1A2C | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, 34H LEU PRJ OAR | ic50 = 0.5 uM | 22.99, 605.757 |
1A4W | 1.8 | HOMO SAPIENS | ENZYME 3.4.21.5 | QWE, NA | Ki = 1.2 uM | 614.802, 22.99 |
1AD8 | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, NA, MDL | Ki = 247 nM | 1129.21, 22.99, 564.547 |
1AE8 | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, AZL, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 221.208, 419.518, 1129.21 |
1AFE | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, ALZ | | 221.208, 1129.21, 334.413 |
1AIX | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | T19 | | 567.44 |
1AWF | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | GR4, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 0.97 uM | 736.843, 1129.21 |
1BCU | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | PRL | Kd = 0.53 mM | 209.247 |
1BHX | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | R56, ASP PHE GLU GLU ILE | Ki = 0.145 uM | 468.593, 648.646 |
1C1U | 1.75 | HOMO SAPIENS | ENZYME 3.4.21.5 | ZN, NA, BAI | | 65.409, 22.99, 290.323 |
1C1V | 1.98 | HOMO SAPIENS | ENZYME 3.4.21.5 | ZN, NA, BAB | Ki = 0.023 uM | 65.409, 22.99, 335.386 |
1C1W | 1.9 | HOMO SAPIENS | ENZYME 3.4.21.5 | ZN, NA, BAH | | 65.409, 22.99, 366.377 |
1C4U | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, IH1 | Ki = 0.043 nM | 22.99, 581.483 |
1C4V | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, IH2 | Ki = 0.016 nM | 22.99, 528.645 |
1C5L | 1.47 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, CA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 22.99, 40.078, 1129.21 |
1C5N | 1.5 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, ESI, CA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 20 uM | 22.99, 303.143, 40.078, 1129.21 |
1C5O | 1.9 | HOMO SAPIENS | ENZYME 3.4.21.5 | BAM, NA | Ki = 320 uM | 121.16, 22.99 |
1D3D | 2.04 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, NA, BZT | Ka = 1240000000 M^-1 | 221.208, 22.99, 591.601 |
1D3P | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, NA, BT3 | Ka = 24300000 M^-1 | 221.208, 22.99, 543.719 |
1D4P | 2.07 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, NA, BPP | Ka = 2000000 M^-1 | 221.208, 22.99, 360.452 |
1D6W | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 00R | Ki = 1100 nM | 22.99, 1129.21, 527.596 |
1D9I | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 00P | Ki = 0.78 nM | 22.99, 1129.21, 475.561 |
1EB1 | 1.8 | SYNTHETIC CONSTRUCT | ENZYME 3.4.21.5 | ZAL PRO MMO, ASP TYR GLU PRO ILE PRO GLU GLU ALA PHE | Ki = 37 pM | 424.59, 1205.24 |
1ETR | 2.2 | BOS TAURUS | ENZYME 3.4.21.5 | MIT | | 509.642 |
1ETS | 2.3 | BOS TAURUS | ENZYME 3.4.21.5 | MID | Ki = 6 nM | 521.631 |
1ETT | 2.5 | BOS TAURUS | ENZYME 3.4.21.5 | 4QQ | Ki = 1.3 uM | 428.548 |
1FPC | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | 0ZI | Ki = 0.1 uM | 503.681 |
1G30 | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | T87 | Ki = 140 nM | 525.602 |
1G32 | 1.9 | HOMO SAPIENS | ENZYME 3.4.21.5 | R11 | Ki = 780 nM | 423.513 |
1G37 | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | PHE GLU ALA ILE PRO ALA GLU TYR LEU, 110 | | 1050.18, 574.689 |
1GHV | 1.85 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, 120 | Ki = 45 uM | 22.99, 254.267 |
1GHW | 1.75 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, BMZ | Ki = 4 uM | 22.99, 253.279 |
