383 |
70 | 4OAC | ADP | 0.00000004683 | 0.69263 |
71 | 3ALN | ANP | 0.00000007264 | 0.69186 |
72 | 3TTI | KBI | 0.00000003264 | 0.69182 |
73 | 3CY2 | MB9 | 0.0000002543 | 0.69158 |
74 | 4IDT | T28 | 0.00000007738 | 0.69049 |
75 | 3F7Z | 34O | 0.0000001825 | 0.6896 |
76 | 2JLD | AG1 | 0.000000001153 | 0.68954 |
77 | 4MWH | ATP | 0.00000002529 | 0.68896 |
78 | 4MWH | ATP | 0.00000002529 | 0.68896 |
79 | 4OH4 | ANP | 0.00000004225 | 0.68644 |
80 | 3BI6 | 396 | 0.00000001959 | 0.68627 |
81 | 3SRV | S19 | 0.0000001442 | 0.6857 |
82 | 3H9R | TAK | 0.0000005055 | 0.68541 |
83 | 3BRB | ADP | 0.0000006048 | 0.68116 |
84 | 2B9J | ADP | 0.0000001195 | 0.68106 |
85 | 2JLD | AG1 | 0.000000001007 | 0.67886 |
86 | 3FI3 | JK2 | 0.00000006217 | 0.67839 |
87 | 3BRB | ADP | 0.000000759 | 0.67579 |
88 | 3ZOS | 0LI | 0.0000003389 | 0.67559 |
89 | 4I94 | ANP | 0.0000002377 | 0.67464 |
90 | 4IZY | 1J2 | 0.00000005256 | 0.67399 |
91 | 1OPK | P16 | 0.00000003647 | 0.67379 |
92 | 4GW8 | 3RA | 0.0000006053 | 0.67151 |
93 | 4F99 | ADP | 0.0000001913 | 0.67086 |
94 | 4X0M | 3WA | 0.000001958 | 0.67083 |
95 | 2B9I | ADP | 0.0000001346 | 0.67017 |
96 | 2O2U | 738 | 0.0000002939 | 0.66994 |
97 | 3IGO | ANP | 0.00000004449 | 0.66979 |
98 | 2H8H | H8H | 0.0000001372 | 0.66977 |
99 | 2OID | ANP | 0.00000009404 | 0.66975 |
100 | 4BHN | BH9 | 0.00000002168 | 0.66946 |
101 | 2P2H | 994 | 0.0000003109 | 0.66869 |
102 | 4C2V | YJA | 0.000000003822 | 0.66814 |
103 | 4MQ1 | 2C3 | 0.00000007037 | 0.66802 |
104 | 2QCS | ANP | 0.00000001159 | 0.66756 |
105 | 2JLD | AG1 | 0.000000001366 | 0.66741 |
106 | 1Q8Y | ADE | 0.000001088 | 0.66725 |
107 | 4F9A | ADP | 0.0000002343 | 0.66645 |
108 | 1CM8 | ANP | 0.0000002383 | 0.66609 |
109 | 1CM8 | ANP | 0.000000245 | 0.66548 |
110 | 3M2W | L8I | 0.0000005341 | 0.6653 |
111 | 3JPV | 1DR | 0.000001834 | 0.66455 |
112 | 4MQ1 | 2C3 | 0.0000001253 | 0.66377 |
113 | 4MKC | 4MK | 0.00000008975 | 0.66304 |
114 | 2RIO | ADP | 0.0000002889 | 0.66191 |
115 | 4N70 | 2HX | 0.0000006261 | 0.6617 |
116 | 4OA2 | ADP | 0.0000001439 | 0.66088 |
117 | 4CNH | 3U9 | 0.0000002313 | 0.65866 |
118 | 4MQ1 | 2C3 | 0.00000008274 | 0.65733 |
119 | 3FHI | ANP | 0.00000002248 | 0.65514 |
120 | 4H3P | ANP | 0.0000002764 | 0.65487 |
121 | 4MQ1 | 2C3 | 0.0000001338 | 0.65486 |
122 | 3IDB | ANP | 0.00000006686 | 0.65446 |
123 | 3EKK | GS2 | 0.00000007014 | 0.65352 |
124 | 2OID | ANP | 0.0000006187 | 0.65345 |
125 | 4X2J | 3WN | 0.0000006224 | 0.65332 |
126 | 4X2K | 3WO | 0.0000006224 | 0.65332 |
