1A2C | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, 34H LEU PRJ OAR | ic50 = 0.5 uM | 22.99, 605.757 |
1A4W | 1.8 | HOMO SAPIENS | ENZYME 3.4.21.5 | QWE, NA | Ki = 1.2 uM | 614.802, 22.99 |
1AD8 | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, MDL, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 247 nM | 22.99, 564.547, 1129.21 |
1AE8 | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, AZL, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 221.208, 419.518, 1129.21 |
1AFE | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, ALZ | | 221.208, 1129.21, 334.413 |
1AIX | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | T19 | | 567.44 |
1AWF | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | GR4, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 0.97 uM | 736.843, 1129.21 |
1BCU | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | PRL | Kd = 0.53 mM | 209.247 |
1BHX | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | R56, ASP PHE GLU GLU ILE | Ki = 0.145 uM | 468.593, 648.646 |
1C1U | 1.75 | HOMO SAPIENS | ENZYME 3.4.21.5 | ZN, NA, BAI | | 65.409, 22.99, 290.323 |
1C1V | 1.98 | HOMO SAPIENS | ENZYME 3.4.21.5 | ZN, NA, BAB | Ki = 0.023 uM | 65.409, 22.99, 335.386 |
1C1W | 1.9 | HOMO SAPIENS | ENZYME 3.4.21.5 | ZN, NA, BAH | | 65.409, 22.99, 366.377 |
1C4U | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, IH1 | Ki = 0.043 nM | 22.99, 581.483 |
1C4V | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, IH2 | Ki = 0.016 nM | 22.99, 528.645 |
1C5L | 1.47 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, CA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 22.99, 40.078, 1129.21 |
1C5N | 1.5 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, ESI, CA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 20 uM | 22.99, 303.143, 40.078, 1129.21 |
1C5O | 1.9 | HOMO SAPIENS | ENZYME 3.4.21.5 | BAM, NA | Ki = 320 uM | 121.16, 22.99 |
1D3D | 2.04 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, NA, BZT | Ka = 1240000000 M^-1 | 221.208, 22.99, 591.601 |
1D3P | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, NA, BT3 | Ka = 24300000 M^-1 | 221.208, 22.99, 543.719 |
1D4P | 2.07 | HOMO SAPIENS | ENZYME 3.4.21.5 | BPP, NAG, NA | Ka = 2000000 M^-1 | 360.452, 221.208, 22.99 |
1D6W | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 00R | Ki = 1100 nM | 22.99, 1129.21, 527.596 |
1D9I | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 00P | Ki = 0.78 nM | 22.99, 1129.21, 475.561 |
1EB1 | 1.8 | SYNTHETIC CONSTRUCT | ENZYME 3.4.21.5 | ZAL PRO MMO, ASP TYR GLU PRO ILE PRO GLU GLU ALA PHE | Ki = 37 pM | 424.59, 1205.24 |
1ETR | 2.2 | BOS TAURUS | ENZYME 3.4.21.5 | MIT | | 509.642 |
1ETS | 2.3 | BOS TAURUS | ENZYME 3.4.21.5 | MID | Ki = 6 nM | 521.631 |
1ETT | 2.5 | BOS TAURUS | ENZYME 3.4.21.5 | 4QQ | Ki = 1.3 uM | 428.548 |
1FPC | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | 0ZI | Ki = 0.1 uM | 503.681 |
1G30 | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | T87 | Ki = 140 nM | 525.602 |
1G32 | 1.9 | HOMO SAPIENS | ENZYME 3.4.21.5 | R11 | Ki = 780 nM | 423.513 |
1G37 | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | PHE GLU ALA ILE PRO ALA GLU TYR LEU, 110 | | 1050.18, 574.689 |
1GHV | 1.85 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, 120 | Ki = 45 uM | 22.99, 254.267 |
1GHW | 1.75 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, BMZ | Ki = 4 uM | 22.99, 253.279 |
1GHY | 1.85 | HOMO SAPIENS | ENZYME 3.4.21.5 | ZN, NA, CA, 121 | Ki = 0.008 uM | 65.409, 22.99, 40.078, 254.267 |
1H8D | 1.4 | HOMO SAPIENS | ENZYME 3.4.21.5 | PHW, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 805.851, 1129.21 |
