3AV9 | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, SER ALA LYS ILE ASP ASN LEU ASP, CL, ACY | ic50 = 435 uM | 96.063, 858.948, 35.453, 60.052 |
3AVA | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, CL, ALA LEU LYS ILE ASP ASN LEU ASP, ACY | ic50 = 39.7 uM | 96.063, 35.453, 885.03, 60.052 |
3AVB | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, SER LEU LYS ILE ASP ASN LEU ASP, CL, ACY | ic50 = 85.2 uM | 96.063, 901.029, 35.453, 60.052 |
3AVC | 1.77 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, SER ASP LYS ILE ASP ASN LEU ASP, CL, ACY | | 96.063, 901.949, 35.453, 60.052 |
3AVF | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, CL, ASP LEU LYS ILE ASP ASN LEU ASP, ACY | ic50 = 295 uM | 96.063, 35.453, 928.031, 60.052 |
3AVG | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, CL, ALA ASP LYS ILE ASP ASN LEU ASP, ACY | | 96.063, 35.453, 885.95, 60.052 |
3AVH | 1.88 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, CL, ALA ARG LYS ILE ASP ASN LEU ASP, ACY | | 96.063, 35.453, 929.067, 60.052 |
3AVI | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, SER LEU LYS ILE ASP ASN MET ASP, CL, ACY | | 96.063, 919.068, 35.453, 60.052 |
3AVJ | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, CL, ALA LEU LYS ILE ASP ASN MET ASP, ACY | | 96.063, 35.453, 903.069, 60.052 |
3AVK | 1.75 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | ACY, SO4, SER LEU LYS ILE ASP ASN GLU ASP, CL | | 60.052, 96.063, 915.976, 35.453 |
3AVL | 1.88 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, CL, ALA THR LYS ILE ASP ASN LEU ASP, ACY | ic50 = 65.8 uM | 96.063, 35.453, 872.975, 60.052 |
3AVM | 1.88 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | CL, SO4, ACY, SER ARG LYS ILE ASP ASN LEU ASP | | 35.453, 96.063, 60.052, 945.066 |
3AVN | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, SER HIS LYS ILE ASP ASN LEU ASP, CL, ACY | | 96.063, 925.011, 35.453, 60.052 |
3BC4 | 1.82 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | LLG, DMS | Ki = 4.5 uM | 229.274, 78.133 |
3BGB | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | LJG, CL | Ki = 0.9 uM | 525.728, 35.453 |
3BGC | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | LJH, CL | Ki = 9.6 uM | 593.76, 35.453 |
3CYW | 1.4 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | 017, GOL, CL | Ki = 17 nM | 547.664, 92.094, 35.453 |
3D1X | 1.05 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ROC, GOL, CL | Ki = 2.2 nM | 670.841, 92.094, 35.453 |
3D1Y | 1.05 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ROC, NA, CL | Ki = 6 nM | 670.841, 22.99, 35.453 |
3D1Z | 1.3 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | CL, ACY, 017 | Ki = 1.6 nM | 35.453, 60.052, 547.664 |
3D20 | 1.05 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | CL, 017, NA | Ki = 5 nM | 35.453, 547.664, 22.99 |
3DJK | 1 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | NA, G55, CL | Ki = 26 pM | 22.99, 550.664, 35.453 |
3DK1 | 1.07 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | NA, G05, CL | Ki = 0.18 nM | 22.99, 576.701, 35.453 |
3DOL | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | PO4, GWI | | 94.971, 574.432 |
3I8W | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | GOL, CL, CB5 | Ki = 4.9 nM | 92.094, 35.453, 323.749 |
3K2P | 2.04 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.1.26.4 | MN, JTH | Kd = 6 uM | 54.938, 180.2 |
3KDB | 1.66 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | GOL, 006 | Kd = 0.14 nM | 92.094, 631.782 |
3KDC | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | JZP, GOL, CL | Kd = 0.52 nM | 672.618, 92.094, 35.453 |
3KDD | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | JZQ, GOL | Kd = 3.45 nM | 639.709, 92.094 |
3LAK | 2.3 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | SO4, KR1, CL | | 96.063, 421.424, 35.453 |
3LP1 | 2.23 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | NVP, MN, LP8 | | 266.298, 54.938, 246.262 |
3N3I | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ROC | | 670.841 |
3SPK | 1.24 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | TPV | ic50 = 3.02 nM | 602.664 |
3ST5 | 1.45 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | G89, CL | Ki = 5 pM | 576.701, 35.453 |
3T3C | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | SO4, BME, 017 | Ki = 0.059 nM | 96.063, 78.133, 547.664 |
3TKG | 1.36 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ROC, PHE, GOL, CL | | 670.841, 165.189, 92.094, 35.453 |
3TKW | 1.55 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | PHE, NA, GOL, CL, 017 | | 165.189, 22.99, 92.094, 35.453, 547.664 |
3TL9 | 1.32 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ROC, PHE, NA, GOL, CL | | 670.841, 165.189, 22.99, 92.094, 35.453 |
4DFG | 1.23 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | NA, CL, 0JV | Ki = 1.8 pM | 22.99, 35.453, 633.753 |
4DKO | 1.98 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | NAG, EPE, 0LM | Kd = 0.3 uM | 221.208, 238.305, 369.861 |
4DKP | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | NAG, EPE, 0LL | Kd = 1.9 uM | 221.208, 238.305, 347.771 |
4DKQ | 1.89 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | NAG, EPE, 0LK | Kd = 0.25 uM | 221.208, 238.305, 389.811 |
