5L2R | 2.05 | LEISHMANIA MAJOR | ENZYME 4.2.1.2 | PEG, SF4, GOL, MLA, LMR | ic50 = 9.8 mM | 106.12, 351.64, 92.094, 104.061, 134.087 |
2R8Q | 1.5 | LEISHMANIA MAJOR | ENZYME 3.1.4.17 | ZN, MG, IBM | ic50 = 580 uM | 65.409, 24.305, 222.244 |
3MHU | 1.85 | LEISHMANIA MAJOR | ENZYME 1.3.3.1 | SO4, GOL, FMN, EJZ | Ki = 212.93 uM | 96.063, 92.094, 456.344, 201.094 |
4UCP | 1.5 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | 9X3, MYA | Kd = 200 uM | 220.311, 977.89 |
4UCM | 2.32 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | X6W, MYA | Kd = 180 uM | 201.268, 977.89 |
2YB0 | 2.28 | LEISHMANIA MAJOR | ENZYME 3.6.1.23 | DUR, SO4 | Kd = 140 uM | 228.202, 96.063 |
3MJY | 1.96 | LEISHMANIA MAJOR | ENZYME 1.3.3.1 | SO4, IJZ, GOL, FMN | Ki = 82.8 uM | 96.063, 171.111, 92.094, 456.344 |
5L4N | 2.35 | LEISHMANIA MAJOR | ENZYME 1.5.1.33 | GOL, ACT, PGE, NDP, PEG, 6QT, EDO | ic50 = 57 uM | 92.094, 59.044, 150.173, 745.421, 106.12, 256.253, 62.068 |
6MSN | 1.59 | LEISHMANIA MAJOR | ENZYME 4.2.1.2 | JYD, SF4 | Ki = 8.9 uM | 150.153, 351.64 |
2YAZ | 2.4 | LEISHMANIA MAJOR | ENZYME 3.6.1.23 | UMP, SO4, MG | Kd = 7.3 uM | 308.182, 96.063, 24.305 |
6MSO | 2.05 | LEISHMANIA MAJOR | ENZYME 4.2.1.2 | JYD, SF4, 1PE, GOL | Ki = 3 uM | 150.153, 351.64, 238.278, 92.094 |
6QD9 | 1.46 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MYA, MG, HWT | ic50 = 2.7 uM | 977.89, 24.305, 332.467 |
6SWX | 1.95 | LEISHMANIA MAJOR | ENZYME 6.1.1.10 | LWN | ic50 = 2.06 uM | 348.307 |
4CYN | 1.4 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MG, A6M, MYA | Ki = 1406 nM | 24.305, 407.333, 977.89 |
6QDF | 1.49 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MYA, MG, HWN | ic50 = 1.2 uM | 977.89, 24.305, 388.573 |
4UXH | 2.4 | LEISHMANIA MAJOR | ENZYME 2.7.1.21 | T5A, ZN | ic50 = 1.1 uM | 891.354, 65.409 |
4CGM | 1.7 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MG, CWZ, MYA | ic50 = 1.02 uM | 24.305, 440.603, 977.89 |
2YAY | 1.86 | LEISHMANIA MAJOR | ENZYME 3.6.1.23 | DUP, CA | Kd = 0.8 uM | 467.157, 40.078 |
6QDC | 1.4 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MYA, MG, HXE | ic50 = 0.62 uM | 977.89, 24.305, 358.504 |
4CGN | 1.69 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | 7AH, MG, MYA | ic50 = 0.55 uM | 351.417, 24.305, 977.89 |
4JZB | 1.9 | LEISHMANIA MAJOR | ENZYME 2.5.1.1 | IPE, NA, CA, P2H | Kd = 342.5 nM | 246.092, 22.99, 40.078, 360.216 |
4CGO | 1.3 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MYA, MG, 6KV | ic50 = 0.299 uM | 977.89, 24.305, 344.478 |
6QDA | 1.6 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MYA, MG, HWZ | ic50 = 0.24 uM | 977.89, 24.305, 338.45 |
4JZX | 1.8 | LEISHMANIA MAJOR | ENZYME 2.5.1.1 | 476, IPE, CA | Kd = 198.6 nM | 324.227, 246.092, 40.078 |
4K10 | 2.3 | LEISHMANIA MAJOR | ENZYME 2.5.1.1 | MES, NI9, NA, PEG, ACT, MG | Kd = 119.5 nM | 195.237, 302.111, 22.99, 106.12, 59.044, 24.305 |