127 | 2OXY | K17 | 0.000003736 | 0.65327 |
128 | 4BHN | BH9 | 0.0000001023 | 0.65306 |
129 | 4FL3 | ANP | 0.0000001031 | 0.6529 |
130 | 4I94 | ANP | 0.0000004544 | 0.65208 |
131 | 2PVF | ACP | 0.0000004603 | 0.6518 |
132 | 4MBI | 26K | 0.000001454 | 0.65123 |
133 | 3EQR | T74 | 0.0000000419 | 0.64995 |
134 | 3ALN | ANP | 0.0000001712 | 0.64982 |
135 | 3THB | 3TA | 0.000000002008 | 0.64923 |
136 | 3THB | 3TA | 0.000000002008 | 0.64923 |
137 | 2OXY | K17 | 0.000003848 | 0.64917 |
138 | 3VRY | B43 | 0.00000004479 | 0.64867 |
139 | 4F1M | ACP | 0.0000008052 | 0.64761 |
140 | 2VAG | V25 | 0.0000003921 | 0.64744 |
141 | 4CCU | AWF | 0.0000005925 | 0.64632 |
142 | 3FHR | P4O | 0.0000002897 | 0.64629 |
143 | 3GQI | ACP | 0.0000004154 | 0.64621 |
144 | 4BFM | ANP | 0.0000002052 | 0.64611 |
145 | 3ZRM | ZRM | 0.0000004399 | 0.64499 |
146 | 3KRL | KRL | 0.0000001547 | 0.64475 |
147 | 4NWM | 2P5 | 0.0000001176 | 0.64333 |
148 | 4F9A | ADP | 0.0000007037 | 0.64259 |
149 | 2WU6 | DKI | 0.0000001382 | 0.64014 |
150 | 2WQN | ADP | 0.00000166 | 0.63964 |
151 | 2QLU | ADE | 0.000005709 | 0.63843 |
152 | 1VJY | 460 | 0.00000005779 | 0.63744 |
153 | 4QTB | 38Z | 0.00000003115 | 0.63657 |
154 | 4H3P | ANP | 0.0000006571 | 0.63646 |
155 | 3UYT | 0CK | 0.0000004667 | 0.63634 |
156 | 3ALN | ANP | 0.000002854 | 0.63563 |
157 | 3VRY | B43 | 0.00000004676 | 0.6352 |
158 | 4AT3 | LTI | 0.000001017 | 0.63461 |
159 | 3MB6 | 01I | 0.000007214 | 0.63456 |
160 | 4EUU | BX7 | 0.00000006779 | 0.63445 |
161 | 3EQR | T74 | 0.00000006943 | 0.634 |
162 | 3EQR | T74 | 0.00000006943 | 0.634 |
163 | 4QTB | 38Z | 0.00000003712 | 0.63339 |
164 | 4F1T | H52 | 0.000008776 | 0.63193 |
165 | 2X2M | X2M | 0.0000003069 | 0.63099 |
166 | 4I6H | 1C8 | 0.0000008885 | 0.63004 |
167 | 4KBA | 1QM | 0.0000009314 | 0.62904 |
168 | 4KBA | 1QM | 0.0000009314 | 0.62904 |
169 | 3PP0 | 03Q | 0.0000002713 | 0.62682 |
170 | 4F9B | 0SY | 0.000009786 | 0.62672 |
171 | 4K1B | 1OC | 0.00000152 | 0.62588 |
172 | 3GC8 | B45 | 0.0000004182 | 0.62477 |
173 | 3GNI | ATP | 0.000000614 | 0.62369 |
174 | 4DCE | 0JF | 0.0000004583 | 0.62293 |
175 | 4OAV | ACP | 0.00000175 | 0.62282 |
176 | 4H3Q | ANP | 0.0000003344 | 0.6227 |
177 | 3SXS | PP2 | 0.000000647 | 0.62261 |
178 | 4K33 | ACP | 0.0000009695 | 0.6211 |
179 | 1Q8Y | ADP | 0.0000007114 | 0.62067 |
180 | 3BU5 | ATP | 0.000001409 | 0.62024 |
181 | 2EVA | ADN | 0.00000006249 | 0.61824 |
182 | 3SXF | BK5 | 0.00000001824 | 0.61786 |
183 | 4KBC | 1QJ | 0.000004415 | 0.6175 |