1GHY | 1.85 | HOMO SAPIENS | ENZYME 3.4.21.5 | ZN, NA, CA, 121 | Ki = 0.008 uM | 65.409, 22.99, 40.078, 254.267 |
1H8D | 1.4 | HOMO SAPIENS | ENZYME 3.4.21.5 | PHW, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 805.851, 1129.21 |
1H8I | 1.75 | HOMO SAPIENS | ENZYME 3.4.21.5 | PHV, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 637.66, 1129.21 |
1HAG | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 221.208, 1129.21 |
1HAH | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 221.208, 1129.21 |
1HXE | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | RB, ASP PHE GLU GLU ILE PRO GLY GLU TYR LEU | | 85.468, 1192.27 |
1HXF | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | ASP PHE GLU GLU ILE PRO GLY GLU TYR LEU | | 1192.27 |
1JWT | 2.5 | HOMO SAPIENS | ENZYME 3.4.21.5 | BLI | Ki = 14 nM | 492.592 |
1K21 | 1.86 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG NAG, NA, IGN | Ki = 4.2 nM | 408.404, 22.99, 438.564 |
1K22 | 1.93 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG NAG, NA, MEL | Ki = 4 nM | 408.404, 22.99, 429.513 |
1KTS | 2.4 | HOMO SAPIENS | ENZYME 3.4.21.5 | C24 | Ki = 4.5 nM | 499.564 |
1KTT | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | C02 | ic50 = 1.5 uM | 419.499 |
1MU6 | 1.99 | HOMO SAPIENS | ENZYME 3.4.21.5 | CDA | Ki = 4.2 nM | 432.399 |
1MU8 | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | CDB | Ki = 1 nM | 448.442 |
1MUE | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | CDD | Ki = 2.3 nM | 467.829 |
1NL2 | 2.3 | BOS TAURUS | ENZYME 3.4.21.5 | NAG NAG, NAG, LPS, CL, CA | | 408.404, 221.208, 485.549, 35.453, 40.078 |
1NM6 | 1.8 | HOMO SAPIENS | ENZYME 3.4.21.5 | L86 | Ki = 0.09 nM | 509.043 |
1NRS | 2.4 | HOMO SAPIENS | ENZYME 3.4.21.5 | LEU ASP PRO ARG | | 484.578 |
1NT1 | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | T76 | Ki = 1.3 nM | 505.006 |
1NY2 | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, ARG PRO PRO GLY PHE | | 1129.21, 558.684 |
1NZQ | 2.18 | HOMO SAPIENS | ENZYME 3.4.21.5 | 162 | ic50 = 11 nM | 456.538 |
1O0D | 2.44 | HOMO SAPIENS | ENZYME 3.4.21.5 | 163 | ic50 = 6.2 nM | 456.538 |
1O2G | 1.58 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, 696 | Ki = 0.76 uM | 22.99, 327.379 |
1O5G | 1.75 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, CR9, CA | Ki = 11 uM | 22.99, 382.431, 40.078 |
1OYT | 1.67 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, FSN, CA | Ki = 0.057 uM | 22.99, 407.461, 40.078 |
1QBV | 1.8 | HOMO SAPIENS | ENZYME 3.4.21.5 | PPX | Ki = 4100 nM | 381.471 |
1QHR | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 157 | | 1129.21, 226.315 |
1QJ1 | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 166 | ic50 = 9 nM | 1129.21, 382.453 |
1QJ6 | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 167 | ic50 = 18 nM | 1129.21, 396.479 |
1QJ7 | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | GR1, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | ic50 = 18 nM | 465.585, 1129.21 |
1RIW | 2.04 | HOMO SAPIENS | ENZYME 3.4.21.5 | OSC, NAG, NA | ic50 = 28 nM | 616.75, 221.208, 22.99 |
1SB1 | 1.9 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, ASP PHE GLU GLU ILE PRO GLU GLU TYS, 165 | Ki = 128 nM | 22.99, 1229.22, 569.739 |
1SL3 | 1.81 | HOMO SAPIENS | ENZYME 3.4.21.5 | 170 | Ki = 1.4 pM | 552.321 |
1T4U | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | 81A | | 483.558 |
1T4V | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | 14A | Ki = 0.021 uM | 394.896 |
