4MW2 | 2.3 | TRYPANOSOMA BRUCEI | ENZYME 6.1.1.10 | 2E9, MET, DMS, GOL, SO4 | | 379.904, 149.211, 78.133, 92.094, 96.063 |
4MWB | 2.31 | TRYPANOSOMA BRUCEI | ENZYME 6.1.1.10 | 2EK, SO4, DMS, GOL | | 364.314, 96.063, 78.133, 92.094 |
4MWE | 2.45 | TRYPANOSOMA BRUCEI | ENZYME 6.1.1.10 | 2EN, SO4, DMS, GOL, MET | | 419.968, 96.063, 78.133, 92.094, 149.211 |
4MVY | 2.31 | TRYPANOSOMA BRUCEI | ENZYME 6.1.1.10 | 387, DMS, GOL | | 368.258, 78.133, 92.094 |
4MW0 | 2.2 | TRYPANOSOMA BRUCEI | ENZYME 6.1.1.10 | 392, DMS, GOL | | 368.258, 78.133, 92.094 |
4RXE | 2.5 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | 3YQ, MG | ic50 = 230 nM | 282.128, 24.305 |
4MWD | 2.25 | TRYPANOSOMA BRUCEI | ENZYME 6.1.1.10 | 43E, ACP, SO4, GOL, DMS | | 358.286, 505.208, 96.063, 92.094, 78.133 |
4BQH | 1.75 | TRYPANOSOMA BRUCEI | ENZYME 2.7.7.23 | 9VU, SO4 | Kd = 2.58 uM | 404.211, 96.063 |
5FSX | 2 | TRYPANOSOMA BRUCEI | NON-ENZYME OTHER | ADP, GOL | Ka = 540 M^-1 | 427.201, 92.094 |
5K50 | 2.26 | TRYPANOSOMA BRUCEI | ENZYME 1.1.1.103 | ALO, ACT, NAD, GOL | | 119.119, 59.044, 663.425, 92.094 |
5FSY | 1.7 | TRYPANOSOMA BRUCEI | NON-ENZYME OTHER | AR6 | Ka = 790000 M^-1 | 559.316 |
3JQG | 1.9 | TRYPANOSOMA BRUCEI | ENZYME 1.5.1.33 | AX6, NAP | Ki = 18 uM | 262.331, 743.405 |
4MW1 | 2.49 | TRYPANOSOMA BRUCEI | ENZYME 6.1.1.10 | DMS, 44F, GOL | | 78.133, 353.867, 92.094 |
4DKB | 1.83 | TRYPANOSOMA BRUCEI | ENZYME 3.6.1.23 | DUN, CA | | 387.177, 40.078 |
3CVN | 2 | TRYPANOSOMA BRUCEI | NON-ENZYME SIGNAL_HORMONE | EDO, ARG ASP ARG ALA ALA LYS LEU | | 62.068, 558.705 |
16PK | 1.6 | TRYPANOSOMA BRUCEI | ENZYME 2.7.2.3 | EPE, BIS | | 238.305, 633.276 |
3QCP | 2.3 | TRYPANOSOMA BRUCEI | ENZYME 1.8.3.2 | FAD | | 785.55 |
6GXQ | 1.96 | TRYPANOSOMA BRUCEI | ENZYME 3.1.4.- | FFZ, MG, GAI, GOL, ZN | Ki = 0.00000079 M | 455.548, 24.305, 59.07, 92.094, 65.409 |
5G2B | 1.83 | TRYPANOSOMA BRUCEI | ENZYME 3.1.4.- | FMT, GOL, ZN, GAI, LQY, MG | Ki = 0.1 uM | 46.025, 92.094, 65.409, 59.07, 528.642, 24.305 |
6RFW | 2.18 | TRYPANOSOMA BRUCEI | ENZYME 3.1.4.- | FMT, K1Q, GAI, ZN, GOL, MG | Ki = 0.00000079 M | 46.025, 487.565, 59.07, 65.409, 92.094, 24.305 |
6RFN | 2.29 | TRYPANOSOMA BRUCEI | ENZYME 3.1.4.- | FMT, MG, GAI, ZN, GOL, K3W | Ki = 0.00000079 M | 46.025, 24.305, 59.07, 65.409, 92.094, 471.548 |
6RGK | 2.03 | TRYPANOSOMA BRUCEI | ENZYME 3.1.4.- | FMT, MG, GOL, GAI, K3N, ZN | | 46.025, 24.305, 92.094, 59.07, 477.638, 65.409 |
6P5R | 2.45 | TRYPANOSOMA BRUCEI | NON-ENZYME OTHER | GDP | | 443.201 |
3CVP | 2 | TRYPANOSOMA BRUCEI | NON-ENZYME SIGNAL_HORMONE | GLY THR LEU SER ASN ARG ALA SER LYS LEU | | 559.665 |
