1Y63 | 1.7 | LEISHMANIA MAJOR | NON-ENZYME OTHER | NA, MN, BR, ADP | | 22.99, 54.938, 79.904, 427.201 |
4JZB | 1.9 | LEISHMANIA MAJOR | ENZYME 2.5.1.1 | IPE, NA, CA, P2H | Kd = 342.5 nM | 246.092, 22.99, 40.078, 360.216 |
4K10 | 2.3 | LEISHMANIA MAJOR | ENZYME 2.5.1.1 | MES, NI9, NA, PEG, ACT, MG | Kd = 119.5 nM | 195.237, 302.111, 22.99, 106.12, 59.044, 24.305 |
2CJE | 2.34 | LEISHMANIA MAJOR | ENZYME 3.6.1.23 | DUN, MG | | 387.177, 24.305 |
2R8Q | 1.5 | LEISHMANIA MAJOR | ENZYME 3.1.4.17 | IBM, ZN, MG | ic50 = 580 uM | 222.244, 65.409, 24.305 |
2X77 | 2.1 | LEISHMANIA MAJOR | NON-ENZYME OTHER | MG, GDP | | 24.305, 443.201 |
2YAZ | 2.4 | LEISHMANIA MAJOR | ENZYME 3.6.1.23 | UMP, SO4, MG | Kd = 7.3 uM | 308.182, 96.063, 24.305 |
3KFL | 2 | LEISHMANIA MAJOR | ENZYME 6.1.1.10 | ZN, POP, MG, ME8, FMT, EDO | | 65.409, 175.959, 24.305, 478.417, 46.025, 62.068 |
4C7H | 1.4 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | EN5, ENF, COA, MG, DMS, MYA | | 511.741, 722.096, 767.534, 24.305, 78.133, 977.89 |
4C7I | 1.3 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | JJ1, MG, DMS, MYA | | 512.726, 24.305, 78.133, 977.89 |
4CGL | 1.48 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MG, MYA, A6K | ic50 = 0.031 uM | 24.305, 977.89, 407.333 |
4CGM | 1.7 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MG, CWZ, MYA | ic50 = 1.02 uM | 24.305, 440.603, 977.89 |
4CGN | 1.69 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | 7AH, MG, MYA | ic50 = 0.55 uM | 351.417, 24.305, 977.89 |
4CGO | 1.3 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MYA, MG, 6KV | ic50 = 0.299 uM | 977.89, 24.305, 344.478 |
4CGP | 1.4 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MG, MYA | | 24.305, 977.89 |
4CYN | 1.4 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MG, A6M, MYA | Ki = 1406 nM | 24.305, 407.333, 977.89 |
4CYO | 1.5 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MG, UEK, MYA | Ki = 1.6 nM | 24.305, 558.471, 977.89 |
4CYP | 1.55 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MG, A62, MYA | | 24.305, 408.318, 977.89 |
4CYQ | 1.65 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MG, YAU, MYA | Ki = 59 nM | 24.305, 559.456, 977.89 |
5A27 | 1.37 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MG, TUT, MYA | Ki = 0.02 uM | 24.305, 401.887, 977.89 |
5A28 | 1.48 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | TUQ, MG, MYA | Ki = 0.01 uM | 401.89, 24.305, 977.89 |
5G20 | 1.52 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | DMS, QBY, MG, MYA | | 78.133, 408.513, 24.305, 977.89 |
5G21 | 1.5 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MG, YN4, MYA | | 24.305, 477.579, 977.89 |
6QD9 | 1.46 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MYA, MG, HWT | ic50 = 2.7 uM | 977.89, 24.305, 332.467 |
