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6PJN | 1.98 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | OQP, SO4 | Ki = 7.3 nM | 609.71, 96.063 |
2F80 | 1.45 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | CL, 017, SO4 | Ki = 6.6 nM | 35.453, 547.664, 96.063 |
5IVS | 1.46 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 6EF, CL | ic50 = 6.1 nM | 650.763, 35.453 |
2AZ8 | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 3TL | ic50 = 6 nM | 909.077 |
1NPV | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | L27 | ic50 = 5.7 nM | 595.685 |
4L1A | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | AB1 | ic50 = 5.39 nM | 628.801 |
1B6L | 1.75 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, PI4 | Ki = 5 nM | 96.063, 545.671 |
2CEN | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 4AH | Ki = 5 nM | 679.804 |
2HS2 | 1.22 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | DMS, CL, 017 | Ki = 4.9 nM | 78.133, 35.453, 547.664 |
2FDD | 1.58 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 385 | ic50 = 4.8 nM | 703.823 |
1HWR | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 216 | Ki = 4.7 nM | 406.517 |
2QCI | 1.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 065, CL, ACT, NA | Ki = 4.6 nM | 576.658, 35.453, 59.044, 22.99 |
3NU5 | 1.29 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, CL, ACT, 478 | Ki = 4.5 nM | 22.99, 35.453, 59.044, 505.627 |
6DJ2 | 1.36 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | AB1, CL, NA | Ki = 4.5 nM | 628.801, 35.453, 22.99 |
4GZF | 2.05 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ILO VAL DC0 GLU ALA NLE | ic50 = 4.4 nM | 832.057 |
3ZPU | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | M8B, CL | Ki = 4.2 nM | 742.743, 35.453 |
1LZQ | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | BME, 0ZQ | Ki = 4.1 nM | 78.133, 687.825 |
1B6M | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, PI6 | Ki = 4 nM | 96.063, 596.757 |
1MTR | 1.75 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, PI6 | Ki = 4 nM | 96.063, 596.757 |
1ZPA | 2.02 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | A83 | Ki = 4 nM | 720.878 |
3OXC | 1.16 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, ROC, FMT | Ki = 3.9 nM | 96.063, 670.841, 46.025 |
1BWB | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 146 | Ki = 3.8 nM | 824.924 |
1HTG | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | G37 | ic50 = 3.8 nM | 761.931 |
3U7S | 2.05 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | BME, 017 | Ki = 3700 pM | 78.133, 547.664 |
5KQX | 2.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ROC | Ki = 3.6 nM | 670.841 |
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