1E7W | 1.75 | LEISHMANIA MAJOR | ENZYME 1.5.1.33 | NDP, MTX, EDO | | 745.421, 454.439, 62.068 |
1E92 | 2.2 | LEISHMANIA MAJOR | ENZYME 1.5.1.33 | NAP, HBI, EDO | | 743.405, 239.231, 62.068 |
1XTP | 1.94 | LEISHMANIA MAJOR | ENZYME TRANSFERASES | SAI | | 431.306 |
1Y63 | 1.7 | LEISHMANIA MAJOR | NON-ENZYME OTHER | NA, MN, BR, ADP | | 22.99, 54.938, 79.904, 427.201 |
2BF7 | 2.4 | LEISHMANIA MAJOR | ENZYME 1.5.1.33 | NAP, HBI, EDO | | 743.405, 239.231, 62.068 |
2CJE | 2.34 | LEISHMANIA MAJOR | ENZYME 3.6.1.23 | MG, DUN | | 24.305, 387.177 |
2HFU | 2 | LEISHMANIA MAJOR | ENZYME 2.7.1.36 | MEV | | 147.149 |
2OEG | 2.3 | LEISHMANIA MAJOR | ENZYME 2.7.7.9 | UPG | | 566.302 |
2R8Q | 1.5 | LEISHMANIA MAJOR | ENZYME 3.1.4.17 | ZN, MG, IBM | ic50 = 580 uM | 65.409, 24.305, 222.244 |
2WSA | 1.6 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MYA, 646 | Kd = 1 nM | 977.89, 495.425 |
2X77 | 2.1 | LEISHMANIA MAJOR | NON-ENZYME OTHER | GDP, MG | | 443.201, 24.305 |
2YAY | 1.86 | LEISHMANIA MAJOR | ENZYME 3.6.1.23 | DUP, CA | Kd = 0.8 uM | 467.157, 40.078 |
2YAZ | 2.4 | LEISHMANIA MAJOR | ENZYME 3.6.1.23 | UMP, SO4, MG | Kd = 7.3 uM | 308.182, 96.063, 24.305 |
2YB0 | 2.28 | LEISHMANIA MAJOR | ENZYME 3.6.1.23 | SO4, DUR | Kd = 140 uM | 96.063, 228.202 |
3H4V | 2.4 | LEISHMANIA MAJOR | ENZYME 1.5.1.33 | NAP, DVP | Ki = 0.1 uM | 743.405, 436.467 |
3KFL | 2 | LEISHMANIA MAJOR | ENZYME 6.1.1.10 | ZN, POP, MG, ME8, FMT, EDO | | 65.409, 175.959, 24.305, 478.417, 46.025, 62.068 |
3MHU | 1.85 | LEISHMANIA MAJOR | ENZYME 1.3.3.1 | SO4, GOL, FMN, EJZ | Ki = 212.93 uM | 96.063, 92.094, 456.344, 201.094 |
3MJY | 1.96 | LEISHMANIA MAJOR | ENZYME 1.3.3.1 | SO4, IJZ, GOL, FMN | Ki = 82.8 uM | 96.063, 171.111, 92.094, 456.344 |
3NGU | 2.29 | LEISHMANIA MAJOR | ENZYME 2.7.4.6 | ADP | | 427.201 |
3OH0 | 2.15 | LEISHMANIA MAJOR | ENZYME 2.7.7.64 | UTP, GOL | | 484.141, 92.094 |
3OH1 | 2.18 | LEISHMANIA MAJOR | ENZYME 2.7.7.64 | UGB, GOL | | 580.285, 92.094 |
3OH2 | 2.14 | LEISHMANIA MAJOR | ENZYME 2.7.7.64 | GOL, GDU | | 92.094, 566.302 |
3OH3 | 2.03 | LEISHMANIA MAJOR | ENZYME 2.7.7.64 | UAD, GOL | | 536.276, 92.094 |
3OH4 | 2.21 | LEISHMANIA MAJOR | ENZYME 2.7.7.64 | UPG, GOL | | 566.302, 92.094 |
3TQ0 | 1.9 | LEISHMANIA MAJOR | ENZYME 1.3.3.1 | SO4, NI, GOL, FUM, FMN | | 96.063, 58.693, 92.094, 116.072, 456.344 |
4A2Z | 2.31 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | VIQ, MYA, GOL, CL | | 337.437, 977.89, 92.094, 35.453 |
4A30 | 1.5 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | QMI, MYA, GOL, CL | | 413.118, 977.89, 92.094, 35.453 |
