13PK | 2.5 | TRYPANOSOMA BRUCEI | ENZYME 2.7.2.3 | PO4, MG, ADP, 3PG | | 94.971, 24.305, 427.201, 186.057 |
16PK | 1.6 | TRYPANOSOMA BRUCEI | ENZYME 2.7.2.3 | EPE, BIS | | 238.305, 633.276 |
1F3T | 2 | TRYPANOSOMA BRUCEI | ENZYME 4.1.1.17 | PLP PUT | | 316.274 |
1GY8 | 2 | TRYPANOSOMA BRUCEI | ENZYME 5.1.3.2 | UDP, NAD | | 404.161, 663.425 |
1VBJ | 2.1 | TRYPANOSOMA BRUCEI | ENZYME 1.1.1.188 | NAP, CIT | | 743.405, 192.124 |
1XDN | 1.2 | TRYPANOSOMA BRUCEI | ENZYME LIGASES | MG, ATP | | 24.305, 507.181 |
2B4G | 1.95 | TRYPANOSOMA BRUCEI | ENZYME 1.3.99.11 | ORO, GOL, FMN, BR | | 156.096, 92.094, 456.344, 79.904 |
2B51 | 2.05 | TRYPANOSOMA BRUCEI | NON-ENZYME TRANSCRIPT_TRANSLATE | UTP, MN | | 484.141, 54.938 |
2B56 | 1.97 | TRYPANOSOMA BRUCEI | NON-ENZYME TRANSCRIPT_TRANSLATE | UTP, U5P, MG | | 484.141, 324.181, 24.305 |
2EWG | 2.48 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | PGO, MG, M0N | | 76.094, 24.305, 322.148 |
2F2T | 1.7 | TRYPANOSOMA BRUCEI | ENZYME 2.4.2.6 | SO4, GOL, 5IQ | | 96.063, 92.094, 144.173 |
2F62 | 1.5 | TRYPANOSOMA BRUCEI | ENZYME 2.4.2.6 | SO4, GOL, 12M | | 96.063, 92.094, 136.191 |
2F64 | 1.6 | TRYPANOSOMA BRUCEI | ENZYME 2.4.2.6 | SO4, GOL, 12Q | | 96.063, 92.094, 159.185 |
2F67 | 1.6 | TRYPANOSOMA BRUCEI | ENZYME 2.4.2.6 | SO4, GOL, 12B | | 96.063, 92.094, 169.179 |
2I19 | 2.28 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | MG, 1BY | | 24.305, 282.128 |
2IKF | 2 | TRYPANOSOMA BRUCEI | ENZYME 2.7.7.52 | UTP, MG | | 484.141, 24.305 |
2NOM | 2.4 | TRYPANOSOMA BRUCEI | ENZYME 2.7.7.52 | MG, DUT | | 24.305, 468.142 |
2P1C | 2.45 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | MG, GG3, BME, ACT | Ki = 21 nM | 24.305, 381.298, 78.133, 59.044 |
2PTY | 2 | TRYPANOSOMA BRUCEI | ENZYME 4.2.1.11 | ZN, PEP, EDO | | 65.409, 168.042, 62.068 |
2PTZ | 1.65 | TRYPANOSOMA BRUCEI | ENZYME 4.2.1.11 | PAH, EDO, ZN | | 155.047, 62.068, 65.409 |
2PU0 | 1.9 | TRYPANOSOMA BRUCEI | ENZYME 4.2.1.11 | ZN, PAH, EDO | | 65.409, 155.047, 62.068 |
2PU1 | 1.8 | TRYPANOSOMA BRUCEI | ENZYME 4.2.1.11 | ZN, FSG, EDO | | 65.409, 173.037, 62.068 |
2Q0C | 2.2 | TRYPANOSOMA BRUCEI | ENZYME 2.7.7.52 | MG, CTP | | 24.305, 483.156 |
2Q0D | 2 | TRYPANOSOMA BRUCEI | ENZYME 2.7.7.52 | MG, ATP | | 24.305, 507.181 |
2Q0E | 2.1 | TRYPANOSOMA BRUCEI | ENZYME 2.7.7.52 | MG, GTP | | 24.305, 523.18 |
2Q0F | 2.4 | TRYPANOSOMA BRUCEI | ENZYME 2.7.7.52 | UTP, U5P, MG | | 484.141, 324.181, 24.305 |
2Q0G | 2.3 | TRYPANOSOMA BRUCEI | ENZYME 2.7.7.52 | UPU, MG, CL | | 550.367, 24.305, 35.453 |
2WOI | 2.1 | TRYPANOSOMA BRUCEI | ENZYME 1.8.1.12 | FAD, CL, NA | | 785.55, 35.453, 22.99 |
