1RQI | 2.42 | ESCHERICHIA COLI | ENZYME 2.5.1.10 | MG, IPR, DST, DPO | | 24.305, 248.108, 262.158, 173.943 |
1RQJ | 1.95 | ESCHERICHIA COLI | ENZYME 2.5.1.10 | IPE, RIS, MG | | 246.092, 283.112, 24.305 |
1YHL | 1.95 | TRYPANOSOMA CRUZI | ENZYME 2.5.1.10 | SO4, RIS, MG, DMA | | 96.063, 283.112, 24.305, 246.092 |
1YHM | 2.5 | TRYPANOSOMA CRUZI | ENZYME 2.5.1.10 | MG, AHD, IPE, SO4 | ic50 = 147 uM | 24.305, 245.064, 246.092, 96.063 |
1YQ7 | 2.2 | HOMO SAPIENS | ENZYME 2.5.1.10 | RIS, PO4, MG | | 283.112, 94.971, 24.305 |
1YV5 | 2 | HOMO SAPIENS | ENZYME 2.5.1.10 | RIS, PO4, MG | | 283.112, 94.971, 24.305 |
1ZW5 | 2.3 | HOMO SAPIENS | ENZYME 2.5.1.10 | IPE, ZOL, MG | | 246.092, 272.09, 24.305 |
2EWG | 2.48 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | PGO, MG, M0N | | 76.094, 24.305, 322.148 |
2F8C | 2.2 | HOMO SAPIENS | ENZYME 2.5.1.10 | ZOL, PO4, MG | | 272.09, 94.971, 24.305 |
2F92 | 2.15 | HOMO SAPIENS | ENZYME 2.5.1.10 | ZN, PO4, AHD | | 65.409, 94.971, 245.064 |
2F94 | 1.94 | HOMO SAPIENS | ENZYME 2.5.1.10 | ZN, PO4, BFQ | | 65.409, 94.971, 319.229 |
2F9K | 2.06 | HOMO SAPIENS | ENZYME 2.5.1.10 | ZOL, ZN, PO4 | | 272.09, 65.409, 94.971 |
2I19 | 2.28 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | MG, 1BY | | 24.305, 282.128 |
2OPM | 2.4 | HOMO SAPIENS | ENZYME 2.5.1.10 | PO4, NI9, MG | | 94.971, 302.111, 24.305 |
2P1C | 2.45 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | MG, GG3, BME, ACT | Ki = 21 nM | 24.305, 381.298, 78.133, 59.044 |
3DYG | 2.1 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | NI9, MPD, MG, BME, ACT | | 302.111, 118.174, 24.305, 78.133, 59.044 |
3DYH | 1.94 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | MG, 721 | | 24.305, 340.227 |
3EFQ | 2 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | MG, 714 | | 24.305, 396.333 |
3EGT | 2 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | MG, 722 | Ki = 1.26 nM | 24.305, 382.306 |
3IBA | 2.4 | TRYPANOSOMA CRUZI | ENZYME 2.5.1.10 | IPE, ZOL, SO4, MG | | 246.092, 272.09, 96.063, 24.305 |
3ICK | 2.4 | TRYPANOSOMA CRUZI | ENZYME 2.5.1.10 | IPE, SO4, MG, M0N, ACY | | 246.092, 96.063, 24.305, 322.148, 60.052 |
3ICM | 2.2 | TRYPANOSOMA CRUZI | ENZYME 2.5.1.10 | IPE, SO4, P2H, MG | | 246.092, 96.063, 360.216, 24.305 |
3ICN | 2.4 | TRYPANOSOMA CRUZI | ENZYME 2.5.1.10 | IPE, SO4, NI9, MG | | 246.092, 96.063, 302.111, 24.305 |
3ICZ | 2.15 | TRYPANOSOMA CRUZI | ENZYME 2.5.1.10 | PB6, MG, IPE | | 322.211, 24.305, 246.092 |
3N1V | 2.18 | HOMO SAPIENS | ENZYME 2.5.1.10 | PO4, 3N1 | ic50 > 500 uM | 94.971, 240.706 |
