1E7W | 1.75 | LEISHMANIA MAJOR | ENZYME 1.5.1.33 | NDP, MTX, EDO | | 745.421, 454.439, 62.068 |
1E92 | 2.2 | LEISHMANIA MAJOR | ENZYME 1.5.1.33 | NAP, HBI, EDO | | 743.405, 239.231, 62.068 |
1XTP | 1.94 | LEISHMANIA MAJOR | ENZYME TRANSFERASES | SAI | | 431.306 |
1Y63 | 1.7 | LEISHMANIA MAJOR | NON-ENZYME OTHER | NA, MN, BR, ADP | | 22.99, 54.938, 79.904, 427.201 |
2BF7 | 2.4 | LEISHMANIA MAJOR | ENZYME 1.5.1.33 | NAP, HBI, EDO | | 743.405, 239.231, 62.068 |
2CJE | 2.34 | LEISHMANIA MAJOR | ENZYME 3.6.1.23 | DUN, MG | | 387.177, 24.305 |
2HFU | 2 | LEISHMANIA MAJOR | ENZYME 2.7.1.36 | MEV | | 147.149 |
2OEG | 2.3 | LEISHMANIA MAJOR | ENZYME 2.7.7.9 | UPG | | 566.302 |
2R8Q | 1.5 | LEISHMANIA MAJOR | ENZYME 3.1.4.17 | ZN, MG, IBM | ic50 = 580 uM | 65.409, 24.305, 222.244 |
2WSA | 1.6 | LEISHMANIA MAJOR | ENZYME 2.3.1.97 | MYA, 646 | Kd = 1 nM | 977.89, 495.425 |
2X77 | 2.1 | LEISHMANIA MAJOR | NON-ENZYME OTHER | MG, GDP | | 24.305, 443.201 |
2YAY | 1.86 | LEISHMANIA MAJOR | ENZYME 3.6.1.23 | DUP, CA | Kd = 0.8 uM | 467.157, 40.078 |
2YAZ | 2.4 | LEISHMANIA MAJOR | ENZYME 3.6.1.23 | UMP, SO4, MG | Kd = 7.3 uM | 308.182, 96.063, 24.305 |
2YB0 | 2.28 | LEISHMANIA MAJOR | ENZYME 3.6.1.23 | SO4, DUR | Kd = 140 uM | 96.063, 228.202 |
3H4V | 2.4 | LEISHMANIA MAJOR | ENZYME 1.5.1.33 | NAP, DVP | Ki = 0.1 uM | 743.405, 436.467 |
3KFL | 2 | LEISHMANIA MAJOR | ENZYME 6.1.1.10 | ZN, POP, MG, ME8, FMT, EDO | | 65.409, 175.959, 24.305, 478.417, 46.025, 62.068 |
3MHU | 1.85 | LEISHMANIA MAJOR | ENZYME 1.3.3.1 | SO4, GOL, FMN, EJZ | Ki = 212.93 uM | 96.063, 92.094, 456.344, 201.094 |
3MJY | 1.96 | LEISHMANIA MAJOR | ENZYME 1.3.3.1 | SO4, IJZ, GOL, FMN | Ki = 82.8 uM | 96.063, 171.111, 92.094, 456.344 |
3NGU | 2.29 | LEISHMANIA MAJOR | ENZYME 2.7.4.6 | ADP | | 427.201 |
3OH0 | 2.15 | LEISHMANIA MAJOR | ENZYME 2.7.7.64 | GOL, UTP | | 92.094, 484.141 |
3OH1 | 2.18 | LEISHMANIA MAJOR | ENZYME 2.7.7.64 | UGB, GOL | | 580.285, 92.094 |
3OH2 | 2.14 | LEISHMANIA MAJOR | ENZYME 2.7.7.64 | GOL, GDU | | 92.094, 566.302 |
3OH3 | 2.03 | LEISHMANIA MAJOR | ENZYME 2.7.7.64 | UAD, GOL | | 536.276, 92.094 |
3OH4 | 2.21 | LEISHMANIA MAJOR | ENZYME 2.7.7.64 | UPG, GOL | | 566.302, 92.094 |
3TQ0 | 1.9 | LEISHMANIA MAJOR | ENZYME 1.3.3.1 | SO4, NI, GOL, FUM, FMN | | 96.063, 58.693, 92.094, 116.072, 456.344 |