1TA2 | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | 176 | Ki = 3 nM | 496.428 |
1TA6 | 1.9 | HOMO SAPIENS | ENZYME 3.4.21.5 | 177 | Ki = 0.74 nM | 479.012 |
1TB6 | 2.5 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, NAG NAG FUC, NAG NAG BMA MAN MAN, NAG NAG BMA, MPD, GU4 GU6 GU0 GU5 GU8 GU9 GU8 GU9 GU8 GU9 GU8 GU5 GU1 GU6 GU2 GU3 | | 221.208, 570.545, 118.174 |
1TMT | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, DPN PRO ARG | | 221.208, 419.506 |
1TOM | 1.8 | HOMO SAPIENS | ENZYME 3.4.21.5 | MIN | Ki = 5 nM | 386.531 |
1TWX | 2.4 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, ASP PHE GLU GLU ILE PRO GLY GLU TYS LEU | | 221.208, 1286.31 |
1UMA | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, IN2, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 221.208, 218.254, 1129.21 |
1UVT | 2.5 | BOS TAURUS | ENZYME 3.4.21.5 | I48 | Ki = 0.023 uM | 384.472 |
1VR1 | 1.9 | HOMO SAPIENS | ENZYME 3.4.21.5 | ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 1129.21 |
1VZQ | 1.54 | HOMO SAPIENS | ENZYME 3.4.21.5 | SHY, NA, CA | Ki = 36 nM | 448.471, 22.99, 40.078 |
1W7G | 1.65 | HOMO SAPIENS | ENZYME 3.4.21.5 | MIU | Ki ~ 13 uM | 507.573 |
1WAY | 2.02 | HOMO SAPIENS | ENZYME 3.4.21.5 | L02, DMS, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | ic50 = 400 uM | 261.75, 78.133, 1129.21 |
1WBG | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | L03, DMS, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | ic50 = 1 mM | 225.698, 78.133, 1129.21 |
1XM1 | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | GAH, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 767.961, 1129.21 |
1XMN | 1.85 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG NAG, NAG NDG, NAG NAG BMA MAN MAN, IDS SGN IDS SGN IDS SGN, SGN IDS SGN IDS SGN, NA, GOL, 0G6 | | 408.404, 1722.33, 1468.16, 22.99, 92.094, 453.986 |
1YCP | 2.5 | BOS TAURUS | ENZYME 3.4.21.5 | TYR GLY VAL ARG GLY PRO | | |
1YPE | 1.81 | HOMO SAPIENS | ENZYME 3.4.21.5 | UIP, NA, GOL, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 8 nM | 446.541, 22.99, 92.094, 1129.21 |
1YPG | 1.8 | HOMO SAPIENS | ENZYME 3.4.21.5 | UIR, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 10 nM | 458.552, 1129.21 |
1YPJ | 1.78 | HOMO SAPIENS | ENZYME 3.4.21.5 | UIB, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 95 nM | 448.557, 1129.21 |
1YPK | 1.78 | HOMO SAPIENS | ENZYME 3.4.21.5 | CCR, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 601.714, 1129.21 |
1YPL | 1.85 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, GOL, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, RA8 | Ki = 10.6 uM | 22.99, 92.094, 1129.21, 494.651 |
1YPM | 1.85 | HOMO SAPIENS | ENZYME 3.4.21.5 | RA4, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 1.9 uM | 489.568, 1129.21 |
1Z71 | 1.8 | HOMO SAPIENS | ENZYME 3.4.21.5 | L17 | Ki = 0.66 nM | 497.322 |
1ZGI | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | 382, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 4.6 uM | 439.461, 1129.21 |
1ZGV | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 501 | ic50 ~ 1 uM | 1129.21, 344.842 |
1ZRB | 1.9 | HOMO SAPIENS | ENZYME 3.4.21.5 | 062 | Ki = 0.77 nM | 492.954 |
2A2X | 2.44 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA9 | ic50 = 20.2 nM | 446.543 |
2ANK | 2.46 | HOMO SAPIENS | ENZYME 3.4.21.5 | N12 | ic50 = 47.3 nM | 472.58 |
2ANM | 2.4 | HOMO SAPIENS | ENZYME 3.4.21.5 | CDO | ic50 = 1.8 nM | 456.538 |
