Searching for Source: 'HUMAN IMMUNODEFICIENCY VIRUS TYPE 1';
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3AV9 1.7 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.7 SO4, SER ALA LYS ILE ASP ASN LEU ASP, CL, ACY ic50 = 435 uM 96.063, 858.948, 35.453, 60.052
3AVA 1.7 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.7 SO4, CL, ALA LEU LYS ILE ASP ASN LEU ASP, ACY ic50 = 39.7 uM 96.063, 35.453, 885.03, 60.052
3AVB 1.85 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.7 SO4, SER LEU LYS ILE ASP ASN LEU ASP, CL, ACY ic50 = 85.2 uM 96.063, 901.029, 35.453, 60.052
3AVC 1.77 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.7 SO4, SER ASP LYS ILE ASP ASN LEU ASP, CL, ACY 96.063, 901.949, 35.453, 60.052
3AVF 1.7 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.7 SO4, CL, ASP LEU LYS ILE ASP ASN LEU ASP, ACY ic50 = 295 uM 96.063, 35.453, 928.031, 60.052
3AVG 1.7 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.7 SO4, CL, ALA ASP LYS ILE ASP ASN LEU ASP, ACY 96.063, 35.453, 885.95, 60.052
3AVH 1.88 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.7 SO4, CL, ALA ARG LYS ILE ASP ASN LEU ASP, ACY 96.063, 35.453, 929.067, 60.052
3AVI 1.7 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.7 SO4, SER LEU LYS ILE ASP ASN MET ASP, CL, ACY 96.063, 919.068, 35.453, 60.052
3AVJ 1.7 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.7 SO4, CL, ALA LEU LYS ILE ASP ASN MET ASP, ACY 96.063, 35.453, 903.069, 60.052
3AVK 1.75 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.7 ACY, SO4, SER LEU LYS ILE ASP ASN GLU ASP, CL 60.052, 96.063, 915.976, 35.453
3AVL 1.88 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.7 SO4, CL, ALA THR LYS ILE ASP ASN LEU ASP, ACY ic50 = 65.8 uM 96.063, 35.453, 872.975, 60.052
3AVM 1.88 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.7 CL, SO4, ACY, SER ARG LYS ILE ASP ASN LEU ASP 35.453, 96.063, 60.052, 945.066
3AVN 2.1 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.7 SO4, SER HIS LYS ILE ASP ASN LEU ASP, CL, ACY 96.063, 925.011, 35.453, 60.052
3BC4 1.82 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 LLG, DMS Ki = 4.5 uM 229.274, 78.133
3BGB 1.9 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 LJG, CL Ki = 0.9 uM 525.728, 35.453
3BGC 1.8 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 LJH, CL Ki = 9.6 uM 593.76, 35.453
3CYW 1.4 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 017, GOL, CL Ki = 17 nM 547.664, 92.094, 35.453
3D1X 1.05 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 ROC, GOL, CL Ki = 2.2 nM 670.841, 92.094, 35.453
3D1Y 1.05 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 ROC, NA, CL Ki = 6 nM 670.841, 22.99, 35.453
3D1Z 1.3 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 CL, ACY, 017 Ki = 1.6 nM 35.453, 60.052, 547.664
3D20 1.05 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 CL, 017, NA Ki = 5 nM 35.453, 547.664, 22.99
3DJK 1 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 NA, G55, CL Ki = 26 pM 22.99, 550.664, 35.453
3DK1 1.07 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 NA, G05, CL Ki = 0.18 nM 22.99, 576.701, 35.453
3DOL 2.5 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.49 PO4, GWI 94.971, 574.432
3I8W 1.7 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 GOL, CL, CB5 Ki = 4.9 nM 92.094, 35.453, 323.749
3K2P 2.04 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.1.26.4 MN, JTH Kd = 6 uM 54.938, 180.2
3KDB 1.66 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 GOL, 006 Kd = 0.14 nM 92.094, 631.782
3KDC 2.2 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 JZP, GOL, CL Kd = 0.52 nM 672.618, 92.094, 35.453
3KDD 1.8 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 JZQ, GOL Kd = 3.45 nM 639.709, 92.094
3LAK 2.3 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.49 SO4, KR1, CL 96.063, 421.424, 35.453
3LP1 2.23 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.49 NVP, MN, LP8 266.298, 54.938, 246.262
3N3I 2.5 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 ROC 670.841
3SPK 1.24 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 TPV ic50 = 3.02 nM 602.664
3ST5 1.45 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 G89, CL Ki = 5 pM 576.701, 35.453
3T3C 2.1 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 SO4, BME, 017 Ki = 0.059 nM 96.063, 78.133, 547.664
3TKG 1.36 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 ROC, PHE, GOL, CL 670.841, 165.189, 92.094, 35.453
3TKW 1.55 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 PHE, NA, GOL, CL, 017 165.189, 22.99, 92.094, 35.453, 547.664
3TL9 1.32 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 ROC, PHE, NA, GOL, CL 670.841, 165.189, 22.99, 92.094, 35.453
4DFG 1.23 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 NA, CL, 0JV Ki = 1.8 pM 22.99, 35.453, 633.753
4DKO 1.98 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 NON-ENZYME OTHER NAG, EPE, 0LM Kd = 0.3 uM 221.208, 238.305, 369.861
4DKP 1.8 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 NON-ENZYME OTHER NAG, EPE, 0LL Kd = 1.9 uM 221.208, 238.305, 347.771
4DKQ 1.89 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 NON-ENZYME OTHER NAG, EPE, 0LK Kd = 0.25 uM 221.208, 238.305, 389.811
