1ETT | 2.5 | BOS TAURUS | ENZYME 3.4.21.5 | 4QQ | Ki = 1.3 uM | 428.548 |
1JWT | 2.5 | HOMO SAPIENS | ENZYME 3.4.21.5 | BLI | Ki = 14 nM | 492.592 |
1TB6 | 2.5 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, NAG NAG FUC, NAG NAG BMA MAN MAN, NAG NAG BMA, MPD, GU4 GU6 GU0 GU5 GU8 GU9 GU8 GU9 GU8 GU9 GU8 GU5 GU1 GU6 GU2 GU3 | | 221.208, 570.545, 118.174 |
1UVT | 2.5 | BOS TAURUS | ENZYME 3.4.21.5 | I48 | Ki = 0.023 uM | 384.472 |
1YCP | 2.5 | BOS TAURUS | ENZYME 3.4.21.5 | TYR GLY VAL ARG GLY PRO | | |
2JH5 | 2.5 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, CA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 895 | Ki = 367 nM | 22.99, 40.078, 1129.21, 447.957 |
2PKS | 2.5 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, G44, ASP PHE GLU GLU ILE PRO GLY GLU TYS LEU | ic50 = 11 uM | 22.99, 344.41, 1286.31 |
3BF6 | 2.5 | HOMO SAPIENS | ENZYME 3.4.21.5 | SVR, PHE PRO ARG | ic50 = 40 uM | 1297.28, 404.515 |
3HAT | 2.5 | HOMO SAPIENS | ENZYME 3.4.21.5 | MBN ABN RNG GLY VAL ARG | | 456.548 |
3TU7 | 2.49 | HOMO SAPIENS | ENZYME 3.4.21.5 | 0BM | Ki = 8.17 nM | 478.608 |
2ANK | 2.46 | HOMO SAPIENS | ENZYME 3.4.21.5 | N12 | ic50 = 47.3 nM | 472.58 |
1O0D | 2.44 | HOMO SAPIENS | ENZYME 3.4.21.5 | 163 | ic50 = 6.2 nM | 456.538 |
2A2X | 2.44 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA9 | ic50 = 20.2 nM | 446.543 |
2FEQ | 2.44 | HOMO SAPIENS | ENZYME 3.4.21.5 | 34P | ic50 = 1.39 nM | 464.582 |
2FES | 2.42 | HOMO SAPIENS | ENZYME 3.4.21.5 | 3SP | ic50 = 0.98 nM | 463.594 |
1KTS | 2.4 | HOMO SAPIENS | ENZYME 3.4.21.5 | C24 | Ki = 4.5 nM | 499.564 |
1NRS | 2.4 | HOMO SAPIENS | ENZYME 3.4.21.5 | LEU ASP PRO ARG | | 484.578 |
1TWX | 2.4 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, ASP PHE GLU GLU ILE PRO GLY GLU TYS LEU | | 221.208, 1286.31 |
2ANM | 2.4 | HOMO SAPIENS | ENZYME 3.4.21.5 | CDO | ic50 = 1.8 nM | 456.538 |
2H9T | 2.4 | HOMO SAPIENS | ENZYME 3.4.21.5 | SVR, PHE PRO ARG | | 1297.28, 404.515 |
4HFP | 2.4 | HOMO SAPIENS | ENZYME 3.4.21.5 | 15U, NA | Kd = 42 nM | 508.634, 22.99 |
1BHX | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | R56, ASP PHE GLU GLU ILE | Ki = 0.145 uM | 468.593, 648.646 |
1D9I | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 00P | Ki = 0.78 nM | 22.99, 1129.21, 475.561 |
1ETS | 2.3 | BOS TAURUS | ENZYME 3.4.21.5 | MID | Ki = 6 nM | 521.631 |
1FPC | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | 0ZI | Ki = 0.1 uM | 503.681 |
1HAH | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 221.208, 1129.21 |
1NL2 | 2.3 | BOS TAURUS | ENZYME 3.4.21.5 | NAG NAG, NAG, LPS, CL, CA | | 408.404, 221.208, 485.549, 35.453, 40.078 |
1NY2 | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, ARG PRO PRO GLY PHE | | 1129.21, 558.684 |
1TA2 | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | 176 | Ki = 3 nM | 496.428 |
1XM1 | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | GAH, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 767.961, 1129.21 |
3BIU | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, NA, 10U | | 221.208, 22.99, 371.477 |
6GWE | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | ODB, NAG, NA, EDO | Ki = 42 nM | 666.834, 221.208, 22.99, 62.068 |
2C90 | 2.25 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, DMS, C1M | ic50 = 330 uM | 22.99, 78.133, 180.594 |
2ZFP | 2.25 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, 19U | Ki = 6.8 uM | 22.99, 323.818 |
2JH6 | 2.21 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, CA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 894 | Ki = 17 nM | 22.99, 40.078, 1129.21, 449.973 |
1AWF | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | GR4, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 0.97 uM | 736.843, 1129.21 |
1ETR | 2.2 | BOS TAURUS | ENZYME 3.4.21.5 | MIT | | 509.642 |
1QHR | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 157 | | 1129.21, 226.315 |
1QJ6 | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 167 | ic50 = 18 nM | 1129.21, 396.479 |
1QJ7 | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | GR1, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | ic50 = 18 nM | 465.585, 1129.21 |
1TMT | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, DPN PRO ARG | | 221.208, 419.506 |
1WBG | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, L03, DMS | ic50 = 1 mM | 1129.21, 225.698, 78.133 |
1ZGI | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | 382, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 4.6 uM | 439.461, 1129.21 |
1ZGV | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 501 | ic50 ~ 1 uM | 1129.21, 344.842 |
2C8Y | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, DMS, C3M | | 22.99, 78.133, 370.465 |
2C93 | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, DMS, C4M | ic50 = 12 uM | 22.99, 78.133, 392.512 |
2HGT | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | DPN PRO ARG | | 419.506 |
2ZF0 | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, 51U | | 22.99, 365.469 |
3BEF | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, ASN ASP LYS TYR GLU PRO PHE TRP GLU | | 221.208, 1210.29 |
3EGK | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, M18 | Ki = 22 uM | 22.99, 410.892 |