3WQQ | 2.25 | PLASMODIUM FALCIPARUM | ENZYME 1.1.1.267 | IB3, CA, NDP, MG | ic50 = 0.01 uM | 287.249, 40.078, 745.421, 24.305 |
3WQR | 1.97 | PLASMODIUM FALCIPARUM | ENZYME 1.1.1.267 | CA, LSX, NDP, MG | ic50 = 0.02 uM | 40.078, 303.248, 745.421, 24.305 |
3WQS | 2.35 | PLASMODIUM FALCIPARUM | ENZYME 1.1.1.267 | KBK, NDP, MG | ic50 = 0.05 uM | 305.221, 745.421, 24.305 |
4GAE | 2.3 | PLASMODIUM FALCIPARUM | ENZYME 1.1.1.267 | ACT, FOB, FOQ, EDO, CL, NDP, MN | Ki = 0.013 uM, Ki = 0.013 uM | 59.044, 274.21, 274.21, 62.068, 35.453, 745.421, 54.938 |
4KP7 | 2 | PLASMODIUM FALCIPARUM | ENZYME 1.1.1.267 | NAP, 1UQ, MN3 | ic50 = 9.4 nM | 743.405, 291.261, 54.938 |
4Y67 | 1.6 | PLASMODIUM FALCIPARUM | ENZYME 1.1.1.267 | MN, RC5 | ic50 = 0.117 uM | 54.938, 315.302 |
1CET | 2.05 | PLASMODIUM FALCIPARUM | ENZYME 1.1.1.27 | CLQ | Ki = 1.3 mM | 319.872 |
1LDG | 1.74 | PLASMODIUM FALCIPARUM | ENZYME 1.1.1.27 | NAI, OXM | | 665.441, 89.05 |
1T24 | 1.7 | PLASMODIUM FALCIPARUM | ENZYME 1.1.1.27 | OXQ, NAD, GOL | ic50 = 0.65 uM | 130.059, 663.425, 92.094 |
1T25 | 1.9 | PLASMODIUM FALCIPARUM | ENZYME 1.1.1.27 | NAI, GOL, GAG | ic50 = 1.1 uM | 665.441, 92.094, 129.071 |
1T26 | 1.8 | PLASMODIUM FALCIPARUM | ENZYME 1.1.1.27 | NAI, GBD | ic50 = 0.14 uM | 665.441, 146.125 |
1T2C | 2.01 | PLASMODIUM FALCIPARUM | ENZYME 1.1.1.27 | NAI, GOL | | 665.441, 92.094 |
1T2D | 1.1 | PLASMODIUM FALCIPARUM | ENZYME 1.1.1.27 | OXL, NAD, GOL | | 88.019, 663.425, 92.094 |
1T2E | 1.85 | PLASMODIUM FALCIPARUM | ENZYME 1.1.1.27 | OXM, NAI, GOL | | 89.05, 665.441, 92.094 |
1U4O | 1.7 | PLASMODIUM FALCIPARUM | ENZYME 1.1.1.27 | NDD, MPD | | 216.19, 118.174 |
1U4S | 2 | PLASMODIUM FALCIPARUM | ENZYME 1.1.1.27 | BIH | | 288.297 |
1U5A | 1.8 | PLASMODIUM FALCIPARUM | ENZYME 1.1.1.27 | BIK | | 204.179 |
2A94 | 1.5 | PLASMODIUM FALCIPARUM | ENZYME 1.1.1.27 | AP0 | | 666.469 |
4PLZ | 1.05 | PLASMODIUM FALCIPARUM | ENZYME 1.1.1.27 | NAI, OXM | | 665.441, 89.05 |
6R8G | 2 | PLASMODIUM FALCIPARUM | ENZYME 1.1.1.37 | NAD, JUT, NA | Kd = 172 uM | 663.425, 212.219, 22.99 |
3JQQ | 2.2 | PLASMODIUM FALCIPARUM | ENZYME 1.18.1.2 | FAD, A2P | Ki = 2.9 uM | 785.55, 427.201 |
3JQR | 2.3 | PLASMODIUM FALCIPARUM | ENZYME 1.18.1.2 | FAD | | 785.55 |
2B4R | 2.25 | PLASMODIUM FALCIPARUM | ENZYME 1.2.1.12 | NAD, GOL, AES | | 663.425, 92.094, 203.234 |
2B4T | 2.5 | PLASMODIUM FALCIPARUM | ENZYME 1.2.1.12 | NAD, AES | | 663.425, 203.234 |
1NHG | 2.43 | PLASMODIUM FALCIPARUM | ENZYME 1.3.1.9 | TCL, NAD | Ki = 0.05 uM | 289.542, 663.425 |
1NHW | 2.35 | PLASMODIUM FALCIPARUM | ENZYME 1.3.1.9 | TCC, NAD | Ki = 14.3 uM | 254.112, 663.425 |
