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4TSX | 1.94 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | SO4, LF0 | Kd = 10.3 uM | 96.063, 405.486 |
6VLM | 2.32 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | R2D | ic50 = 10 uM | 342.799 |
4EJL | 2.45 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | IOP, DMS, GOL, PEG | Kd = 7.2 uM | 189.211, 78.133, 92.094, 106.12 |
4EJK | 1.79 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | IOP, IVA VAL VAL STA ALA STA | Kd = 5.3 uM | 189.211, 696.992 |
6EB1 | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | J3M | ic50 = 4.65 uM | 467.556 |
1SGU | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | MK1 | Ki = 4235 nM | 613.789 |
4EJ8 | 2.35 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | EDO, 1F1, DMS | Kd = 4.1 uM | 62.068, 161.157, 78.133 |
2XDE | 1.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | NON-ENZYME OTHER | 1B0 | Kd = 3.42 uM | 425.522 |
4U7V | 1.38 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | BME, 3EN | Ki = 3.2 uM | 78.133, 524.675 |
1QS4 | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | MG, 100 | ic50 = 2.3 uM | 24.305, 289.677 |
2PQZ | 1.55 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | G0G, CL | Ki = 2.15 uM | 561.715, 35.453 |
1GNN | 2.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | U0E | Ki = 2100 nM | 596.762 |
2AVM | 1.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, ACY, 2NC | Ki = 2 uM | 92.094, 60.052, 770.983 |
1XL2 | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, CL, 189 | Ki = 1.5 uM | 92.094, 35.453, 577.777 |
2R3T | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | G4G, CL | Ki = 1.4 uM | 647.764, 35.453 |
2HNY | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.49 | PO4, NVP, MG | ic50 = 1165 nM | 94.971, 266.298, 24.305 |
1ZLF | 2.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 0ZR | Ki = 1000 nM | 702.84 |
2R43 | 1.58 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, G3G, CL | Ki = 1 uM | 92.094, 591.744, 35.453 |
1SH9 | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | RIT | Ki = 932 nM | 720.944 |
4INB | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | NON-ENZYME OTHER | NA, 1F6 | ic50 = 0.89 uM | 22.99, 419.397 |
1MEU | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | DMP | Ki = 0.8 uM | 566.687 |
4HVP | 2.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 2NC | Ki = 0.78 uM | 770.983 |
2QNQ | 2.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | QN3, CL | Ki = 0.77 uM | 630.605, 35.453 |
2FGV | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | QNC ASN HPH DIQ NTB, PO4 | Kd = 760 nM | 670.855, 94.971 |
6OPZ | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | 017 | Ki = 759.2 nM | 547.664 |
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