1H8I | 1.75 | HOMO SAPIENS | ENZYME 3.4.21.5 | PHV, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 637.66, 1129.21 |
1HAG | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 221.208, 1129.21 |
1HAH | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 221.208, 1129.21 |
1HXE | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | RB, ASP PHE GLU GLU ILE PRO GLY GLU TYR LEU | | 85.468, 1192.27 |
1HXF | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | ASP PHE GLU GLU ILE PRO GLY GLU TYR LEU | | 1192.27 |
1JWT | 2.5 | HOMO SAPIENS | ENZYME 3.4.21.5 | BLI | Ki = 14 nM | 492.592 |
1K21 | 1.86 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG NAG, NA, IGN | Ki = 4.2 nM | 408.404, 22.99, 438.564 |
1K22 | 1.93 | HOMO SAPIENS | ENZYME 3.4.21.5 | MEL, NAG NAG, NA | Ki = 4 nM | 429.513, 408.404, 22.99 |
1KTS | 2.4 | HOMO SAPIENS | ENZYME 3.4.21.5 | C24 | Ki = 4.5 nM | 499.564 |
1KTT | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | C02 | ic50 = 1.5 uM | 419.499 |
1MU6 | 1.99 | HOMO SAPIENS | ENZYME 3.4.21.5 | CDA | Ki = 4.2 nM | 432.399 |
1MU8 | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | CDB | Ki = 1 nM | 448.442 |
1MUE | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | CDD | Ki = 2.3 nM | 467.829 |
1NL2 | 2.3 | BOS TAURUS | ENZYME 3.4.21.5 | NAG NAG, NAG, LPS, CL, CA | | 408.404, 221.208, 485.549, 35.453, 40.078 |
1NM6 | 1.8 | HOMO SAPIENS | ENZYME 3.4.21.5 | L86 | Ki = 0.09 nM | 509.043 |
1NRS | 2.4 | HOMO SAPIENS | ENZYME 3.4.21.5 | LEU ASP PRO ARG | | 484.578 |
1NT1 | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | T76 | Ki = 1.3 nM | 505.006 |
1NY2 | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, ARG PRO PRO GLY PHE | | 1129.21, 558.684 |
1NZQ | 2.18 | HOMO SAPIENS | ENZYME 3.4.21.5 | 162 | ic50 = 11 nM | 456.538 |
1O0D | 2.44 | HOMO SAPIENS | ENZYME 3.4.21.5 | 163 | ic50 = 6.2 nM | 456.538 |
1O2G | 1.58 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, 696 | Ki = 0.76 uM | 22.99, 327.379 |
1O5G | 1.75 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, CR9, CA | Ki = 11 uM | 22.99, 382.431, 40.078 |
1OYT | 1.67 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, FSN, CA | Ki = 0.057 uM | 22.99, 407.461, 40.078 |
1QBV | 1.8 | HOMO SAPIENS | ENZYME 3.4.21.5 | PPX | Ki = 4100 nM | 381.471 |
1QHR | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 157 | | 1129.21, 226.315 |
1QJ1 | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 166 | ic50 = 9 nM | 1129.21, 382.453 |
1QJ6 | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 167 | ic50 = 18 nM | 1129.21, 396.479 |
1QJ7 | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | GR1, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | ic50 = 18 nM | 465.585, 1129.21 |
1RIW | 2.04 | HOMO SAPIENS | ENZYME 3.4.21.5 | OSC, NAG, NA | ic50 = 28 nM | 616.75, 221.208, 22.99 |
1SB1 | 1.9 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, ASP PHE GLU GLU ILE PRO GLU GLU TYS, 165 | Ki = 128 nM | 22.99, 1229.22, 569.739 |
1SL3 | 1.81 | HOMO SAPIENS | ENZYME 3.4.21.5 | 170 | Ki = 1.4 pM | 552.321 |
1T4U | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | 81A | | 483.558 |
1T4V | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | 14A | Ki = 0.021 uM | 394.896 |
1TA2 | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | 176 | Ki = 3 nM | 496.428 |
1TA6 | 1.9 | HOMO SAPIENS | ENZYME 3.4.21.5 | 177 | Ki = 0.74 nM | 479.012 |
1TB6 | 2.5 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, NAG NAG FUC, NAG NAG BMA MAN MAN, NAG NAG BMA, MPD, GU4 GU6 GU0 GU5 GU8 GU9 GU8 GU9 GU8 GU9 GU8 GU5 GU1 GU6 GU2 GU3 | | 221.208, 570.545, 118.174 |
