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1YTH | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACE SER LEU ASN PHE | 520.563 | |
1ZJ7 | 1.93 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 0ZT | Ki = 86 nM | 703.824 |
1ZLF | 2.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 0ZR | Ki = 1000 nM | 702.84 |
1ZP8 | 2.02 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | AB2 | Ki = 1.7 nM | 663.784 |
1ZPA | 2.02 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | A83 | Ki = 4 nM | 720.878 |
1ZSF | 1.98 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 0ZS | Ki = 0.12 nM | 703.824 |
1ZSR | 2.06 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 0ZT | Ki = 0.15 nM | 703.824 |
1ZTZ | 2.15 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | CB5, ALA GLY ALA ALA | Ki = 66 nM | 323.749, 273.313 |
2A1E | 1.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, IPF, GOL, DMS, CL, ACT | 22.99, 905.092, 92.094, 78.133, 35.453, 59.044 | |
2A4F | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | AAU | 641.71 | |
2AID | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | THK, CL | Ki = 15 uM | 452.048, 35.453 |
2AQU | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | DR7 | Ki = 0.48 nM | 704.855 |
2AVM | 1.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, ACY, 2NC | Ki = 2 uM | 92.094, 60.052, 770.983 |
2AVO | 1.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, MK1, GOL, DMS, ACY | Ki = 1.4 nM | 96.063, 613.789, 92.094, 78.133, 60.052 |
2AVS | 1.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, PO4, MK1, DMS, ACY | Ki = 27 nM | 96.063, 94.971, 613.789, 78.133, 60.052 |
2AVV | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | MK1, CL, ACY | Ki = 0.55 nM | 613.789, 35.453, 60.052 |
2AZ8 | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 3TL | ic50 = 6 nM | 909.077 |
2AZ9 | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 3TL | ic50 = 22 nM | 909.077 |
2AZB | 2.03 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 3TL | ic50 = 64 nM | 909.077 |
2AZC | 2.01 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 3TL | ic50 = 183 nM | 909.077 |
2BB9 | 1.35 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | AKC | ic50 = 0.44 nM | 625.711 |
2BBB | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | HH1 | ic50 = 2.4 nM | 623.738 |
2BE2 | 2.43 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.49 | GLC FRU, R22, MN, GOL | ic50 = 0.002 uM | 340.281, 481.347, 54.938, 92.094 |
2BPV | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 1IN | Ki = 21.2 nM | 621.81 |
2BPY | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 3IN | Ki = 39.8 nM | 727.336 |
2BPZ | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 3IN | Ki = 39.8 nM | 727.336 |
2BQV | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | A1A | Ki = 9 nM | 588.694 |
2CEJ | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 1AH | Ki = 2.4 nM | 681.617 |
2CEM | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 2AH | Ki = 12 nM | 679.804 |
2CEN | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 4AH | Ki = 5 nM | 679.804 |
2F3K | 1.6 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | RO1, PO4 | Kd = 0.95 nM | 711.911, 94.971 |
2F80 | 1.45 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, CL, 017 | Ki = 6.6 nM | 96.063, 35.453, 547.664 |
2F81 | 1.25 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, GOL, CL, 017 | Ki = 0.03 nM | 22.99, 92.094, 35.453, 547.664 |
2F8G | 1.22 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, GOL, CL, ACY, 017 | Ki = 2 nM | 22.99, 92.094, 35.453, 60.052, 547.664 |
2FDD | 1.58 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 385 | ic50 = 4.8 nM | 703.823 |
2FGU | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | QNC ASN HPH DIQ NTB, PO4 | Kd = 0.66 nM | 670.855, 94.971 |
2FGV | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | QNC ASN HPH DIQ NTB, PO4 | Kd = 760 nM | 670.855, 94.971 |
2FLE | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, AI | Ki = 14 nM | 92.094, 801.029 |
2FNS | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, ARG GLN ALA ASN PHE LEU GLY LYS ILE ASN, ACT | 94.971, 647.754, 59.044 | |
2FNT | 1.44 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, ARG GLN VAL ASN PHE LEU GLY LYS ILE ASN, ACT | 94.971, 675.808, 59.044 | |
2FXD | 1.6 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, DR7, ACT | ic50 = 12 nM | 96.063, 704.855, 59.044 |
2FXE | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, GOL, DR7, ACT | 96.063, 92.094, 704.855, 59.044 | |
2HB3 | 1.35 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, GRL, GOL, CL | Ki = 0.0045 nM | 22.99, 560.702, 92.094, 35.453 |
2HND | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.49 | PO4, NVP, MG | 94.971, 266.298, 24.305 | |
2HNY | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.49 | PO4, NVP, MG | ic50 = 1165 nM | 94.971, 266.298, 24.305 |
2HS1 | 0.84 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | DMS, CL, 017 | Ki = 3.3 nM | 78.133, 35.453, 547.664 |
2HS2 | 1.22 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | DMS, CL, 017 | Ki = 4.9 nM | 78.133, 35.453, 547.664 |
2I0A | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, MUI, GOL | Ki = 0.004 nM | 94.971, 637.743, 92.094 |
2I0D | 1.95 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, MUT, ACT | Ki = 0.0008 nM | 94.971, 637.743, 59.044 |
2I4D | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | QFI | Ki = 2.1 pM | 672.681 |
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