1GHY | 1.85 | HOMO SAPIENS | ENZYME 3.4.21.5 | ZN, NA, CA, 121 | Ki = 0.008 uM | 65.409, 22.99, 40.078, 254.267 |
1C1U | 1.75 | HOMO SAPIENS | ENZYME 3.4.21.5 | ZN, NA, BAI | | 65.409, 22.99, 290.323 |
1C1W | 1.9 | HOMO SAPIENS | ENZYME 3.4.21.5 | ZN, NA, BAH | | 65.409, 22.99, 366.377 |
1C1V | 1.98 | HOMO SAPIENS | ENZYME 3.4.21.5 | ZN, NA, BAB | Ki = 0.023 uM | 65.409, 22.99, 335.386 |
1EB1 | 1.8 | SYNTHETIC CONSTRUCT | ENZYME 3.4.21.5 | ZAL PRO MMO, ASP TYR GLU PRO ILE PRO GLU GLU ALA PHE | Ki = 37 pM | 424.59, 1205.24 |
5AHG | 1.24 | HOMO SAPIENS | ENZYME 3.4.21.5 | Y4L, PO4, NAG, GOL, NA, DMS | | 234.703, 94.971, 221.208, 92.094, 22.99, 78.133 |
5AFY | 1.12 | HOMO SAPIENS | ENZYME 3.4.21.5 | WCE, PO4, NA, TYS, GOL, NAG, DMS | | 155.582, 94.971, 22.99, 261.252, 92.094, 221.208, 78.133 |
2BDY | 1.61 | HOMO SAPIENS | ENZYME 3.4.21.5 | UNB, NA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | ic50 = 0.017 uM | 502.585, 22.99, 1129.21 |
1YPG | 1.8 | HOMO SAPIENS | ENZYME 3.4.21.5 | UIR, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 10 nM | 458.552, 1129.21 |
1YPE | 1.81 | HOMO SAPIENS | ENZYME 3.4.21.5 | UIP, NA, GOL, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 8 nM | 446.541, 22.99, 92.094, 1129.21 |
1YPJ | 1.78 | HOMO SAPIENS | ENZYME 3.4.21.5 | UIB, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 95 nM | 448.557, 1129.21 |
5AFZ | 1.53 | HOMO SAPIENS | ENZYME 3.4.21.5 | TYS, PO4, NA, UET, NAG | Kd = 0.16 uM | 261.252, 94.971, 22.99, 507.605, 221.208 |
1YCP | 2.5 | BOS TAURUS | ENZYME 3.4.21.5 | TYR GLY VAL ARG GLY PRO | | |
1G30 | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | T87 | Ki = 140 nM | 525.602 |
1NT1 | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | T76 | Ki = 1.3 nM | 505.006 |
1AIX | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | T19 | | 567.44 |
3C1K | 1.84 | HOMO SAPIENS | ENZYME 3.4.21.5 | T15 | Ki = 0.36 nM | 542.65 |
2H9T | 2.4 | HOMO SAPIENS | ENZYME 3.4.21.5 | SVR, PHE PRO ARG | | 1297.28, 404.515 |
3BF6 | 2.5 | HOMO SAPIENS | ENZYME 3.4.21.5 | SVR, PHE PRO ARG | ic50 = 40 uM | 1297.28, 404.515 |
2GDE | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | SN3, NA, ASP PHE GLU GLU ILE PRO GLY GLU TYS LEU | ic50 = 5.7 nM | 667.172, 22.99, 1286.31 |
1VZQ | 1.54 | HOMO SAPIENS | ENZYME 3.4.21.5 | SHY, NA, CA | Ki = 36 nM | 448.471, 22.99, 40.078 |
4UFD | 1.43 | HOMO SAPIENS | ENZYME 3.4.21.5 | S49, NAG, NA, PO4, GOL | | 547.668, 221.208, 22.99, 94.971, 92.094 |
1HXE | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | RB, ASP PHE GLU GLU ILE PRO GLY GLU TYR LEU | | 85.468, 1192.27 |
1YPL | 1.85 | HOMO SAPIENS | ENZYME 3.4.21.5 | RA8, NA, GOL, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 10.6 uM | 494.651, 22.99, 92.094, 1129.21 |
1YPM | 1.85 | HOMO SAPIENS | ENZYME 3.4.21.5 | RA4, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 1.9 uM | 489.568, 1129.21 |
1BHX | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | R56, ASP PHE GLU GLU ILE | Ki = 0.145 uM | 468.593, 648.646 |
1G32 | 1.9 | HOMO SAPIENS | ENZYME 3.4.21.5 | R11 | Ki = 780 nM | 423.513 |