2WOV | 2.5 | TRYPANOSOMA BRUCEI | ENZYME 1.8.1.12 | NDP, NA, FAD | | 745.421, 22.99, 785.55 |
2WOW | 2.2 | TRYPANOSOMA BRUCEI | ENZYME 1.8.1.12 | NDP, GCG, FAD | | 745.421, 723.862, 785.55 |
2WP6 | 2.5 | TRYPANOSOMA BRUCEI | ENZYME 1.8.1.12 | WP6, FAD, CL | ic50 = 0.93 uM | 346.853, 785.55, 35.453 |
2WPC | 2.1 | TRYPANOSOMA BRUCEI | ENZYME 1.8.1.12 | WP7, NA, FAD, CL | ic50 = 0.42 uM | 462.971, 22.99, 785.55, 35.453 |
2WPE | 2.1 | TRYPANOSOMA BRUCEI | ENZYME 1.8.1.12 | MRD, WPE, MPD, NA, FAD, CL | ic50 = 0.86 uM | 118.174, 393.866, 118.174, 22.99, 785.55, 35.453 |
2WPF | 1.9 | TRYPANOSOMA BRUCEI | ENZYME 1.8.1.12 | WPF, FAD, CL, BR | ic50 = 0.23 uM | 355.904, 785.55, 35.453, 79.904 |
3BJE | 1.44 | TRYPANOSOMA BRUCEI | ENZYME 2.4.2.- | URA, R1P, CA | | 112.087, 230.11, 40.078 |
3CV0 | 2 | TRYPANOSOMA BRUCEI | NON-ENZYME SIGNAL_HORMONE | PHE ASN GLU LEU SER HIS LEU, EDO | | 666.733, 62.068 |
3CVL | 2.15 | TRYPANOSOMA BRUCEI | NON-ENZYME SIGNAL_HORMONE | HIS GLU GLU LEU ALA LYS LEU | | 571.696 |
3CVN | 2 | TRYPANOSOMA BRUCEI | NON-ENZYME SIGNAL_HORMONE | EDO, ARG ASP ARG ALA ALA LYS LEU | | 62.068, 558.705 |
3CVP | 2 | TRYPANOSOMA BRUCEI | NON-ENZYME SIGNAL_HORMONE | GLY THR LEU SER ASN ARG ALA SER LYS LEU | | 559.665 |
3DYG | 2.1 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | NI9, MPD, MG, BME, ACT | | 302.111, 118.174, 24.305, 78.133, 59.044 |
3DYH | 1.94 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | MG, 721 | | 24.305, 340.227 |
3E7F | 2.2 | TRYPANOSOMA BRUCEI | ENZYME 3.1.1.17 | ZN, 6PG | | 65.409, 276.135 |
3EB9 | 2 | TRYPANOSOMA BRUCEI | ENZYME 3.1.1.17 | ZN, FLC | | 65.409, 189.1 |
3EFQ | 2 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | MG, 714 | | 24.305, 396.333 |
3EGT | 2 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | MG, 722 | Ki = 1.26 nM | 24.305, 382.306 |
3HIY | 2.3 | TRYPANOSOMA BRUCEI | ENZYME UNCLASSIFIED | UTP, MG | | 484.141, 24.305 |
3HJ1 | 1.95 | TRYPANOSOMA BRUCEI | ENZYME UNCLASSIFIED | UTP | | 484.141 |
3JQ6 | 1.8 | TRYPANOSOMA BRUCEI | ENZYME 1.5.1.33 | DTT, NAP, DX1 | Ki = 3.3 uM | 154.251, 743.405, 246.312 |
3JQ7 | 1.8 | TRYPANOSOMA BRUCEI | ENZYME 1.5.1.33 | NAP, DX2, DTT, ACT | Ki = 1.2 uM | 743.405, 253.263, 154.251, 59.044 |
3JQ8 | 1.95 | TRYPANOSOMA BRUCEI | ENZYME 1.5.1.33 | NAP, DX3, DTT | Ki > 35 uM | 743.405, 206.248, 154.251 |
3JQ9 | 2.3 | TRYPANOSOMA BRUCEI | ENZYME 1.5.1.33 | NAP, AX1 | Ki = 0.4 uM | 743.405, 295.253 |
3JQA | 1.9 | TRYPANOSOMA BRUCEI | ENZYME 1.5.1.33 | NAP, DX4 | | 743.405, 167.192 |