184 | 4AG8 | AXI | 0.00000003586 | 0.61699 |
185 | 2NRU | T12 | 0.000002505 | 0.61505 |
186 | 3PP0 | 03Q | 0.000000196 | 0.61455 |
187 | 3UZP | 0CK | 0.000001905 | 0.61382 |
188 | 4F1O | ACP | 0.000005195 | 0.61381 |
189 | 4FOC | 0UU | 0.000002735 | 0.61314 |
190 | 4CQE | CQE | 0.0000005464 | 0.61301 |
191 | 2CSN | CKI | 0.0000002203 | 0.61236 |
192 | 3GC8 | B45 | 0.0000006136 | 0.61072 |
193 | 2QU6 | 857 | 0.0000003557 | 0.60917 |
194 | 4F9B | 0SY | 0.00002072 | 0.60718 |
195 | 1ZY5 | ANP | 0.000004001 | 0.60488 |
196 | 4KBC | 1QJ | 0.000007784 | 0.60466 |
197 | 4KBC | 1QJ | 0.000007784 | 0.60466 |
198 | 2QU6 | 857 | 0.0000008453 | 0.6044 |
199 | 4AOI | 4K0 | 0.000005837 | 0.60373 |
200 | 2A19 | ANP | 0.00001137 | 0.60364 |
201 | 4JX7 | 1N6 | 0.000008357 | 0.60305 |
202 | 4KBA | 1QM | 0.000004353 | 0.60305 |
203 | 4NFN | 2KC | 0.000004368 | 0.60298 |
204 | 3VHE | 42Q | 0.0000001469 | 0.60297 |
205 | 4CD0 | AWJ | 0.000001248 | 0.6028 |
206 | 3UYT | 0CK | 0.000002346 | 0.60266 |
207 | 3ZBF | VGH | 0.00000633 | 0.60193 |
208 | 3UZP | 0CK | 0.000002476 | 0.60154 |
209 | 3UZP | 0CK | 0.000002476 | 0.60154 |
210 | 3BQC | EMO | 0.000001355 | 0.60114 |
211 | 4CNH | 3U9 | 0.00001304 | 0.60046 |
212 | 4QTC | 38Z | 0.0000005687 | 0.60023 |
213 | 2NRU | T12 | 0.000003614 | 0.6002 |
214 | 2Y6O | 1N1 | 0.000001449 | 0.5998 |
215 | 4CLJ | 5P8 | 0.000005177 | 0.59929 |
216 | 4TWC | 37J | 0.000005232 | 0.59907 |
217 | 1XKK | FMM | 0.00000002326 | 0.59884 |
218 | 4CQE | CQE | 0.000001621 | 0.59755 |
219 | 2P2I | 608 | 0.0000009215 | 0.59675 |
220 | 2P2I | 608 | 0.0000009748 | 0.59566 |
221 | 2XVD | AS6 | 0.000000316 | 0.59453 |
222 | 3RI1 | 3RH | 0.0000005825 | 0.59413 |
223 | 2HK5 | 1BM | 0.000002656 | 0.59372 |
224 | 4AT5 | MUJ | 0.000002029 | 0.59304 |
225 | 2NRU | T12 | 0.000003828 | 0.59246 |
226 | 1XR1 | ANP | 0.000004061 | 0.59123 |
227 | 4F0F | ACP | 0.00001047 | 0.59079 |
228 | 4DCE | 0JF | 0.0000032 | 0.5899 |
229 | 4KBA | 1QM | 0.00001524 | 0.58946 |
230 | 1ZP9 | ATP | 0.000008661 | 0.58813 |
231 | 4TW9 | 386 | 0.000008809 | 0.58776 |
232 | 3PVW | QRX | 0.000000827 | 0.58756 |
233 | 4RLL | E91 | 0.00005141 | 0.58574 |
234 | 1ZTH | ADP | 0.00002511 | 0.58531 |
235 | 4PMT | 31Y | 0.00000541 | 0.58524 |
236 | 4NWM | 2P5 | 0.000000006058 | 0.58371 |
237 | 1ZP9 | ATP | 0.00001119 | 0.58257 |
238 | 1ZTH | ADP | 0.00003022 | 0.58102 |
239 | 3UYT | 0CK | 0.000006744 | 0.58065 |
240 | 4HNF | 16W | 0.00003138 | 0.58015 |
241 | 1ULE | GLA GAL NAG | 0.00006909 | 0.58007 |
