1A2C | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, 34H LEU PRJ OAR | ic50 = 0.5 uM | 22.99, 605.757 |
1A4W | 1.8 | HOMO SAPIENS | ENZYME 3.4.21.5 | QWE, NA | Ki = 1.2 uM | 614.802, 22.99 |
1AD8 | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, MDL, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 247 nM | 22.99, 564.547, 1129.21 |
1AE8 | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | AZL, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, NAG | | 419.518, 1129.21, 221.208 |
1AFE | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, ALZ | | 221.208, 1129.21, 334.413 |
1AIX | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | T19 | | 567.44 |
1AWF | 2.2 | HOMO SAPIENS | ENZYME 3.4.21.5 | GR4, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 0.97 uM | 736.843, 1129.21 |
1BCU | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | PRL | Kd = 0.53 mM | 209.247 |
1BHX | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | R56, ASP PHE GLU GLU ILE | Ki = 0.145 uM | 468.593, 648.646 |
1C1U | 1.75 | HOMO SAPIENS | ENZYME 3.4.21.5 | ZN, NA, BAI | | 65.409, 22.99, 290.323 |
1C1V | 1.98 | HOMO SAPIENS | ENZYME 3.4.21.5 | ZN, NA, BAB | Ki = 0.023 uM | 65.409, 22.99, 335.386 |
1C1W | 1.9 | HOMO SAPIENS | ENZYME 3.4.21.5 | ZN, NA, BAH | | 65.409, 22.99, 366.377 |
1C4U | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, IH1 | Ki = 0.043 nM | 22.99, 581.483 |
1C4V | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, IH2 | Ki = 0.016 nM | 22.99, 528.645 |
1C5L | 1.47 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, CA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 22.99, 40.078, 1129.21 |
1C5N | 1.5 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, ESI, CA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | Ki = 20 uM | 22.99, 303.143, 40.078, 1129.21 |
1C5O | 1.9 | HOMO SAPIENS | ENZYME 3.4.21.5 | BAM, NA | Ki = 320 uM | 121.16, 22.99 |
1D3D | 2.04 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, NA, BZT | Ka = 1240000000 M^-1 | 221.208, 22.99, 591.601 |
1D3P | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | BT3, NAG, NA | Ka = 24300000 M^-1 | 543.719, 221.208, 22.99 |
1D4P | 2.07 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, NA, BPP | Ka = 2000000 M^-1 | 221.208, 22.99, 360.452 |
1D6W | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 00R | Ki = 1100 nM | 22.99, 1129.21, 527.596 |
1D9I | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, 00P | Ki = 0.78 nM | 22.99, 1129.21, 475.561 |
1EB1 | 1.8 | SYNTHETIC CONSTRUCT | ENZYME 3.4.21.5 | ZAL PRO MMO, ASP TYR GLU PRO ILE PRO GLU GLU ALA PHE | Ki = 37 pM | 424.59, 1205.24 |
1ETR | 2.2 | BOS TAURUS | ENZYME 3.4.21.5 | MIT | | 509.642 |
1ETS | 2.3 | BOS TAURUS | ENZYME 3.4.21.5 | MID | Ki = 6 nM | 521.631 |
1ETT | 2.5 | BOS TAURUS | ENZYME 3.4.21.5 | 4QQ | Ki = 1.3 uM | 428.548 |
1FPC | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | 0ZI | Ki = 0.1 uM | 503.681 |
1G30 | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | T87 | Ki = 140 nM | 525.602 |
1G32 | 1.9 | HOMO SAPIENS | ENZYME 3.4.21.5 | R11 | Ki = 780 nM | 423.513 |
1G37 | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | PHE GLU ALA ILE PRO ALA GLU TYR LEU, 110 | | 1050.18, 574.689 |
1GHV | 1.85 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, 120 | Ki = 45 uM | 22.99, 254.267 |
1GHW | 1.75 | HOMO SAPIENS | ENZYME 3.4.21.5 | NA, BMZ | Ki = 4 uM | 22.99, 253.279 |
1GHY | 1.85 | HOMO SAPIENS | ENZYME 3.4.21.5 | ZN, NA, CA, 121 | Ki = 0.008 uM | 65.409, 22.99, 40.078, 254.267 |
1H8D | 1.4 | HOMO SAPIENS | ENZYME 3.4.21.5 | PHW, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 805.851, 1129.21 |
1H8I | 1.75 | HOMO SAPIENS | ENZYME 3.4.21.5 | ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU, PHV | | 1129.21, 637.66 |
1HAG | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 221.208, 1129.21 |
1HAH | 2.3 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG, ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU | | 221.208, 1129.21 |
1HXE | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | RB, ASP PHE GLU GLU ILE PRO GLY GLU TYR LEU | | 85.468, 1192.27 |
1HXF | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | ASP PHE GLU GLU ILE PRO GLY GLU TYR LEU | | 1192.27 |
1JWT | 2.5 | HOMO SAPIENS | ENZYME 3.4.21.5 | BLI | Ki = 14 nM | 492.592 |
1K21 | 1.86 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG NAG, NA, IGN | Ki = 4.2 nM | 408.404, 22.99, 438.564 |
1K22 | 1.93 | HOMO SAPIENS | ENZYME 3.4.21.5 | NAG NAG, NA, MEL | Ki = 4 nM | 408.404, 22.99, 429.513 |
1KTS | 2.4 | HOMO SAPIENS | ENZYME 3.4.21.5 | C24 | Ki = 4.5 nM | 499.564 |
1KTT | 2.1 | HOMO SAPIENS | ENZYME 3.4.21.5 | C02 | ic50 = 1.5 uM | 419.499 |
1MU6 | 1.99 | HOMO SAPIENS | ENZYME 3.4.21.5 | CDA | Ki = 4.2 nM | 432.399 |
1MU8 | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | CDB | Ki = 1 nM | 448.442 |
1MUE | 2 | HOMO SAPIENS | ENZYME 3.4.21.5 | CDD | Ki = 2.3 nM | 467.829 |
1NL2 | 2.3 | BOS TAURUS | ENZYME 3.4.21.5 | NAG NAG, NAG, LPS, CL, CA | | 408.404, 221.208, 485.549, 35.453, 40.078 |
1NM6 | 1.8 | HOMO SAPIENS | ENZYME 3.4.21.5 | L86 | Ki = 0.09 nM | 509.043 |
1NRS | 2.4 | HOMO SAPIENS | ENZYME 3.4.21.5 | LEU ASP PRO ARG | | 484.578 |