13PK | 2.5 | TRYPANOSOMA BRUCEI | ENZYME 2.7.2.3 | PO4, MG, ADP, 3PG | | 94.971, 24.305, 427.201, 186.057 |
16PK | 1.6 | TRYPANOSOMA BRUCEI | ENZYME 2.7.2.3 | EPE, BIS | | 238.305, 633.276 |
1F3T | 2 | TRYPANOSOMA BRUCEI | ENZYME 4.1.1.17 | PLP PUT | | 316.274 |
1GY8 | 2 | TRYPANOSOMA BRUCEI | ENZYME 5.1.3.2 | UDP, NAD | | 404.161, 663.425 |
1VBJ | 2.1 | TRYPANOSOMA BRUCEI | ENZYME 1.1.1.188 | NAP, CIT | | 743.405, 192.124 |
1XDN | 1.2 | TRYPANOSOMA BRUCEI | ENZYME LIGASES | MG, ATP | | 24.305, 507.181 |
2B4G | 1.95 | TRYPANOSOMA BRUCEI | ENZYME 1.3.99.11 | FMN, BR, ORO, GOL | | 456.344, 79.904, 156.096, 92.094 |
2B51 | 2.05 | TRYPANOSOMA BRUCEI | NON-ENZYME TRANSCRIPT_TRANSLATE | UTP, MN | | 484.141, 54.938 |
2B56 | 1.97 | TRYPANOSOMA BRUCEI | NON-ENZYME TRANSCRIPT_TRANSLATE | UTP, U5P, MG | | 484.141, 324.181, 24.305 |
2EWG | 2.48 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | PGO, MG, M0N | | 76.094, 24.305, 322.148 |
2F2T | 1.7 | TRYPANOSOMA BRUCEI | ENZYME 2.4.2.6 | SO4, GOL, 5IQ | | 96.063, 92.094, 144.173 |
2F62 | 1.5 | TRYPANOSOMA BRUCEI | ENZYME 2.4.2.6 | SO4, GOL, 12M | | 96.063, 92.094, 136.191 |
2F64 | 1.6 | TRYPANOSOMA BRUCEI | ENZYME 2.4.2.6 | SO4, GOL, 12Q | | 96.063, 92.094, 159.185 |
2F67 | 1.6 | TRYPANOSOMA BRUCEI | ENZYME 2.4.2.6 | SO4, GOL, 12B | | 96.063, 92.094, 169.179 |
2I19 | 2.28 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | MG, 1BY | | 24.305, 282.128 |
2IKF | 2 | TRYPANOSOMA BRUCEI | ENZYME 2.7.7.52 | UTP, MG | | 484.141, 24.305 |
2NOM | 2.4 | TRYPANOSOMA BRUCEI | ENZYME 2.7.7.52 | DUT, MG | | 468.142, 24.305 |
2P1C | 2.45 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | MG, GG3, BME, ACT | Ki = 21 nM | 24.305, 381.298, 78.133, 59.044 |
2PTY | 2 | TRYPANOSOMA BRUCEI | ENZYME 4.2.1.11 | ZN, PEP, EDO | | 65.409, 168.042, 62.068 |
2PTZ | 1.65 | TRYPANOSOMA BRUCEI | ENZYME 4.2.1.11 | ZN, PAH, EDO | | 65.409, 155.047, 62.068 |
2PU0 | 1.9 | TRYPANOSOMA BRUCEI | ENZYME 4.2.1.11 | ZN, PAH, EDO | | 65.409, 155.047, 62.068 |
2PU1 | 1.8 | TRYPANOSOMA BRUCEI | ENZYME 4.2.1.11 | ZN, FSG, EDO | | 65.409, 173.037, 62.068 |
2Q0C | 2.2 | TRYPANOSOMA BRUCEI | ENZYME 2.7.7.52 | MG, CTP | | 24.305, 483.156 |
2Q0D | 2 | TRYPANOSOMA BRUCEI | ENZYME 2.7.7.52 | MG, ATP | | 24.305, 507.181 |
2Q0E | 2.1 | TRYPANOSOMA BRUCEI | ENZYME 2.7.7.52 | MG, GTP | | 24.305, 523.18 |
2Q0F | 2.4 | TRYPANOSOMA BRUCEI | ENZYME 2.7.7.52 | UTP, U5P, MG | | 484.141, 324.181, 24.305 |