2BDY | 1.61 | HOMO SAPIENS | ENZYME 3.4.21.5 | UNB, NA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | ic50 = 0.017 uM | 502.585, 22.99, 1129.21 |
2C8W | 1.96 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, C7M | ic50 = 3.7 nM | 22.99, 546.061 |
2C8X | 2.17 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, DMS, C5M | ic50 = 220 nM | 22.99, 78.133, 517.08 |
2C8Y | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, DMS, C3M | | 22.99, 78.133, 370.465 |
2C8Z | 2.14 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, DMS, C2A | ic50 > 1 mM | 22.99, 78.133, 141.598 |
2C90 | 2.25 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, DMS, C1M | ic50 = 330 uM | 22.99, 78.133, 180.594 |
2C93 | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, DMS, C4M | ic50 = 12 uM | 22.99, 78.133, 392.512 |
2CF8 | 1.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | ESH, CA, NA | Ki = 0.008 uM | 451.004, 40.078, 22.99 |
2CF9 | 1.79 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, CA, 348 | Ki = 0.015 uM | 22.99, 40.078, 446.584 |
2CN0 | 1.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, F25, CA | Ki = 22 nM | 22.99, 444.493, 40.078 |
2FEQ | 2.44 | HOMO SAPIENS | ENZYME 3.4.21.5 | 34P | ic50 = 1.39 nM | 464.582 |
2FES | 2.42 | HOMO SAPIENS | ENZYME 3.4.21.5 | 3SP | ic50 = 0.98 nM | 463.594 |
2GDE | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | SN3, NA, ASP PHE GLU GLU ILE PRO GLY GLU TYS LEU | ic50 = 5.7 nM | 667.172, 22.99, 1286.31 |
2H9T | 2.4 | HOMO SAPIENS | ENZYME 3.4.21.5 | SVR, PHE PRO ARG | | 1297.28, 404.515 |
2HGT | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | DPN PRO ARG | | 419.506 |
2JH0 | 1.7 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, CA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 701 | Ki = 2 nM | 22.99, 40.078, 1129.21, 461.983 |
2JH5 | 2.5 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, CA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 895 | Ki = 367 nM | 22.99, 40.078, 1129.21, 447.957 |
2JH6 | 2.21 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, CA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 894 | Ki = 17 nM | 22.99, 40.078, 1129.21, 449.973 |
2PKS | 2.5 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, G44, ASP PHE GLU GLU ILE PRO GLY GLU TYS LEU | ic50 = 11 uM | 22.99, 344.41, 1286.31 |
2R2M | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | I50 | Ki = 47.1 nM | 443.851 |
2UUF | 1.26 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, CA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 22.99, 40.078, 1129.21 |
2UUJ | 1.32 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, CA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 896 | | 22.99, 40.078, 1129.21, 355.474 |
2UUK | 1.39 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, CA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 897 | | 22.99, 40.078, 1129.21, 454.605 |
2V3H | 1.79 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, I25, CA | | 22.99, 426.552, 40.078 |
2V3O | 1.79 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, I26, CA | | 22.99, 444.542, 40.078 |
2ZC9 | 1.58 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, 22U | Ki = 180 nM | 22.99, 385.887 |
2ZDA | 1.73 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, NA, 32U | | 94.971, 22.99, 394.49 |
2ZDV | 1.72 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, NA, 37U | | 94.971, 22.99, 369.433 |
