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1GNM | 2.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | U0E | Ki = 560 nM | 596.762 |
6O57 | 1.71 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | 2NC, FMT | Ki = 514 nM | 770.983, 46.025 |
6O5A | 1.67 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | GOL, 2NC | Ki = 514 nM | 92.094, 770.983 |
2ZGA | 1.65 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | YDP | Ki = 0.48 uM | 603.753 |
3CKT | 1.65 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | YDP, CL | Ki = 0.48 uM | 603.753, 35.453 |
6EB2 | 2.49 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | J3P | ic50 = 0.48 uM | 547.644 |
1BDQ | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | IM1 | Ki = 460 nM | 534.69 |
1HBV | 2.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GAN | Ki = 430 nM | 585.778 |
1RTH | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.49 | U05 | ic50 = 0.4 uM | 298.297 |
2QNP | 1.41 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | QN2, CL | Ki = 0.39 uM | 813.508, 35.453 |
3BVB | 1.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, GOL, CL, 017 | Ka = 3170000 M^-1 | 22.99, 92.094, 35.453, 547.664 |
3BVA | 1.05 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, 2NC | Ka = 3300000 M^-1 | 92.094, 770.983 |
2PWC | 1.78 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, G3G, CL | Ki = 0.27 uM | 92.094, 591.744, 35.453 |
4RZ8 | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | NON-ENZYME OTHER | EPE, NAG, 3ZM | ic50 ~ 270 nM | 238.305, 221.208, 444.978 |
2PWR | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, G4G, CL | Ki = 0.26 uM | 92.094, 647.764, 35.453 |
4EYR | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | RIT | ic50 = 237 nM | 720.944 |
4XRQ | 1.95 | HUMAN IMMUNODEFICIENCY VIRUS 1 | NON-ENZYME OTHER | 1B0 | Kd = 0.232 uM | 425.522 |
4LH5 | 2.19 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | LF0, MG | ic50 = 0.23 uM | 405.486, 24.305 |
5OI8 | 2.35 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | 9VN, SO4, MG | ic50 = 0.21 uM | 413.573, 96.063, 24.305 |
5OI5 | 2.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | MG, 9VK | ic50 = 0.19 uM | 24.305, 413.573 |
2AZC | 2.01 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 3TL | ic50 = 183 nM | 909.077 |
4J5J | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 478, CL | Ka = 5610000 M^-1 | 505.627, 35.453 |
6OPX | 2.03 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | 017 | Ki = 172.7 nM | 547.664 |
5OI2 | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | SO4, 9VN, MG | ic50 = 0.17 uM | 96.063, 413.573, 24.305 |
5OIA | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | 9VK, SO4, MG | ic50 = 0.17 uM | 413.573, 96.063, 24.305 |
6UM8 | 2.33 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | PEG, 1PE, SO4, QCG | Ki = 0.17 uM | 106.12, 238.278, 96.063, 503.565 |
6OPY | 2.13 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | 017 | Ki = 156.4 nM | 547.664 |
2PYM | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 1UN | Kd = 150 nM | 567.782 |
1HTF | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | G26 | ic50 = 148 nM | 574.734 |
3AID | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ARQ | Ki = 137 nM | 504.64 |
2R3W | 1.92 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | G3G, CL | Ki = 0.128 uM | 591.744, 35.453 |
1K6V | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | XN2, ACT | Kd = 120 nM | 670.837, 59.044 |
2UY0 | 1.76 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | HV1 | Ki = 120 nM | 723.653 |
1A9M | 2.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | U0E | Ki = 119 nM | 596.762 |
1TCX | 2.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | IM1 | Ki = 112 nM | 534.69 |
1ODW | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 0E8 | Ki = 100 nM | 543.695 |
1VRU | 2.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.49 | AAP | ic50 = 0.1 uM | 351.227 |
1ZJ7 | 1.93 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 0ZT | Ki = 86 nM | 703.824 |
1VRT | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.49 | NVP, MG | ic50 = 0.08 uM | 266.298, 24.305 |
6O48 | 1.46 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | FMT, GOL, 0Q4, NA, CL | Ki = 75 nM | 46.025, 92.094, 833.053, 22.99, 35.453 |
2QNN | 1.48 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | QN1, GOL, CL | Ki = 0.07 uM | 783.76, 92.094, 35.453 |
1ZTZ | 2.15 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | CB5, ALA GLY ALA ALA | Ki = 66 nM | 323.749, 273.313 |
2Q63 | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 1UN | Kd = 66 nM | 567.782 |
1T7J | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACT, 478 | Kd = 0.000000064 M | 59.044, 505.627 |
2AZB | 2.03 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 3TL | ic50 = 64 nM | 909.077 |
2PSV | 1.75 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | MUV, ACT, PO4 | Ki = 58 nM | 477.574, 59.044, 94.971 |
1MRX | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | K57 | Kd = 55 nM | 527.675 |
6OGP | 1.53 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | EDO, MJD | ic50 = 0.055 uM | 62.068, 692.77 |
2QHZ | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, MZ2 | Ki = 53 nM | 94.971, 606.6 |
2QI1 | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, MZ4 | Ki = 50 nM | 94.971, 582.688 |
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