4DKR 1.8 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 NON-ENZYME OTHER NAG, EPE, 0LJ Kd = 0.3 uM 221.208, 238.305, 389.811
4DMN 2.45 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.7 SO4, ARS, 0L9 ic50 = 2.3 uM 96.063, 74.922, 420.684
4E1M 1.9 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.49 TQ2 ic50 = 215 nM 377.476
4E1N 2 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.7 TQX ic50 = 19 nM 437.503
4FE6 2 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 0TQ Ki < 0.1 nM 642.763
4G1Q 1.51 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.49 MG, EDO, SO4, T27 24.305, 62.068, 96.063, 366.419
4HDB 1.49 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 G52, CL, NA Ki = 8.9 nM 604.712, 35.453, 22.99
4HDF 1.29 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 G52, CL Ki = 3.2 nM 604.712, 35.453
4HDP 1.22 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 NA, G52, CL Ki = 30.9 nM 22.99, 604.712, 35.453
4HE9 1.06 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 G52, CL, NA Ki = 3.5 nM 604.712, 35.453, 22.99
4HEG 1.46 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 G52 Ki = 1.2 nM 604.712
4I53 2.5 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 NON-ENZYME OTHER FMT, ASN ILE THR GLY LEU LEU LEU LEU ARG ASP, 1C1, NAG Kd = 110 nM 46.025, 404.846, 221.208
4I54 2.5 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 NON-ENZYME OTHER EPE, 1C1, NAG Kd = 110 nM 238.305, 404.846, 221.208
4I8W 1.96 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 G07 Ki = 12.7 pM 576.658
4I8Z 1.75 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 G08 Ki = 8.9 pM 575.674
4ICL 1.8 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.49 MG, T27, DMS, 14N 24.305, 366.419, 78.133, 220.268
4ID1 1.87 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.7 SO4, LF0 96.063, 405.486
4ID5 1.95 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.49 MG, T27, 1FF, DMS 24.305, 366.419, 202.209, 78.133
4IDK 2.1 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.49 T27, 1FE, DMS, MG 366.419, 206.201, 78.133, 24.305
4IFV 2.05 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.49 DMS, T27, MG, FMQ 78.133, 366.419, 24.305, 206.216
4IFY 2.1 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.49 MG, 1FD, T27, DMS 24.305, 191.15, 366.419, 78.133
4IG0 2.5 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.49 1FG, DMS 362.425, 78.133
4IG3 1.95 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.49 T27, DMS, J94 366.419, 78.133, 382.387
4JLH 2.09 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.7 SO4, 0L9 ic50 = 15.6 uM 96.063, 420.684
4K4P 2.31 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 NO3, 3TL 62.005, 909.077
4K4R 1.8 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 27B, BR, NO3, 3TL, DMS 251.076, 79.904, 62.005, 909.077, 78.133
4KFB 1.85 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.49 T27, DMS, 1QP 366.419, 78.133, 190.199
4KO0 1.95 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.49 SO4, JLJ, EDO 96.063, 310.35, 62.068
4NX4 1.5 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 NON-ENZYME OTHER CL, ZN, JPR 35.453, 65.409, 381.92
4NYF 1.9 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.7 CD, 4BI Kd = 49 nM 112.411, 383.868
4O0J 2.05 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.7 LF8, SO4 ic50 = 13 uM 451.985, 96.063
4O55 2.24 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.7 SO4, LF9 ic50 = 5.03 uM 96.063, 463.956
4O5B 2.37 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.7 SO4, LF9 96.063, 463.956
4OBD 1.9 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 ARG PRO GLY ASN PHE PHE GLN ASN ARG PRO, EDO, GOL 851.919, 62.068, 92.094
4OBF 1.68 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 ACT, PO4, GOL, ARG PRO GLY ASN PHE LEU GLN ASN ARG PRO, EDO 59.044, 94.971, 92.094, 789.916, 62.068
4OBG 1.78 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 ARG PRO GLY ASN PHE LEU GLN SER ARG PRO, PO4, EDO, GOL 975.119, 94.971, 62.068, 92.094
4OBH 1.85 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 ACT, PO4, GOL, EDO, ARG PRO GLY ASN PHE PHE GLN SER ARG PRO 59.044, 94.971, 92.094, 62.068, 938.057
4OBJ 1.75 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 GOL, ARG PRO GLY ASN PHE LEU GLN ASN ARG PRO, ACT, EDO 92.094, 789.916, 59.044, 62.068
4OBK 1.65 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 ACT, EDO, ARG PRO GLY ASN PHE PHE GLN ASN ARG PRO, GOL 59.044, 62.068, 851.919, 92.094
4OJR 1.82 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.7 SO4, 2SQ, CAC 96.063, 453.503, 136.989
4Q5M 1.8 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 ROC 670.841
4QAG 1.71 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.1.26.4 F95, MN ic50 = 4.8 uM 236.178, 54.938
4ZIP 1.11 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 3.4.23.16 G64, GOL, NA, CL Ki = 0.21 nM 690.849, 92.094, 22.99, 35.453
5HGP 1.95 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 NON-ENZYME OTHER BHC 342.169
6UL5 2.23 HUMAN IMMUNODEFICIENCY VIRUS TYPE 1 ENZYME 2.7.7.49 QAG, MG, EDO, SO4 ic50 = 36.2 nM 441.48, 24.305, 62.068, 96.063
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