2ZF0 | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, 51U | | 22.99, 365.469 |
2ZFP | 2.25 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, 19U | Ki = 6.8 uM | 22.99, 323.818 |
2ZGB | 1.6 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, 21U | Ki = 0.54 uM | 22.99, 351.871 |
2ZGX | 1.8 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, 29U | Ki = 180 nM | 22.99, 331.413 |
2ZHQ | 1.96 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, 27U | Ki = 0.75 uM | 22.99, 378.467 |
2ZI2 | 1.65 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, BEN, 24U | Ki = 5.7 uM | 22.99, 120.152, 316.398 |
2ZNK | 1.8 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, 31U | Ki = 0.02 uM | 22.99, 359.466 |
2ZO3 | 1.7 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, 33U | Ki = 0.1 nM | 22.99, 469.578 |
3BEF | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | ASN ASP LYS TYR GLU PRO PHE TRP GLU, NAG | | 1210.29, 221.208 |
3BF6 | 2.5 | HOMO SAPIENS | ENZYME 3.4.21.5 | SVR, PHE PRO ARG | ic50 = 40 uM | 1297.28, 404.515 |
3BIU | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, NA, 10U | | 221.208, 22.99, 371.477 |
3BIV | 1.8 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, 11U | | 221.208, 385.503 |
3BV9 | 1.8 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, IOD, GOL, DAR OIC PRO DAL 4PH NH2 | Ki = 4.4 uM | 22.99, 126.904, 92.094, 661.893 |
3C1K | 1.84 | HOMO SAPIENS | ENZYME 3.4.21.5 | T15 | Ki = 0.36 nM | 542.65 |
3DA9 | 1.8 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, ASP PHE GLU GLU ILE PRO GLY GLU PTR, 44U | Kd = 3.1 uM | 22.99, 1157.07, 379.495 |
3DHK | 1.73 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, 23U | Ki = 47 nM | 22.99, 461.983 |
3DUX | 1.6 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, 64U | Ki = 100 nM | 22.99, 391.935 |
3EGK | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, M18 | Ki = 22 uM | 22.99, 410.892 |
3F68 | 1.75 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, 91U | Ki = 8.7 uM | 22.99, 433.971 |
3HAT | 2.5 | HOMO SAPIENS | ENZYME 3.4.21.5 | MBN ABN RNG GLY VAL ARG | | 456.548 |
3P17 | 1.43 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, NAG, NA, 99P | Ki = 33.4 uM | 94.971, 221.208, 22.99, 352.43 |
3PMA | 2.2 | BOS TAURUS | ENZYME 3.4.21.5 | GU4 YYJ, NA, CIT | | 974.737, 22.99, 192.124 |
3PO1 | 1.65 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, MKY, ASP PHE GLU GLU ILE PRO GLY GLU TYS LEU, ACT | Kd = 95 uM | 22.99, 294.33, 1286.31, 59.044 |
3QTO | 1.52 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, NAG, NA, GOL, 10P | Ki = 74.8 uM | 94.971, 221.208, 22.99, 92.094, 367.465 |
3QTV | 1.63 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, NAG, NA, GOL, 06P | Ki = 22.5 uM | 94.971, 221.208, 22.99, 92.094, 367.465 |
3QWC | 1.75 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, NA, GOL, 98P | Ki = 55.4 uM | 221.208, 22.99, 92.094, 401.91 |
3QX5 | 1.35 | HOMO SAPIENS | ENZYME 3.4.21.5 | GOL, 02P, PO4, NAG, NA | Ki = 63.5 uM | 92.094, 401.91, 94.971, 221.208, 22.99 |
3SHA | 1.52 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, P97, NAG, NA, GOL | Ki = 2.6 uM | 94.971, 386.875, 221.208, 22.99, 92.094 |
3SHC | 1.9 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, NA, B01 | Ki = 1.9 uM | 221.208, 22.99, 386.875 |
3SI3 | 1.55 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, NAG, NA, GOL, B03 | Ki = 69.3 uM | 94.971, 221.208, 22.99, 92.094, 352.43 |