2Q0G | 2.3 | TRYPANOSOMA BRUCEI | ENZYME 2.7.7.52 | UPU, MG, CL | | 550.367, 24.305, 35.453 |
2WOI | 2.1 | TRYPANOSOMA BRUCEI | ENZYME 1.8.1.12 | NA, FAD, CL | | 22.99, 785.55, 35.453 |
2WOV | 2.5 | TRYPANOSOMA BRUCEI | ENZYME 1.8.1.12 | NDP, NA, FAD | | 745.421, 22.99, 785.55 |
2WOW | 2.2 | TRYPANOSOMA BRUCEI | ENZYME 1.8.1.12 | NDP, GCG, FAD | | 745.421, 723.862, 785.55 |
2WP6 | 2.5 | TRYPANOSOMA BRUCEI | ENZYME 1.8.1.12 | WP6, FAD, CL | ic50 = 0.93 uM | 346.853, 785.55, 35.453 |
2WPC | 2.1 | TRYPANOSOMA BRUCEI | ENZYME 1.8.1.12 | WP7, NA, FAD, CL | ic50 = 0.42 uM | 462.971, 22.99, 785.55, 35.453 |
2WPE | 2.1 | TRYPANOSOMA BRUCEI | ENZYME 1.8.1.12 | MPD, NA, FAD, CL, WPE, MRD | ic50 = 0.86 uM | 118.174, 22.99, 785.55, 35.453, 393.866, 118.174 |
2WPF | 1.9 | TRYPANOSOMA BRUCEI | ENZYME 1.8.1.12 | WPF, FAD, CL, BR | ic50 = 0.23 uM | 355.904, 785.55, 35.453, 79.904 |
3BJE | 1.44 | TRYPANOSOMA BRUCEI | ENZYME 2.4.2.- | URA, R1P, CA | | 112.087, 230.11, 40.078 |
3CV0 | 2 | TRYPANOSOMA BRUCEI | NON-ENZYME SIGNAL_HORMONE | PHE ASN GLU LEU SER HIS LEU, EDO | | 666.733, 62.068 |
3CVL | 2.15 | TRYPANOSOMA BRUCEI | NON-ENZYME SIGNAL_HORMONE | HIS GLU GLU LEU ALA LYS LEU | | 571.696 |
3CVN | 2 | TRYPANOSOMA BRUCEI | NON-ENZYME SIGNAL_HORMONE | ARG ASP ARG ALA ALA LYS LEU, EDO | | 558.705, 62.068 |
3CVP | 2 | TRYPANOSOMA BRUCEI | NON-ENZYME SIGNAL_HORMONE | GLY THR LEU SER ASN ARG ALA SER LYS LEU | | 559.665 |
3DYG | 2.1 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | NI9, MPD, MG, BME, ACT | | 302.111, 118.174, 24.305, 78.133, 59.044 |
3DYH | 1.94 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | MG, 721 | | 24.305, 340.227 |
3E7F | 2.2 | TRYPANOSOMA BRUCEI | ENZYME 3.1.1.17 | ZN, 6PG | | 65.409, 276.135 |
3EB9 | 2 | TRYPANOSOMA BRUCEI | ENZYME 3.1.1.17 | ZN, FLC | | 65.409, 189.1 |
3EFQ | 2 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | 714, MG | | 396.333, 24.305 |
3EGT | 2 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | MG, 722 | Ki = 1.26 nM | 24.305, 382.306 |
3HIY | 2.3 | TRYPANOSOMA BRUCEI | ENZYME UNCLASSIFIED | UTP, MG | | 484.141, 24.305 |
3HJ1 | 1.95 | TRYPANOSOMA BRUCEI | ENZYME UNCLASSIFIED | UTP | | 484.141 |
3JQ6 | 1.8 | TRYPANOSOMA BRUCEI | ENZYME 1.5.1.33 | NAP, DX1, DTT | Ki = 3.3 uM | 743.405, 246.312, 154.251 |
3JQ7 | 1.8 | TRYPANOSOMA BRUCEI | ENZYME 1.5.1.33 | NAP, DX2, DTT, ACT | Ki = 1.2 uM | 743.405, 253.263, 154.251, 59.044 |
3JQ8 | 1.95 | TRYPANOSOMA BRUCEI | ENZYME 1.5.1.33 | NAP, DX3, DTT | Ki > 35 uM | 743.405, 206.248, 154.251 |