3N45 | 1.88 | HOMO SAPIENS | ENZYME 2.5.1.10 | ZOL, PO4, MG, 3N3 | | 272.09, 94.971, 24.305, 297.305 |
3N46 | 2.35 | HOMO SAPIENS | ENZYME 2.5.1.10 | ZOL, PO4, MG, 3N5 | | 272.09, 94.971, 24.305, 297.305 |
3N49 | 2.5 | HOMO SAPIENS | ENZYME 2.5.1.10 | PO4, 3N4 | ic50 = 7 uM | 94.971, 242.293 |
3N5H | 2.2 | HOMO SAPIENS | ENZYME 2.5.1.10 | PO4, GO0 | ic50 = 2 uM | 94.971, 288.084 |
3N5J | 2.35 | HOMO SAPIENS | ENZYME 2.5.1.10 | PO4, GO1 | ic50 = 6 uM | 94.971, 288.084 |
3N6K | 2.25 | HOMO SAPIENS | ENZYME 2.5.1.10 | PO4, BFH | Kd = 180 nM | 94.971, 269.252 |
4DEM | 1.85 | HOMO SAPIENS | ENZYME 2.5.1.10 | YS4, MG | ic50 = 28 nM | 402.276, 24.305 |
4DWB | 2.1 | TRYPANOSOMA CRUZI | ENZYME 2.5.1.10 | NA, 0M7, SO4, ACT, IPE, MG | ic50 = 1840 nM | 22.99, 275.176, 96.063, 59.044, 246.092, 24.305 |
4DWG | 2.01 | TRYPANOSOMA CRUZI | ENZYME 2.5.1.10 | NA, PEG, ACT, MG, 0M8, SO4 | ic50 = 58 nM | 22.99, 106.12, 59.044, 24.305, 303.23, 96.063 |
4DXJ | 2.35 | TRYPANOSOMA CRUZI | ENZYME 2.5.1.10 | IPE, PGE, SO4, PEG, 0M9, MG, ACT | ic50 = 38 nM | 246.092, 150.173, 96.063, 106.12, 247.123, 24.305, 59.044 |
4H5C | 2.02 | HOMO SAPIENS | ENZYME 2.5.1.10 | YS4, PO4, MG | | 402.276, 94.971, 24.305 |
4H5D | 2.02 | HOMO SAPIENS | ENZYME 2.5.1.10 | YS4, POP, MG | Kd = 0.58 uM | 402.276, 175.959, 24.305 |
4H5E | 2.04 | HOMO SAPIENS | ENZYME 2.5.1.10 | YS4, MG, IPR | Kd = 0.86 uM | 402.276, 24.305, 248.108 |
4LFV | 2 | HOMO SAPIENS | ENZYME 2.5.1.10 | YS4, CL, PO4, MG | | 402.276, 35.453, 94.971, 24.305 |
4LPG | 2.35 | HOMO SAPIENS | ENZYME 2.5.1.10 | PO4, 1MV | Kd = 55.6 uM | 94.971, 415.298 |
4LPH | 2.3 | HOMO SAPIENS | ENZYME 2.5.1.10 | PO4, YL3 | Kd = 9.2 uM | 94.971, 335.318 |
4P0V | 2.4 | HOMO SAPIENS | ENZYME 2.5.1.10 | MG, 1WO, ZOL | | 24.305, 314.419, 272.09 |
4P0W | 2.41 | HOMO SAPIENS | ENZYME 2.5.1.10 | 1XH, ZOL, MG | | 312.446, 272.09, 24.305 |
4P0X | 2.5 | HOMO SAPIENS | ENZYME 2.5.1.10 | 1WO | | 314.419 |
4QXS | 1.9 | HOMO SAPIENS | ENZYME 2.5.1.10 | WC1, PO4, GOL | ic50 = 1.1 uM | 451.39, 94.971, 92.094 |
4RXA | 2.2 | HOMO SAPIENS | ENZYME 2.5.1.10 | 3F2, PO4 | ic50 = 1.8 uM | 528.604, 94.971 |
4RXC | 2.31 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | HRX, MG | ic50 ~ 33 uM | 297.139, 24.305 |
4RXD | 2 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | RIS, MG | ic50 = 300 nM | 283.112, 24.305 |
4RXE | 2.5 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | 3YQ, MG | ic50 = 230 nM | 282.128, 24.305 |
4UMJ | 1.85 | PSEUDOMONAS AERUGINOSA | ENZYME 2.5.1.10 | BFQ, MG | ic50 = 2.7 uM | 319.229, 24.305 |