5L8C | 2.01 | TRYPANOSOMA BRUCEI | ENZYME 3.1.4.- | GOL, GAI, FMT, 908, PEG, MG, ZN | Ki = 100 nM | 92.094, 59.07, 46.025, 474.552, 106.12, 24.305, 65.409 |
5K4Y | 1.77 | TRYPANOSOMA BRUCEI | ENZYME 1.1.1.103 | GOL, NA, CL, ACT, NAD | | 92.094, 22.99, 35.453, 59.044, 663.425 |
5K4Q | 2.3 | TRYPANOSOMA BRUCEI | ENZYME 1.1.1.103 | GOL, SO4, NAD | | 92.094, 96.063, 663.425 |
3CVL | 2.15 | TRYPANOSOMA BRUCEI | NON-ENZYME SIGNAL_HORMONE | HIS GLU GLU LEU ALA LYS LEU | | 571.696 |
4RXC | 2.31 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | HRX, MG | ic50 ~ 33 uM | 297.139, 24.305 |
3TIK | 2.05 | TRYPANOSOMA BRUCEI | ENZYME 1.14.13.70 | JKF, HEM | | 505.943, 616.487 |
6RB6 | 1.9 | TRYPANOSOMA BRUCEI | ENZYME 3.1.4.- | JX2, MG, ZN, FMT, EDO, GAI | | 499.601, 24.305, 65.409, 46.025, 62.068, 59.07 |
4MW5 | 2.35 | TRYPANOSOMA BRUCEI | ENZYME 6.1.1.10 | MET, SO4, 415, GOL, DMS | | 149.211, 96.063, 347.839, 92.094, 78.133 |
2I19 | 2.28 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | MG, 1BY | | 24.305, 282.128 |
3EFQ | 2 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | MG, 714 | | 24.305, 396.333 |
3DYH | 1.94 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | MG, 721 | | 24.305, 340.227 |
3EGT | 2 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | MG, 722 | Ki = 1.26 nM | 24.305, 382.306 |
1XDN | 1.2 | TRYPANOSOMA BRUCEI | ENZYME LIGASES | MG, ATP | | 24.305, 507.181 |
2Q0D | 2 | TRYPANOSOMA BRUCEI | ENZYME 2.7.7.52 | MG, ATP | | 24.305, 507.181 |
3DYG | 2.1 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | MG, BME, ACT, NI9, MPD | | 24.305, 78.133, 59.044, 302.111, 118.174 |
2Q0G | 2.3 | TRYPANOSOMA BRUCEI | ENZYME 2.7.7.52 | MG, CL, UPU | | 24.305, 35.453, 550.367 |
2Q0C | 2.2 | TRYPANOSOMA BRUCEI | ENZYME 2.7.7.52 | MG, CTP | | 24.305, 483.156 |
2NOM | 2.4 | TRYPANOSOMA BRUCEI | ENZYME 2.7.7.52 | MG, DUT | | 24.305, 468.142 |
5G5V | 1.8 | TRYPANOSOMA BRUCEI | ENZYME 3.1.4.- | MG, FMT, ZN, EDO, GAI, 8Z4 | Ki = 200 nM | 24.305, 46.025, 65.409, 62.068, 59.07, 487.59 |
2P1C | 2.45 | TRYPANOSOMA BRUCEI | ENZYME 2.5.1.10 | MG, GG3, BME, ACT | Ki = 21 nM | 24.305, 381.298, 78.133, 59.044 |
2Q0E | 2.1 | TRYPANOSOMA BRUCEI | ENZYME 2.7.7.52 | MG, GTP | | 24.305, 523.18 |
2WPE | 2.1 | TRYPANOSOMA BRUCEI | ENZYME 1.8.1.12 | MRD, WPE, MPD, NA, FAD, CL | ic50 = 0.86 uM | 118.174, 393.866, 118.174, 22.99, 785.55, 35.453 |
3OTX | 1.55 | TRYPANOSOMA BRUCEI | ENZYME 2.7.1.20 | NA, AP5 | ic50 = 29.4 uM | 22.99, 916.367 |
4DK4 | 1.9 | TRYPANOSOMA BRUCEI | ENZYME 3.6.1.23 | NA, DUN, CA | | 22.99, 387.177, 40.078 |
2WOI | 2.1 | TRYPANOSOMA BRUCEI | ENZYME 1.8.1.12 | NA, FAD, CL | | 22.99, 785.55, 35.453 |
5K4W | 1.72 | TRYPANOSOMA BRUCEI | ENZYME 1.1.1.103 | NA, GOL, NAI, THR | | 22.99, 92.094, 665.441, 119.119 |