3JQB | 2.4 | TRYPANOSOMA BRUCEI | ENZYME 1.5.1.33 | NAP, DX6, DTT | Ki = 0.96 uM | 743.405, 254.287, 154.251 |
3JQC | 1.8 | TRYPANOSOMA BRUCEI | ENZYME 1.5.1.33 | NAP, JU2 | Ki = 3.9 uM | 743.405, 254.044 |
3JQD | 1.6 | TRYPANOSOMA BRUCEI | ENZYME 1.5.1.33 | NAP, DX7, ACT | Ki = 0.71 uM | 743.405, 251.243, 59.044 |
3JQE | 2 | TRYPANOSOMA BRUCEI | ENZYME 1.5.1.33 | NAP, DX8, ACT | Ki = 0.36 uM | 743.405, 281.269, 59.044 |
3JQF | 1.6 | TRYPANOSOMA BRUCEI | ENZYME 1.5.1.33 | NAP, D1D, GOL, AX2, DTT, ACT | | 743.405, 152.235, 92.094, 126.12, 154.251, 59.044 |
3JQG | 1.9 | TRYPANOSOMA BRUCEI | ENZYME 1.5.1.33 | NAP, AX6 | Ki = 18 uM | 743.405, 262.331 |
3OTX | 1.55 | TRYPANOSOMA BRUCEI | ENZYME 2.7.1.20 | NA, AP5 | ic50 = 29.4 uM | 22.99, 916.367 |
3QCP | 2.3 | TRYPANOSOMA BRUCEI | ENZYME 1.8.3.2 | FAD | | 785.55 |
3TIK | 2.05 | TRYPANOSOMA BRUCEI | ENZYME 1.14.13.70 | JKF, HEM | | 505.943, 616.487 |
3ZS7 | 2 | TRYPANOSOMA BRUCEI | ENZYME 2.7.1.35 | PO4, ATP | | 94.971, 507.181 |
4BQH | 1.75 | TRYPANOSOMA BRUCEI | ENZYME 2.7.7.23 | 9VU, SO4 | Kd = 2.58 uM | 404.211, 96.063 |
4DK4 | 1.9 | TRYPANOSOMA BRUCEI | ENZYME 3.6.1.23 | NA, DUN, CA | | 22.99, 387.177, 40.078 |
4DKB | 1.83 | TRYPANOSOMA BRUCEI | ENZYME 3.6.1.23 | DUN, CA | | 387.177, 40.078 |
4DL8 | 1.7 | TRYPANOSOMA BRUCEI | ENZYME 3.6.1.23 | UMP AF3 PO4, NA, MG | | 485.113, 22.99, 24.305 |
4DLC | 1.76 | TRYPANOSOMA BRUCEI | ENZYME 3.6.1.23 | MGF, MG, UMP | | 81.3, 24.305, 308.182 |
4MVY | 2.31 | TRYPANOSOMA BRUCEI | ENZYME 6.1.1.10 | 387, DMS, GOL | | 368.258, 78.133, 92.094 |
4MW0 | 2.2 | TRYPANOSOMA BRUCEI | ENZYME 6.1.1.10 | 392, DMS, GOL | | 368.258, 78.133, 92.094 |
4MW1 | 2.49 | TRYPANOSOMA BRUCEI | ENZYME 6.1.1.10 | DMS, 44F, GOL | | 78.133, 353.867, 92.094 |
4MW2 | 2.3 | TRYPANOSOMA BRUCEI | ENZYME 6.1.1.10 | 2E9, MET, DMS, GOL, SO4 | | 379.904, 149.211, 78.133, 92.094, 96.063 |
4MW4 | 2.5 | TRYPANOSOMA BRUCEI | ENZYME 6.1.1.10 | SO4, 2EB, MET, GOL, DMS | | 96.063, 465.737, 149.211, 92.094, 78.133 |
4MW5 | 2.35 | TRYPANOSOMA BRUCEI | ENZYME 6.1.1.10 | DMS, MET, SO4, 415, GOL | | 78.133, 149.211, 96.063, 347.839, 92.094 |
4MWB | 2.31 | TRYPANOSOMA BRUCEI | ENZYME 6.1.1.10 | 2EK, SO4, DMS, GOL | | 364.314, 96.063, 78.133, 92.094 |
4MWD | 2.25 | TRYPANOSOMA BRUCEI | ENZYME 6.1.1.10 | 43E, ACP, SO4, GOL, DMS | | 358.286, 505.208, 96.063, 92.094, 78.133 |
4MWE | 2.45 | TRYPANOSOMA BRUCEI | ENZYME 6.1.1.10 | MET, 2EN, SO4, DMS, GOL | | 149.211, 419.968, 96.063, 78.133, 92.094 |
4RXC | 2.31 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | HRX, MG | ic50 ~ 33 uM | 297.139, 24.305 |