1TMT | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, DPN PRO ARG | | 221.208, 419.506 |
1TOM | 1.8 | HOMO SAPIENS | ENZYME 3.4.21.5 | MIN | Ki = 5 nM | 386.531 |
1TWX | 2.4 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, ASP PHE GLU GLU ILE PRO GLY GLU TYS LEU | | 221.208, 1286.31 |
1UMA | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, IN2, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 221.208, 218.254, 1129.21 |
1UVT | 2.5 | BOS TAURUS | ENZYME 3.4.21.5 | I48 | Ki = 0.023 uM | 384.472 |
1VR1 | 1.9 | HOMO SAPIENS | ENZYME 3.4.21.5 | ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 1129.21 |
1VZQ | 1.54 | HOMO SAPIENS | ENZYME 3.4.21.5 | SHY, NA, CA | Ki = 36 nM | 448.471, 22.99, 40.078 |
1W7G | 1.65 | HOMO SAPIENS | ENZYME 3.4.21.5 | MIU | Ki ~ 13 uM | 507.573 |
1WAY | 2.02 | HOMO SAPIENS | ENZYME 3.4.21.5 | L02, DMS, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | ic50 = 400 uM | 261.75, 78.133, 1129.21 |
1WBG | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | L03, DMS, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | ic50 = 1 mM | 225.698, 78.133, 1129.21 |
1XM1 | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | GAH, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 767.961, 1129.21 |
1XMN | 1.85 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG NAG, NAG NDG, NAG NAG BMA MAN MAN, IDS SGN IDS SGN IDS SGN, SGN IDS SGN IDS SGN, NA, GOL, 0G6 | | 408.404, 1722.33, 1468.16, 22.99, 92.094, 453.986 |
1YCP | 2.5 | BOS TAURUS | ENZYME 3.4.21.5 | TYR GLY VAL ARG GLY PRO | | |
1YPE | 1.81 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, GOL, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, UIP | Ki = 8 nM | 22.99, 92.094, 1129.21, 446.541 |
1YPG | 1.8 | HOMO SAPIENS | ENZYME 3.4.21.5 | UIR, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 10 nM | 458.552, 1129.21 |
1YPJ | 1.78 | HOMO SAPIENS | ENZYME 3.4.21.5 | UIB, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 95 nM | 448.557, 1129.21 |
1YPK | 1.78 | HOMO SAPIENS | ENZYME 3.4.21.5 | CCR, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 601.714, 1129.21 |
1YPL | 1.85 | HOMO SAPIENS | ENZYME 3.4.21.5 | RA8, NA, GOL, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 10.6 uM | 494.651, 22.99, 92.094, 1129.21 |
1YPM | 1.85 | HOMO SAPIENS | ENZYME 3.4.21.5 | RA4, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 1.9 uM | 489.568, 1129.21 |
1Z71 | 1.8 | HOMO SAPIENS | ENZYME 3.4.21.5 | L17 | Ki = 0.66 nM | 497.322 |
1ZGI | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | 382, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 4.6 uM | 439.461, 1129.21 |
1ZGV | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 501 | ic50 ~ 1 uM | 1129.21, 344.842 |
1ZRB | 1.9 | HOMO SAPIENS | ENZYME 3.4.21.5 | 062 | Ki = 0.77 nM | 492.954 |
2A2X | 2.44 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA9 | ic50 = 20.2 nM | 446.543 |
2ANK | 2.46 | HOMO SAPIENS | ENZYME 3.4.21.5 | N12 | ic50 = 47.3 nM | 472.58 |
2ANM | 2.4 | HOMO SAPIENS | ENZYME 3.4.21.5 | CDO | ic50 = 1.8 nM | 456.538 |
2BDY | 1.61 | HOMO SAPIENS | ENZYME 3.4.21.5 | UNB, NA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | ic50 = 0.017 uM | 502.585, 22.99, 1129.21 |
2C8W | 1.96 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, C7M | ic50 = 3.7 nM | 22.99, 546.061 |
2C8X | 2.17 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, DMS, C5M | ic50 = 220 nM | 22.99, 78.133, 517.08 |
2C8Y | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, DMS, C3M | | 22.99, 78.133, 370.465 |