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4DJO | 1.78 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, MK5, GOL, ACT | Ki = 0.003 nM | 94.971, 618.57, 92.094, 59.044 |
4DJQ | 1.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, M86 | Ki = 0.048 nM | 94.971, 576.705 |
4DJP | 1.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, M73 | Ki = 0.028 nM | 94.971, 564.691 |
3GI5 | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, K62 | Ki = 0.006 nM | 94.971, 651.727 |
3GI4 | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, K60, ACT | Ki = 0.016 nM | 94.971, 677.688, 59.044 |
3S53 | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, IOD, 017 | Ki = 0.23 nM | 94.971, 126.904, 547.664 |
2QD7 | 1.11 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, GOL, DMS, 065 | Ki = 0.8 nM | 94.971, 92.094, 78.133, 576.658 |
4DQC | 1.94 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, GOL, 017 | 94.971, 92.094, 547.664 | |
4DQB | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, EDO, DMS, 017 | 94.971, 62.068, 78.133, 547.664 | |
3GI6 | 1.84 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, D78 | Ki = 0.006 nM | 94.971, 663.704 |
1MT9 | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, ARG PRO GLY ASN PHE LEU GLN SER ARG PRO | 94.971, 975.119 | |
2FNT | 1.44 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, ARG GLN VAL ASN PHE LEU GLY LYS ILE ASN, ACT | 94.971, 675.808, 59.044 | |
2FNS | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, ARG GLN ALA ASN PHE LEU GLY LYS ILE ASN, ACT | 94.971, 647.754, 59.044 | |
1T7I | 1.35 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, ACT, 017 | 94.971, 59.044, 547.664 | |
2Q5K | 1.95 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, AB1 | Ki = 0.005 nM | 94.971, 628.801 |
3R4B | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, 74T | 94.971, 755.987 | |
4Q1X | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, 017, GOL | Ki = 7 pM | 94.971, 547.664, 92.094 |
1T3R | 1.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, 017 | Ki = 14 pM | 94.971, 547.664 |
1HOS | 2.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PHP | Ki = 2.8 nM | 770.85 |
3OU4 | 1.6 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | PHE ASN PHE PRO GLN ILE THR | 865.986 | |
6UM8 | 2.33 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | PEG, 1PE, SO4, QCG | Ki = 0.17 uM | 106.12, 238.278, 96.063, 503.565 |
6PU8 | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | P3V | 563.663 | |
6PJG | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ORV | Ki = 0.019 nM | 569.646 |
6PJM | 1.93 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | OQV, SO4 | Ki = 0.013 nM | 611.726, 96.063 |
6PJN | 1.98 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | OQP, SO4 | Ki = 7.3 nM | 609.71, 96.063 |
6PJK | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | OQD, SO4 | Ki = 0.055 nM | 611.726, 96.063 |
6PJO | 1.95 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | OQ7, SO4 | Ki = 0.161 nM | 623.736, 96.063 |
6PJE | 1.92 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | OPJ, SO4 | Ki = 46 nM | 609.71, 96.063 |
6PJF | 1.94 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | OP7, SO4 | Ki = 0.235 nM | 623.736, 96.063 |
6PJI | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | OO4, SO4 | Ki = 0.571 nM | 595.683, 96.063 |
4CHN | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | ONZ, ACT, EDO, GOL, SO4 | 223.182, 59.044, 62.068, 92.094, 96.063 | |
4CK1 | 1.75 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | OM1, CL, EDO, ACT, SO4 | 449.476, 35.453, 62.068, 59.044, 96.063 | |
4CF0 | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | O5U, ACT, SO4 | 510.579, 59.044, 96.063 | |
4CEZ | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | O3N, CL, SO4, GOL | 550.643, 35.453, 96.063, 92.094 | |
4CE9 | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | O3N, ACY, SO4, GOL | 550.643, 60.052, 96.063, 92.094 | |
2PK6 | 1.45 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | O33, GOL | Kd = 13 pM | 771.945, 92.094 |
4CGI | 2.07 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | NZL, ACT, SO4 | Kd = 752 uM | 424.49, 59.044, 96.063 |
4CGJ | 2.15 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | NZL, ACT, SO4 | 424.49, 59.044, 96.063 | |
4CK2 | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | NVU, SO4, ACT | 177.157, 96.063, 59.044 | |
1VRT | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.49 | NVP, MG | ic50 = 0.08 uM | 266.298, 24.305 |
1AJV | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NMB | Ki = 19.1 nM | 574.687 |
1G2K | 1.95 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NM1 | Ki = 11 nM | 631.738 |
6OYD | 1.46 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NKA | ic50 = 0.12 nM | 674.78 |
6OYR | 1.54 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NJY | ic50 = 0.29 nM | 674.78 |
6OXO | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NJM, SO4 | 562.675, 96.063 | |
6OY2 | 1.99 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NJJ, SO4 | 620.754, 96.063 | |
6OXZ | 1.96 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NJG, SO4 | 606.727, 96.063 | |
6OXR | 2.04 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NJA | 576.701 | |
6OY0 | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NJ7, SO4 | 606.727, 96.063 | |
6OXS | 1.99 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NJ4 | 576.701 |
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