4RXD | 2 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | RIS, MG | ic50 = 300 nM | 283.112, 24.305 |
4RXE | 2.5 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | 3YQ, MG | ic50 = 230 nM | 282.128, 24.305 |
5AFX | 2.39 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | PVZ, MG | ic50 = 1.2 uM | 399.337, 24.305 |
5FSX | 2 | TRYPANOSOMA BRUCEI | NON-ENZYME OTHER | ADP, GOL | Ka = 540 M^-1 | 427.201, 92.094 |
5FSY | 1.7 | TRYPANOSOMA BRUCEI | NON-ENZYME OTHER | AR6 | Ka = 790000 M^-1 | 559.316 |
5FUV | 2.3 | TRYPANOSOMA BRUCEI | ENZYME 2.7.1.21 | PO4, THM, ZN, GOL | | 94.971, 242.229, 65.409, 92.094 |
5FUW | 2.2 | TRYPANOSOMA BRUCEI | ENZYME 2.7.1.21 | PO4, THM, QBT, ZN | | 94.971, 242.229, 324.224, 65.409 |
5FUX | 2.2 | TRYPANOSOMA BRUCEI | ENZYME 2.7.1.21 | MG, PO4, ZN, QBT | | 24.305, 94.971, 65.409, 324.224 |
5G2B | 1.83 | TRYPANOSOMA BRUCEI | ENZYME 3.1.4.- | GOL, ZN, GAI, LQY, MG, FMT | Ki = 0.1 uM | 92.094, 65.409, 59.07, 528.642, 24.305, 46.025 |
5G57 | 1.73 | TRYPANOSOMA BRUCEI | ENZYME 3.1.4.- | PEG, 6M5, FMT, MG, ZN, GOL, GAI | Ki = 4 nM | 106.12, 584.708, 46.025, 24.305, 65.409, 92.094, 59.07 |
5G5V | 1.8 | TRYPANOSOMA BRUCEI | ENZYME 3.1.4.- | 8Z4, MG, FMT, ZN, EDO, GAI | Ki = 200 nM | 487.59, 24.305, 46.025, 65.409, 62.068, 59.07 |
5I49 | 1.8 | TRYPANOSOMA BRUCEI | ENZYME TRANSFERASES | ZN, MG, 2KH | | 65.409, 24.305, 483.156 |
5IDO | 2.2 | TRYPANOSOMA BRUCEI | ENZYME TRANSFERASES | UTP, MG, ZN | | 484.141, 24.305, 65.409 |
5K4Q | 2.3 | TRYPANOSOMA BRUCEI | ENZYME 1.1.1.103 | GOL, SO4, NAD | | 92.094, 96.063, 663.425 |
5K4U | 1.9 | TRYPANOSOMA BRUCEI | ENZYME 1.1.1.103 | NAD, ACT, GOL | | 663.425, 59.044, 92.094 |
5K4V | 2.2 | TRYPANOSOMA BRUCEI | ENZYME 1.1.1.103 | NA, NAD, GOL, ACT | | 22.99, 663.425, 92.094, 59.044 |
5K4W | 1.72 | TRYPANOSOMA BRUCEI | ENZYME 1.1.1.103 | NA, GOL, NAI, THR | | 22.99, 92.094, 665.441, 119.119 |
5K4Y | 1.77 | TRYPANOSOMA BRUCEI | ENZYME 1.1.1.103 | GOL, NA, CL, ACT, NAD | | 92.094, 22.99, 35.453, 59.044, 663.425 |
5K50 | 2.26 | TRYPANOSOMA BRUCEI | ENZYME 1.1.1.103 | ACT, NAD, GOL, ALO | | 59.044, 663.425, 92.094, 119.119 |
5L8C | 2.01 | TRYPANOSOMA BRUCEI | ENZYME 3.1.4.- | PEG, MG, ZN, GOL, GAI, FMT, 908 | Ki = 100 nM | 106.12, 24.305, 65.409, 92.094, 59.07, 46.025, 474.552 |
5L8Y | 2.14 | TRYPANOSOMA BRUCEI | ENZYME 3.1.4.- | ZN, GAI, FMT, CVA, GOL, MG | Ki = 400 nM | 65.409, 59.07, 46.025, 572.694, 92.094, 24.305 |
5L9H | 2.25 | TRYPANOSOMA BRUCEI | ENZYME 3.1.4.- | ZN, FMT, CVL, GOL, MG | ic50 = 0.4 uM | 65.409, 46.025, 492.57, 92.094, 24.305 |
6E4P | 1.95 | TRYPANOSOMA BRUCEI | NON-ENZYME OTHER | U U U U | | |