3SI4 | 1.27 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, NAG, NA, GOL, B04 | Ki = 132.2 uM | 94.971, 221.208, 22.99, 92.094, 367.465 |
3SV2 | 1.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | P05, PO4, NAG, NA, GOL | Ki = 64 uM | 352.43, 94.971, 221.208, 22.99, 92.094 |
3TU7 | 2.49 | HOMO SAPIENS | ENZYME 3.4.21.5 | 0BM | Ki = 8.17 nM | 478.608 |
3U8O | 1.28 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, NA, MRD, IOD, DPN PRO DAR DTH NH2, CL | Ki = 0.92 uM | 221.208, 22.99, 118.174, 126.904, 521.643, 35.453 |
3U8R | 1.47 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, NA, MRD, MPD, IOD, DPN PRO DAR ILE NH2, CL | Ki = 7.7 uM | 221.208, 22.99, 118.174, 118.174, 126.904, 533.698, 35.453 |
3U8T | 1.86 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, NA, MPD, IOD, DPN PRO DAR CYS NH2, CL | Ki = 16.5 uM | 221.208, 22.99, 118.174, 126.904, 523.683, 35.453 |
3UTU | 1.55 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, 1TS | Ki = 0.012 nM | 22.99, 680.174 |
3VXE | 1.25 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, DPN PRO ARG | | 221.208, 419.506 |
4AX9 | 1.9 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, NA, N5N | Ki = 0.00027 uM | 221.208, 22.99, 558.65 |
4BAH | 1.94 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, MEL, NA | Ki = 2.01 nM | 221.208, 429.513, 22.99 |
4BAK | 1.94 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, M67, NA | Ki = 1.22 nM | 221.208, 470.608, 22.99 |
4BAM | 1.88 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, NA, MM9 | Ki = 1.14 nM | 221.208, 22.99, 456.581 |
4BAN | 1.87 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, NA, M6S | Ki = 2.43 nM | 221.208, 22.99, 442.554 |
4BAO | 1.87 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG NAG, NA, MVF, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 4.29 nM | 408.404, 22.99, 428.528, 1129.21 |
4BAQ | 1.89 | HOMO SAPIENS | ENZYME 3.4.21.5 | M4Z, NAG, NA | Ki = 0.98 nM | 456.581, 221.208, 22.99 |
4HFP | 2.4 | HOMO SAPIENS | ENZYME 3.4.21.5 | 15U, NA | Kd = 42 nM | 508.634, 22.99 |
4LOY | 1.77 | HOMO SAPIENS | ENZYME 3.4.21.5 | 6XS, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, NAG, NA | | 620.544, 1129.21, 221.208, 22.99 |
4LXB | 1.61 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, 7R9, NAG | ic50 = 7 nM | 22.99, 648.142, 221.208 |
4UD9 | 1.12 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, NAG, FQI, PO4, TYS, DMS, GOL, EDO | Kd = 475 uM | 22.99, 221.208, 161.609, 94.971, 261.252, 78.133, 92.094, 62.068 |
4UDW | 1.16 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, NAG, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU GLN, N6L, NA, GOL | Kd = 0.27 uM | 94.971, 221.208, 420.332, 22.99, 92.094 |
4UE7 | 1.13 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, MRZ, EDO, DMS, GOL, NA, PO4, IOD | Kd = 107 uM | 221.208, 127.188, 62.068, 78.133, 92.094, 22.99, 94.971, 126.904 |
4UEH | 1.16 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, NAG, NA, BEN, GOL | Kd = 355 uM | 94.971, 221.208, 22.99, 120.152, 92.094 |
4UFD | 1.43 | HOMO SAPIENS | ENZYME 3.4.21.5 | S49, NAG, NA, PO4, GOL | | 547.668, 221.208, 22.99, 94.971, 92.094 |
4UFE | 1.59 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, NAG, NA, 3ZD | | 94.971, 221.208, 22.99, 521.631 |
4UFF | 1.55 | HOMO SAPIENS | ENZYME 3.4.21.5 | 6V2, NAG, PO4, NA | | 521.631, 221.208, 94.971, 22.99 |