242 | 4KBA | 1QM | 0.000009946 | 0.57868 |
243 | 1ZTH | ADP | 0.0000339 | 0.57836 |
244 | 4KNB | 1RU | 0.00001988 | 0.57659 |
245 | 4AT4 | T6E | 0.000006323 | 0.57596 |
246 | 4ASE | AV9 | 0.000001285 | 0.5741 |
247 | 3QUP | LUN | 0.00001689 | 0.57364 |
248 | 4HNF | 16W | 0.00001722 | 0.57322 |
249 | 3E8N | ATP | 0.00000002344 | 0.57218 |
250 | 3E8N | VRA | 0.00000002344 | 0.57218 |
251 | 3E8N | VRA | 0.00000002344 | 0.57218 |
252 | 3E8N | ATP | 0.00000002344 | 0.57218 |
253 | 4MK0 | 29X | 0.000003295 | 0.57204 |
254 | 4KNB | 1RU | 0.00002601 | 0.57063 |
255 | 4PMM | 31V | 0.000006189 | 0.57063 |
256 | 4TWC | 37J | 0.00001101 | 0.57041 |
257 | 4ORK | GDP | 0.00003612 | 0.56993 |
258 | 3UYT | 0CK | 0.00001135 | 0.56979 |
259 | 1ZP9 | ATP | 0.0000271 | 0.56972 |
260 | 1ZP9 | ATP | 0.00002803 | 0.56898 |
261 | 3ORK | AGS | 0.000002995 | 0.56857 |
262 | 4FOB | 0US | 0.000005668 | 0.56685 |
263 | 2NRU | T12 | 0.00001063 | 0.56533 |
264 | 4LRJ | ANP | 0.00002489 | 0.56523 |
265 | 4IWD | 1JC | 0.0000004509 | 0.56395 |
266 | 4WHZ | 3NL | 0.0000001206 | 0.56378 |
267 | 4C2V | YJA | 0.000001029 | 0.56345 |
268 | 3RE4 | TO1 | 0.00002723 | 0.56328 |
269 | 1ZTH | ADP | 0.00005074 | 0.56224 |
270 | 2XB7 | GUI | 0.0000001047 | 0.56184 |
271 | 3ZOS | 0LI | 0.000002508 | 0.56177 |
272 | 4LRJ | ANP | 0.00002979 | 0.56133 |
273 | 4C2W | ANP | 0.0001516 | 0.56053 |
274 | 3TDV | GDP | 0.00002377 | 0.56015 |
275 | 4ORK | GDP | 0.00003338 | 0.55886 |
276 | 4ORK | GDP | 0.00002717 | 0.55731 |
277 | 3TDV | GDP | 0.00002853 | 0.55627 |
278 | 3RI1 | 3RH | 0.000004482 | 0.55588 |
279 | 4LOO | SB4 | 0.00003054 | 0.55482 |
280 | 1Y57 | MPZ | 0.00001158 | 0.55274 |
281 | 4KNB | 1RU | 0.00007755 | 0.55264 |
282 | 4KNB | 1RU | 0.00005872 | 0.5526 |
283 | 4Q5H | ANP | 0.00003519 | 0.55181 |
284 | 3RE4 | TO1 | 0.0001086 | 0.55142 |
285 | 4ITH | RCM | 0.00004839 | 0.5508 |
286 | 4PNI | KQQ | 0.00000432 | 0.54708 |
287 | 4CYI | ATP | 0.00002616 | 0.5469 |
288 | 2CFM | AMP | 0.0001327 | 0.54678 |
289 | 2XNM | WGZ | 0.000003649 | 0.5456 |
290 | 4E93 | GUI | 0.000002354 | 0.54453 |
291 | 4ITH | RCM | 0.0000653 | 0.5443 |
292 | 3WG3 | A2G GAL NAG FUC | 0.0003035 | 0.54406 |
293 | 4F4P | 0SB | 0.000000214 | 0.54309 |
294 | 3LKM | AMP | 0.00004181 | 0.54259 |
295 | 2PZI | AXX | 0.0001301 | 0.54093 |
296 | 4CYI | ATP | 0.0000478 | 0.5398 |
297 | 4CYI | ATP | 0.0000495 | 0.53907 |
298 | 2PZI | AXX | 0.0001509 | 0.53756 |
299 | 3U6H | 03X | 0.000001364 | 0.5372 |
300 | 4DEH | 0JK |