4DKR | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | NAG, EPE, 0LJ | Kd = 0.3 uM | 221.208, 238.305, 389.811 |
4DMN | 2.45 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, ARS, 0L9 | ic50 = 2.3 uM | 96.063, 74.922, 420.684 |
4E1M | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | TQ2 | ic50 = 215 nM | 377.476 |
4E1N | 2 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | TQX | ic50 = 19 nM | 437.503 |
4FE6 | 2 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | 0TQ | Ki < 0.1 nM | 642.763 |
4G1Q | 1.51 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | MG, EDO, SO4, T27 | | 24.305, 62.068, 96.063, 366.419 |
4HDB | 1.49 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | G52, CL, NA | Ki = 8.9 nM | 604.712, 35.453, 22.99 |
4HDF | 1.29 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | G52, CL | Ki = 3.2 nM | 604.712, 35.453 |
4HDP | 1.22 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | NA, G52, CL | Ki = 30.9 nM | 22.99, 604.712, 35.453 |
4HE9 | 1.06 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | G52, CL, NA | Ki = 3.5 nM | 604.712, 35.453, 22.99 |
4HEG | 1.46 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | G52 | Ki = 1.2 nM | 604.712 |
4I53 | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | FMT, ASN ILE THR GLY LEU LEU LEU LEU ARG ASP, 1C1, NAG | Kd = 110 nM | 46.025, 404.846, 221.208 |
4I54 | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | EPE, 1C1, NAG | Kd = 110 nM | 238.305, 404.846, 221.208 |
4I8W | 1.96 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | G07 | Ki = 12.7 pM | 576.658 |
4I8Z | 1.75 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | G08 | Ki = 8.9 pM | 575.674 |
4ICL | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | MG, T27, DMS, 14N | | 24.305, 366.419, 78.133, 220.268 |
4ID1 | 1.87 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, LF0 | | 96.063, 405.486 |
4ID5 | 1.95 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | MG, T27, 1FF, DMS | | 24.305, 366.419, 202.209, 78.133 |
4IDK | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | T27, 1FE, DMS, MG | | 366.419, 206.201, 78.133, 24.305 |
4IFV | 2.05 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | DMS, T27, MG, FMQ | | 78.133, 366.419, 24.305, 206.216 |
4IFY | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | MG, 1FD, T27, DMS | | 24.305, 191.15, 366.419, 78.133 |
4IG0 | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | 1FG, DMS | | 362.425, 78.133 |
4IG3 | 1.95 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | T27, DMS, J94 | | 366.419, 78.133, 382.387 |
4JLH | 2.09 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, 0L9 | ic50 = 15.6 uM | 96.063, 420.684 |
4K4P | 2.31 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | NO3, 3TL | | 62.005, 909.077 |
4K4R | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | 27B, BR, NO3, 3TL, DMS | | 251.076, 79.904, 62.005, 909.077, 78.133 |
4KFB | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | T27, DMS, 1QP | | 366.419, 78.133, 190.199 |
4KO0 | 1.95 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | SO4, JLJ, EDO | | 96.063, 310.35, 62.068 |
4NX4 | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | CL, ZN, JPR | | 35.453, 65.409, 381.92 |
4NYF | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | CD, 4BI | Kd = 49 nM | 112.411, 383.868 |
4O0J | 2.05 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | LF8, SO4 | ic50 = 13 uM | 451.985, 96.063 |
4O55 | 2.24 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, LF9 | ic50 = 5.03 uM | 96.063, 463.956 |
4O5B | 2.37 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, LF9 | | 96.063, 463.956 |
4OBD | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ARG PRO GLY ASN PHE PHE GLN ASN ARG PRO, EDO, GOL | | 851.919, 62.068, 92.094 |
4OBF | 1.68 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ACT, PO4, GOL, ARG PRO GLY ASN PHE LEU GLN ASN ARG PRO, EDO | | 59.044, 94.971, 92.094, 789.916, 62.068 |
4OBG | 1.78 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ARG PRO GLY ASN PHE LEU GLN SER ARG PRO, PO4, EDO, GOL | | 975.119, 94.971, 62.068, 92.094 |
4OBH | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ACT, PO4, GOL, EDO, ARG PRO GLY ASN PHE PHE GLN SER ARG PRO | | 59.044, 94.971, 92.094, 62.068, 938.057 |
4OBJ | 1.75 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | GOL, ARG PRO GLY ASN PHE LEU GLN ASN ARG PRO, ACT, EDO | | 92.094, 789.916, 59.044, 62.068 |
4OBK | 1.65 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ACT, EDO, ARG PRO GLY ASN PHE PHE GLN ASN ARG PRO, GOL | | 59.044, 62.068, 851.919, 92.094 |
4OJR | 1.82 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.7 | SO4, 2SQ, CAC | | 96.063, 453.503, 136.989 |
4Q5M | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | ROC | | 670.841 |
4QAG | 1.71 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.1.26.4 | F95, MN | ic50 = 4.8 uM | 236.178, 54.938 |
4ZIP | 1.11 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 3.4.23.16 | G64, GOL, NA, CL | Ki = 0.21 nM | 690.849, 92.094, 22.99, 35.453 |
5HGP | 1.95 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | NON-ENZYME OTHER | BHC | | 342.169 |
6UL5 | 2.23 | HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 | ENZYME 2.7.7.49 | QAG, MG, EDO, SO4 | ic50 = 36.2 nM | 441.48, 24.305, 62.068, 96.063 |