1A4W | 1.8 | HOMO SAPIENS | ENZYME 3.4.21.5 | QWE, NA | Ki = 1.2 uM | 614.802, 22.99 |
6ZV8 | 1.7 | HOMO SAPIENS | ENZYME 3.4.21.5 | QQT, GLY ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, NAG | ic50 = 0.7 nM | 491.94, 221.208 |
6ZUW | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | QQK, GLY ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, NAG | ic50 = 0.4 nM | 502.002, 221.208 |
6ZUN | 1.79 | HOMO SAPIENS | ENZYME 3.4.21.5 | QQ5, GLY ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, NAG | ic50 = 10 nM | 429.897, 221.208 |
1BCU | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | PRL | Kd = 0.53 mM | 209.247 |
1QBV | 1.8 | HOMO SAPIENS | ENZYME 3.4.21.5 | PPX | Ki = 4100 nM | 381.471 |
3SHA | 1.52 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, P97, NAG, NA, GOL | Ki = 2.6 uM | 94.971, 386.875, 221.208, 22.99, 92.094 |
3SI4 | 1.27 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, NAG, NA, GOL, B04 | Ki = 132.2 uM | 94.971, 221.208, 22.99, 92.094, 367.465 |
3SI3 | 1.55 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, NAG, NA, GOL, B03 | Ki = 69.3 uM | 94.971, 221.208, 22.99, 92.094, 352.43 |
3QTO | 1.52 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, NAG, NA, GOL, 10P | Ki = 74.8 uM | 94.971, 221.208, 22.99, 92.094, 367.465 |
3QTV | 1.63 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, NAG, NA, GOL, 06P | Ki = 22.5 uM | 94.971, 221.208, 22.99, 92.094, 367.465 |
4UFG | 1.65 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, NAG, NA, D6J | | 94.971, 221.208, 22.99, 549.684 |
4UEH | 1.16 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, NAG, NA, BEN, GOL | Kd = 355 uM | 94.971, 221.208, 22.99, 120.152, 92.094 |
3P17 | 1.43 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, NAG, NA, 99P | Ki = 33.4 uM | 94.971, 221.208, 22.99, 352.43 |
4UFE | 1.59 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, NAG, NA, 3ZD | | 94.971, 221.208, 22.99, 521.631 |
4UDW | 1.16 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, NAG, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU GLN, N6L, NA, GOL | Kd = 0.27 uM | 94.971, 221.208, 420.332, 22.99, 92.094 |
4UFF | 1.55 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, NA, 6V2, NAG | | 94.971, 22.99, 521.631, 221.208 |
2ZDV | 1.72 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, NA, 37U | | 94.971, 22.99, 369.433 |
2ZDA | 1.73 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, NA, 32U | | 94.971, 22.99, 394.49 |
5AF9 | 1.18 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, EDO, NA, NAG, SJR, GOL, DMS | Kd = 1003 uM | 94.971, 62.068, 22.99, 221.208, 228.247, 92.094, 78.133 |
1H8D | 1.4 | HOMO SAPIENS | ENZYME 3.4.21.5 | PHW, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 805.851, 1129.21 |
1H8I | 1.75 | HOMO SAPIENS | ENZYME 3.4.21.5 | PHV, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 637.66, 1129.21 |
1G37 | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | PHE GLU ALA ILE PRO ALA GLU TYR LEU, 110 | | 1050.18, 574.689 |