3AV9 | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, SER ALA LYS ILE ASP ASN LEU ASP, CL, ACY | ic50 = 435 uM | 96.063, 858.948, 35.453, 60.052 |
3AVF | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, CL, ASP LEU LYS ILE ASP ASN LEU ASP, ACY | ic50 = 295 uM | 96.063, 35.453, 928.031, 60.052 |
3AVB | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, SER LEU LYS ILE ASP ASN LEU ASP, CL, ACY | ic50 = 85.2 uM | 96.063, 901.029, 35.453, 60.052 |
3AVL | 1.88 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, CL, ALA THR LYS ILE ASP ASN LEU ASP, ACY | ic50 = 65.8 uM | 96.063, 35.453, 872.975, 60.052 |
3AVA | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, CL, ALA LEU LYS ILE ASP ASN LEU ASP, ACY | ic50 = 39.7 uM | 96.063, 35.453, 885.03, 60.052 |
4JLH | 2.09 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, 0L9 | ic50 = 15.6 uM | 96.063, 420.684 |
4O0J | 2.05 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | LF8, SO4 | ic50 = 13 uM | 451.985, 96.063 |
3BGC | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | LJH, CL | Ki = 9.6 uM | 593.76, 35.453 |
3K2P | 2.04 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.1.26.4 | MN, JTH | Kd = 6 uM | 54.938, 180.2 |
4O55 | 2.24 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, LF9 | ic50 = 5.03 uM | 96.063, 463.956 |
4QAG | 1.71 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.1.26.4 | MN, F95 | ic50 = 4.8 uM | 54.938, 236.178 |
3BC4 | 1.82 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | LLG, DMS | Ki = 4.5 uM | 229.274, 78.133 |
4DMN | 2.45 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, ARS, 0L9 | ic50 = 2.3 uM | 96.063, 74.922, 420.684 |
4DKP | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | NAG, EPE, 0LL | Kd = 1.9 uM | 221.208, 238.305, 347.771 |
3BGB | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | LJG, CL | Ki = 0.9 uM | 525.728, 35.453 |
4DKO | 1.98 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | NAG, EPE, 0LM | Kd = 0.3 uM | 221.208, 238.305, 369.861 |
4DKR | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | NAG, EPE, 0LJ | Kd = 0.3 uM | 221.208, 238.305, 389.811 |
4DKQ | 1.89 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | NAG, EPE, 0LK | Kd = 0.25 uM | 221.208, 238.305, 389.811 |
4E1M | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | TQ2 | ic50 = 215 nM | 377.476 |
4I53 | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | 1C1, NAG, FMT, ASN ILE THR GLY LEU LEU LEU LEU ARG ASP | Kd = 110 nM | 404.846, 221.208, 46.025 |
4I54 | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | EPE, 1C1, NAG | Kd = 110 nM | 238.305, 404.846, 221.208 |
4NYF | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | CD, 4BI | Kd = 49 nM | 112.411, 383.868 |
6UL5 | 2.23 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | QAG, MG, EDO, SO4 | ic50 = 36.2 nM | 441.48, 24.305, 62.068, 96.063 |
4HDP | 1.22 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | NA, G52, CL | Ki = 30.9 nM | 22.99, 604.712, 35.453 |
4E1N | 2 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | TQX | ic50 = 19 nM | 437.503 |
3CYW | 1.4 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | GOL, CL, 017 | Ki = 17 nM | 92.094, 35.453, 547.664 |
4HDB | 1.49 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | G52, CL, NA | Ki = 8.9 nM | 604.712, 35.453, 22.99 |
3D1Y | 1.05 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ROC, NA, CL | Ki = 6 nM | 670.841, 22.99, 35.453 |
3D20 | 1.05 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | CL, 017, NA | Ki = 5 nM | 35.453, 547.664, 22.99 |
3I8W | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | GOL, CL, CB5 | Ki = 4.9 nM | 92.094, 35.453, 323.749 |
4HE9 | 1.06 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | G52, CL, NA | Ki = 3.5 nM | 604.712, 35.453, 22.99 |
3KDD | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | JZQ, GOL | Kd = 3.45 nM | 639.709, 92.094 |
4HDF | 1.29 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | G52, CL | Ki = 3.2 nM | 604.712, 35.453 |
3SPK | 1.24 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | TPV | ic50 = 3.02 nM | 602.664 |
3D1X | 1.05 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ROC, GOL, CL | Ki = 2.2 nM | 670.841, 92.094, 35.453 |
3D1Z | 1.3 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | CL, ACY, 017 | Ki = 1.6 nM | 35.453, 60.052, 547.664 |
4HEG | 1.46 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | G52 | Ki = 1.2 nM | 604.712 |
3KDC | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | CL, JZP, GOL | Kd = 0.52 nM | 35.453, 672.618, 92.094 |
4ZIP | 1.11 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | G64, GOL, NA, CL | Ki = 0.21 nM | 690.849, 92.094, 22.99, 35.453 |
3DK1 | 1.07 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | NA, G05, CL | Ki = 0.18 nM | 22.99, 576.701, 35.453 |
3KDB | 1.66 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | GOL, 006 | Kd = 0.14 nM | 92.094, 631.782 |
4FE6 | 2 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | 0TQ | Ki < 0.1 nM | 642.763 |
3T3C | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | SO4, BME, 017 | Ki = 0.059 nM | 96.063, 78.133, 547.664 |
3DJK | 1 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | NA, G55, CL | Ki = 26 pM | 22.99, 550.664, 35.453 |
4I8W | 1.96 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | G07 | Ki = 12.7 pM | 576.658 |
4I8Z | 1.75 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | G08 | Ki = 8.9 pM | 575.674 |
3ST5 | 1.45 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | G89, CL | Ki = 5 pM | 576.701, 35.453 |
4DFG | 1.23 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | NA, CL, 0JV | Ki = 1.8 pM | 22.99, 35.453, 633.753 |
3AVC | 1.77 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, SER ASP LYS ILE ASP ASN LEU ASP, CL, ACY | | 96.063, 901.949, 35.453, 60.052 |
3AVG | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, CL, ALA ASP LYS ILE ASP ASN LEU ASP, ACY | | 96.063, 35.453, 885.95, 60.052 |