3AV9 | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, SER ALA LYS ILE ASP ASN LEU ASP, CL, ACY | ic50 = 435 uM | 96.063, 858.948, 35.453, 60.052 |
3AVA | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, CL, ALA LEU LYS ILE ASP ASN LEU ASP, ACY | ic50 = 39.7 uM | 96.063, 35.453, 885.03, 60.052 |
3AVB | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, SER LEU LYS ILE ASP ASN LEU ASP, CL, ACY | ic50 = 85.2 uM | 96.063, 901.029, 35.453, 60.052 |
3AVC | 1.77 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, SER ASP LYS ILE ASP ASN LEU ASP, CL, ACY | | 96.063, 901.949, 35.453, 60.052 |
3AVF | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, CL, ASP LEU LYS ILE ASP ASN LEU ASP, ACY | ic50 = 295 uM | 96.063, 35.453, 928.031, 60.052 |
3AVG | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, CL, ALA ASP LYS ILE ASP ASN LEU ASP, ACY | | 96.063, 35.453, 885.95, 60.052 |
3AVH | 1.88 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, CL, ALA ARG LYS ILE ASP ASN LEU ASP, ACY | | 96.063, 35.453, 929.067, 60.052 |
3AVI | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, SER LEU LYS ILE ASP ASN MET ASP, CL, ACY | | 96.063, 919.068, 35.453, 60.052 |
3AVJ | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, CL, ALA LEU LYS ILE ASP ASN MET ASP, ACY | | 96.063, 35.453, 903.069, 60.052 |
3AVK | 1.75 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | ACY, SO4, SER LEU LYS ILE ASP ASN GLU ASP, CL | | 60.052, 96.063, 915.976, 35.453 |
3AVL | 1.88 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, CL, ALA THR LYS ILE ASP ASN LEU ASP, ACY | ic50 = 65.8 uM | 96.063, 35.453, 872.975, 60.052 |
3AVM | 1.88 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, SER ARG LYS ILE ASP ASN LEU ASP, CL, ACY | | 96.063, 945.066, 35.453, 60.052 |
3AVN | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, SER HIS LYS ILE ASP ASN LEU ASP, CL, ACY | | 96.063, 925.011, 35.453, 60.052 |
3BC4 | 1.82 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | LLG, DMS | Ki = 4.5 uM | 229.274, 78.133 |
3BGB | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | LJG, CL | Ki = 0.9 uM | 525.728, 35.453 |
3BGC | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | LJH, CL | Ki = 9.6 uM | 593.76, 35.453 |
3CYW | 1.4 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | GOL, CL, 017 | Ki = 17 nM | 92.094, 35.453, 547.664 |
3D1X | 1.05 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ROC, GOL, CL | Ki = 2.2 nM | 670.841, 92.094, 35.453 |
3D1Y | 1.05 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ROC, NA, CL | Ki = 6 nM | 670.841, 22.99, 35.453 |
3D1Z | 1.3 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | CL, ACY, 017 | Ki = 1.6 nM | 35.453, 60.052, 547.664 |
3D20 | 1.05 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | CL, 017, NA | Ki = 5 nM | 35.453, 547.664, 22.99 |
3DJK | 1 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | NA, G55, CL | Ki = 26 pM | 22.99, 550.664, 35.453 |
3DK1 | 1.07 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | NA, G05, CL | Ki = 0.18 nM | 22.99, 576.701, 35.453 |
3DOL | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | PO4, GWI | | 94.971, 574.432 |
3I8W | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | GOL, CL, CB5 | Ki = 4.9 nM | 92.094, 35.453, 323.749 |
3K2P | 2.04 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.1.26.4 | MN, JTH | Kd = 6 uM | 54.938, 180.2 |
3KDB | 1.66 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | GOL, 006 | Kd = 0.14 nM | 92.094, 631.782 |
3KDC | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | JZP, GOL, CL | Kd = 0.52 nM | 672.618, 92.094, 35.453 |
3KDD | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | JZQ, GOL | Kd = 3.45 nM | 639.709, 92.094 |
3LAK | 2.3 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | SO4, KR1, CL | | 96.063, 421.424, 35.453 |
3LP1 | 2.23 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | NVP, MN, LP8 | | 266.298, 54.938, 246.262 |
3N3I | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ROC | | 670.841 |
3SPK | 1.24 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | TPV | ic50 = 3.02 nM | 602.664 |
3ST5 | 1.45 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | G89, CL | Ki = 5 pM | 576.701, 35.453 |
3T3C | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | SO4, BME, 017 | Ki = 0.059 nM | 96.063, 78.133, 547.664 |
3TKG | 1.36 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ROC, PHE, GOL, CL | | 670.841, 165.189, 92.094, 35.453 |
3TKW | 1.55 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | PHE, NA, GOL, CL, 017 | | 165.189, 22.99, 92.094, 35.453, 547.664 |
3TL9 | 1.32 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ROC, PHE, NA, GOL, CL | | 670.841, 165.189, 22.99, 92.094, 35.453 |
4DFG | 1.23 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | NA, CL, 0JV | Ki = 1.8 pM | 22.99, 35.453, 633.753 |
4DKO | 1.98 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | NAG, EPE, 0LM | Kd = 0.3 uM | 221.208, 238.305, 369.861 |
4DKP | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | NAG, EPE, 0LL | Kd = 1.9 uM | 221.208, 238.305, 347.771 |
4DKQ | 1.89 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | NAG, EPE, 0LK | Kd = 0.25 uM | 221.208, 238.305, 389.811 |
4DKR | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | NAG, EPE, 0LJ | Kd = 0.3 uM | 221.208, 238.305, 389.811 |
4DMN | 2.45 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, ARS, 0L9 | ic50 = 2.3 uM | 96.063, 74.922, 420.684 |
4E1M | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | TQ2 | ic50 = 215 nM | 377.476 |
4E1N | 2 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | TQX | ic50 = 19 nM | 437.503 |
4FE6 | 2 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | 0TQ | Ki < 0.1 nM | 642.763 |
4G1Q | 1.51 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | MG, EDO, SO4, T27 | | 24.305, 62.068, 96.063, 366.419 |
4HDB | 1.49 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | G52, CL, NA | Ki = 8.9 nM | 604.712, 35.453, 22.99 |
4HDF | 1.29 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | G52, CL | Ki = 3.2 nM | 604.712, 35.453 |