4A31 | 2.09 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MYA, GOL, 2CB | | 977.89, 92.094, 407.534 |
4A32 | 2.2 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MYA, GOL, 2CD | | 977.89, 92.094, 495.465 |
4A33 | 2.4 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | PS8, MYA | | 495.425, 977.89 |
4C7H | 1.4 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MYA, EN5, ENF, COA, MG, DMS | | 977.89, 511.741, 722.096, 767.534, 24.305, 78.133 |
4C7I | 1.3 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | JJ1, MG, DMS, MYA | | 512.726, 24.305, 78.133, 977.89 |
4CGL | 1.48 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MG, MYA, A6K | ic50 = 0.031 uM | 24.305, 977.89, 407.333 |
4CGM | 1.7 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MG, CWZ, MYA | ic50 = 1.02 uM | 24.305, 440.603, 977.89 |
4CGN | 1.69 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | 7AH, MG, MYA | ic50 = 0.55 uM | 351.417, 24.305, 977.89 |
4CGO | 1.3 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MYA, MG, 6KV | ic50 = 0.299 uM | 977.89, 24.305, 344.478 |
4CGP | 1.4 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MG, MYA | | 24.305, 977.89 |
4CYN | 1.4 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MG, A6M, MYA | Ki = 1406 nM | 24.305, 407.333, 977.89 |
4CYO | 1.5 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MG, UEK, MYA | Ki = 1.6 nM | 24.305, 558.471, 977.89 |
4CYP | 1.55 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MG, A62, MYA | | 24.305, 408.318, 977.89 |
4CYQ | 1.65 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MG, YAU, MYA | Ki = 59 nM | 24.305, 559.456, 977.89 |
4EF8 | 1.56 | LEISHMANIA MAJOR | ENZYME 1.3.3.1 | SO4, GOL, FMN, 0FI | | 96.063, 92.094, 456.344, 137.202 |
4EF9 | 1.6 | LEISHMANIA MAJOR | ENZYME 1.3.3.1 | SO4, GOL, FMN, 4NF | | 96.063, 92.094, 456.344, 182.2 |
4JZB | 1.9 | LEISHMANIA MAJOR | ENZYME 2.5.1.1 | IPE, NA, CA, P2H | Kd = 342.5 nM | 246.092, 22.99, 40.078, 360.216 |
4JZX | 1.8 | LEISHMANIA MAJOR | ENZYME 2.5.1.1 | 476, IPE, CA | Kd = 198.6 nM | 324.227, 246.092, 40.078 |
4K10 | 2.3 | LEISHMANIA MAJOR | ENZYME 2.5.1.1 | NI9, NA, PEG, ACT, MG, MES | Kd = 119.5 nM | 302.111, 22.99, 106.12, 59.044, 24.305, 195.237 |
4UCM | 2.32 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | X6W, MYA | Kd = 180 uM | 201.268, 977.89 |
4UCN | 1.8 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | JRB, MYA | | 177.246, 977.89 |
4UCP | 1.5 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | 9X3, MYA | Kd = 200 uM | 220.311, 977.89 |
4UXH | 2.4 | LEISHMANIA MAJOR | ENZYME 2.7.1.21 | T5A, ZN | ic50 = 1.1 uM | 891.354, 65.409 |