3N3I | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ROC | | 670.841 |
4Q5M | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ROC | | 670.841 |
4FE6 | 2 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | 0TQ | Ki < 0.1 nM | 642.763 |
4HEG | 1.46 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | G52 | Ki = 1.2 nM | 604.712 |
3SPK | 1.24 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | TPV | ic50 = 3.02 nM | 602.664 |
4I8W | 1.96 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | G07 | Ki = 12.7 pM | 576.658 |
4I8Z | 1.75 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | G08 | Ki = 8.9 pM | 575.674 |
4E1N | 2 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | TQX | ic50 = 19 nM | 437.503 |
4E1M | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | TQ2 | ic50 = 215 nM | 377.476 |
5HGP | 1.95 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | BHC | | 342.169 |
4DKO | 1.98 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | NAG, EPE, 0LM | Kd = 0.3 uM | 221.208, 238.305, 369.861 |
4DKP | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | NAG, EPE, 0LL | Kd = 1.9 uM | 221.208, 238.305, 347.771 |
4DKQ | 1.89 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | NAG, EPE, 0LK | Kd = 0.25 uM | 221.208, 238.305, 389.811 |
4DKR | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | NAG, EPE, 0LJ | Kd = 0.3 uM | 221.208, 238.305, 389.811 |
4I54 | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | NAG, EPE, 1C1 | Kd = 110 nM | 221.208, 238.305, 404.846 |
4NYF | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | 4BI, CD | Kd = 49 nM | 383.868, 112.411 |
4ID1 | 1.87 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, LF0 | | 96.063, 405.486 |
4JLH | 2.09 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, 0L9 | ic50 = 15.6 uM | 96.063, 420.684 |
4O0J | 2.05 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | LF8, SO4 | ic50 = 13 uM | 451.985, 96.063 |
4O55 | 2.24 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, LF9 | ic50 = 5.03 uM | 96.063, 463.956 |
4O5B | 2.37 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, LF9 | | 96.063, 463.956 |
4OJR | 1.82 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, 2SQ, CAC | | 96.063, 453.503, 136.989 |
3DOL | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | PO4, GWI | | 94.971, 574.432 |
3KDB | 1.66 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | GOL, 006 | Kd = 0.14 nM | 92.094, 631.782 |
3KDD | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | JZQ, GOL | Kd = 3.45 nM | 639.709, 92.094 |
3BC4 | 1.82 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | LLG, DMS | Ki = 4.5 uM | 229.274, 78.133 |
3T3C | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | SO4, BME, 017 | Ki = 0.059 nM | 96.063, 78.133, 547.664 |
4IG0 | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | 1FG, DMS | | 362.425, 78.133 |
4IG3 | 1.95 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | J94, T27, DMS | | 382.387, 366.419, 78.133 |
4KFB | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | T27, DMS, 1QP | | 366.419, 78.133, 190.199 |
4DMN | 2.45 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, ARS, 0L9 | ic50 = 2.3 uM | 96.063, 74.922, 420.684 |
4KO0 | 1.95 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | SO4, JLJ, EDO | | 96.063, 310.35, 62.068 |
4OBD | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ARG PRO GLY ASN PHE PHE GLN ASN ARG PRO, EDO, GOL | | 851.919, 62.068, 92.094 |
4OBG | 1.78 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ARG PRO GLY ASN PHE LEU GLN SER ARG PRO, PO4, EDO, GOL | | 975.119, 94.971, 62.068, 92.094 |
4K4P | 2.31 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | NO3, 3TL | | 62.005, 909.077 |
4K4R | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | 27B, BR, NO3, 3TL, DMS | | 251.076, 79.904, 62.005, 909.077, 78.133 |
4OBF | 1.68 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ACT, PO4, GOL, ARG PRO GLY ASN PHE LEU GLN ASN ARG PRO, EDO | | 59.044, 94.971, 92.094, 789.916, 62.068 |
4OBH | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ACT, PO4, GOL, EDO, ARG PRO GLY ASN PHE PHE GLN SER ARG PRO | | 59.044, 94.971, 92.094, 62.068, 938.057 |
4OBJ | 1.75 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | GOL, ARG PRO GLY ASN PHE LEU GLN ASN ARG PRO, ACT, EDO | | 92.094, 789.916, 59.044, 62.068 |
4OBK | 1.65 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ACT, EDO, ARG PRO GLY ASN PHE PHE GLN ASN ARG PRO, GOL | | 59.044, 62.068, 851.919, 92.094 |
3K2P | 2.04 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.1.26.4 | JTH, MN | Kd = 6 uM | 180.2, 54.938 |
3LP1 | 2.23 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | NVP, MN, LP8 | | 266.298, 54.938, 246.262 |
4QAG | 1.71 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.1.26.4 | MN, F95 | ic50 = 4.8 uM | 54.938, 236.178 |
4I53 | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | FMT, ASN ILE THR GLY LEU LEU LEU LEU ARG ASP, 1C1, NAG | Kd = 110 nM | 46.025, 404.846, 221.208 |
3AV9 | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, SER ALA LYS ILE ASP ASN LEU ASP, CL, ACY | ic50 = 435 uM | 96.063, 858.948, 35.453, 60.052 |
3AVA | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | ALA LEU LYS ILE ASP ASN LEU ASP, ACY, SO4, CL | ic50 = 39.7 uM | 885.03, 60.052, 96.063, 35.453 |
3AVB | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, SER LEU LYS ILE ASP ASN LEU ASP, CL, ACY | ic50 = 85.2 uM | 96.063, 901.029, 35.453, 60.052 |
3AVC | 1.77 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, SER ASP LYS ILE ASP ASN LEU ASP, CL, ACY | | 96.063, 901.949, 35.453, 60.052 |
3AVF | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, CL, ASP LEU LYS ILE ASP ASN LEU ASP, ACY | ic50 = 295 uM | 96.063, 35.453, 928.031, 60.052 |
3AVG | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, CL, ALA ASP LYS ILE ASP ASN LEU ASP, ACY | | 96.063, 35.453, 885.95, 60.052 |