4UFG | 1.65 | HOMO SAPIENS | ENZYME 3.4.21.5 | PO4, NAG, NA, D6J | | 94.971, 221.208, 22.99, 549.684 |
4YES | 1.5 | HOMO SAPIENS | ENZYME 3.4.21.5 | MG, GOL, 45S, NAG | Ki = 9.6 nM | 24.305, 92.094, 374.865, 221.208 |
5AF9 | 1.18 | HOMO SAPIENS | ENZYME 3.4.21.5 | EDO, NA, NAG, SJR, GOL, DMS, PO4 | Kd = 1003 uM | 62.068, 22.99, 221.208, 228.247, 92.094, 78.133, 94.971 |
5AFY | 1.12 | HOMO SAPIENS | ENZYME 3.4.21.5 | WCE, PO4, NA, TYS, GOL, NAG, DMS | | 155.582, 94.971, 22.99, 261.252, 92.094, 221.208, 78.133 |
5AFZ | 1.53 | HOMO SAPIENS | ENZYME 3.4.21.5 | TYS, PO4, NA, UET, NAG | Kd = 0.16 uM | 261.252, 94.971, 22.99, 507.605, 221.208 |
5AHG | 1.24 | HOMO SAPIENS | ENZYME 3.4.21.5 | Y4L, PO4, NAG, GOL, NA, DMS | | 234.703, 94.971, 221.208, 92.094, 22.99, 78.133 |
6EO8 | 1.94 | HOMO SAPIENS | ENZYME 3.4.21.5 | 2FN, DMS | Ki = 100 nM | 696.208, 78.133 |
6EO9 | 1.84 | HOMO SAPIENS | ENZYME 3.4.21.5 | 2OJ, DMS | Ki = 160 nM | 864.355, 78.133 |
6GBW | 1.45 | HOMO SAPIENS | ENZYME 3.4.21.5 | EU5, NA, NAG, DMS | Ki = 3.51 nM | 578.127, 22.99, 221.208, 78.133 |
6GWE | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | ODB, NAG, NA, EDO | Ki = 42 nM | 666.834, 221.208, 22.99, 62.068 |
6ROT | 1.34 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, PO4, KDQ, NA, DMS | Ki = 483.63 nM | 221.208, 94.971, 479.977, 22.99, 78.133 |
6T3Q | 1.33 | HOMO SAPIENS | ENZYME 3.4.21.5 | GOL, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU GLN, PO4, M6Q, NAG, NA | Ki = 379 nM | 92.094, 94.971, 367.445, 221.208, 22.99 |
6T4A | 1.31 | HOMO SAPIENS | ENZYME 3.4.21.5 | GOL, NAG, PO4, J5K, NA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU GLN | Ki = 140 nM | 92.094, 221.208, 94.971, 367.445, 22.99 |
6TDT | 1.53 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, NA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU GLN, PO4, DMS, LXW | Ki = 1213 nM | 221.208, 22.99, 94.971, 78.133, 428.526 |
6ZUG | 1.8 | HOMO SAPIENS | ENZYME 3.4.21.5 | GLY ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, QPW, NAG | ic50 = 12 nM | 457.95, 221.208 |
6ZUH | 1.7 | HOMO SAPIENS | ENZYME 3.4.21.5 | DMS, GLY ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, N6H, NAG | ic50 = 27 nM | 78.133, 429.897, 221.208 |
6ZUN | 1.79 | HOMO SAPIENS | ENZYME 3.4.21.5 | QQ5, GLY ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, NAG | ic50 = 10 nM | 429.897, 221.208 |
6ZUU | 1.94 | HOMO SAPIENS | ENZYME 3.4.21.5 | GLY ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, QQN, NAG | ic50 = 3900 nM | 429.897, 221.208 |
6ZUW | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | QQK, GLY ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, NAG | ic50 = 0.4 nM | 502.002, 221.208 |
6ZUX | 1.94 | HOMO SAPIENS | ENZYME 3.4.21.5 | GLY ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, QQE, NAG | ic50 = 4 nM | 473.949, 221.208 |
6ZV7 | 1.94 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, GLY ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, QQW | ic50 = 6 nM | 221.208, 473.949 |
6ZV8 | 1.7 | HOMO SAPIENS | ENZYME 3.4.21.5 | QQT, GLY ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, NAG | ic50 = 0.7 nM | 491.94, 221.208 |
7KME | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, ACE 0BN CHG PRR LEU PRO NH2 | Ki = 40 uM | 22.99, 1129.21, 540.709 |
8KME | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | ACE 0BN CHG MLY LEU PRO NH2, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, NA | Ki = 8 uM | 1129.21, 22.99 |