1NNU | 2.5 | PLASMODIUM FALCIPARUM | ENZYME 1.3.1.9 | TCT, NAD | Ki = 0.15 uM | 286.71, 663.425 |
1UH5 | 2.2 | PLASMODIUM FALCIPARUM | ENZYME 1.3.1.9 | TCL, NAD | | 289.542, 663.425 |
1V35 | 2.5 | PLASMODIUM FALCIPARUM | ENZYME 1.3.1.9 | NAI | Ki = 96 pM | 665.441 |
1VRW | 2.4 | PLASMODIUM FALCIPARUM | ENZYME 1.3.1.9 | NAI | | 665.441 |
2FOI | 2.5 | PLASMODIUM FALCIPARUM | ENZYME 1.3.1.9 | NAD, JPA | ic50 = 440 nM | 663.425, 345.219 |
2NQ8 | 2.5 | PLASMODIUM FALCIPARUM | ENZYME 1.3.1.9 | ZID | ic50 = 320 nM | 768.519 |
2O2Y | 2.2 | PLASMODIUM FALCIPARUM | ENZYME 1.3.1.9 | TCL, SO4, NAD, CL | Ki = 0.4 nM | 289.542, 96.063, 663.425, 35.453 |
2OL4 | 2.26 | PLASMODIUM FALCIPARUM | ENZYME 1.3.1.9 | NAD, JPN | ic50 = 440 nM | 663.425, 373.272 |
2OOS | 2.1 | PLASMODIUM FALCIPARUM | ENZYME 1.3.1.9 | NAD, JPJ | ic50 = 76 nM | 663.425, 359.246 |
3AM3 | 2.5 | PLASMODIUM FALCIPARUM | ENZYME 1.3.1.9 | TCL, NAD | Ki = 28 nM | 289.542, 663.425 |
3AM4 | 2.3 | PLASMODIUM FALCIPARUM | ENZYME 1.3.1.9 | NAD, FT1 | ic50 = 97 nM | 663.425, 283.107 |
3AM5 | 2.05 | PLASMODIUM FALCIPARUM | ENZYME 1.3.1.9 | TCL, NAD | Ki = 38 nM | 289.542, 663.425 |
3LT0 | 1.96 | PLASMODIUM FALCIPARUM | ENZYME 1.3.1.9 | NAD, FT1 | Ki = 0.18 uM | 663.425, 283.107 |
3LT1 | 2.2 | PLASMODIUM FALCIPARUM | ENZYME 1.3.1.9 | NAD, FT2 | Ki = 0.32 uM | 663.425, 303.568 |
3LT2 | 2.5 | PLASMODIUM FALCIPARUM | ENZYME 1.3.1.9 | NAD, FT3 | Ki = 0.38 uM | 663.425, 285.123 |
3LT4 | 2.25 | PLASMODIUM FALCIPARUM | ENZYME 1.3.1.9 | NAD, FB4 | Ki = 0.1 uM | 663.425, 270.111 |
4IGE | 2.15 | PLASMODIUM FALCIPARUM | ENZYME 1.3.1.9 | GOL, NAD, CHJ, SO4 | ic50 = 0.25 uM | 92.094, 663.425, 302.709, 96.063 |
4IGF | 2.3 | PLASMODIUM FALCIPARUM | ENZYME 1.3.1.9 | CHV, GOL, NAD, SO4 | ic50 = 6 uM | 304.682, 92.094, 663.425, 96.063 |
1TV5 | 2.4 | PLASMODIUM FALCIPARUM | ENZYME 1.3.5.2 | SO4, ORO, N8E, FMN, A26 | Ki ~ 1000 nM | 96.063, 156.096, 350.491, 456.344, 270.207 |
3O8A | 2.3 | PLASMODIUM FALCIPARUM | ENZYME 1.3.5.2 | ORO, O8A, LDA, FMN | ic50 = 0.022 uM | 156.096, 381.372, 229.402, 456.344 |
4CQ8 | 1.98 | PLASMODIUM FALCIPARUM | ENZYME 1.3.5.2 | FMN, ORO, JBW | ic50 = 0.08 uM | 456.344, 156.096, 322.384 |
4ORM | 2.07 | PLASMODIUM FALCIPARUM | ENZYME 1.3.5.2 | FMN, 2V6, SO4, GOL, ORO | ic50 = 0.0018 uM | 456.344, 397.226, 96.063, 92.094, 156.096 |
4RX0 | 2.25 | PLASMODIUM FALCIPARUM | ENZYME 1.3.5.2 | FMN, GOL, D65, ORO | | 456.344, 92.094, 415.332, 156.096 |
5DEL | 2.2 | PLASMODIUM FALCIPARUM | ENZYME 1.3.5.2 | GOL, ORO, D59, LDA, FMN | ic50 = 16 nM | 92.094, 156.096, 325.147, 229.402, 456.344 |