6QDA | 1.6 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MYA, MG, HWZ | ic50 = 0.24 uM | 977.89, 24.305, 338.45 |
6QDB | 1.4 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MYA, MG, HWQ | | 977.89, 24.305, 330.451 |
6QDC | 1.4 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MYA, MG, HXE | ic50 = 0.62 uM | 977.89, 24.305, 358.504 |
6QDD | 1.65 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MG, DMS, HXW, MYA | | 24.305, 78.133, 368.499, 977.89 |
6QDE | 1.45 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MYA, MG, HWW | | 977.89, 24.305, 388.573 |
6QDF | 1.49 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MYA, MG, HWN | ic50 = 1.2 uM | 977.89, 24.305, 388.573 |
6QDG | 1.98 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MYA, MG, HXN | | 977.89, 24.305, 405.335 |
6QDH | 1.45 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | HXQ, MYA, HZ5, HZ8, MG | | 500.66, 977.89, 203.262, 313.44, 24.305 |
4A2Z | 2.31 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | GOL, CL, VIQ, MYA | | 92.094, 35.453, 337.437, 977.89 |
4A30 | 1.5 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | QMI, MYA, GOL, CL | | 413.118, 977.89, 92.094, 35.453 |
2YAY | 1.86 | LEISHMANIA MAJOR | ENZYME 3.6.1.23 | DUP, CA | Kd = 0.8 uM | 467.157, 40.078 |
4JZX | 1.8 | LEISHMANIA MAJOR | ENZYME 2.5.1.1 | 476, IPE, CA | Kd = 198.6 nM | 324.227, 246.092, 40.078 |
6VJC | 1.8 | LEISHMANIA MAJOR | ENZYME 2.5.1.1 | PEG, ACT, IPR, 476, CA | | 106.12, 59.044, 248.108, 324.227, 40.078 |
6W7I | 2.1 | LEISHMANIA MAJOR | ENZYME 2.5.1.1 | ACT, PEG, IPR, 476, CA | | 59.044, 106.12, 248.108, 324.227, 40.078 |
6WW1 | 2.05 | LEISHMANIA MAJOR | ENZYME 2.5.1.1 | ACT, IPR, 476, CA | | 59.044, 248.108, 324.227, 40.078 |
5NTH | 2.5 | LEISHMANIA MAJOR | ENZYME 3.4.11.- | BB2, BCT, MN | | 385.498, 61.017, 54.938 |
3TQ0 | 1.9 | LEISHMANIA MAJOR | ENZYME 1.3.3.1 | SO4, NI, GOL, FUM, FMN | | 96.063, 58.693, 92.094, 116.072, 456.344 |
5L4N | 2.35 | LEISHMANIA MAJOR | ENZYME 1.5.1.33 | PEG, 6QT, EDO, GOL, ACT, PGE, NDP | ic50 = 57 uM | 106.12, 256.253, 62.068, 92.094, 59.044, 150.173, 745.421 |
1E7W | 1.75 | LEISHMANIA MAJOR | ENZYME 1.5.1.33 | NDP, MTX, EDO | | 745.421, 454.439, 62.068 |
1E92 | 2.2 | LEISHMANIA MAJOR | ENZYME 1.5.1.33 | NAP, HBI, EDO | | 743.405, 239.231, 62.068 |
2BF7 | 2.4 | LEISHMANIA MAJOR | ENZYME 1.5.1.33 | NAP, HBI, EDO | | 743.405, 239.231, 62.068 |
4UXH | 2.4 | LEISHMANIA MAJOR | ENZYME 2.7.1.21 | T5A, ZN | ic50 = 1.1 uM | 891.354, 65.409 |
3MHU | 1.85 | LEISHMANIA MAJOR | ENZYME 1.3.3.1 | EJZ, SO4, GOL, FMN | Ki = 212.93 uM | 201.094, 96.063, 92.094, 456.344 |
3MJY | 1.96 | LEISHMANIA MAJOR | ENZYME 1.3.3.1 | SO4, IJZ, GOL, FMN | Ki = 82.8 uM | 96.063, 171.111, 92.094, 456.344 |
3OH0 | 2.15 | LEISHMANIA MAJOR | ENZYME 2.7.7.64 | UTP, GOL | | 484.141, 92.094 |
3OH1 | 2.18 | LEISHMANIA MAJOR | ENZYME 2.7.7.64 | UGB, GOL | | 580.285, 92.094 |