1K6T | 2.25 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | XN1, ACT | Kd = 24 nM | 627.816, 59.044 |
1K6V | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | XN2, ACT | Kd = 120 nM | 670.837, 59.044 |
1KJ7 | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PRO ALA THR ILE MET MET GLN ARG GLY ASN, ACT | | 892.138, 59.044 |
1KJF | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ARG PRO GLY ASN PHE LEU GLN SER ARG PRO, ACT | | 975.119, 59.044 |
1KJG | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GLY ALA GLU THR PHE TYR VAL ASP GLY ALA, ACT | | 968.995, 59.044 |
1KJH | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ILE ARG LYS ILE LEU PHE LEU ASP GLY ILE, ACT | | 1146.42, 59.044 |
1LZQ | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | BME, 0ZQ | Ki = 4.1 nM | 78.133, 687.825 |
1M0B | 2.45 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, 0ZQ | Ki = 1.53 nM | 92.094, 687.825 |
1MER | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | DMQ | Ki = 10 nM | 536.664 |
1MES | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | DMP | Ki = 20 nM | 566.687 |
1MET | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | DMP | Ki = 0.4 nM | 566.687 |
1MEU | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | DMP | Ki = 0.8 uM | 566.687 |
1MRW | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | K57 | Kd = 0.2 nM | 527.675 |
1MRX | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | K57 | Kd = 55 nM | 527.675 |
1MSM | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | JE2 | Kd = 33 pM | 575.718 |
1MSN | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | JE2 | Kd < 1 nM | 575.718 |
1MT7 | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | VAL SER GLN ASN TYR PRO ILE VAL GLN ASN, ACT | | 904.056, 59.044 |
1MT8 | 2.15 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | LYS ALA ARG VAL LEU ALA GLU ALA MET SER, ACT | | 916.136, 59.044 |
1MT9 | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, ARG PRO GLY ASN PHE LEU GLN SER ARG PRO | | 94.971, 975.119 |
1MTB | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | QNC ASN HPH DIQ NTB | | 670.855 |
1MTR | 1.75 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, PI6 | Ki = 4 nM | 96.063, 596.757 |
1N49 | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | RIT | | 720.944 |
1NH0 | 1.03 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, KI2 PHE GLU GLU NH2, BME | Ki = 0.18 nM | 96.063, 732.767, 78.133 |
1NPA | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 3NH | ic50 = 2 nM | 629.743 |
1NPV | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | L27 | ic50 = 5.7 nM | 595.685 |
1NPW | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | LGZ | ic50 = 2 nM | 625.711 |
1ODW | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 0E8 | Ki = 100 nM | 543.695 |
1ODX | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 0E8 | | 543.695 |
1OHR | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 1UN | Ki = 2 nM | 567.782 |
1PRO | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | A88 | Ki = 5 pM | 583.674 |
1QBR | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | XV6 | Ki = 0.027 nM | 758.908 |
1QBS | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | DMP | Ki = 0.34 nM | 566.687 |
1QBT | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 146 | Ki = 0.024 nM | 824.924 |
1QBU | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 846 | Ki = 0.058 nM | 596.739 |
1RL8 | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | RIT | | 720.944 |
1SDT | 1.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | MK1, CL | Ki = 540 pM | 613.789, 35.453 |
1SDU | 1.25 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, MK1, ACT | Ki = 86 pM | 96.063, 613.789, 59.044 |
1SDV | 1.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | MK1, CL | Ki = 1810 pM | 613.789, 35.453 |
1SGU | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | MK1 | Ki = 4235 nM | 613.789 |
1SH9 | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | RIT | Ki = 932 nM | 720.944 |
1SP5 | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | TYR ASP GLN ILE LEU, DMS, CL, BME | | 649.722, 78.133, 35.453, 78.133 |
1T3R | 1.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, 017 | Ki = 14 pM | 94.971, 547.664 |
1T7I | 1.35 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, ACT, 017 | | 94.971, 59.044, 547.664 |
1T7J | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACT, 478 | Kd = 0.000000064 M | 59.044, 505.627 |
1T7K | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | BH0 | Ki = 1.37 nM | 598.669 |
1TCX | 2.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | IM1 | Ki = 112 nM | 534.69 |
1U8G | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | KI2 PHE GLU GLU NH2 | | 732.767 |
1UPJ | 2.22 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | U01 | | 373.24 |
1VIJ | 2.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | BAY | ic50 = 0.3 nM | 1131.49 |
1VIK | 2.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | BAY | ic50 = 0.3 nM | 1131.49 |