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6PJE | 1.92 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | OPJ, SO4 | Ki = 46 nM | 609.71, 96.063 |
1XL5 | 1.73 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | CL, 190 | Ki = 45 nM | 35.453, 634.597 |
1K6P | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | XN3, ACT | Kd = 44 nM | 656.811, 59.044 |
2QI0 | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | MZ3, PO4 | Ki = 42 nM | 582.706, 94.971 |
3UCB | 1.38 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 017 | Kd = 41 nM | 547.664 |
2BPY | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 3IN | Ki = 39.8 nM | 727.336 |
2BPZ | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 3IN | Ki = 39.8 nM | 727.336 |
6VOD | 1.25 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, T1R, CL, GOL, FMT | ic50 = 38 nM | 22.99, 588.712, 35.453, 92.094, 46.025 |
2R38 | 1.81 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | G4G, CL | Ki = 0.036 uM | 647.764, 35.453 |
1IIQ | 1.83 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, 0ZR | Ki = 33 nM | 92.094, 702.84 |
1K6C | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | MK1, ACT | Kd = 33 nM | 613.789, 59.044 |
2QHY | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, MZ1, ACT | Ki = 33 nM | 94.971, 583.643, 59.044 |
6OTG | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, FMT, 4UY | Ki = 31.4 nM | 92.094, 46.025, 591.716 |
6OGT | 1.21 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | JDY, EDO, GOL | ic50 = 31 nM | 688.83, 62.068, 92.094 |
2AVS | 1.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACY, SO4, PO4, MK1, DMS | Ki = 27 nM | 60.052, 96.063, 94.971, 613.789, 78.133 |
2PYN | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 1UN | Kd = 27 nM | 567.782 |
6OGQ | 1.41 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | JDV, SO4, PEG, GOL | ic50 = 26 nM | 688.83, 96.063, 106.12, 92.094 |
1K6T | 2.25 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | XN1, ACT | Kd = 24 nM | 627.816, 59.044 |
2P3C | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACY, 3TL | Ki = 24 nM | 60.052, 909.077 |
2PSU | 1.93 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, MUU, ACT | Ki = 24 nM | 94.971, 517.638, 59.044 |
6NCJ | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | KJJ, SO4, EDO | ic50 = 0.024 uM | 572.709, 96.063, 62.068 |
6OPW | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | 017, SO4 | Ki = 23.2 nM | 547.664, 96.063 |
2AZ9 | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 3TL | ic50 = 22 nM | 909.077 |
6O5X | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | 0Q4, NA, CL | Ki = 22 nM | 833.053, 22.99, 35.453 |
2BPV | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 1IN | Ki = 21.2 nM | 621.81 |
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